| Compound ID |
Compound Name |
Compound Formula |
|
CP0857655
|
N-(2-((3S,4S)-1-(4-(benzo[d][1,3]dioxol-5-yl)-4-hydroxycyclohexyl)-4-ethoxypyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C29H34F3N3O6
|
4
|
| 1 |
Kd = 0.23 nM
|
|
|
| 2 |
Kd = 0.72 nM
|
|
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| 3 |
Kd = 0.9 nM
|
|
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| 4 |
Kd = 1.2 nM
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CP0544332
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5,6-dimethoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C29H34F6N2O3
|
1
|
| 1 |
Ki = 3.9 nM
|
|
|
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CP0479757
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5-methoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H32F6N2O2
|
1
|
| 1 |
Ki = 6.1 nM
|
|
|
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CP0544333
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(6,7-dihydro-5H-cyclopenta[f][1,3]benzodioxol-7-ylamino)-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H30F6N2O3
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
|
CP0165577
|
(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopropyl-3-(tetrahydro-2H-pyran-4-ylamino)cyclopentanecarboxamide
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|
C23H30F6N2O2
|
1
|
| 1 |
Ki = 6.8 nM
|
|
|
|
CP0395825
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5-chloro-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C27H29ClF6N2O
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0449657
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C29H34F6N2O2
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0395824
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5-hydroxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C27H30F6N2O2
|
1
|
| 1 |
Ki = 29 nM
|
|
|
|
CP0238399
|
(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopropyl-3-(tetrahydro-2H-thiopyran-4-ylamino)cyclopentanecarboxamide
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|
C23H30F6N2OS
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0404369
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-propan-2-yl-3-(1,2,3,4-tetrahydronaphthalen-1-ylamino)cyclopentane-1-carboxamide
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|
C28H32F6N2O
|
1
|
| 1 |
Ki = 33 nM
|
|
|
|
CP0389822
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(5-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H32F6N2O2
|
1
|
| 1 |
Ki = 35 nM
|
|
|
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CP0397124
|
(1S,3R)-3-[(4-amino-2,3-dihydro-1H-inden-1-yl)amino]-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C27H31F6N3O
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0331716
|
(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(2,3-dihydro-1H-inden-1-ylamino)-1-isopropylcyclopentanecarboxamide
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|
C27H30F6N2O
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0524891
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(6-cyano-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H29F6N3O
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0397125
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(6-methyl-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H32F6N2O
|
1
|
| 1 |
Ki = 55 nM
|
|
|
|
CP0449762
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(4-cyano-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C28H29F6N3O
|
1
|
| 1 |
Ki = 70 nM
|
|
|
|
CP0404118
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(4-hydroxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C27H30F6N2O2
|
1
|
| 1 |
Ki = 86 nM
|
|
|
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CP0165578
|
(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(cyclohexylamino)-1-isopropylcyclopentanecarboxamide
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|
C24H32F6N2O
|
1
|
| 1 |
Ki = 110 nM
|
|
|
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CP0461993
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-[(4,5-dimethoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C29H34F6N2O3
|
1
|
| 1 |
Ki = 130 nM
|
|
|
|
CP0404117
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(3-phenylpropylamino)-1-propan-2-ylcyclopentane-1-carboxamide
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|
C27H32F6N2O
|
1
|
| 1 |
Ki = 134 nM
|
|
|
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CP0521838
|
(1S,3R)-3-(benzylamino)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-propan-2-ylcyclopentane-1-carboxamide
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|
C25H28F6N2O
|
1
|
| 1 |
Ki = 437 nM
|
|
|
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CP0444063
|
(1S,3R)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(2-phenylethylamino)-1-propan-2-ylcyclopentane-1-carboxamide
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|
C26H30F6N2O
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
