Brief Information of the Cell Line and Protein
Cell Line ID: CL000053 , COS-7
 Cell Line Info 
Synonyms
Cos-7
COS 7
Cos 7
COS7
Cos7
CV-1 in Origin Simian-7
Category Transformed cell line
Organism
Chlorocebus aethiops (Green monkey)
Cellosaurus ID
CVCL_0224
Protein ID: PT00958 , Cholecystokinin receptor type A
 Protein Info 
Gene Name CCKAR
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P32238
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000053
 Cell Line Info 
 Protein ID: PT00958
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0191267
 Compound Info 
(2R)-2-[[2-(1H-indole-2-carbonylamino)benzoyl]amino]-4-phenylbutanoic acid
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C26H23N3O4
  11
1
Ki = 0.32 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 2.3 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
3
Ki = 3.7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
4
Ki = 3.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
5
Ki = 4.9 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
6
Ki = 5 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
7
Ki = 5.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
8
Ki = 7.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
9
Ki = 19.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
10
Ki = 39.1 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
11
Ki = 522 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0079600
 Compound Info 
2-[[2-(1H-indole-2-carbonylamino)benzoyl]amino]-4-phenylbutanoic acid
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C26H23N3O4
  1
1
Ki = 3.9 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0161714
 Compound Info 
N-(1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl)-1H-indole-2-carboxamide
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C25H20N4O2
  1
1
Ki = 10.4 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0276701
 Compound Info 
(+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-phenylpropanoic acid
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C25H21N3O4
  1
1
Ki = 59.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0285872
 Compound Info 
(2S)-2-[[2-(1H-indole-2-carbonylamino)benzoyl]amino]-4-phenylbutanoic acid
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C26H23N3O4
  1
1
Ki = 973 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS