| Compound ID |
Compound Name |
Compound Formula |
|
CP0504385
|
3-[2-(4-isopropylphenyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-6,6-dimethyl-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C30H30F3N3O3
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0480497
|
3-[2-(4-chlorophenyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-6,6-dimethyl-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C27H23ClF3N3O3
|
1
|
| 1 |
IC50 = 221 nM
|
|
|
|
CP0428615
|
6,6-dimethyl-3-{5-methyl-3-oxo-2-[4-(trifluoromethoxy)phenyl]-2,3-dihydro-1H-pyrazol-4-yl}-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C28H23F6N3O4
|
1
|
| 1 |
IC50 = 337 nM
|
|
|
|
CP0495958
|
3-[2-(4-methyllphenyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-6,6-dimethyl-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C28H26F3N3O3
|
1
|
| 1 |
IC50 = 375 nM
|
|
|
|
CP0485234
|
3-[2-(4-methoxyphenyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-6,6-dimethyl-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C28H26F3N3O4
|
1
|
| 1 |
IC50 = 503 nM
|
|
|
|
CP0515764
|
3-[2-(4-cyanophenyl)-5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl]-6,6-dimethyl-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C28H23F3N4O3
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0857816
|
2-[(1-Methyl-1H-imidazol-4-yl)sulfonyl]-N-[4-(propan-2-yloxy)phenyl]-2-azabicyclo[2.2.2]octane-6-carboxamide
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|
C21H28N4O4S
|
1
|
| 1 |
IC50 = 1510 nM
|
|
|
|
CP0443407
|
6,6-dimethyl-3-(5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione
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|
C27H24F3N3O3
|
1
|
| 1 |
IC50 > 10 nM
|
|
|