Brief Information of the Cell Line and Protein
Cell Line ID: CL000049 , C6
Synonyms
C-6
C 6
RGC-6
RGC6
RGc6
Category Cancer cell line
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_0194
Protein ID: PT06071 , Sodium- and chloride-dependent glycine transporter 2
Gene Name SLC6A5
Organism Rattus norvegicus, Rat
Protein Classification Transporter
Uniprot ID P58295
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000049  Protein ID: PT06071
 
Compound ID Compound Name Compound Formula
CP0410012
5-Biphenyl-4-yl-4-(2-fluorophenyl)-N-methyl-4H-1,2,4-triazol-3-amine
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C21H17FN4
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0373521
3-Biphenyl-4-yl-5-ethyl-4-(2-fluorophenyl)-1,2,4-triazole
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C22H18FN3
 1
1
IC50 = 230 nM
   TI
   LI
   LO
   TS
CP0379616
2-(3-Biphenyl-4-yl-5-methyl-4H-1,2,4-triazole-4-yl)benzonitrile
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C22H16N4
 1
1
IC50 = 260 nM
   TI
   LI
   LO
   TS
CP0379733
3-Biphenyl-4-yl-4-(2-chlorophenyl)-5-methyl-4H-1,2,4-triazole
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C21H16ClN3
 1
1
IC50 = 280 nM
   TI
   LI
   LO
   TS
CP0379732
3-Biphenyl-4-yl-4-(2-fluorophenyl)-5-methyl-4H-1,2,4-triazole
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C21H16FN3
 1
1
IC50 = 340 nM
   TI
   LI
   LO
   TS
CP0425664
3-Biphenyl-4-yl-5-methyl-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
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C22H16F3N3
 1
1
IC50 = 600 nM
   TI
   LI
   LO
   TS
CP0500543
2-(3-(biphenyl-4-yl)-5-methyl-4H-1,2,4-triazol-4-yl)phenol
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C21H17N3O
 1
1
IC50 = 680 nM
   TI
   LI
   LO
   TS
CP0425665
3-Biphenyl-4-yl-5-methyl-4-(2-methylphenyl)-4H-1,2,4-triazole
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C22H19N3
 1
1
IC50 = 780 nM
   TI
   LI
   LO
   TS
CP0511752
3-Biphenyl-4-yl-4-(2-fluorophenyl)-5-methoxy-4H-1,2,4-triazole
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C21H16FN3O
 1
1
IC50 = 990 nM
   TI
   LI
   LO
   TS
CP0389819
3-Biphenyl-4-yl-5-methyl-4-phenyl-4H-1,2,4-triazole
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C21H17N3
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0402966
3-Biphenyl-4-yl-4-(2-methoxy-phenyl)-5-methyl-4H-[1,2,4]triazole
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C22H19N3O
 1
1
IC50 = 1700 nM
   TI
   LI
   LO
   TS
CP0051811
3-Biphenyl-4-yl-4-(2-fluorophenyl)-5-isopropyl-4H-1,2,4-triazole
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C23H20FN3
 1
1
IC50 = 3300 nM
   TI
   LI
   LO
   TS