| Compound ID |
Compound Name |
Compound Formula |
|
CP0868363
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-(4-methylpiperazin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
|
C20H23ClFN7O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0868364
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C15H12Cl2FN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0868365
|
(S)-N-(1-(3-chloro-4-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C17H17ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0868386
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-morpholino-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C19H20ClFN6O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0868389
|
(S)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C18H20N4O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0868397
|
(S)-2-(3-oxo-5-(piperidin-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C22H24F3N5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0868429
|
(S)-N-(1-(4-chlorophenyl)ethyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C16H14ClFN4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870162
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870163
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870164
|
(S)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H16F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870165
|
(S)-2-(5-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H17FN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870166
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C16H13Cl2FN4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870167
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-cyano-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C17H13ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870168
|
(S)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(3-fluoro-4-methylphenyl)ethyl)acetamide
Show/Hide
|
C17H16F2N4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870175
|
2-(7-((R)-3-hydroxypiperidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-((S)-1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C22H24F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870178
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(5,7-dimethyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C17H17ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870298
|
(S)-2-(8-((2,2-difluoroethyl)amino)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C19H21F2N5O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870300
|
(S)-N-(1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H13F4N5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870301
|
(S)-2-(6-chloro-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C16H13ClF3N5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870302
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C15H13ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870303
|
(S)-N-(1-(3,4-dichlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C16H14Cl2N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870306
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-(oxetan-3-ylamino)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C19H19ClFN5O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870311
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0870314
|
(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H18N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870328
|
(S)-2-(8-amino-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H19N5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870330
|
(S)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H14F4N4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870331
|
(S)-2-(5-(3-hydroxyazetidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C20H20F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870332
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(5-morpholino-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C20H21ClFN5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0870333
|
(S)-2-(7-(4-hydroxypiperidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C22H24F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0871619
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C16H13ClF2N4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0882473
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C15H13ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0882481
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-cyclopropyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C18H17ClFN5O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0882483
|
(S)-N-(1-(3-fluoro-4-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C16H16FN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0882488
|
(S)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethyl)phenyl)ethyl)acetamide
Show/Hide
|
C17H14F4N4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0882489
|
(S)-2-(7-(oxetan-3-yloxy)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C20H19F3N4O5
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0887598
|
(S)-2-(7-(4-methoxypiperidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C23H26F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0887600
|
(S)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C16H17N5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0887602
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C15H12Cl2FN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0887603
|
(S)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C16H13ClF3N5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0887623
|
(S)-N-(1-(4-chloro-2-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H16ClN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0898608
|
(S)-2-(8-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C18H20N4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0898609
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-methoxy-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0898611
|
(S)-2-(8-(methylamino)-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H17F3N6O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0898647
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-cyclopropyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C18H17ClFN5O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0903305
|
(S)-N-(1-(3-fluoro-4-methylphenyl)ethyl)-2-(8-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C17H18FN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903316
|
(S)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H19N5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903319
|
(S)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C18H17F3N4O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0903320
|
(S)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C18H20N4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0903344
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-iodo-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C15H12ClFIN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903345
|
(S)-N-(1-(4-chloro-3-fluorophenyl)propyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903346
|
(S)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H19N5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903351
|
(S)-N-(1-(4-chloro-2-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C17H17ClN4O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903352
|
(S)-2-(6-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C18H17F3N4O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0903353
|
2-(7-((S)-3-hydroxypiperidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-((S)-1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C22H24F3N5O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0911968
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-8-(piperidin-1-yl)-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
|
C20H22ClFN6O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0911969
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C17H16ClFN4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0914628
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C16H14ClFN4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0914629
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C15H12ClF2N5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0914630
|
(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H15F3N4O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0914631
|
(S)-2-(5-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C18H17F3N4O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0914632
|
(S)-N-(1-(3,4-dichlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C15H13Cl2N5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0914633
|
(S)-N-(1-(4-chloro-3-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H16ClN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0914714
|
(S)-N-(1-(4-chlorophenyl)ethyl)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H16ClN5O2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0928247
|
(S)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C17H17FN4O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0928248
|
(S)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C18H17F3N4O4
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0928249
|
(S)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C18H17F3N4O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0942934
|
N-((S)-1-(4-chloro-3-fluorophenyl)ethyl)-2-(5-(3-methylmorpholino)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C21H23ClFN5O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0942936
|
(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-morpholino-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C20H21ClFN5O3
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1
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| 1 |
EC50 < 1 nM
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CP0943033
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methoxy-6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C17H17ClFN5O3
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1
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| 1 |
EC50 < 1 nM
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CP0943680
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(S)-2-(8-((2,2-difluoroethyl)amino)-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C18H17F5N6O3
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1
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| 1 |
EC50 = 1 nM
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CP0943681
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
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C15H13ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0943685
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(5-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H17ClN4O3
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1
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| 1 |
EC50 = 1 nM
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CP0943688
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-chloro-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C15H12Cl2FN5O2
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1
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| 1 |
EC50 < 1 nM
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CP0943693
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethyl)phenyl)ethyl)acetamide
Show/Hide
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C17H15F3N4O2
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1
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| 1 |
EC50 = 1 nM
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CP0943697
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(S)-N-(1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H15F3N4O3
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1
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| 1 |
EC50 = 1 nM
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CP0943701
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(S)-2-(6-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C18H20N4O3
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1
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| 1 |
EC50 < 1 nM
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CP0944300
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClFN5O3
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1
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| 1 |
EC50 < 1 nM
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CP0944921
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H16ClFN4O3
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1
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| 1 |
EC50 < 1 nM
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CP0944922
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(S)-2-(5-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C18H20N4O3
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1
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| 1 |
EC50 = 1 nM
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CP0952677
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(S)-N-(1-(4-chloro-3-fluorophenyl)-2-methylpropyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C17H17ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0954292
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(S)-N-(1-(4-cyclopropyl-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C18H18FN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0954293
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7,8-dimethyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C17H17ClFN5O2
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1
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| 1 |
EC50 < 1 nM
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CP0954296
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(S)-2-(8-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C17H17ClN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0955703
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-7-phenyl-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C22H18ClFN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0955713
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClFN5O3
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1
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| 1 |
EC50 < 1 nM
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CP0955715
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H16ClN5O3
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1
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| 1 |
EC50 = 1 nM
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CP0955716
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-cyano-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H13ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0955718
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(S)-2-(7-morpholino-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C21H22F3N5O4
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1
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| 1 |
EC50 = 1 nM
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CP0955719
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(S)-N-(1-(3-chloro-4-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C16H16ClN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0955720
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(R)-N-((S)-1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)propanamide
Show/Hide
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C16H15ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0955722
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(S)-2-(3-oxo-7-(piperidin-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C22H24F3N5O3
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1
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| 1 |
EC50 < 1 nM
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CP0956031
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(S)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C18H20N4O2
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1
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| 1 |
EC50 < 1 nM
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CP0956045
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(S)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(5-fluoro-6-methylpyridin-3-yl)ethyl)acetamide
Show/Hide
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C16H15ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0956049
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(S)-2-(8-(methylamino)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C18H21N5O2
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1
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| 1 |
EC50 < 1 nM
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CP0957611
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(S)-2-(8-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C17H17FN4O2
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1
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| 1 |
EC50 = 1 nM
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CP0958445
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClFN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0958448
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(S)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C17H17ClN4O2
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1
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| 1 |
EC50 = 1 nM
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CP0958688
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClFN5O2
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1
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| 1 |
EC50 < 1 nM
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CP0958689
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-(oxetan-3-ylamino)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
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C18H18ClFN6O3
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1
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| 1 |
EC50 = 1 nM
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CP0958693
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(S)-2-(6-bromo-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C17H17BrN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0958694
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(S)-2-(8-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H16F3N5O3
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1
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| 1 |
EC50 = 1 nM
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CP0960975
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(S)-N-(1-(4-chloro-3-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H17ClN4O2
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1
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| 1 |
EC50 = 1 nM
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CP0961050
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-(oxetan-3-ylamino)-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C18H18ClFN6O3
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1
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| 1 |
EC50 = 1 nM
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CP0962195
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(S)-2-(7-chloro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H14ClF3N4O3
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1
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| 1 |
EC50 < 1 nM
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CP0962196
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-iodo-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C16H13ClFIN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0962207
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-(methylamino)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
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C16H16ClFN6O2
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1
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| 1 |
EC50 < 1 nM
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CP0962208
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0963502
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(S)-N-(1-(3-fluoro-4-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C16H16FN5O2
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1
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| 1 |
EC50 = 1 nM
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CP0964630
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(5-(3,3-difluoroazetidin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C19H17ClF3N5O2
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1
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| 1 |
EC50 < 1 nM
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CP0967444
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(R)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C16H14ClFN4O2
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1
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| 1 |
EC50 < 1 nM
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CP0870174
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(S)-N-(1-(4-cyclopropyl-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C18H18FN5O2
|
1
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| 1 |
EC50 = 10 nM
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CP0870308
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N-(1-(4-(difluoromethoxy)phenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H16F2N4O3
|
1
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| 1 |
EC50 = 10 nM
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CP0870309
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-(6-methyl-1,6-diazaspiro[3.3]heptan-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C22H24ClFN6O2
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1
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| 1 |
EC50 = 10 nM
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CP0870310
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(S)-N-(1-(4-cyclopropylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C18H19N5O2
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1
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| 1 |
EC50 = 10 nM
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CP0882485
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(6-cyclopropyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C18H17ClFN5O2
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1
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| 1 |
EC50 = 10 nM
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CP0887599
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(S)-N-(1-mesitylethyl)-2-(7-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C20H24N4O3
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1
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| 1 |
EC50 = 10 nM
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CP0887604
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(S)-2-(8-iodo-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C16H13F3IN5O3
|
1
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| 1 |
EC50 = 10 nM
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CP0903303
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C15H14ClN5O2
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1
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| 1 |
EC50 = 10 nM
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CP0943682
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(S)-N-(1-(3,4-dichlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C15H13Cl2N5O2
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1
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| 1 |
EC50 = 10 nM
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CP0943683
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(5-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C16H15ClFN5O2
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1
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| 1 |
EC50 = 10 nM
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CP0943687
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C16H14F3N5O3
|
1
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| 1 |
EC50 = 10 nM
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CP0944302
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-8-(1,6-diazaspiro[3.3]heptan-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C21H22ClFN6O2
|
1
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| 1 |
EC50 = 10 nM
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CP0955712
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(3-oxo-8-(piperazin-1-yl)-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
|
C19H21ClFN7O2
|
1
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| 1 |
EC50 = 10 nM
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CP0958446
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(S)-N-(1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C17H15F4N5O3
|
1
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| 1 |
EC50 = 10 nM
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CP0966350
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(S)-N-(1-(3-chloro-4-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C16H16ClN5O2
|
1
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| 1 |
EC50 = 10 nM
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CP0868395
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(S)-2-(8-(oxetan-3-ylamino)-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C19H19F3N6O4
|
1
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| 1 |
EC50 >= 100 nM
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CP0868396
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(S)-2-(6-methoxy-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H16F3N5O4
|
1
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| 1 |
EC50 >= 100 nM
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CP0870171
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(S)-N-(1-(3-fluoro-4-(trifluoromethoxy)phenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C16H13F4N5O3
|
1
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| 1 |
EC50 >= 100 nM
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CP0870177
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
|
C15H13ClFN5O2
|
1
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| 1 |
EC50 >= 100 nM
|
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CP0870299
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2-(3-oxo-8-(pyrrolidin-3-yl)-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-((S)-1-(p-tolyl)ethyl)acetamide
Show/Hide
|
C21H25N5O2
|
1
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| 1 |
EC50 >= 100 nM
|
|
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CP0870312
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(S)-2-(3-oxo-6-(piperidin-1-yl)-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C21H23F3N6O3
|
1
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| 1 |
EC50 >= 100 nM
|
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CP0870313
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(S)-2-(5-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
|
C17H16F3N5O3
|
1
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| 1 |
EC50 >= 100 nM
|
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CP0882478
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N-(1-(4-chlorophenyl)cyclopropyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
|
C16H14ClN5O2
|
1
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| 1 |
EC50 >= 100 nM
|
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CP0887597
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(5-(4-methylpiperazin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
|
C21H24ClFN6O2
|
1
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| 1 |
EC50 >= 100 nM
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CP0887601
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(S)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
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C17H16F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0903218
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C16H17N5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0903313
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(6-methoxy-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C16H16ClN5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0903315
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C15H14ClN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0903317
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(S)-N-(1-(4-isopropoxyphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
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C19H22N4O3
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1
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| 1 |
EC50 >= 100 nM
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CP0903318
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(2-(trifluoromethyl)pyrimidin-5-yl)ethyl)acetamide
Show/Hide
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C15H13F3N6O2
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1
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| 1 |
EC50 >= 100 nM
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CP0903347
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(S)-N-(1-(4-chloro-2-methylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H16ClN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0903354
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2-(8-(1-methylpyrrolidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-((S)-1-(p-tolyl)ethyl)acetamide
Show/Hide
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C22H27N5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0914624
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N-(1-(3-chlorophenyl)cyclopropyl)-2-(3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)acetamide
Show/Hide
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C16H14ClN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0914625
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(S)-N-(1-(4-(difluoromethoxy)-3-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H14F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0914626
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(S)-N-(1-(4-cyclopropylphenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C18H19N5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0922696
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(S)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H16F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0922697
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(7-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C16H15ClFN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0942927
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(S)-2-(8-(difluoromethyl)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H14F5N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0942938
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(S)-N-(1-(4-fluorophenyl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C16H15FN4O2
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1
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| 1 |
EC50 >= 100 nM
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CP0942939
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N-(1-(3-chlorophenyl)cyclopropyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H14ClFN4O2
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1
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| 1 |
EC50 >= 100 nM
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CP0943678
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(S)-N-(1-(4-chloro-3-fluorophenyl)ethyl)-2-(8-((1-methylazetidin-3-yl)oxy)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)acetamide
Show/Hide
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C19H20ClFN6O3
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1
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| 1 |
EC50 >= 100 nM
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CP0943686
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(S)-2-(5-(4-methylpiperazin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C22H25F3N6O3
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1
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| 1 |
EC50 >= 100 nM
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CP0944920
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N-(1-(5-chloro-3-fluoropyridin-2-yl)ethyl)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C15H13ClFN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0954290
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(S)-2-(7-(4-methylpiperazin-1-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C22H25F3N6O3
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1
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| 1 |
EC50 >= 100 nM
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CP0955702
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(S)-2-(6-cyclopropyl-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C19H18F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0955714
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(S)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H16F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0955717
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(S)-2-(3-oxo-5-(piperazin-1-yl)-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C21H23F3N6O3
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1
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| 1 |
EC50 >= 100 nM
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CP0956046
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N-(1-(4-chlorophenyl)cyclopropyl)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)acetamide
Show/Hide
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C17H14ClFN4O2
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1
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| 1 |
EC50 >= 100 nM
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CP0956047
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(5,7-dimethyl-3-oxo-[1,2,4]triazolo[4,3-c]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C17H18ClN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0956048
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(S)-2-(6-fluoro-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C16H13F4N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0958447
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(S)-N-(1-(4-chlorophenyl)ethyl)-2-(5,7-dimethyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)acetamide
Show/Hide
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C17H18ClN5O2
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1
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| 1 |
EC50 >= 100 nM
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CP0958695
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(S)-2-(6-methyl-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C17H16F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0958696
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C16H14F3N5O3
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1
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| 1 |
EC50 >= 100 nM
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CP0960360
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(S)-2-(8-(azetidin-3-yloxy)-3-oxo-[1,2,4]triazolo[4,3-a]pyrazin-2(3H)-yl)-N-(1-(4-chloro-3-fluorophenyl)ethyl)acetamide
Show/Hide
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C18H18ClFN6O3
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1
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| 1 |
EC50 >= 100 nM
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CP0961754
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(S)-2-(7-((1-methylazetidin-3-yl)oxy)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
Show/Hide
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C21H22F3N5O4
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1
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| 1 |
EC50 >= 100 nM
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CP0962194
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(S)-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-2(3H)-yl)-N-(1-(p-tolyl)ethyl)acetamide
Show/Hide
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C16H17N5O2
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1
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| 1 |
EC50 >= 100 nM
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