| Compound ID |
Compound Name |
Compound Formula |
|
CP0222241
|
US9073922, 87
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|
C19H18FN3O
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0265963
|
US9073922, 101
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|
C21H20FN3O3
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0143255
|
US9073922, 226
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|
C21H20FN3O3
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0341118
|
US9073922, 215
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|
C21H21FN4O2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0726326
|
(1r,4r)-4-(4-(5-fluoro-4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexanecarboxylic acid
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|
C26H27F2N3O3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0965399
|
(1s,4s)-4-(4-(5-fluoro-4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexanecarboxylic acid
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|
C26H27F2N3O3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0962478
|
1-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)cyclohex-3-enyl)piperidine-4-carboxylic acid
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|
C27H29F2N3O3
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0968689
|
2-((1r,4r)-4-(4-(5-fluoro-4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexyl)acetic acid
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|
C27H29F2N3O3
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0567168
|
US9796708, Example 228
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|
C22H23FN4O5S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0773151
|
(1s,4s)-4-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexanecarboxylic acid
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|
C26H28FN3O3
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0128822
|
US9073922, 288
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|
C27H30FN3O3
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0265979
|
US9073922, 119
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|
C20H20FN3O3S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0914334
|
(1r,4r)-4-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexanecarboxylic acid
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|
C26H28FN3O3
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0132970
|
US9073922, 289
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|
C27H30FN3O3
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0565903
|
US9073922, 241
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|
C25H28FN3O3
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0968691
|
2-(4-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)cyclohex-3-enyl)piperazin-1-yl)acetic acid
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|
C26H29FN4O3
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0961574
|
4-[4-(5-fluoro-2-methoxy-phenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-N-methylsulfonyl-cyclohex-3-ene-1-carboxamide
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|
C22H22FN3O4S
|
1
|
| 1 |
IC50 = 660 nM
|
|
|
|
CP0962662
|
2-(1-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)cyclohex-3-enyl)piperidin-4-yl)acetic acid
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|
C26H28FN3O3
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0965400
|
2-((1s,4s)-4-(4-(5-fluoro-4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dihydropyridin-1(2H)-yl)cyclohexyl)acetic acid
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|
C27H30FN3O3
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0578436
|
(4-{4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2H)-yl}piperidin-1-yl)acetic acid
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|
C26H29FN4O3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0963886
|
2-[[4-[4-(5-fluoro-2-methoxy-phenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]cyclohex-3-en-1-yl]amino]acetic acid
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|
C22H22FN3O3
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0697060
|
US9073922, 219
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|
C21H19FN2O3
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0968690
|
2-(4-(4-(4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl)cyclohex-3-enyl)piperidin-1-yl)acetic acid
Show/Hide
|
C27H30FN3O3
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
