General Information of the Compound
Compound ID
CP0943680
Compound Name
(S)-2-(8-((2,2-difluoroethyl)amino)-3-oxo-[1,2,4]triazolo[4,3-b]pyridazin-2(3H)-yl)-N-(1-(4-(trifluoromethoxy)phenyl)ethyl)acetamide
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Structure
Formula
C18H17F5N6O3
Molecular Weight
460.363
Canonical SMILES
C[C@H](NC(=O)Cn1nc2c(NCC(F)F)ccnn2c1=O)c1ccc(OC(F)(F)F)cc1
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InChI
InChI=1S/C18H17F5N6O3/c1-10(11-2-4-12(5-3-11)32-18(21,22)23)26-15(30)9-28-17(31)29-16(27-28)13(6-7-25-29)24-8-14(19)20/h2-7,10,14,24H,8-9H2,1H3,(H,26,30)/t10-/m0/s1
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InChIKey
JZXTXRQFIPRKQR-JTQLQIEISA-N
Physicochemical Property
logP
2.344
Rotatable Bonds
8
Heavy Atom Count
32
Polar Areas
102.55
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 148156995
ChEMBL ID
CHEMBL4792896
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT06789, Probable G-protein coupled receptor 139
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 1 nM
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