| Compound ID |
Compound Name |
Compound Formula |
|
CP0198695
|
(S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluoromethyl)phenylsulfonamido)piperidine-1-carbonyl)pyrrolidine-1-carboxylate
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|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0074574
|
5-(benzenesulfonyl)-N-[1-[6-(dimethylamino)pyridine-3-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C26H27F3N4O5S2
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0265625
|
tert-butyl (3R)-3-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylate
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|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0074305
|
4-{[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]sulfonyl}benzoic acid
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|
C25H23F3N2O8S3
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0147968
|
5-(benzenesulfonyl)-N-[1-(pyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H22F3N3O5S2
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0108523
|
5-(benzenesulfonyl)-N-[1-(6-morpholin-4-ylpyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C28H29F3N4O6S2
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0151328
|
5-(Phenylsulfonyl)-2-(trifluoromethyl)-N-(1-{[6-(trifluoromethyl)pyridin-3-yl]carbonyl}piperidin-4-yl)benzenesulfonamide
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|
C25H21F6N3O5S2
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0265624
|
5-(benzenesulfonyl)-N-[1-(6-chloropyridine-3-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H21ClF3N3O5S2
|
1
|
| 1 |
EC50 = 140 nM
|
|
|
|
CP0212062
|
tert-butyl (3S)-3-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]pyrrolidine-1-carboxylate
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|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0265626
|
5-(Phenylsulfonyl)-N-[1-(piperidin-4-ylcarbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H28F3N3O5S2
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0168224
|
5-(benzenesulfonyl)-N-[1-(3-cyanophenyl)sulfonylpiperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C25H22F3N3O6S3
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0181362
|
3-{[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]sulfonyl}benzoic acid
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|
C25H23F3N2O8S3
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0254325
|
5-(benzenesulfonyl)-N-[1-[4-(dimethylamino)benzoyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C27H28F3N3O5S2
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0151329
|
5-(Phenylsulfonyl)-N-[1-(piperidin-4-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C25H30F3N3O5S2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0212060
|
(R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluoromethyl)phenylsulfonamido)piperidine-1-carbonyl)pyrrolidine-1-carboxylate
Show/Hide
|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0328999
|
5-(Phenylsulfonyl)-N-[1-(phenylsulfonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H23F3N2O6S3
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0157377
|
5-(Phenylsulfonyl)-N-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H22F3N3O5S2
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0181363
|
4-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]-sulfonyl}amino)piperidin-1-yl]benzoic acid
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|
C25H23F3N2O6S2
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0212056
|
5-(Phenylsulfonyl)-N-{1-[(6-pyrrolidin-1-ylpyridin-3-yl)carbonyl]piperidin-4-yl}-2-(trifluoromethyl)benzenesulfonamide
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|
C28H29F3N4O5S2
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0108522
|
5-(benzenesulfonyl)-N-(1-benzoylpiperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
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|
C25H23F3N2O5S2
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0192098
|
2-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]-sulfonyl}amino)piperidin-1-yl]acetamide
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|
C20H22F3N3O5S2
|
1
|
| 1 |
EC50 = 310 nM
|
|
|
|
CP0265627
|
(S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbonyl)piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
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|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0307969
|
3-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]benzoic acid
Show/Hide
|
C25H23F3N2O6S2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0265629
|
5-(Phenylsulfonyl)-N-{1-[(3R)-pyrrolidin-3-ylcarbonyl]-piperidin-4-yl}-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0192099
|
4-Oxo-4-[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)-phenyl]sulfonyl}amino)piperidin-1-yl]butanoic acid
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|
C22H23F3N2O7S2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0212059
|
tert-butyl 4-[2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]-2-oxoethyl]piperidine-1-carboxylate
Show/Hide
|
C30H38F3N3O7S2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0108524
|
tert-butyl 4-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]piperidine-1-carboxylate
Show/Hide
|
C29H36F3N3O7S2
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0074576
|
2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidin-1-yl]acetic acid
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|
C20H21F3N2O6S2
|
1
|
| 1 |
EC50 = 570 nM
|
|
|
|
CP0192162
|
5-Oxo-5-[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)-phenyl]sulfonyl}amino)piperidin-1-yl]pentanoic acid
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|
C23H25F3N2O7S2
|
1
|
| 1 |
EC50 = 570 nM
|
|
|
|
CP0095572
|
5-(Phenylsulfonyl)-N-[1-(pyridin-2-ylcarbonyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C24H22F3N3O5S2
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0108526
|
5-(benzenesulfonyl)-N-[1-(3-hydroxy-3-methylbutyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H29F3N2O5S2
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
|
CP0265628
|
5-(Phenylsulfonyl)-N-{1-[(3S)-pyrrolidin-3-ylcarbonyl]-piperidin-4-yl}-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0192160
|
(R)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbonyl)piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
|
CP0212064
|
5-(benzenesulfonyl)-N-[1-(3-hydroxypropyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C21H25F3N2O5S2
|
1
|
| 1 |
EC50 = 850 nM
|
|
|
|
CP0300648
|
5-(benzenesulfonyl)-N-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H22ClF3N2O5S2
|
1
|
| 1 |
EC50 = 870 nM
|
|
|
|
CP0265623
|
5-(Phenylsulfonyl)-2-(trifluoromethyl)-N-{1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}benzenesulfonamide
Show/Hide
|
C26H22F6N2O5S2
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
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CP0151330
|
3-[4-({[5-(Phenylsulfonyl)-2-(trifluoromethyl)phenyl]-sulfonyl}amino)piperidin-1-yl]propanoic acid
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|
C21H23F3N2O6S2
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
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CP0168223
|
5-(Phenylsulfonyl)-N-(1-{[3-(2H-tetrazol-5-yl)phenyl]-sulfonyl}piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H23F3N6O6S3
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
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CP0317086
|
5-(benzenesulfonyl)-N-[1-(4-chlorobenzoyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H22ClF3N2O5S2
|
1
|
| 1 |
EC50 = 1800 nM
|
|
|
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CP0191420
|
5-(benzenesulfonyl)-N-[1-(2-chlorobenzoyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H22ClF3N2O5S2
|
1
|
| 1 |
EC50 = 1900 nM
|
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|
