| Compound ID |
Compound Name |
Compound Formula |
|
CP0467692
|
2-[4-(trifluoromethoxy)phenyl]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C13H5F6N3O2S
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0451004
|
2-(propylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C9H9F3N4OS
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0405396
|
2-(4-methylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C13H8F3N3OS
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0405395
|
2-phenyl-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C12H6F3N3OS
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0405397
|
2-(3-methoxyanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C13H9F3N4O2S
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0471775
|
2-(3,5-dimethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H10F3N3OS
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0451005
|
2-(3-nitrophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C12H5F3N4O3S
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0482624
|
2-(4-methoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C13H8F3N3O2S
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0482625
|
7-(trifluoromethyl)-2-[3-(trifluoromethyl)phenyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C13H5F6N3OS
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0563374
|
2-(4-aminoanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C12H8F3N5OS
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0563494
|
2-(butylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C10H11F3N4OS
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0482621
|
2-(3-fluorophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
Show/Hide
|
C12H5F4N3OS
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0432301
|
2-(3,5-dimethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H10F3N3O3S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0482617
|
2-(pentylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C11H13F3N4OS
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0432302
|
2-(4-ethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
Show/Hide
|
C14H10F3N3O2S
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0467693
|
2-(prop-2-enylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C9H7F3N4OS
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
|
CP0429927
|
3-[5-oxo-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-2-yl]benzonitrile
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|
C13H5F3N4OS
|
1
|
| 1 |
IC50 = 1120 nM
|
|
|
|
CP0482622
|
2-(3-phenylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C18H10F3N3OS
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
|
CP0482619
|
2-(3,4-dimethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H10F3N3OS
|
1
|
| 1 |
IC50 = 1750 nM
|
|
|
|
CP0471820
|
2-(4-ethoxyanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H11F3N4O2S
|
1
|
| 1 |
IC50 = 2020 nM
|
|
|
|
CP0451003
|
2-[amino(methyl)amino]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C7H6F3N5OS
|
1
|
| 1 |
IC50 = 2220 nM
|
|
|
|
CP0482618
|
2-[2-(dimethylamino)ethylamino]-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C10H12F3N5OS
|
1
|
| 1 |
IC50 = 3750 nM
|
|
|
|
CP0471819
|
2-(4-ethylphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H10F3N3OS
|
1
|
| 1 |
IC50 = 4550 nM
|
|
|
|
CP0455729
|
2-(dibutylamino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C14H19F3N4OS
|
1
|
| 1 |
IC50 = 4630 nM
|
|
|
|
CP0467691
|
2-(4-propan-2-ylanilino)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
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|
C15H13F3N4OS
|
1
|
| 1 |
IC50 = 31500 nM
|
|
|
|
CP0036918
|
(2S)-2-amino-3-phenylpropanoic acid
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|
C9H11NO2
|
1
|
| 1 |
IC50 = 80200 nM
|
|
|
|
CP0432303
|
2-(2-ethoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
Show/Hide
|
C14H10F3N3O2S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0467694
|
2-(2-fluorophenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
Show/Hide
|
C12H5F4N3OS
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0482620
|
2-(2-methoxyphenyl)-7-(trifluoromethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
Show/Hide
|
C13H8F3N3O2S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
