Brief Information of the Cell Line and Protein
Cell Line ID: CL000063 , Hep-G2
Synonyms
HEP-G2
Hep G2
HEP G2
HepG2
HEPG2
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0027
Protein ID: PT06172 , Mothers against decapentaplegic homolog 3
Gene Name SMAD3
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P84022
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000063  Protein ID: PT06172
 
Compound ID Compound Name Compound Formula
CP0416037
MLS002703014
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C24H34O9
 1
1
Potency ~ 4.1 nM
   TI
   LI
   LO
   TS
CP0888980
SID92763369
   Show/Hide
C11H13N3O4S
 1
1
Potency ~ 16.4 nM
   TI
   LI
   LO
   TS
CP0851790
SID14719315
   Show/Hide
C12H17N5O6
 1
1
Potency ~ 18.4 nM
   TI
   LI
   LO
   TS
CP0433892
4-[2-(3,5-dimethyl-5-oxidanyl-2-oxidanylidene-cyclohexyl)-2-oxidanyl-ethyl]piperidine-2,6-dione
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C15H23NO5
 1
1
Potency ~ 20.6 nM
   TI
   LI
   LO
   TS
CP0905782
SID92763404
   Show/Hide
C12H13N5O4
 1
1
Potency ~ 25.9 nM
   TI
   LI
   LO
   TS
CP0884597
SID56422424
   Show/Hide
C29H43ClN2O5
 1
1
Potency ~ 32.6 nM
   TI
   LI
   LO
   TS
CP0411307
4-amino-7-(3,4-dihydroxy-5-methylol-tetrahydrofuran-2-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide;hydrate
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C12H15N5O5
 1
1
Potency ~ 36.6 nM
   TI
   LI
   LO
   TS
CP0846860
SID92763334
   Show/Hide
C16H24O4
 1
1
Potency ~ 73.1 nM
   TI
   LI
   LO
   TS
CP0853620
SID92763371
   Show/Hide
C22H24N2O8S
 1
1
Potency ~ 82 nM
   TI
   LI
   LO
   TS
CP0378346
(2E,10E)-12,15-dihydroxy-7-methyl-8-oxabicyclo[11.3.0]hexadeca-2,10-dien-9-one
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C16H24O4
 1
1
Potency ~ 103.2 nM
   TI
   LI
   LO
   TS
CP0438388
1,2,3,4,7-pentahydroxy-2,3,4,4a,5,11b-hexahydro-1H-[1,3]dioxolo[4,5-j]phenanthridin-6-one
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C14H15NO8
 1
1
Potency ~ 103.2 nM
   TI
   LI
   LO
   TS
CP0064739
2-(6-AMINO-2-FLUORO-PURIN-9-YL)-5-HYDROXYMETHYL-TETRAHYDRO-FURAN-3,4-DIOL
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C10H12FN5O4
 1
1
Potency ~ 115.8 nM
   TI
   LI
   LO
   TS
CP0079091
Anisomycin from Streptomyces griseolus
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C14H19NO4
 1
1
Potency ~ 145.8 nM
   TI
   LI
   LO
   TS
CP0061146
(2R,3S,4S,5R)-2-(6-amino-2-fluoro-9-purinyl)-5-(hydroxymethyl)oxolane-3,4-diol
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C10H12FN5O4
 1
1
Potency ~ 183.6 nM
   TI
   LI
   LO
   TS
CP0921060
SID92763413
   Show/Hide
C25H34O10
 1
1
Potency ~ 206 nM
   TI
   LI
   LO
   TS
CP0921168
SID99355952
   Show/Hide
C14H10Br2N2O2
 1
1
Potency ~ 206 nM
   TI
   LI
   LO
   TS
CP0664710
SID49681823
   Show/Hide
C27H30ClNO11
 1
1
Potency ~ 326.4 nM
   TI
   LI
   LO
   TS
CP0856702
SID93577483
   Show/Hide
C11H14N4O5
 1
1
Potency ~ 326.4 nM
   TI
   LI
   LO
   TS
CP0081887
4-((1R,3S,5S,8R,10R,11R,13R,14S,17R)-1,5,11,14-tetrahydroxy-10-(hydroxymethyl)-13-methyl-3-((2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyl-tetrahydro-2H-pyran-2-yloxy)-hexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)furan-2(5H)-one
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C29H44O12
 1
1
Potency ~ 366.3 nM
   TI
   LI
   LO
   TS
CP0900419
SID89850929
   Show/Hide
C24H29NO6
 1
1
Potency ~ 410.9 nM
   TI
   LI
   LO
   TS
CP0908037
SID56463667
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C16H18ClNO4
 1
1
Potency ~ 410.9 nM
   TI
   LI
   LO
   TS
CP0103674
(S)-10-Amino-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione
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C20H17N3O4
 1
1
Potency ~ 461.1 nM
   TI
   LI
   LO
   TS
CP0888629
SID92763894
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C13H18N4O4
 1
1
Potency ~ 461.1 nM
   TI
   LI
   LO
   TS
CP0914548
SID92764800
   Show/Hide
C24H25ClN4O5
 1
1
Potency ~ 461.1 nM
   TI
   LI
   LO
   TS
CP0961461
SID93577122
   Show/Hide
C13H9BrN2O
 1
1
Potency ~ 517.4 nM
   TI
   LI
   LO
   TS
CP0649513
SID50086453
   Show/Hide
C11H10BrClN2OS
 1
1
Potency ~ 580.5 nM
   TI
   LI
   LO
   TS
CP0849486
SID92763868
   Show/Hide
C28H28O9
 1
1
Potency ~ 580.5 nM
   TI
   LI
   LO
   TS
CP0883527
SID85272968
   Show/Hide
C52H84N8O12
 1
1
Potency ~ 651.3 nM
   TI
   LI
   LO
   TS
CP0732771
SID24781162
   Show/Hide
C14H10N6O3
 1
1
Potency ~ 730.8 nM
   TI
   LI
   LO
   TS
CP0695950
SID17517432
   Show/Hide
C12H13BrN2OS
 1
1
Potency ~ 819.9 nM
   TI
   LI
   LO
   TS
CP0832055
SID49823646
   Show/Hide
C23H19FN4O
 1
1
Potency ~ 819.9 nM
   TI
   LI
   LO
   TS
CP0893353
SID49731728
   Show/Hide
C19H18N2O3S
 1
1
Potency ~ 819.9 nM
   TI
   LI
   LO
   TS
CP0921312
SID103050197
   Show/Hide
C20H19N5S
 1
1
Potency ~ 819.9 nM
   TI
   LI
   LO
   TS
CP0647880
SID24837215
   Show/Hide
C20H14N2O4S2
 1
1
Potency ~ 1032.3 nM
   TI
   LI
   LO
   TS
CP0342820
2-Chloro-N-[2,2,2-trifluoro-1-(6-nitro-benzothiazol-2-ylamino)-1-trifluoromethyl-ethyl]-benzamide
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C17H9ClF6N4O3S
 1
1
Potency ~ 1158.2 nM
   TI
   LI
   LO
   TS
CP0382380
3-(4-hydroxyphenyl)-2-[(E)-2-(5-nitro-2-furanyl)ethenyl]-4-quinazolinone
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C20H13N3O5
 1
1
Potency ~ 1158.2 nM
   TI
   LI
   LO
   TS
CP0912873
SID99494713
   Show/Hide
C23H20N4O4S
 1
1
Potency ~ 1299.5 nM
   TI
   LI
   LO
   TS
CP0956783
SID17511441
   Show/Hide
C19H18ClN3O2
 1
1
Potency ~ 1299.5 nM
   TI
   LI
   LO
   TS
CP0838198
SID49824120
   Show/Hide
C22H14F5N3O5
 1
1
Potency ~ 1458.1 nM
   TI
   LI
   LO
   TS
CP0907963
SID92764525
   Show/Hide
C17H19N5O5
 1
1
Potency ~ 1458.1 nM
   TI
   LI
   LO
   TS
CP0101250
2-[5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-yl]-2-(3-chlorophenyl)acetonitrile
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C18H8ClF6N3
 1
1
Potency ~ 1636 nM
   TI
   LI
   LO
   TS
CP0873847
SID92763435
   Show/Hide
C29H49N7O5
 1
1
Potency ~ 1636 nM
   TI
   LI
   LO
   TS
CP0967364
SID24813603
   Show/Hide
C18H14N2O4
 1
1
Potency ~ 1636 nM
   TI
   LI
   LO
   TS
CP0912442
SID121285141
   Show/Hide
C51H82N8O12
 1
1
Potency ~ 1835.6 nM
   TI
   LI
   LO
   TS
CP0961320
SID49641120
   Show/Hide
C17H14FNO
 1
1
Potency ~ 1835.6 nM
   TI
   LI
   LO
   TS
CP0110873
(3E,5E)-3,5-bis(3,4,5-trimethoxybenzylidene)tetrahydropyran-4-one
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C25H28O8
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0176736
4,9-diketo-2-methyl-N-p-anisyl-benzo[f]benzofuran-3-carboxamide
   Show/Hide
C22H17NO5
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0316762
3-(9-acridinylamino)-1-propanol
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C16H16N2O
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0330165
1-(2,3-Dihydro-indol-1-yl)-2-[5-(quinolin-8-yloxymethyl)-[1,3,4]oxadiazol-2-ylsulfanyl]-ethanone
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C22H18N4O3S
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0685484
SID49667054
   Show/Hide
C13H11ClN4
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0860634
SID92763810
   Show/Hide
C23H34O4
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0867358
5-(hydroxymethyl)quinolin-8-ol
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C10H9NO2
 1
1
Potency ~ 2059.6 nM
   TI
   LI
   LO
   TS
CP0646631
SID14732208
   Show/Hide
C24H27N3O5S
 1
1
Potency ~ 2310.9 nM
   TI
   LI
   LO
   TS
CP0735944
SID17514054
   Show/Hide
C19H18O2
 1
1
Potency ~ 2310.9 nM
   TI
   LI
   LO
   TS
CP0861454
PEUCEDANIN
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C15H14O4
 1
1
Potency ~ 2310.9 nM
   TI
   LI
   LO
   TS
CP0912483
SID103051216
   Show/Hide
C20H23N5OS
 1
1
Potency ~ 2310.9 nM
   TI
   LI
   LO
   TS
CP0230507
3-Methyl-1-(3-nitro-phenylamino)-benzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile
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C19H13N5O2
 1
1
Potency ~ 2592.9 nM
   TI
   LI
   LO
   TS
CP0846632
SID92763326
   Show/Hide
C14H16N8O6S
 1
1
Potency ~ 2592.9 nM
   TI
   LI
   LO
   TS
CP0851436
SID92763407
   Show/Hide
C23H33NO6
 1
1
Potency ~ 2592.9 nM
   TI
   LI
   LO
   TS
CP0885671
SID92763409
   Show/Hide
C12H14BrN5O5
 1
1
Potency ~ 2592.9 nM
   TI
   LI
   LO
   TS
CP0888384
SID14722899
   Show/Hide
C17H13ClN6O3
 1
1
Potency ~ 2592.9 nM
   TI
   LI
   LO
   TS
CP0232948
2-[(4-methoxy-6-methyl-2-quinazolinyl)amino]-1H-quinazolin-4-one
   Show/Hide
C18H15N5O2
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0336974
MLS000591280
   Show/Hide
C16H9F6N5O3S
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0450693
MLS001249435
   Show/Hide
C15H10ClI2NO3
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0668204
SID49727208
   Show/Hide
C13H9N3O4S
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0874727
SID92764840
   Show/Hide
C19H22ClN3O2
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0908502
SID47199821
   Show/Hide
C15H10FNO
 1
1
Potency ~ 2909.3 nM
   TI
   LI
   LO
   TS
CP0125193
2-[(3,4-difluorophenyl)sulfonylamino]-N-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]benzamide
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C23H17F2N3O4S2
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0370047
MLS000563453
   Show/Hide
C19H24O7
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0728030
SID26666845
   Show/Hide
C19H12Cl2N4O4
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0826479
SID49735130
   Show/Hide
C20H27N9O3
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0852866
SID49648722
   Show/Hide
C27H41NO5
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0876247
SID49716130
   Show/Hide
C23H18N2O5S
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0881324
SID87235992
   Show/Hide
C22H22F3N3O5
 1
1
Potency ~ 3264.3 nM
   TI
   LI
   LO
   TS
CP0024184
3-nitro-N-[3-(3-piperidin-1-ylsulfonylanilino)quinoxalin-2-yl]benzenesulfonamide
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C25H24N6O6S2
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0043376
3-(phenylcarbonyl)-2-(trifluoromethyl)benzo[f][1]benzofuran-4,9-dione
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C20H9F3O4
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0222600
5-nitro-2-(4-pyrimidinylthio)thiazole
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C7H4N4O2S2
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0667245
4-amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-7H-pyrrolo[2,3-d]pyrimidine-5-carbothioamide
   Show/Hide
C12H15N5O4S
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0721224
SID24827835
   Show/Hide
C16H11NO4
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0728848
SID17512572
   Show/Hide
C24H20N2O4
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0871668
SID50107430
   Show/Hide
C15H17N5O5
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0877012
SID103159016
   Show/Hide
C23H28N4S
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0884469
SID49823714
   Show/Hide
C16H11ClN4O2S2
 1
1
Potency ~ 3662.6 nM
   TI
   LI
   LO
   TS
CP0064538
6,8-bis(bromanyl)-4-piperidin-1-yl-quinazoline
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C13H13Br2N3
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0301198
MLS001077534
   Show/Hide
C22H29N3O3S
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0423819
1-[(3-ethyl-9,10-dimethoxy-2,3,4,6,7,11b-hexahydro-1H-benzo[a]quinolizin-2-yl)methyl]-2,3,4,9-tetrahydro-1H-beta-carbolin-6-ol
   Show/Hide
C29H37N3O3
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0647944
DNDI1417941
   Show/Hide
C20H14N2O3S2
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0667433
SID24823947
   Show/Hide
C15H12N2O4S
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0732354
SID49670187
   Show/Hide
C24H29IN2O
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0788846
SID24822421
   Show/Hide
C13H9N3O6S
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0867359
SID92763751
   Show/Hide
C18H12N2O2
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0882090
SID85199724
   Show/Hide
C23H18N2O4S
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0904013
SID17508788
   Show/Hide
C21H17ClN4O2S
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0924105
MMV1164554
   Show/Hide
C16H8ClF3N4
 1
1
Potency ~ 4109.5 nM
   TI
   LI
   LO
   TS
CP0134143
6-amino-7-bromo-quinoline-5,8-quinone
   Show/Hide
C9H5BrN2O2
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0210430
3-(7-Chloro-4-nitro-benzo[1,2,5]oxadiazol-5-ylamino)-phenol
   Show/Hide
C12H7ClN4O4
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0297612
4-[(7-chloranyl-4-nitro-1,3-dihydro-2,1,3-benzoxadiazol-5-yl)imino]cyclohexa-2,5-dien-1-one
   Show/Hide
C12H7ClN4O4
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0450711
(phenylmethyl) N-[4-[phenylmethoxycarbonyl-[3-[(phenylmethyl)amino]propyl]amino]butyl]-N-[3-[(phenylmethyl)amino]propyl]carbamate
   Show/Hide
C40H50N4O4
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0837136
SID24805492
   Show/Hide
C14H16N4O
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0846007
SID56323601
   Show/Hide
C15H15N3O6S2
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0850014
SID103060936
   Show/Hide
C31H32FN3O3
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0879219
SID92764022
   Show/Hide
C27H34N2O2
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0881126
SID92764784
   Show/Hide
C18H22BrClN2O6
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0885641
SID56463219
   Show/Hide
C22H30ClN7O5
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0886494
SID92763760
   Show/Hide
C13H10N2O2S
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0913432
SID103060880
   Show/Hide
C22H19N3O4S
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0942601
SID121286569
   Show/Hide
C18H18O4
 1
1
Potency ~ 4610.9 nM
   TI
   LI
   LO
   TS
CP0073975
2-(4-methylphenyl)sulfonyl-5-nitro-pyridine
   Show/Hide
C12H10N2O4S
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0163189
(7-Chloro-4-nitro-benzo[1,2,5]oxadiazol-5-yl)-pyridin-2-yl-amine
   Show/Hide
C11H6ClN5O3
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0201622
(4S)-1-[(1S)-1-benzyl-2-[(2R)-2-[[(5S)-5-(4-hydroxybenzyl)-2-thioxo-imidazolidin-1-yl]methyl]pyrrolidino]ethyl]-4-(4-hydroxybenzyl)-3-phenethyl-imidazolidine-2-thione
   Show/Hide
C42H49N5O2S2
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0209442
6-(1H-Benzoimidazol-2-ylsulfanylmethyl)-2-(4-methyl-quinazolin-2-ylamino)-pyrimidin-4-ol
   Show/Hide
C21H17N7OS
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0307648
(Z)-2-(1,3-benzothiazol-2-yl)-N-(4-chlorophenyl)-3-(3-hydroxyphenyl)-2-propenamide
   Show/Hide
C22H15ClN2O2S
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0448780
2-N,2-N-dimethyl-6-[(1-naphthalen-1-yltetrazol-5-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine
   Show/Hide
C17H17N9S
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0640109
SID24822906
   Show/Hide
C22H17N3O4S2
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0673712
SID144204738
   Show/Hide
C13H13ClN2O
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0688004
SID92764049
   Show/Hide
C14H16N8O5S
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0766081
SID22415655
   Show/Hide
C16H11ClFNO
 1
1
Potency ~ 5173.5 nM
   TI
   LI
   LO
   TS
CP0044759
3-Hydroxy-naphthalene-2-carboxylic acid (3-nitro-phenyl)-amide
   Show/Hide
C17H12N2O4
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0152322
2-amino-1-[3-(2-furoyloxy)propyl]pyrrolo[3,2-b]quinoxaline-3-carboxylic acid ethyl ester
   Show/Hide
C21H20N4O5
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0233022
1-(4,9-diketo-2-methyl-benzo[f]benzofuran-3-carbonyl)isonipecotic acid ethyl ester
   Show/Hide
C22H21NO6
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0432819
1-[3,5-bis(2,2,2-trifluoroethoxy)phenyl]-3-(4-fluorophenyl)urea
   Show/Hide
C17H13F7N2O3
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0793949
SID22408051
   Show/Hide
C27H22N2O3S
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0864511
MMV1507428
   Show/Hide
C17H10ClF3N4O2S
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0911188
SID51090672
   Show/Hide
C17H20ClN3O6S
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0914832
Dolastatin 12
   Show/Hide
C50H80N8O11
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0914840
SID92764783
   Show/Hide
C16H18Cl2N2O5
 1
1
Potency ~ 5804.8 nM
   TI
   LI
   LO
   TS
CP0001360
(Z)-2-(6-methyl-1H-benzimidazol-2-yl)-3-(5-nitro-2-furanyl)-2-propenenitrile
   Show/Hide
C15H10N4O3
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0010841
1-(3-Ethylsulfanyl-[1,2,4]thiadiazol-5-yl)-3-(3-fluoro-phenyl)-urea
   Show/Hide
C11H11FN4OS2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0046109
6-(2-furanyl)-3-methyl-4-oxo-1,5,6,7-tetrahydroindole-2-carboxylic acid ethyl ester
   Show/Hide
C16H17NO4
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0077704
2-[[(2S,3R,5R,6S,8R,9R)-2-[(1S)-2-keto-1-methyl-2-(1H-pyrrol-2-yl)ethyl]-3,5,9-trimethyl-1,7-dioxaspiro[5.5]undecan-8-yl]methyl]-5-(methylamino)-1,3-benzoxazole-4-carboxylic acid
   Show/Hide
C29H37N3O6
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0103089
5-chloranyl-N-[4-[ethyl(phenyl)sulfamoyl]phenyl]-2-methylsulfonyl-pyrimidine-4-carboxamide
   Show/Hide
C20H19ClN4O5S2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0168400
5-chloranyl-N-[4-[methyl(phenyl)sulfamoyl]phenyl]-2-methylsulfonyl-pyrimidine-4-carboxamide
   Show/Hide
C19H17ClN4O5S2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0262349
MLS000526265
   Show/Hide
C15H13N5O3S2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0281007
5,6-bis(chloranyl)-2-[3-(trifluoromethyl)phenyl]-1H-imidazo[4,5-b]pyrazine
   Show/Hide
C12H5Cl2F3N4
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0304717
2-chloranyl-3-(1H-indazol-6-ylamino)naphthalene-1,4-dione
   Show/Hide
C17H10ClN3O2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0394351
1-(3-Chloro-phenyl)-3-(5-pyridin-4-yl-[1,3,4]thiadiazol-2-yl)-urea
   Show/Hide
C14H10ClN5OS
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0712321
SID22411020
   Show/Hide
C23H21Cl3N4O3S
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0725241
SID17513439
   Show/Hide
C22H18N2O2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0758987
SID24823466
   Show/Hide
C26H21N3O3
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0789868
SID24823986
   Show/Hide
C12H17N5O4
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0851488
SID47195856
   Show/Hide
C14H15BrN4S2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0865859
SID121283973
   Show/Hide
C44H53N5O3S2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0893384
SID87336891
   Show/Hide
C38H47ClN4O6
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0912481
SID99495111
   Show/Hide
C30H30ClN3O2
 1
1
Potency ~ 6513.1 nM
   TI
   LI
   LO
   TS
CP0103145
4-cyano-3-methyl-5-[[2-(o-tolyl)quinoline-4-carbonyl]amino]thiophene-2-carboxylic acid isopropyl ester
   Show/Hide
C27H23N3O3S
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0168183
(E)-4,4-dimethyl-1-(3-nitrophenyl)-2-(1,2,4-triazol-1-yl)-1-penten-3-one
   Show/Hide
C15H16N4O3
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0169356
MLS001003501
   Show/Hide
C15H11FN4OS2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0196797
5-chloranyl-2-ethylsulfonyl-N-[4-[methyl(phenyl)sulfamoyl]phenyl]pyrimidine-4-carboxamide
   Show/Hide
C20H19ClN4O5S2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0247735
(4S)-3-[2-(4-ethoxyphenyl)ethyl]-4-[(4-hydroxyphenyl)methyl]-1-[(2S)-1-(4-hydroxyphenyl)-3-[(2R)-2-[[(5S)-5-(2-methylpropyl)-2-sulfanylidene-1-imidazolidinyl]methyl]-1-pyrrolidinyl]propan-2-yl]-2-imidazolidinethione
   Show/Hide
C41H55N5O3S2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0278383
2-amino-N-[3,5-bis(trifluoromethyl)phenyl]-5-bromo-3-pyridinesulfonamide
   Show/Hide
C13H8BrF6N3O2S
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0303476
1,1'-[3-(2-naphthylsulfonyl)-1,2-propanediyl]dipiperidine
   Show/Hide
C23H32N2O2S
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0311336
(6-chloro-2-phenyl-benzotriazol-5-yl)amine
   Show/Hide
C12H9ClN4
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0312438
MLS000738149
   Show/Hide
C18H14ClNO2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0338169
5-chloranyl-2-ethylsulfonyl-N-[4-(3-methylpiperidin-1-yl)sulfonylphenyl]pyrimidine-4-carboxamide
   Show/Hide
C19H23ClN4O5S2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0434618
2-benzylsulfonyl-5-chloro-N-(2-ethoxyphenyl)pyrimidine-4-carboxamide
   Show/Hide
C20H18ClN3O4S
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0665416
SID17505483
   Show/Hide
C21H19ClN2O6
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0709752
SID51087137
   Show/Hide
C30H35ClN4O4S2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0743168
CO-ADD:0136616
   Show/Hide
C19H13ClN2O2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0810838
SID22411045
   Show/Hide
C24H22ClF3N4O3S
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0817966
SID49819127
   Show/Hide
C11H10Cl2N2OS
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0893458
SID92763659
   Show/Hide
C39H57N5OS2
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0947421
SID103162505
   Show/Hide
C16H18N4OS
 1
1
Potency ~ 7307.8 nM
   TI
   LI
   LO
   TS
CP0041688
2-nitro-N-(8-quinolinyl)benzenesulfonamide
   Show/Hide
C15H11N3O4S
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0064184
C.I. Azoic Coupling Component 23
   Show/Hide
C19H16ClNO4
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0075660
1,2-bis(5-bromo-2-hydroxyphenyl)ethane-1,2-dione
   Show/Hide
C14H8Br2O4
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0136865
4-cyano-3-methyl-5-[(2-phenylquinoline-4-carbonyl)amino]thiophene-2-carboxylic acid methyl ester
   Show/Hide
C24H17N3O3S
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0222675
2-[(5-chloranylthiophen-2-yl)sulfonylamino]-N-[2-(phenylmethyl)phenyl]benzamide
   Show/Hide
C24H19ClN2O3S2
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0286350
2-(benzenesulfonyl)-5-nitropyridine
   Show/Hide
C11H8N2O4S
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0489814
2,6-bis(fluoranyl)-3-nitro-N-(12-oxidanylidene-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazolin-2-yl)benzamide
   Show/Hide
C20H16F2N4O4
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0539531
(3-chlorophenyl)-[4-(2-sec-butoxy-4-pyridyl)pyrimidin-2-yl]amine
   Show/Hide
C19H19ClN4O
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0737953
2-[5,7-bis(trifluoromethyl)-1,8-naphthyridin-2-yl]-2-(4-chlorophenyl)acetonitrile
   Show/Hide
C18H8ClF6N3
 1
1
Potency ~ 8199.5 nM
   TI
   LI
   LO
   TS
CP0101833
'2-(4-AMINO-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-HYDROXYMETHYL-TETRAHYDRO-FURAN-3,4-DIOL
   Show/Hide
C11H14N4O4
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0104621
(5-acetamido-4-acetyloxy-2,1,3-benzoxadiazol-7-yl) acetate
   Show/Hide
C12H11N3O6
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0167831
5-chloranyl-N-[4-(2-ethylpiperidin-1-yl)sulfonylphenyl]-2-methylsulfonyl-pyrimidine-4-carboxamide
   Show/Hide
C19H23ClN4O5S2
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0250533
1-[3-(diethylsulfamoyl)phenyl]-3-[3-(trifluoromethyl)phenyl]urea
   Show/Hide
C18H20F3N3O3S
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0370678
5-chloranyl-2-ethylsulfonyl-N-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]pyrimidine-4-carboxamide
   Show/Hide
C19H23ClN4O5S2
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0394132
4-(3-aminophenyl)-N-(4-methoxyphenyl)-2-pyrimidinamine
   Show/Hide
C17H16N4O
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0395730
1-[5-(2-Ethylsulfanyl-ethyl)-[1,3,4]thiadiazol-2-yl]-3-(3-trifluoromethyl-phenyl)-urea
   Show/Hide
C14H15F3N4OS2
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0907197
SID99359305
   Show/Hide
C36H45Cl2FN4O5
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0910141
SID87349217
   Show/Hide
C35H37F3N4O4
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0965991
SID92763899
   Show/Hide
C13H8FNO
 1
1
Potency ~ 9200 nM
   TI
   LI
   LO
   TS
CP0053259
MLS001029919
   Show/Hide
C18H18ClNO3
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0143227
2-chloranyl-3-[[4-(dimethylamino)phenyl]amino]naphthalene-1,4-dione
   Show/Hide
C18H15ClN2O2
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0195353
2-[(E)-1-(benzenesulfonyl)-2-(3-methylphenyl)ethenyl]-1H-benzimidazole
   Show/Hide
C22H18N2O2S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0239508
3-[1-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrazol-5-yl]-[2-(trifluoromethyloxy)phenyl]methyl]piperidin-4-yl]-1H-benzimidazol-2-one
   Show/Hide
C29H26F3N7O4
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0298422
(E)-2-(benzenesulfonyl)-3-[5-(4-bromophenyl)-2-furanyl]-N-(3-pyridinylmethyl)-2-propenamide
   Show/Hide
C25H19BrN2O4S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0350532
1-[3-[(2-chlorophenyl)sulfamoyl]-4-(1-pyrrolidinyl)phenyl]-3-(4-fluorophenyl)urea
   Show/Hide
C23H22ClFN4O3S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0351387
2-[1-(4-tert-Butyl-benzenesulfonyl)-piperidin-4-yl]-5-chloro-1H-benzoimidazole
   Show/Hide
C22H26ClN3O2S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0412928
2-benzylsulfonyl-5-chloro-N-(2,5-dimethoxyphenyl)pyrimidine-4-carboxamide
   Show/Hide
C20H18ClN3O5S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0514312
MLS000721625
   Show/Hide
C25H27N3O2
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0741895
SID22410259
   Show/Hide
C22H22ClN3O6S3
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0791790
SID3714949
   Show/Hide
C18H15N5O
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0826229
SID22410885
   Show/Hide
C19H17ClN2O5S2
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0852863
SID14747000
   Show/Hide
C16H17N3O5S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0852864
SID50085535
   Show/Hide
C23H26N2O3
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0856388
SID121284955
   Show/Hide
C26H25N7O3S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0857963
SID92763381
   Show/Hide
C20H22N6O6S
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0867354
SID103073968
   Show/Hide
C19H14F3N5O
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0883001
SID92763360
   Show/Hide
C36H45BrN4O6
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0898681
SID57265093
   Show/Hide
C22H21ClN2O3
 1
1
Potency ~ 10322.5 nM
   TI
   LI
   LO
   TS
CP0074040
7-bromanyl-N-(2-methoxyphenyl)-3-oxidanyl-naphthalene-2-carboxamide
   Show/Hide
C18H14BrNO3
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0105199
MLS000057468
   Show/Hide
C13H10N2O2S2
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0208795
MLS000418668
   Show/Hide
C24H21N3O4S2
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0338278
5,5-dimethyl-2,6-dihydropyrazolo[4,3-d][3]benzazepin-3-one
   Show/Hide
C13H13N3O
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0388557
2-benzyl-N-[2-methyl-4-(4-methylpiperazin-1-yl)phenyl]-3,4-dihydro-1H-benzo[b][1,6]naphthyridine-10-carboxamide
   Show/Hide
C32H35N5O
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0413146
MLS000418648
   Show/Hide
C23H18FN3O3S2
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0541559
4-(4-morpholinyl)-7-nitro-3-oxido-2,1,3-benzoxadiazol-3-ium
   Show/Hide
C10H10N4O5
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0701515
SID49674835
   Show/Hide
C22H21ClN2O2
 1
1
Potency ~ 11582.1 nM
   TI
   LI
   LO
   TS
CP0128019
4-[(2-benzylsulfonyl-5-chloro-pyrimidine-4-carbonyl)amino]benzoic acid ethyl ester
   Show/Hide
C21H18ClN3O5S
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0252497
1-(2,4-Difluoro-phenyl)-3-(3-propylsulfanyl-[1,2,4]thiadiazol-5-yl)-urea
   Show/Hide
C12H12F2N4OS2
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0350357
MLS000539021
   Show/Hide
C25H23F3N6O
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0397213
2-[2-hydroxyethyl-(7-nitro-3-oxidanidyl-2,1,3-benzoxadiazol-3-ium-4-yl)amino]ethanol
   Show/Hide
C10H12N4O6
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0413913
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-keto-N-[4-(4-methoxyphenyl)-5-methyl-thiazol-2-yl]pyrrolidine-3-carboxamide
   Show/Hide
C24H23N3O5S
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0665704
SID17515143
   Show/Hide
C14H12N2O3S
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0782145
SID24780125
   Show/Hide
C20H21N5O
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0796052
SID22411700
   Show/Hide
C25H26ClN3O2
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0809495
SID24791749
   Show/Hide
C19H17ClN2O4S2
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0847687
SID49674104
   Show/Hide
C18H22F2N2OS
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0856584
SID49649794
   Show/Hide
C15H16ClN3O
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0879706
SID121283276
   Show/Hide
C19H18N6O4
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0891795
SID99360007
   Show/Hide
C27H18ClN3O3
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0894862
SID49725329
   Show/Hide
C16H18N2O5S2
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0895843
SID92764348
   Show/Hide
C18H16N2O3
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0896044
2-cyclopropyl-N'-(3,4-dichlorophenyl)-2-oxoacetohydrazonoyl cyanide
   Show/Hide
C12H9Cl2N3O
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0918086
SID92763664
   Show/Hide
C41H55N5O3S2
 1
1
Potency ~ 12995.3 nM
   TI
   LI
   LO
   TS
CP0133378
4-[5-[1-(furan-2-ylcarbonyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl]-N-(phenylmethyl)benzenesulfonamide
   Show/Hide
C25H24N4O5S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0156082
(4S,9S,10S,12E)-9,10,18-trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),12,15,17-tetraene-2,8-dione
   Show/Hide
C19H24O7
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0204212
1-(5-nitro-1,3-thiazol-2-yl)-3-phenyl-urea
   Show/Hide
C10H8N4O3S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0303240
MLS000718916
   Show/Hide
C19H21ClN4O5
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0379337
MLS001006742
   Show/Hide
C22H18N4O2
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0439074
MLS001172437
   Show/Hide
C18H19F3N4S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0665407
SID22402031
   Show/Hide
C24H20FN3O5S2
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0691324
SID24824109
   Show/Hide
C15H12N4O5S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0715643
SID49715950
   Show/Hide
C14H9N3O6
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0728921
SID14745805
   Show/Hide
C21H16N2O3S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0755622
SID49824643
   Show/Hide
C13H11N5O3S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0852858
SID87336901
   Show/Hide
C40H45ClN4O5
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0859493
SID121285115
   Show/Hide
C29H34N6
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0864851
SID92764852
   Show/Hide
C20H25ClN4O
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0875509
SID49731807
   Show/Hide
C19H16ClN3O4S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0881130
SID85257296
   Show/Hide
C18H12F6N2O3S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0881139
4-(4-chlorophenyl)-1-((3-(4-methoxyphenyl)-1H-pyrazol-4-yl)methyl)piperidin-4-ol
   Show/Hide
C22H24ClN3O2
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0893354
SID93577509
   Show/Hide
C13H9N3O3
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0907404
SID121283728
   Show/Hide
C12H8Cl2N2O4S
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0912446
SID121285088
   Show/Hide
C28H36N6
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0912770
SID26726452
   Show/Hide
C21H21ClFN3O
 1
1
Potency ~ 14581 nM
   TI
   LI
   LO
   TS
CP0007251
MLS000673919
   Show/Hide
C21H22N2O3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0039752
MLS002693850
   Show/Hide
C17H11NO3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0041629
3-[[7-(1,3-benzothiazol-2-ylsulfanyl)-4-nitro-2,1,3-benzoxadiazol-5-yl]amino]propan-1-ol
   Show/Hide
C16H13N5O4S2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0064482
MLS001121514
   Show/Hide
C15H17BrN4O3S2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0140235
Furan-2-carboxylic acid [1-butyl-3-(toluene-4-sulfonyl)-1H-pyrrolo[2,3-b]quinoxalin-2-yl]-amide
   Show/Hide
C26H24N4O4S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0142018
4-[(4-methylbenzyl)amino]phenol
   Show/Hide
C14H15NO
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0162679
(9-amino-7-ethoxy-acridin-3-yl)-p-anisyl-amine
   Show/Hide
C23H23N3O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0211433
4-(3-oxo-5-phenyl-1H-pyrazol-2-yl)benzoic acid ethyl ester
   Show/Hide
C18H16N2O3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0285852
2-methyl-4,9-dioxo-3-benzo[f]benzofurancarboxylic acid ethyl ester
   Show/Hide
C16H12O5
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0336408
MLS001007696
   Show/Hide
C19H19N3O2S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0342063
5-(3-thienyl)-3-({[4-(trifluoromethyl)phenyl]sulfonyl}amino)thiophene-2-carboxamide
   Show/Hide
C16H11F3N2O3S3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0371129
2-(4-fluorobenzyl)-5-(4-fluorobenzyl)oxy-3,4-dihydroisocarbostyril
   Show/Hide
C23H19F2NO2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0401614
(4S)-1-benzyl-4-(4-bromophenyl)-2-(2-methoxyethylamino)-6-methyl-4H-pyrimidine-5-carboxylic acid methyl ester
   Show/Hide
C23H26BrN3O3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0407127
5-N-[3-methoxy-5-[[3-(trifluoromethyl)phenyl]carbamoyl]phenyl]-1H-imidazole-4,5-dicarboxamide
   Show/Hide
C20H16F3N5O4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0410047
2-N-(3-aminopropyl)-4-N-cyclohexyl-5-nitropyrimidine-2,4,6-triamine
   Show/Hide
C13H23N7O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0419043
5-chloranyl-N-(4-fluorophenyl)-2-[(2-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
   Show/Hide
C19H15ClFN3O3S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0423820
5-nitro-2-[3-(trifluoromethyl)phenyl]sulfonyl-pyridine
   Show/Hide
C12H7F3N2O4S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0480151
MLS001095214
   Show/Hide
C21H22ClN3O4S2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0514946
5-Methyl-3-phenyl-isoxazole-4-carboxylic acid (5-nitro-thiazol-2-yl)-amide
   Show/Hide
C14H10N4O4S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0693739
SID87338259
   Show/Hide
C20H22N4O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0712020
SID26732535
   Show/Hide
C31H38N4O6
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0846471
SID49647990
   Show/Hide
C22H15FN2O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0852862
SID860222
   Show/Hide
C20H21N3O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0855399
SID74373554
   Show/Hide
C26H32F3N3O2S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0857410
SID49648347
   Show/Hide
C17H18N4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0860959
SID85301986
   Show/Hide
C31H35F3N4O3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0862823
SID121286317
   Show/Hide
C32H22N4O4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0867314
SID17515747
   Show/Hide
C27H28F2N4OS
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0867352
SID92764801
   Show/Hide
C18H24ClNO3
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0872951
SID87340817
   Show/Hide
C22H16N2O5S2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0877016
SID49666013
   Show/Hide
C16H11ClN2O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0877017
SID103076267
   Show/Hide
C21H14ClF3N2O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0883158
SID87349266
   Show/Hide
C42H50N4O7
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0883350
SID49675188
   Show/Hide
C26H30N2O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0887475
SID103050902
   Show/Hide
C22H22N4S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0887830
SID92764440
   Show/Hide
C16H12ClNOS
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0895497
SID92764520
   Show/Hide
C25H19N3O4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0905584
SID26731845
   Show/Hide
C21H10Cl2N4O4S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0910023
SID87349215
   Show/Hide
C37H48N4O4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0918164
SID121284980
   Show/Hide
C27H27N7O2
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0921524
SID121285615
   Show/Hide
C22H17ClN4
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0956960
SID87349570
   Show/Hide
C30H30F3N3O6S
 1
1
Potency ~ 16360.1 nM
   TI
   LI
   LO
   TS
CP0010267
1-[3-chloro-4-(difluoromethoxy)phenyl]-3-(4-nitrophenyl)urea
   Show/Hide
C14H10ClF2N3O4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0066114
1,2-diphenylguanidine
   Show/Hide
C13H13N3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0100533
2-(4-methylphenyl)sulfanyl-N-(5-nitro-2-oxidanyl-phenyl)ethanamide
   Show/Hide
C15H14N2O4S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0122613
1-(4-chlorophenyl)-3-(5-nitro-3-thienyl)urea
   Show/Hide
C11H8ClN3O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0152790
1-chloranyl-7,8-bis(fluoranyl)-3-methyl-pyrido[1,2-a]benzimidazole-4-carbonitrile
   Show/Hide
C13H6ClF2N3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0168365
4-methyl-2-nitro-N-(8-quinolinyl)benzenesulfonamide
   Show/Hide
C16H13N3O4S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0307977
1-[(2,4-dimethoxyphenyl)-(4-morpholinyl)methyl]-2-naphthalenol
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C23H25NO4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0342064
5-nitro-N-[3-(2-thenoylamino)phenyl]-2-furamide
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C16H11N3O5S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0352385
2-[(2-{[(4-chlorophenyl)sulfonyl]amino}phenyl)sulfanyl]-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]acetamide
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C17H12ClF3N4O3S3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0411697
5-chloranyl-N-(3,4-dimethylphenyl)-2-[(2-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
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C21H20ClN3O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0442869
(4S)-1-[(1S)-1-benzyl-2-[2-[[(5S)-5-(4-hydroxybenzyl)-2-thioxo-imidazolidin-1-yl]methyl]pyrrolidino]ethyl]-4-(4-hydroxybenzyl)-3-phenethyl-imidazolidine-2-thione
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C42H49N5O2S2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0447540
1-{phenyl[(phenylacetyl)amino]methyl}-2-naphthyl acetate
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C27H23NO3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0454217
(2-Pyridin-3-yl-quinazolin-4-yl)-p-tolyl-amine
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C20H16N4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0464215
2-(dimethylamino)-3-(4-methylphenyl)sulfanyl-naphthalene-1,4-dione
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C19H17NO2S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0465662
2-phenyl-2-(phenylthio)-N-[4-(sec-butylsulfamoyl)phenyl]acetamide
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C24H26N2O3S2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0488520
(3S)-5-methyl-6'-(4-methylbenzoyl)-7'-(3-nitrophenyl)spiro[1H-indole-3,5'-3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole]-2-one
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C28H25N3O4S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0514313
Cyclohexanecarboxylic acid [(2-hydroxy-naphthalen-1-yl)-p-tolyl-methyl]-amide
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C25H27NO2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0521877
1-(3-chlorophenyl)-3-methyl-6-(trifluoromethyl)-2H-pyrazolo[3,4-d]pyrimidin-4-one
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C13H8ClF3N4O
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0633379
SID22403046
   Show/Hide
C12H12ClN5O2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0679680
SID26725587
   Show/Hide
C23H14ClF3N4O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0725062
SID24269432
   Show/Hide
C20H18N4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0781141
SID17413725
   Show/Hide
C22H21N3O6S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0789708
SID49713768
   Show/Hide
C28H30N4O4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0803430
SID152199723
   Show/Hide
C17H20Cl3NO3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0811176
SID14735752
   Show/Hide
C16H14Cl3NO2S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0818283
SID24833068
   Show/Hide
C21H15ClN2O4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0834821
SID87334302
   Show/Hide
C24H20O6
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0848128
SID87341456
   Show/Hide
C24H26N2O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0849482
SID17413346
   Show/Hide
C20H16ClNO4S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0849494
SID49646446
   Show/Hide
C25H26Cl2N2O3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0850047
SID24787304
   Show/Hide
C20H25BrN4OS
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0852872
SID24841667
   Show/Hide
C25H28F3NO4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0852913
SID99359829
   Show/Hide
C19H12Cl2N2O4S2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0856749
SID99456131
   Show/Hide
C28H21N3O3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0857469
SID47200316
   Show/Hide
C27H31Cl2N5O2S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0864799
SID103060596
   Show/Hide
C19H18N4S2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0865634
SID121283926
   Show/Hide
C39H57N5OS2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0867232
SID103060464
   Show/Hide
C26H28Cl2N2O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0875901
SID87336745
   Show/Hide
C31H32ClF3N4O4
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0876881
SID49821941
   Show/Hide
C18H18ClN5O2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0884735
SID17506356
   Show/Hide
C22H20ClN3O5S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0885181
SID103158874
   Show/Hide
C16H14F3N5S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0887478
MMV1527628
   Show/Hide
C18H15ClN2O2S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0887479
SID87336770
   Show/Hide
C34H43ClN4O5
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0887480
SID56316824
   Show/Hide
C18H19ClN4O5
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0887491
SID47196203
   Show/Hide
C19H24ClNO
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0887505
SID121285447
   Show/Hide
C27H27N7O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0907695
SID121284977
   Show/Hide
C28H26F3N7O3
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0908476
SID103163450
   Show/Hide
C21H23FN4O4S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0908501
SID103159064
   Show/Hide
C22H22N2O3S
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0912023
SID93576846
   Show/Hide
C34H54O7
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0960198
SID17416119
   Show/Hide
C23H18BrClFN3OS2
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0964108
SID92764692
   Show/Hide
C23H25N5O
 1
1
Potency ~ 18356.4 nM
   TI
   LI
   LO
   TS
CP0123190
2-methyl-3-(4-methylpiperidin-1-yl)carbonyl-benzo[f][1]benzofuran-4,9-dione
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C20H19NO4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0133489
2-(3-chloro-N-(2-chloro-1-oxoethyl)-4-methoxyanilino)-N-(2-phenylethyl)-2-thiophen-2-ylacetamide
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C23H22Cl2N2O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0208501
(1E)-1-[amino-[(4,6-dimethyl-2-quinazolinyl)amino]methylidene]-3-cyclohexylurea
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C18H24N6O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0209480
MLS000583250
   Show/Hide
C16H13Cl2N3O2S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0235358
4-[4-(2,3-dimethylphenyl)piperazin-1-yl]carbonyl-2,9-dimethyl-pyrido[3,4-b]indol-1-one
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C26H28N4O2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0267931
2-[(2-methoxybenzyl)thio]-4-(4-nitrophenyl)-1H-imidazole
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C17H15N3O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0295533
MLS000394969
   Show/Hide
C22H21ClN2O3S2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0314204
2,3,4,7,8,9,10,11-octahydro-1H-cyclohepta[4,5]thieno[2,3-b]quinolin-12-amine
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C16H20N2S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0342437
2-[2-(2,4-dimethylanilino)-2-keto-ethyl]cinchoninic acid
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C20H18N2O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0352158
(E)-2-(1H-benzimidazol-2-yl)-3-(3-chlorophenyl)-1-phenyl-2-propen-1-one
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C22H15ClN2O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0352683
1-[2-(4-tert-butylphenoxy)ethyl]-3-phenyl-thiourea
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C19H24N2OS
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0356857
2-[4-[3-(1,3-benzodioxol-5-yl)-5-(3-thienyl)isoxazol-4-yl]phenyl]cinchoninic acid
   Show/Hide
C30H18N2O5S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0465581
(5S)-1-[2-(3-fluorophenyl)ethyl]-5-(2-methylpropyl)-N-phenyl-4,5-dihydroimidazol-2-amine
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C21H26FN3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0480417
1-[3-[[2-(2-thenylamino)thieno[3,2-d]pyrimidin-4-yl]amino]propyl]-2-pyrrolidone
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C18H21N5OS2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0481019
MLS002222506
   Show/Hide
C27H36N2O2S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0531291
5-fluoranyl-N-[4-(4-fluorophenyl)-1,2,5-oxadiazol-3-yl]-3-methyl-1-benzofuran-2-carboxamide
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C18H11F2N3O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0554232
MLS000051884
   Show/Hide
C20H15NO5S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0663417
SID17503792
   Show/Hide
C31H32FN3O5
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0663436
MMV1652527
   Show/Hide
C28H28N4O2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0690364
SID17416047
   Show/Hide
C23H19Br2N3OS2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0694682
SID47200506
   Show/Hide
C22H25NO4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0702740
SID49825561
   Show/Hide
C19H14ClNO4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0727884
SID26661687
   Show/Hide
C18H14N2O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0736424
SID24788030
   Show/Hide
C16H12N4O4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0787106
SID17507995
   Show/Hide
C15H10Cl2N4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0787797
SID24835408
   Show/Hide
C19H16N4S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0804936
SID24835534
   Show/Hide
C25H33N3O7S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0815301
SID99245557
   Show/Hide
C21H18ClF3N4O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0843421
SID24822165
   Show/Hide
C12H14ClN3O2S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0846667
SID47204929
   Show/Hide
C15H14ClN3O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0852860
SID56324973
   Show/Hide
C20H23F3N2O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0856924
SID24837069
   Show/Hide
C19H17NO5
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0860381
SID89853212
   Show/Hide
C12H9N3O4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0860633
SID121283940
   Show/Hide
C38H57N5O2S2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0865585
SID87336923
   Show/Hide
C40H48ClN5O5
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0868308
SID121285024
   Show/Hide
C25H28F3N7O2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0868591
SID121283958
   Show/Hide
C39H57N5O2S2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0874958
SID24799044
   Show/Hide
C22H27NO3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0877140
SID51085116
   Show/Hide
C27H28F3N3O2S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0893418
SID87336780
   Show/Hide
C31H34ClF3N4O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0897512
SID87349241
   Show/Hide
C36H37F3N4O4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0899374
SID121284974
   Show/Hide
C28H29N7O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0900498
SID22410719
   Show/Hide
C17H19Cl2N3O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0911987
SID22408208
   Show/Hide
C19H15Cl2NO5
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0912482
SID103059960
   Show/Hide
C23H23Cl2N5O4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0914839
SID103162663
   Show/Hide
C24H20N4O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0918088
SID103073556
   Show/Hide
C21H19N3OS
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0921506
SID85201744
   Show/Hide
C36H41N3O5S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0923552
SID17512513
   Show/Hide
C21H18ClFN2O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0925784
SID99494907
   Show/Hide
C22H27N3O3S
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0926414
SID103050988
   Show/Hide
C14H16N4OS2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0929260
SID81066797
   Show/Hide
C25H38N2O
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0932755
SID121283953
   Show/Hide
C36H53N5OS2
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0948789
SID85146834
   Show/Hide
C27H28N8O4
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0956946
SID57257634
   Show/Hide
C25H30N2O3
 1
1
Potency ~ 20596.2 nM
   TI
   LI
   LO
   TS
CP0076836
(Z)-3-[5-(1H-benzimidazol-2-ylsulfanyl)furan-2-yl]-2-phenyl-prop-2-enenitrile
   Show/Hide
C20H13N3OS
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0163339
1-(3-chlorophenyl)-3-(5-nitro-3-thienyl)urea
   Show/Hide
C11H8ClN3O3S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0233015
1-[2-(4-chlorophenyl)ethyl]-3-(4-nitrophenyl)thiourea
   Show/Hide
C15H14ClN3O2S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0240958
1-(2-methyl-5-propan-2-yl-phenyl)-3-(4-nitrophenyl)urea
   Show/Hide
C17H19N3O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0282196
MLS000595074
   Show/Hide
C20H15N5O7
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0285143
MLS000583603
   Show/Hide
C20H14FN3O2S2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0332609
MLS000083238
   Show/Hide
C20H29N3O5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0336528
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(3-pyridinyl)acetamide
   Show/Hide
C21H23Cl2N3O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0367499
(4S)-1-[(1S)-1-benzyl-2-[2-[[(5S)-5-(4-hydroxybenzyl)-2-thioxo-imidazolidin-1-yl]methyl]pyrrolidino]ethyl]-3-(cyclohexylmethyl)-4-(4-hydroxybenzyl)imidazolidine-2-thione
   Show/Hide
C41H53N5O2S2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0375429
2-benzylsulfonyl-5-chloro-N-piperonyl-pyrimidine-4-carboxamide
   Show/Hide
C20H16ClN3O5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0378911
(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-keto-N-phenyl-3,4,4a,7,8,8a-hexahydroisoquinoline-8-carboxamide
   Show/Hide
C23H22Cl2N2O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0394471
Acetic acid 4-(acetyl-benzenesulfonyl-amino)-2-bromo-naphthalen-1-yl ester
   Show/Hide
C20H16BrNO5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0477178
2-(1,3-benzodioxol-5-yl)-4,5-bis(4-methoxyphenyl)-1H-imidazole
   Show/Hide
C24H20N2O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0561374
4-(4-chlorophenyl)-4-keto-N-[3-[(4-methoxyphenyl)sulfamoyl]phenyl]butyramide
   Show/Hide
C23H21ClN2O5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0665188
SID26658812
   Show/Hide
C23H22FN5O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0669412
SID17511440
   Show/Hide
C21H23N3O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0687731
SID14733888
   Show/Hide
C24H26N2O3S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0709310
Benzoic acid N'-(5-nitro-furan-2-carbonyl)-hydrazide
   Show/Hide
C12H9N3O5
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0712903
SID17513788
   Show/Hide
C21H15N7O3S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0721035
SID24814503
   Show/Hide
C23H16N2O5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0741928
SID24785450
   Show/Hide
C19H29ClN2O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0752530
SID49714039
   Show/Hide
C22H24N4S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0765492
N-[6-[4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl]pyridin-3-yl]thiophene-2-carboxamide
   Show/Hide
C20H18F3N5OS
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0791876
SID24785506
   Show/Hide
C19H16ClN3OS
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0834870
SID87336821
   Show/Hide
C21H20Cl2N4O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0844361
SID49672767
   Show/Hide
C26H29ClN2O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0847686
SID51090288
   Show/Hide
C20H23NO5
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0850012
SID103075676
   Show/Hide
C16H18N4S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0857198
SID87349252
   Show/Hide
C38H46N4O5
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0860331
SID121283937
   Show/Hide
C39H51N5O2S2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0860960
SID89853891
   Show/Hide
C15H11BrFNO3S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0864852
SID49720036
   Show/Hide
C23H26FN3O3S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0865617
SID87336912
   Show/Hide
C36H39ClF3N5O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0867353
SID56462964
   Show/Hide
C22H29N3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0868621
SID121283946
   Show/Hide
C36H59N5OS2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0893419
SID99360689
   Show/Hide
C35H43N3O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0905358
SID121285511
   Show/Hide
C29H33N7O
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0905406
SID22412612
   Show/Hide
C16H15BrN2O2S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0907487
SID57263885
   Show/Hide
C26H25N3O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0907495
3-(4-methoxyphenyl)-5-phenyl-2-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-7(4H)-one
   Show/Hide
C20H14F3N3O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0908478
SID85148524
   Show/Hide
C27H25FN2O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0908871
SID103073666
   Show/Hide
C25H23Cl2N3O3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0909629
SID103060170
   Show/Hide
C27H24N4O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0912447
SID87336911
   Show/Hide
C39H50ClN5O4
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0914176
SID121282560
   Show/Hide
C30H34F3N3O5S
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0917830
SID49649756
   Show/Hide
C20H15Cl2N3O
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0923783
SID56463714
   Show/Hide
C21H26FN3
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0947418
SID99456647
   Show/Hide
C18H20N6OS
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0947851
SID103163397
   Show/Hide
C23H19ClN4O2
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0949423
SID121285003
   Show/Hide
C26H31N7O
 1
1
Potency ~ 23109.3 nM
   TI
   LI
   LO
   TS
CP0031043
N-quinolin-8-ylbenzenesulfonamide
   Show/Hide
C15H12N2O2S
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0044299
4-methoxy-N-((1-(2-(p-tolyloxy)ethyl)-1H-benzo[d]imidazol-2-yl)methyl)aniline
   Show/Hide
C24H25N3O2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0060475
3-(4-chlorophenyl)-1-(3,4-dichlorophenyl)urea
   Show/Hide
C13H9Cl3N2O
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0128204
4-(4-methyl-1-piperazinyl)-7-nitro-3-oxido-2,1,3-benzoxadiazol-3-ium
   Show/Hide
C11H13N5O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0220396
1-chloranyl-3-methyl-pyrido[1,2-a]benzimidazole-4-carbonitrile
   Show/Hide
C13H8ClN3
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0233949
(4-anilino-6-methyl-pyrimidin-2-yl)-benzyl-amine
   Show/Hide
C18H18N4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0296914
1-(3-tert-Butylsulfanyl-[1,2,4]thiadiazol-5-yl)-3-(3-methoxy-phenyl)-urea
   Show/Hide
C14H18N4O2S2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0304621
3-({7-[(5-methyl-1,3,4-thiadiazol-2-yl)thio]-4-nitro-2,1,3-benzoxadiazol-5-yl}amino)propan-1-ol
   Show/Hide
C12H12N6O4S2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0312648
1-(4-butylphenyl)-3-[4-(4-methoxyanilino)phenyl]thiourea
   Show/Hide
C24H27N3OS
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0360886
(E)-3-(3-methoxy-4-oxidanyl-phenyl)-1-(5-nitrofuran-2-yl)prop-2-en-1-one
   Show/Hide
C14H11NO6
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0378026
2-[2-ethoxy-4-(2-nitrovinyl)phenoxy]-N-(2-methylphenyl)acetamide
   Show/Hide
C19H20N2O5
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0389670
N,2-diphenylquinazolin-4-amine
   Show/Hide
C20H15N3
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0395990
MLS002702985
   Show/Hide
C27H27NO6
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0407005
1-Benzyl-5-[3-(3,5-dimethyl-pyrazol-1-yl)-2-hydroxy-propoxy]-2-methyl-1H-indole-3-carboxylic acid ethyl ester
   Show/Hide
C27H31N3O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0426884
(2-chlorophenyl)-[2-(4-pyridyl)quinazolin-4-yl]amine
   Show/Hide
C19H13ClN4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0457985
2-ethyl-N-(5-nitro-1,3-thiazol-2-yl)hexanamide
   Show/Hide
C11H17N3O3S
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0459009
3-cyclohexyl-N-[(1S)-2-[(3S,6R)-3-(4-hydroxybenzyl)-6-p-anisyl-2,3,5,6-tetrahydroimidaz[1,2-a]imidazol-7-yl]-1-methyl-ethyl]propionamide
   Show/Hide
C32H44N4O3
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0501545
MLS000721672
   Show/Hide
C17H18ClN5O
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0646495
SID17409332
   Show/Hide
C24H23N3O3
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0820742
SID49817443
   Show/Hide
C22H29BrN2O5
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0830359
SID104219725
   Show/Hide
C16H15N3O2S
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0836256
SID24818823
   Show/Hide
C22H18Cl2FN3O2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0856907
SID87336744
   Show/Hide
C34H43ClN4O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0857391
SID121283976
   Show/Hide
C42H55N5O2S2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0867351
SID92763643
   Show/Hide
C39H57N5OS2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0882323
SID49670026
   Show/Hide
C21H20ClF3N2O5
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0884607
SID22410579
   Show/Hide
C24H25ClFN3O6S2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0907371
SID121285941
   Show/Hide
C22H19BrN2O
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0908475
SID87336910
   Show/Hide
C38H50ClN5O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0908500
SID56314726
   Show/Hide
C27H28ClFN2O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0911985
SID99360546
   Show/Hide
C8H8N6S
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0912651
SID85201828
   Show/Hide
C37H41N3O5
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0919667
SID121286288
   Show/Hide
C30H23N3O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0921309
SID56319828
   Show/Hide
C24H28N2O4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0923970
SID121286576
   Show/Hide
C17H26ClNO4
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0947850
SID92763655
   Show/Hide
C42H55N5O2S2
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0949424
SID56316010
   Show/Hide
C26H32FN3O4S
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0961319
SID49822535
   Show/Hide
C14H9Cl2N5O
 1
1
Potency ~ 25929 nM
   TI
   LI
   LO
   TS
CP0008489
7-bromo-3,6,6-trimethyl-1-(1,3-thiazol-2-yl)-5,7-dihydroindazol-4-one
   Show/Hide
C13H14BrN3OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0011641
MLS000950003
   Show/Hide
C18H12ClN3O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0041787
(2S)-2-[[4-[[4-[(tert-butoxycarbonylamino)methyl]phenyl]carbamoyl]-1H-imidazole-5-carbonyl]amino]propionic acid tert-butyl ester
   Show/Hide
C24H33N5O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0049067
3-(3,4-dimethoxyphenyl)-1-[(pentafluorophenyl)sulfonyl]-1H-pyrazol-5-amine
   Show/Hide
C17H12F5N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0049956
2,2-bis(4-methylphenyl)-N-(4-nitro-2-oxidanyl-phenyl)cyclopropane-1-carboxamide
   Show/Hide
C24H22N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0089042
MLS000689772
   Show/Hide
C18H14N4O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0099880
2-[2,2,2-Trichloro-1-(2,2-dimethyl-propionylamino)-ethylamino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid methyl ester
   Show/Hide
C16H21Cl3N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0103034
4-(1H-benzimidazol-2-ylsulfanyl)-1-[4-(2,3-dimethylphenyl)piperazin-1-yl]butan-1-one
   Show/Hide
C23H28N4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0105832
(6E)-6-[5-(4-methoxyphenyl)-1,2-dihydropyrazol-3-ylidene]-1-cyclohexa-2,4-dienone
   Show/Hide
C16H14N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0125964
2-benzylsulfonyl-5-chloro-N-[(4-methoxyphenyl)methyl]pyrimidine-4-carboxamide
   Show/Hide
C20H18ClN3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0128579
2,6-ditert-butyl-4-[[4-(2-hydroxyethyl)-1-piperazinyl]-(3-pyridinyl)methyl]phenol
   Show/Hide
C26H39N3O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0152706
(5Z)-5-[5-(3,4-dimethoxyphenyl)-1,2-dihydropyrazol-3-ylidene]-4,7-dimethoxy-1-benzofuran-6-one
   Show/Hide
C21H20N2O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0158407
4-mesyl-3-nitro-benzoic acid [2-(cyclohexanecarbonylamino)-2-keto-ethyl] ester
   Show/Hide
C17H20N2O8S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0166398
4-(4-{[4-(2-methoxyphenyl)-6-(trifluoromethyl)-2-pyrimidinyl]sulfonyl}butanoyl)morpholine
   Show/Hide
C20H22F3N3O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0166456
(methylbenzoprim, MBP) 5-[4-(Benzyl-methyl-amino)-3-nitro-phenyl]-6-ethyl-pyrimidine-2,4-diamine
   Show/Hide
C20H22N6O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0176366
MLS000775269
   Show/Hide
C15H15N3O7S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0196311
4,5-bis(bromanyl)-2-phenyl-pyridazin-3-one
   Show/Hide
C10H6Br2N2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0196826
5-chloranyl-N-(phenylmethyl)-2-(phenylmethyl)sulfonyl-pyrimidine-4-carboxamide
   Show/Hide
C19H16ClN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0210152
5,6-diphenyl-[1,2,5]oxadiazolo[3,4-b]pyrazine
   Show/Hide
C16H10N4O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0217408
(7-chloro-4-nitro-benzofurazan-5-yl)-methyl-amine
   Show/Hide
C7H5ClN4O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0217437
2-Amino-3-bromo-[1,4]naphthoquinone
   Show/Hide
C10H6BrNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0229313
MLS000580606
   Show/Hide
C21H21NO2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0232363
(E)-3-(4,6-dimethylpyrimidin-2-yl)sulfanyl-1-(2-fluorophenyl)prop-2-en-1-one
   Show/Hide
C15H13FN2OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0232374
9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole
   Show/Hide
C18H16N2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0242117
2-[(E)-2-(5-nitrofuran-2-yl)ethenyl]-3-(3-oxidanylpropyl)quinazolin-4-one
   Show/Hide
C17H15N3O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0259331
2-benzylsulfonyl-5-chloro-N-(3-methylphenyl)pyrimidine-4-carboxamide
   Show/Hide
C19H16ClN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0294729
2-[[2-(2,4-dichlorophenyl)-2-(1H-indol-3-yl)ethyl]amino]-1-phenyl-ethanol
   Show/Hide
C24H22Cl2N2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0299461
1-Ethyl-4-hydroxy-2-oxo-1,2-dihydro-quinoline-3-carboxylic acid (1H-benzoimidazol-2-yl)-amide
   Show/Hide
C19H16N4O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0303214
MLS000394779
   Show/Hide
C18H16Cl2N4O3S4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0304162
4-(2-methoxyphenyl)-2-{[4-(2-methylpiperidin-1-yl)-4-oxobutyl]sulfonyl}-6-(trifluoromethyl)pyrimidine
   Show/Hide
C22H26F3N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0304584
3-Methyl-2-[2-(5-nitro-furan-2-yl)-vinyl]-3H-quinazolin-4-one
   Show/Hide
C15H11N3O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0323041
US9320722, CB13
   Show/Hide
C15H19NO4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0330167
2-[(E)-1-(benzenesulfonyl)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-benzimidazole
   Show/Hide
C22H15F3N2O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0338302
4-[(6-bromanyl-1H-benzimidazol-2-yl)amino]-N-(cyclopropylmethyl)benzamide
   Show/Hide
C18H17BrN4O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0340798
3-(2-chloranyl-6-fluoranyl-phenyl)-5-methyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-1,2-oxazole-4-carboxamide
   Show/Hide
C14H7ClF4N4O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0352118
MLS000876826
   Show/Hide
C28H38O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0358944
5-chloranyl-N-(4-fluorophenyl)-2-[(3-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
   Show/Hide
C19H15ClFN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0364127
MLS000391919
   Show/Hide
C15H10N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0375648
2-[(Z)-1-(benzenesulfonyl)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-benzimidazole
   Show/Hide
C22H15F3N2O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0376042
1-(2-methylphenoxy)-3-[[4-[[3-(2-methylphenoxy)-2-oxidanyl-propyl]amino]cyclohexyl]amino]propan-2-ol
   Show/Hide
C26H38N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0377131
4,5,6,7-tetrafluoro-2-methyl-N-[3-(trifluoromethyl)phenyl]-1-benzofuran-3-sulfonamide
   Show/Hide
C16H8F7NO3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0378240
2-[1-(3-bromobenzyl)indol-3-yl]sulfonyl-N-(5-methylisoxazol-3-yl)acetamide
   Show/Hide
C21H18BrN3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0382379
5-chloro-N-[4-(difluoromethoxy)phenyl]-2-(4-methylbenzyl)sulfonyl-pyrimidine-4-carboxamide
   Show/Hide
C20H16ClF2N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0383879
2-(6-benzoxypurin-9-yl)-1-[4-(2,4,6-trimethylbenzyl)piperazino]ethanone
   Show/Hide
C28H32N6O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0386929
4-(2-cyclopropyl-1,3-oxazol-5-yl)-N-methyl-N-(3-methylphenyl)benzenesulfonamide
   Show/Hide
C20H20N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0389679
2-[(3S,6R,8Z,11R)-11-[(4-fluorophenyl)methyl]-5,12-bis(oxidanylidene)-3-phenyl-1-oxa-4-azacyclododec-8-en-6-yl]-N-(2-hydroxyethyl)-N-(phenylmethyl)ethanamide
   Show/Hide
C34H37FN2O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0389714
1-(2-chloranyl-5-piperidin-1-ylsulfonyl-phenyl)-3-(3-chlorophenyl)urea
   Show/Hide
C18H19Cl2N3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0394443
5-nitro-N-[3-(trifluoromethyl)cyclohexyl]-2-furamide
   Show/Hide
C12H13F3N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0394809
1-(4-fluorophenyl)-3-[(2S,3R)-3-methyl-2-[[methyl-[(4-phenoxyphenyl)methyl]amino]methyl]-6-oxidanylidene-5-[(2S)-1-oxidanylpropan-2-yl]-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]urea
   Show/Hide
C36H39FN4O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0401313
3-[(4-chlorophenyl)sulfonyl-methyl-amino]-4-methoxy-N-(4-methoxyphenyl)benzenesulfonamide
   Show/Hide
C21H21ClN2O6S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0401615
(E)-1-(5-nitro-2-furanyl)-3-(3-nitrophenyl)-2-propen-1-one
   Show/Hide
C13H8N2O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0406470
MLS003107001
   Show/Hide
C23H32O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0413626
5-[(4-chlorophenyl)carbamoylamino]-3-methyl-thiophene-2-carboxylic acid ethyl ester
   Show/Hide
C15H15ClN2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0413644
4-[1-(4-chlorophenyl)tetrazol-5-yl]sulfanylthieno[2,3-d]pyrimidine
   Show/Hide
C13H7ClN6S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0418194
4-(2-cyclopropyl-1,3-oxazol-5-yl)-N-(2,6-dimethylphenyl)benzenesulfonamide
   Show/Hide
C20H20N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0423983
5-Nitro-furan-2-carboxylic acid {3-[(furan-2-carbonyl)-amino]-phenyl}-amide
   Show/Hide
C16H11N3O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0429361
1,2-dihydroacenaphthylen-5-yl-[1-[(6-methyl-2-pyridinyl)methyl]-3-piperidinyl]methanone
   Show/Hide
C25H26N2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0431727
2-[2-bromanyl-6-ethoxy-4-[(E)-(4-oxidanylidenechromen-3-ylidene)methyl]phenoxy]-N,N-dimethyl-ethanamide
   Show/Hide
C22H22BrNO5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0439264
1-(4-methyl-3-piperidin-1-ylsulfonyl-phenyl)-3-(phenylmethyl)thiourea
   Show/Hide
C20H25N3O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0442210
3-(benzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-(4-methyl-1,3-benzothiazol-2-yl)propanamide
   Show/Hide
C22H27N3O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0447550
2-[4-(4-chlorophenyl)benzyl]-5-[[1-[2-(1,3-dioxan-2-yl)ethyl]triazol-4-yl]methyl]-1,1-diketo-3-methyl-1,2,5-thiadiazepan-4-one
   Show/Hide
C27H32ClN5O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0449696
5-nitro-N-(3-pyridinyl)-2-thiophenecarboxamide
   Show/Hide
C10H7N3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0449880
(E)-1-(5-nitro-2-furyl)-3-(o-tolyl)prop-2-en-1-one
   Show/Hide
C14H11NO4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0452927
2-[5-[(3,4-dichlorobenzyl)thio]-4-(2-thenyl)-1,2,4-triazol-3-yl]pyridine
   Show/Hide
C19H14Cl2N4S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0454668
(2S)-2-[[4-[(3-chlorophenyl)carbamoyl]-1H-imidazole-5-carbonyl]amino]-3-phenyl-propionic acid tert-butyl ester
   Show/Hide
C24H25ClN4O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0457806
2-(4,6-dimethyl-2-pyrimidinyl)-1-(2-phenylphenyl)guanidine
   Show/Hide
C19H19N5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0460481
(2R,3R)-2,3-bis(phenylmethyl)-1,4-dioxaspiro[4.5]deca-6,9-dien-8-one
   Show/Hide
C22H20O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0461460
5-chloranyl-N-(2,6-dimethylphenyl)-2-[(3-methylphenyl)methylsulfonyl]pyrimidine-4-carboxamide
   Show/Hide
C21H20ClN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0462616
1-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-3-phenyl-urea
   Show/Hide
C20H19N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0464109
5-chloro-2-(3-methylbenzyl)sulfonyl-N-piperonyl-pyrimidine-4-carboxamide
   Show/Hide
C21H18ClN3O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0465515
(E)-3-(3-methylphenyl)-1-(5-nitro-2-furanyl)-2-propen-1-one
   Show/Hide
C14H11NO4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0466288
(2S,3S)-2,3-bis(p-anisyl)-1,4-dioxaspiro[4.5]deca-6,9-dien-8-one
   Show/Hide
C24H24O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0468723
(4-Fluoro-benzyl)-[3-(4-fluoro-phenyl)-3-(4-methoxy-phenyl)-propyl]-amine
   Show/Hide
C23H23F2NO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0487993
1-(3,5-dichlorobenzoyl)-4-[1-[(3-methylphenyl)methoxy]-3-phenylpropan-2-yl]-1,4-diazepan-5-one
   Show/Hide
C29H30Cl2N2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0508565
3-(5-chloranyl-2-oxidanyl-phenyl)-3-phenyl-N-(1-phenylethyl)propanamide
   Show/Hide
C23H22ClNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0508856
3-Fluoro-N-[3-nitro-5-(pyridin-2-ylsulfanyl)-phenyl]-benzamide
   Show/Hide
C18H12FN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0514304
4,5-dihydro-2H-benz[g]indazol-3-yl-(4-piperonylpiperazino)methanone
   Show/Hide
C24H24N4O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0518203
MLS000582357
   Show/Hide
C16H22ClN3OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0521691
2-(2-phenoxyethylsulfonyl)-1H-benzimidazole
   Show/Hide
C15H14N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0650169
SID24793346
   Show/Hide
C17H20ClN3OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0650792
GNF-Pf-1644
   Show/Hide
C26H21FN2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0654225
SID17431493
   Show/Hide
C30H45ClN2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0655489
SID17506455
   Show/Hide
C20H21N3O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0660005
MMV1506686
   Show/Hide
C11H8ClN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0665122
SID16953491
   Show/Hide
C19H13BrN4O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0675150
SID24779760
   Show/Hide
C32H40N2O6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0686021
SID17387498
   Show/Hide
C19H17N3O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0695973
SID857671
   Show/Hide
C19H21ClFNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0700454
SID24821451
   Show/Hide
C15H11N3O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0700998
1-(4-tert-butylphenyl)-3-(5-chloro-2-hydroxyphenyl)propane-1,3-dione
   Show/Hide
C19H19ClO3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0712439
SID17432729
   Show/Hide
C17H12ClN3O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0712828
SID22402539
   Show/Hide
C18H21N7O4S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0718794
SID49822752
   Show/Hide
C11H5ClN4O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0721163
SID24791345
   Show/Hide
C18H14N4O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0724123
SID22416907
   Show/Hide
C19H16N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0724867
SID49733384
   Show/Hide
C23H22N4O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0730773
SID26732040
   Show/Hide
C30H28N4O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0736690
SID85304815
   Show/Hide
C24H22FN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0741660
SID22412900
   Show/Hide
C15H16Cl2N4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0747112
N-(3-chloro-4-morpholinophenyl)-5-nitrofuran-2-carboxamide
   Show/Hide
C15H14ClN3O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0752002
SID17507620
   Show/Hide
C18H15ClF3N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0760000
SID17387029
   Show/Hide
C19H18BrNO3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0768554
SID17517261
   Show/Hide
C24H26N4O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0771055
SID24793086
   Show/Hide
C22H19ClN4O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0773707
SID47202561
   Show/Hide
C19H20ClNO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0781899
SID17505822
   Show/Hide
C29H24N2O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0787778
SID17506577
   Show/Hide
C19H18BrNO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0790724
SID845300
   Show/Hide
C17H20ClNO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0797599
SID26658583
   Show/Hide
C20H20N2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0803128
SID22406672
   Show/Hide
C25H22ClN5O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0803172
SID17504147
   Show/Hide
C18H12BrFN4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0803296
SID17411844
   Show/Hide
C18H15Cl2N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0810524
SID24781522
   Show/Hide
C20H18N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0812816
SID849093
   Show/Hide
C10H9BrN6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0813706
SID22402986
   Show/Hide
C27H25NO3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0814030
SID24816137
   Show/Hide
C14H12N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0816037
SID14738998
   Show/Hide
C24H25ClN2O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0817824
1-cyclohexyl-3-[(Z)-N'-(4-methylquinazolin-2-yl)carbamimidoyl]urea
   Show/Hide
C17H22N6O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0818133
SID24800735
   Show/Hide
C24H26ClN3O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0818149
SID14743084
   Show/Hide
C26H20N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0825094
SID24792667
   Show/Hide
C13H13N3O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0829960
SID24806855
   Show/Hide
C14H15BrN4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0832518
SID24790634
   Show/Hide
C23H36ClNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0847685
SID49734785
   Show/Hide
C27H31BrClN5OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0849483
SID99356804
   Show/Hide
C25H30ClFN4O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0850046
SID99454054
   Show/Hide
C24H25BrN4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0851453
SID17507284
   Show/Hide
C22H16BrN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0852457
SID121283957
   Show/Hide
C38H55N5O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0852859
SID121285261
   Show/Hide
C21H16BrFN2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0852861
SID14728475
   Show/Hide
C30H42N2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0852867
SID49668724
   Show/Hide
C21H17N3O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0856583
SID99495120
   Show/Hide
C17H14Cl2N4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0856926
2-piperidyl-[2-(trifluoromethyl)-6-[4-(trifluoromethyl)phenyl]-4-pyridyl]methanol
   Show/Hide
C19H18F6N2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0857218
SID22415875
   Show/Hide
C21H21ClN2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0857418
SID56315014
   Show/Hide
C22H24ClF3N4O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0858487
SID24815617
   Show/Hide
C21H25ClFN3O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0860347
SID51088780
   Show/Hide
C16H13FN2O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0860961
SID56319613
   Show/Hide
C22H29N5O6S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0864801
SID87341718
   Show/Hide
C25H25NO3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0864849
SID103060209
   Show/Hide
C23H17ClF3N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0864850
SID85268858
   Show/Hide
C24H21N3O9S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0864853
SID26732337
   Show/Hide
C31H31FN2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0865590
SID121285025
   Show/Hide
C28H31N7O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0865637
SID103074105
   Show/Hide
C20H13Cl2FN2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0866000
SID103050345
   Show/Hide
C15H14N4O6S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0866135
SID49731925
   Show/Hide
C23H29N3O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0867315
SID99359317
   Show/Hide
C35H47F3N4O7S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0867355
SID85201294
   Show/Hide
C29H34ClN3O7S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0867356
SID24814804
   Show/Hide
C16H14ClN3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0867357
SID103060265
   Show/Hide
C24H22N2O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0872825
SID49646136
   Show/Hide
C20H23Cl2NO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0873560
SID92764769
   Show/Hide
C15H20ClNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0874987
SID92764858
   Show/Hide
C30H37ClN2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0875071
SID49673483
   Show/Hide
C23H20N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0875072
SID121284600
   Show/Hide
C20H17BrN2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0879388
SID26730101
   Show/Hide
C18H17NO6
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0879609
SID121285472
   Show/Hide
C30H33N7O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0880917
SID99205795
   Show/Hide
C22H26ClN3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0882448
SID103060529
   Show/Hide
C28H30N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0882469
SID56320908
   Show/Hide
C27H30ClNO10
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0883098
SID92764806
   Show/Hide
C28H45BrN2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0884468
SID93576585
   Show/Hide
C21H25N3O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0884471
SID49679576
   Show/Hide
C21H17N3O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0884729
SID26728484
   Show/Hide
C21H25N3O2S3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0884985
SID56316424
   Show/Hide
C24H25ClF3N5O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0885795
SID14746324
   Show/Hide
C14H12Cl2N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0887476
SID87349247
   Show/Hide
C35H39N5O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0887506
SID51085113
   Show/Hide
C27H34F3N3O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0887507
SID99494642
   Show/Hide
C22H26N4O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0887508
SID99360016
   Show/Hide
C27H17F2N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0887585
SID92764802
   Show/Hide
C16H22ClNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0889065
SID99494745
   Show/Hide
C18H21F3N4O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0890127
SID99357067
   Show/Hide
C37H34F6N6O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0890140
SID49667069
   Show/Hide
C18H24N4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0890145
SID22410472
   Show/Hide
C27H21ClN2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0890226
SID92763672
   Show/Hide
C41H53N5O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0893805
SID24790542
   Show/Hide
C19H30N2O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0895406
SID85268652
   Show/Hide
C23H23ClN4O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0898576
SID85200522
   Show/Hide
C35H39FN2O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0899320
SID57261070
   Show/Hide
C23H21FN2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0900383
SID99454868
   Show/Hide
C23H20N4O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0904613
SID22409685
   Show/Hide
C27H33N5O5S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0904621
SID81066753
   Show/Hide
C19H14F3N5O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0905357
SID92764831
   Show/Hide
C17H24ClNO2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0906130
SID92763666
   Show/Hide
C38H55N5O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0906889
SID121285083
   Show/Hide
C30H35N7
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0907488
SID57258776
   Show/Hide
C25H27ClN2O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0907508
SID103163471
   Show/Hide
C23H16ClF4NO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0907583
SID87336924
   Show/Hide
C37H37ClF3N5O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0908148
SID121282828
   Show/Hide
C20H18N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0908462
CO-ADD:0135932
   Show/Hide
C14H10N2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0908463
SID17387361
   Show/Hide
C24H20N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0908464
SID99454630
   Show/Hide
C18H21F3N4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0909083
SID57260737
   Show/Hide
C14H9Br2ClN4O2S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0909326
SID87336768
   Show/Hide
C36H49ClN4O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0909984
SID103076663
   Show/Hide
C19H16ClF2N3O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0910414
SID103162717
   Show/Hide
C30H29Cl2N3O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0910503
SID103163266
   Show/Hide
C21H23NO3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0910530
SID17413607
   Show/Hide
C24H30N2O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0910595
SID26725984
   Show/Hide
C20H18N4O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0911986
SID103050514
   Show/Hide
C25H25ClN2O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0912251
SID17411938
   Show/Hide
C24H26N2O3S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0912252
SID49647966
   Show/Hide
C24H23FN4OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0912448
SID56318036
   Show/Hide
C22H29N5O5S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0912489
SID121283770
   Show/Hide
C37H47N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0917864
SID87345531
   Show/Hide
C38H55N5O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0917873
SID24789165
   Show/Hide
C14H15ClN4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0919856
SID49667170
   Show/Hide
C16H12F3N3O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0920060
SID92764827
   Show/Hide
C34H47Cl3N6O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0921308
SID121282779
   Show/Hide
C22H19ClN2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0921523
SID56315085
   Show/Hide
C27H31N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0923478
SID99356675
   Show/Hide
C23H31ClN4O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0923551
SID121285000
   Show/Hide
C24H29N7OS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0923553
SID85201403
   Show/Hide
C35H38N4O5
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0923835
SID92763957
   Show/Hide
C15H21NOS
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0924001
SID87342346
   Show/Hide
C34H48N4O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0924104
SID92763379
   Show/Hide
C29H33NO10
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0928399
SID46501024
   Show/Hide
C26H30N4O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0940374
SID121283171
   Show/Hide
C11H8N6O
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0945088
SID92763667
   Show/Hide
C39H57N5O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0947417
SID51086189
   Show/Hide
C20H19ClN4O3S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0947858
SID121284993
   Show/Hide
C28H31N7O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0948583
SID17514210
   Show/Hide
C28H25N3O4S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0949816
SID85148538
   Show/Hide
C23H27F3N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0951532
SID92763650
   Show/Hide
C35H57N5OS2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0952404
SID121283950
   Show/Hide
C42H55N5O2S2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0956944
SID56323233
   Show/Hide
C26H22FN3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0956945
SID85201301
   Show/Hide
C32H35N5O6S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0959038
SID92764493
   Show/Hide
C15H12FNO
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0960197
SID121285075
   Show/Hide
C26H28N6S
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0960993
GNF-Pf-2356
   Show/Hide
C20H23ClN4O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0961321
SID85148527
   Show/Hide
C29H26F4N2O4
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0961998
SID103075452
   Show/Hide
C22H16F3N3O3
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0966668
SID47196384
   Show/Hide
C16H18N2O2
 1
1
Potency ~ 29092.9 nM
   TI
   LI
   LO
   TS
CP0056178
4-fluoranyl-N-(4-oxidanyl-3-quinolin-8-ylsulfanyl-naphthalen-1-yl)benzenesulfonamide
   Show/Hide
C25H17FN2O3S2
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0094185
4-methoxy-N-[4-oxidanyl-3-(1H-1,2,4-triazol-5-ylsulfanyl)naphthalen-1-yl]benzenesulfonamide
   Show/Hide
C19H16N4O4S2
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0106324
(4-fluorobenzyl)-(2-phenylquinazolin-4-yl)amine
   Show/Hide
C21H16FN3
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0135396
2-[(7-chloranyl-[1,2,4]triazolo[3,4-c][1,2,4]benzotriazin-1-yl)sulfanyl]-N,N-diethyl-ethanamide
   Show/Hide
C14H15ClN6OS
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0196742
10-phenothiazinecarbothioic acid S-(5-methyl-1,3,4-thiadiazol-2-yl) ester
   Show/Hide
C16H11N3OS3
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0335232
5-[1-(2,5-dimethylphenyl)sulfonyl-4-piperidinyl]-3-[(4-methylphenyl)methyl]-2H-triazolo[4,5-d]pyrimidin-7-one
   Show/Hide
C25H28N6O3S
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0352388
2-benzylsulfonyl-5-chloro-N-(4-fluorophenyl)pyrimidine-4-carboxamide
   Show/Hide
C18H13ClFN3O3S
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0352632
5-[2-(1-cyclohexenyl)ethylsulfamoyl]-2-fluoro-N-(4-methylphenyl)benzamide
   Show/Hide
C22H25FN2O3S
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0378195
3-(4-Phenyl-6-trifluoromethyl-pyrimidine-2-sulfonyl)-propionic acid methyl ester
   Show/Hide
C15H13F3N2O4S
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0378347
4-(4-benzylpiperazin-1-yl)-7-nitro-3-oxido-2,1,3-benzoxadiazol-3-ium
   Show/Hide
C17H17N5O4
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0450694
5-Fluoro-1-(3,4-dideoxy-3-fluoro-6-O-trityl-.beta.-D-glycero-hex-3-enopyranos-2-ulosyl) uracil
   Show/Hide
C29H22F2N2O5
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0841757
SID24822841
   Show/Hide
C18H13ClN2O3
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0848045
SID103075820
   Show/Hide
C26H23F3N4OS
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0852171
SID89855697
   Show/Hide
C17H13NO5
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0872682
SID92764123
   Show/Hide
C11H12N4O4
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0875070
SID51086071
   Show/Hide
C18H18N2O4S2
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0907494
SID87349250
   Show/Hide
C35H42N4O5
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0921189
SID81066866
   Show/Hide
C44H68O13
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS
CP0925810
SID121285482
   Show/Hide
C29H33N7O2
 1
1
Potency ~ 32642.7 nM
   TI
   LI
   LO
   TS