Brief Information of the Compound and Protein
Compound Name
4-methyl-2-(2-methylpropanoylamino)-N-[(2R)-3,3,3-trifluoro-2-[[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]carbamoyl]propyl]-1,3-thiazole-5-carboxamide
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PubChem ID
CID: 162759954
Canonical SMILES
CC(C)C(=O)Nc1nc(C)c(s1)C(=O)NC[C@H](C(=O)N[C@H]1c2ccccc2CN2CCCN2C1=O)C(F)(F)F
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Compound Formula C25H29F3N6O4S
Compound Structure
Protein Name
Signal peptide peptidase-like 2A
Protein Classification
Enzyme
>
Hydrolase
Uniprot ID
Q8TCT8
Gene Name
SPPL2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000043 U2OS Homo sapiens (Human)  1
1
IC50 = 0.5 nM
   TI
   LI
   LO
   TS