| Compound ID |
Compound Name |
Compound Formula |
|
CP0919189
|
(E)-thyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phenylcarbamoyl oxime
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|
C20H25N3O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0430150
|
5-phenyl-2-pyridin-4-yl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
Show/Hide
|
C25H19N5
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0528293
|
5-phenyl-4-(pyridin-2-ylmethylamino)quinazoline-2-carbonitrile
Show/Hide
|
C21H15N5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0532047
|
5-phenyl-N-(pyridin-2-ylmethyl)-2-(1,3-thiazol-5-yl)quinazolin-4-amine
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|
C23H17N5S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0226778
|
5-phenyl-2-pyridin-3-yl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
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|
C25H19N5
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0875972
|
(E)-2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-phenylcarbamoyl oxime
Show/Hide
|
C18H21N3O2
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0463468
|
US10214511, Example 19
Show/Hide
|
C20H15ClN4
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0528292
|
5-phenyl-N-(pyridin-2-ylmethyl)-2-(trifluoromethyl)quinazolin-4-amine
Show/Hide
|
C21H15F3N4
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0213936
|
5-phenyl-N-(pyridin-2-ylmethyl)-2-pyrimidin-5-ylquinazolin-4-amine
Show/Hide
|
C24H18N6
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0424259
|
2-(3,5-dimethyl-1,2-oxazol-4-yl)-5-phenyl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
Show/Hide
|
C25H21N5O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0410404
|
2-(2-methoxypyrimidin-5-yl)-5-phenyl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
Show/Hide
|
C25H20N6O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0420392
|
5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]-1H-pyridin-2-one
Show/Hide
|
C25H19N5O
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0475187
|
2-(5-methoxypyridin-3-yl)-5-phenyl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
Show/Hide
|
C26H21N5O
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0849439
|
(E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-N-phenylhydrazinecarboxamide
Show/Hide
|
C18H22N4O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0853409
|
(E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-1-methylhydrazinecarboxamide
Show/Hide
|
C19H23ClN4O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0536588
|
5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-2-carbonitrile
Show/Hide
|
C26H18N6
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0532922
|
N-(pyridin-2-ylmethyl)-2-pyrimidin-5-yl-5-[4-(trifluoromethyl)phenyl]quinazolin-4-amine
Show/Hide
|
C25H17F3N6
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0430151
|
5-phenyl-2-(1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)quinazolin-4-amine
Show/Hide
|
C23H18N6
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0463594
|
2-cyclopropyl-5-phenyl-N-(pyridin-2-ylmethyl)quinazolin-4-amine
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|
C23H20N4
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0442773
|
1-[1-(3,4-dimethylphenyl)cyclopropyl]-2-[2-(4-methoxyphenyl)ethyl]-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C20H24N5O+
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0881690
|
(E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-N-(3-(trifluoromethyl)phenyl)hydrazinecarbothioamide
Show/Hide
|
C19H21F3N4S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0559363
|
5-(4-fluorophenyl)-N-(pyridin-2-ylmethyl)-2-pyrimidin-5-ylquinazolin-4-amine
Show/Hide
|
C24H17FN6
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0847376
|
(E)-2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-fluorophenylcarbamoyl oxime
Show/Hide
|
C18H20FN3O2
|
1
|
| 1 |
IC50 = 275 nM
|
|
|
|
CP0869684
|
(E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-N-(4-(methylthio)phenyl)hydrazinecarboxamide
Show/Hide
|
C19H24N4OS
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0441863
|
1-(2,3-dimethylphenyl)-2-[2-(4-methoxyphenyl)ethyl]-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C17H20N5O+
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0529635
|
2-[2-(4-methoxyphenyl)ethyl]-1-[1-(4-methylphenyl)cyclopropyl]-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C19H22N5O+
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0881691
|
(E)-2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-4-(methylthio)phenylcarbamoyl oxime
Show/Hide
|
C19H23N3O2S
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0938857
|
(E)-1-(4-((3-ethyl-1,2-dimethyl-6,7-dihydro-1H-indol-4(5H)-ylideneaminooxy)carbonylamino)phenyl)ethanone
Show/Hide
|
C21H25N3O3
|
1
|
| 1 |
IC50 = 368 nM
|
|
|
|
CP0863020
|
(E)-N-(4-chlorophenyl)-2-(2,3-dimethyl-6,7-dihydro-1H-indol-4(5H)-ylidene)hydrazinecarboxamide
Show/Hide
|
C17H19ClN4O
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0927803
|
(E)-N-(4-acetylphenyl)-2-(2,3-diethyl-1-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-1-methylhydrazinecarboxamide
Show/Hide
|
C23H30N4O2
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0441864
|
2-[2-(4-methoxyphenyl)ethyl]-1-[1-(4-methylphenyl)cyclopentyl]-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C21H26N5O+
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0889980
|
(E)-N-(4-chlorophenyl)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)hydrazinecarboxamide
Show/Hide
|
C18H21ClN4O
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0442650
|
1-[1-(4-methylphenyl)cyclopropyl]-2-(3-phenylpropyl)-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C19H22N5+
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0881341
|
(E)-2-methyl-6,7-dihydro-1H-indol-4(5H)-one O-2-(pyridin-2-yl)ethylcarbamoyl oxime
Show/Hide
|
C19H24N4O2
|
1
|
| 1 |
IC50 = 547 nM
|
|
|
|
CP0503196
|
1-(3,4-dichlorophenyl)-2-[2-(4-methoxyphenyl)ethyl]-2H-1,2,3,4,5-pentazol-1-ylium
Show/Hide
|
C15H14Cl2N5O+
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0868731
|
(E)-2-(3-ethyl-2-methyl-6,7-dihydro-1H-indol-4(5H)-ylidene)-N-(3-(pyrrolidin-2-yl)phenyl)hydrazinecarboxamide
Show/Hide
|
C22H29N5O
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0878258
|
(E)-N-(4-chlorophenyl)-2-(6,7-dihydro-1H-indol-4(5H)-ylidene)hydrazinecarboxamide
Show/Hide
|
C15H15ClN4O
|
1
|
| 1 |
IC50 = 5600 nM
|
|
|
