Compound ID |
Compound Name |
Compound Formula |
CP0573199
|
4-[ethyl-[3-[[2-[[4-[2-[4-(methylsulfamoylcarbamoyl)phenyl]ethyl]phenyl]carbamoyl]-6-piperidin-1-ylpyridin-3-yl]carbamoyl]phenyl]sulfonylamino]cyclohexane-1-carboxylic acid
Show/Hide
|
C43H51N7O9S2
|
1
|
1 |
IC50 = 21 nM
|
|
|
CP0572734
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C46H56N6O7
|
1
|
1 |
IC50 = 36 nM
|
|
|
CP0550252
|
4-[3-[4-[[2-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C45H51N5O7
|
1
|
1 |
IC50 = 71 nM
|
|
|
CP0577666
|
4-[2-[4-[[3-[[3-[(4-carboxycyclohexyl)-ethylsulfamoyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C42H47N5O8S
|
1
|
1 |
IC50 = 77 nM
|
|
|
CP0579870
|
4-[3-[4-[[2-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-heptan-4-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid;hydrochloride
Show/Hide
|
C47H56ClN5O7
|
1
|
1 |
IC50 = 78 nM
|
|
|
CP0572733
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-methoxypyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C42H49N5O8
|
1
|
1 |
IC50 = 107 nM
|
|
|
CP0577078
|
4-[2-[4-[[3-[[3-[ethyl-[4-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethylcarbamoyl]cyclohexyl]sulfamoyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C50H64N6O11S
|
1
|
1 |
IC50 = 141 nM
|
|
|
CP0577667
|
4-[2-[4-[[3-[[3-[ethyl-[4-(methylsulfamoylcarbamoyl)cyclohexyl]sulfamoyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C43H51N7O9S2
|
1
|
1 |
IC50 = 147 nM
|
|
|
CP0578367
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-(dimethylamino)pyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C43H52N6O7
|
1
|
1 |
IC50 = 161 nM
|
|
|
CP0577236
|
4-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenoxy]benzoic acid
Show/Hide
|
C44H52N6O8
|
1
|
1 |
IC50 = 162 nM
|
|
|
CP0574536
|
4-[3-[4-[[2-[[3-[[2-[[4-[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethylamino]-4-oxobutanoyl]-methylamino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C53H68N6O10
|
1
|
1 |
IC50 = 166 nM
|
|
|
CP0578502
|
4-[methyl-[2-[[3-[[2-[[4-[2-[4-(methylsulfamoylcarbamoyl)phenyl]ethyl]phenyl]carbamoyl]-6-piperidin-1-ylpyridin-3-yl]carbamoyl]phenyl]methyl-pentan-3-ylamino]ethyl]amino]-4-oxobutanoic acid
Show/Hide
|
C47H60N8O8S
|
1
|
1 |
IC50 = 192 nM
|
|
|
CP0580149
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-(2-methoxyethoxy)pyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C44H53N5O9
|
1
|
1 |
IC50 = 201 nM
|
|
|
CP0573196
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-morpholin-4-ylpyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C45H54N6O8
|
1
|
1 |
IC50 = 205 nM
|
|
|
CP0577077
|
4-[methyl-[2-[[3-[[2-[[4-[2-[4-(methylsulfonylcarbamoyl)phenyl]ethyl]phenyl]carbamoyl]-6-piperidin-1-ylpyridin-3-yl]carbamoyl]phenyl]methyl-pentan-3-ylamino]ethyl]amino]-4-oxobutanoic acid
Show/Hide
|
C47H59N7O8S
|
1
|
1 |
IC50 = 237 nM
|
|
|
CP0970487
|
4-[3-(4-{[2-(3-{[(1r,4r)-4-Carboxycyclohexyl](ethyl)sulfamoyl}benzamido)-1H-indole-3-carbonyl]amino}phenyl)propyl]benzoic acid
Show/Hide
|
C41H42N4O8S
|
1
|
1 |
IC50 = 257 nM
|
|
|
CP0572634
|
4-[3-[4-[[2-[[3-[[2-[carboxymethoxycarbonylsulfamoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C44H50N6O10S
|
1
|
1 |
IC50 = 267 nM
|
|
|
CP0573195
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-chloropyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C41H46ClN5O7
|
1
|
1 |
IC50 = 271 nM
|
|
|
CP0577611
|
4-[3-[4-[[2-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-propan-2-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C43H47N5O7
|
1
|
1 |
IC50 = 356 nM
|
|
|
CP0551939
|
4-[3-[4-[[2-[[3-[[2-[carboxymethylcarbamoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C44H50N6O7
|
1
|
1 |
IC50 = 369 nM
|
|
|
CP0569613
|
4-[3-[4-[[2-[[3-[[2-[[2-[(5-carbamoyl-1H-pyrrol-3-yl)sulfonylamino]acetyl]-methylamino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C48H54N8O8S
|
1
|
1 |
IC50 = 401 nM
|
|
|
CP0969408
|
4-[3-(4-{[2-(3-{[(2-{[(2,5-Dioxohexahydroimidazo[4,5-d]imidazol-1(2H)-yl)acetyl](methyl)amino}ethyl)(pentan-3-yl)amino]methyl}benzamido)-1H-indole-3-carbonyl]amino}phenyl)propyl]benzoic acid
Show/Hide
|
C47H53N9O7
|
1
|
1 |
IC50 = 401 nM
|
|
|
CP0577505
|
4-[[4-[[2-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]methyl]benzoic acid
Show/Hide
|
C43H47N5O7
|
1
|
1 |
IC50 = 448 nM
|
|
|
CP0570247
|
4-[3-[4-[[2-[[3-[[2-[[4-[2-[2-[2-(2-carboxyethoxy)ethoxy]ethoxy]ethylamino]-4-oxobutanoyl]-methylamino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-1H-indole-3-carbonyl]amino]phenyl]propyl]benzoic acid
Show/Hide
|
C54H68N6O11
|
1
|
1 |
IC50 = 535 nM
|
|
|
CP0570244
|
4-[methyl-[2-[pentan-3-yl-[[3-[[3-(phenylcarbamoyl)-1H-indol-2-yl]carbamoyl]phenyl]methyl]amino]ethyl]amino]-4-oxobutanoic acid
Show/Hide
|
C35H41N5O5
|
1
|
1 |
IC50 = 538 nM
|
|
|
CP0573198
|
6-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenoxy]pyridine-3-carboxylic acid
Show/Hide
|
C43H51N7O8
|
1
|
1 |
IC50 = 715 nM
|
|
|
CP0572735
|
6-[[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-piperidin-1-ylpyridine-2-carbonyl]amino]phenoxy]methyl]pyridine-3-carboxylic acid
Show/Hide
|
C44H53N7O8
|
1
|
1 |
IC50 = 744 nM
|
|
|
CP0966273
|
4-{3-[4-({2-[3-({3-[(3-Carboxypropanoyl)(methyl)amino]pyrrolidin-1-yl}methyl)benzamido]-1H-indole-3-carbonyl}amino)phenyl]propyl}benzoic acid hydrochloride
Show/Hide
|
C42H44ClN5O7
|
1
|
1 |
IC50 = 1015 nM
|
|
|
CP0573197
|
4-[2-[4-[[3-[[3-[[2-[3-carboxypropanoyl(methyl)amino]ethyl-pentan-3-ylamino]methyl]benzoyl]amino]-6-(4-methylpiperazin-1-yl)pyridine-2-carbonyl]amino]phenyl]ethyl]benzoic acid
Show/Hide
|
C46H57N7O7
|
1
|
1 |
IC50 = 1342 nM
|
|
|
CP0965430
|
4-{3-[4-({2-[3-({[1-(3-Carboxypropanoyl)pyrrolidin-3-yl](methyl)amino}methyl)benzamido]-1H-indole-3-carbonyl}amino)phenyl]propyl}benzoic acid hydrochloride
Show/Hide
|
C42H44ClN5O7
|
1
|
1 |
IC50 = 2582 nM
|
|
|