| Compound ID |
Compound Name |
Compound Formula |
|
CP0433973
|
[5-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]pyridin-2-yl]methanol
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|
C23H24FN5O
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0440005
|
6-fluoro-1-[1-[6-(6-methylpyridin-3-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C23H24FN5
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0445540
|
2-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]-4-methyl-1,3-thiazole
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|
C21H22FN5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0304175
|
[1-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]imidazol-4-yl]methanol
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|
C21H23FN6O
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0324513
|
6-fluoro-1-[1-[6-(6-methoxypyridin-3-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C23H24FN5O
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0213491
|
[1-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]pyrazol-4-yl]methanol
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|
C21H23FN6O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0392902
|
6-fluoro-1-[1-[6-(5-methylthiophen-2-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C22H23FN4S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0432919
|
5-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]-N-methylpyridine-2-carboxamide
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|
C24H25FN6O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0292970
|
[4-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]phenyl]methanol
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|
C24H25FN4O
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0079592
|
6-fluoro-1-[1-[6-(4-methylimidazol-1-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C21H23FN6
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0445542
|
1-[1-[6-(4-ethoxypyrazol-1-yl)pyridazin-3-yl]piperidin-4-yl]-6-fluoro-2,3-dihydroindole
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|
C22H25FN6O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0392900
|
6-fluoro-1-[1-[6-(4-methylphenyl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C24H25FN4
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0466048
|
2-[1-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]pyrazol-4-yl]ethanol
Show/Hide
|
C22H25FN6O
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0432920
|
2-[4-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]pyrazol-1-yl]-N-methylacetamide
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|
C23H26FN7O
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0560917
|
2-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]-5-methyl-1,3-thiazole
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|
C21H22FN5S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0560916
|
6-fluoro-1-[1-[6-[6-(trifluoromethyl)pyridin-3-yl]pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C23H21F4N5
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0064713
|
BDBM50448680
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|
C21H23FN6
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0443931
|
2-[4-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]pyrazol-1-yl]ethanol
Show/Hide
|
C22H25FN6O
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0505141
|
6-fluoro-1-[1-[6-(4-methylpyrazol-1-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C21H23FN6
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0119637
|
BDBM50448674
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|
C21H21FN6
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0440007
|
6-chloro-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
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|
C21H23ClN6
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0466047
|
1-[1-[6-(1-ethylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-6-fluoro-2,3-dihydroindole
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|
C22H25FN6
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0549748
|
5-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]-N,N-dimethylpyridin-2-amine
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|
C24H27FN6
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0445541
|
1-[1-[6-[1-(2-ethoxyethyl)pyrazol-4-yl]pyridazin-3-yl]piperidin-4-yl]-6-fluoro-2,3-dihydroindole
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|
C24H29FN6O
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0240700
|
1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-6-(trifluoromethyl)-2,3-dihydroindole
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|
C22H23F3N6
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0432921
|
6-fluoro-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]indazole
Show/Hide
|
C20H20FN7
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0217904
|
BDBM50448682
Show/Hide
|
C23H22F2N4
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0440006
|
6-fluoro-1-[1-[6-(1-propylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C23H27FN6
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0505142
|
5-fluoro-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C21H23FN6
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0466038
|
5-chloro-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C21H23ClN6
|
1
|
| 1 |
IC50 = 218 nM
|
|
|
|
CP0313371
|
6-methyl-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C22H26N6
|
1
|
| 1 |
IC50 = 241 nM
|
|
|
|
CP0466070
|
4-[6-[4-(6-fluoro-2,3-dihydroindol-1-yl)piperidin-1-yl]pyridazin-3-yl]benzoic acid
Show/Hide
|
C24H23FN4O2
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0445543
|
6-methoxy-1-[1-[6-(1-methylpyrazol-4-yl)pyridazin-3-yl]piperidin-4-yl]-2,3-dihydroindole
Show/Hide
|
C22H26N6O
|
1
|
| 1 |
IC50 = 407 nM
|
|
|
