Brief Information of the Cell Line and Protein
Cell Line ID: CL000053 , COS-7
Synonyms
Cos-7
COS 7
Cos 7
COS7
Cos7
CV-1 in Origin Simian-7
Category Transformed cell line
Organism
Chlorocebus aethiops (Green monkey)
Cellosaurus ID
CVCL_0224
Protein ID: PT02174 , Melatonin receptor type 1B
Gene Name MTNR1B
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P49286
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000053  Protein ID: PT02174
 
Compound ID Compound Name Compound Formula
CP0060238
N-[2-(6-chloro-5-methoxy-1H-indol-3-yl)ethyl]acetamide
   Show/Hide
C13H15ClN2O2
 1
1
Ki = 0.2 nM
   TI
   LI
   LO
   TS
CP0055675
2-Iodomelatonin
   Show/Hide
C13H15IN2O2
 1
1
Ki = 0.22 nM
   TI
   LI
   LO
   TS
CP0401149
Luzindole,5-Methoxy
   Show/Hide
C20H22N2O2
 1
1
Ki = 0.25 nM
   TI
   LI
   LO
   TS
CP0397235
1-[3-(5-Methoxy-1H-indol-3-yl)piperidino]ethanone
   Show/Hide
C16H20N2O2
 1
1
Ki = 0.8 nM
   TI
   LI
   LO
   TS
CP0114370
4-P-PDOT
   Show/Hide
C19H21NO
 1
1
Ki = 1.5 nM
   TI
   LI
   LO
   TS
CP0415639
N-[2-(6-chloro-5-methoxy-2-methyl-1H-indol-3-yl)ethyl]acetamide
   Show/Hide
C14H17ClN2O2
 1
1
Ki = 2.2 nM
   TI
   LI
   LO
   TS
CP0401148
melatonin, 6-Methoxy
   Show/Hide
C14H18N2O3
 1
1
Ki = 3.5 nM
   TI
   LI
   LO
   TS
CP0260237
CAS_117946-91-5
   Show/Hide
C19H20N2O
 1
1
Ki = 10.2 nM
   TI
   LI
   LO
   TS