| Compound ID |
Compound Name |
Compound Formula |
|
CP0580025
|
(2R)-2-methyl-N'-[2-methyl-5-(2-methylpropanoylamino)pyrazol-3-yl]-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C25H33N7O4
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0578650
|
4-methyl-2-(2-methylpropanoylamino)-N-[(2R)-3,3,3-trifluoro-2-[[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]carbamoyl]propyl]-1,3-thiazole-5-carboxamide
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|
C25H29F3N6O4S
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0579589
|
(2S)-2-cyclobutyl-N'-[2-methyl-5-(2-methylpropanoylamino)pyrazol-3-yl]-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C28H37N7O4
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0546944
|
4-methyl-N-[(2R)-2-methyl-3-oxo-3-[[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]amino]propyl]-2-(2-methylpropanoylamino)-1,3-thiazole-5-carboxamide
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|
C25H32N6O4S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0578315
|
(2R)-N'-[5-(2,2-difluoroethylcarbamoyl)-2-methylpyrazol-3-yl]-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H29F2N7O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0578651
|
(2R)-N'-[4-chloro-2-(2-methylpropanoylamino)-1,3-thiazol-5-yl]-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H29ClN6O4S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0013376
|
N-[(2S,3S)-3-amino-2-hydroxy-3-[4-(trifluoromethoxy)phenyl]propyl]-4-tert-butyl-N-cyclobutylbenzenesulfonamide
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|
C24H31F3N2O4S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0460550
|
(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
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|
C27H28FN5O4
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
