| Compound ID |
Compound Name |
Compound Formula |
|
CP0067951
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C23H27N5O3S
|
2
|
| 1 |
IC50 = 0.3981 nM
|
|
|
| 2 |
IC50 = 1.259 nM
|
|
|
|
CP0065780
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H25Cl2N5O3S
|
3
|
| 1 |
IC50 = 1.995 nM
|
|
|
| 2 |
IC50 = 12.59 nM
|
|
|
| 3 |
IC50 = 19.95 nM
|
|
|
|
CP0419708
|
4-amino-3,5-dichloro-N-[(2R)-4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0445928
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-6-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0519195
|
N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-[4-(trifluoromethyl)piperidin-1-yl]butan-2-yl]-1H-indole-4-sulfonamide
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|
C23H24F3N5O3S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0573785
|
N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-piperidin-1-ylbutan-2-yl]-1H-indole-4-sulfonamide
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|
C22H25N5O3S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0477748
|
N-[4-(2-cyanopyrrol-1-yl)-1-(2-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0563703
|
N-[1-(azepan-1-yl)-4-(2-cyanopyrrol-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 25.12 nM
|
|
|
|
CP0534624
|
2-amino-4,6-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0519194
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]naphthalene-1-sulfonamide
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|
C25H28N4O3S
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0534622
|
4-amino-3,5-dichloro-N-[4-(5-cyanopyrazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C20H24Cl2N6O3S
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0545420
|
4-amino-2,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0573715
|
N-[4-(2-cyanopyrrol-1-yl)-1-(3-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0419712
|
3-amino-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-2,4-dimethylbenzenesulfonamide
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|
C23H31N5O3S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0419704
|
4-amino-3,5-dichloro-N-[4-(2-chlorophenyl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C22H26Cl3N3O3S
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0558400
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1-methylindole-4-sulfonamide
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|
C24H29N5O3S
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0563702
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-hydroxypiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C22H25N5O4S
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0522591
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-piperidin-1-ylbutan-2-yl]benzenesulfonamide
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|
C20H23Cl2N5O3S
|
1
|
| 1 |
IC50 = 158.49 nM
|
|
|
|
CP0447538
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-5-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 199.53 nM
|
|
|
|
CP0419710
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H24Cl2N6O5S
|
2
|
| 1 |
IC50 = 251.19 nM
|
|
|
| 2 |
IC50 = 794.33 nM
|
|
|
|
CP0519198
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-7-sulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0573713
|
4-amino-3,5-dichloro-N-[4-(5-chloropyrazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H24Cl3N5O3S
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0573714
|
4-amino-N-[1-(azepan-1-yl)-4-(2-cyanopyrrol-1-yl)-1-oxobutan-2-yl]-3,5-dichlorobenzenesulfonamide
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|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0509949
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-[4-(trifluoromethyl)piperidin-1-yl]butan-2-yl]benzenesulfonamide
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|
C21H22Cl2F3N5O3S
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0445927
|
4-amino-3,5-dichloro-N-[(2R)-1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H24Cl2N6O5S
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0447537
|
4-amino-3,5-dichloro-N-[4-(2-cyanoimidazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
Show/Hide
|
C20H24Cl2N6O3S
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0534634
|
4-amino-3,5-dichloro-N-[4-(2-chloroimidazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H24Cl3N5O3S
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0427286
|
4-amino-3,5-dichloro-N-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamide
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|
C22H27Cl2N3O3S
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0451606
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(3-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
Show/Hide
|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0558394
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(2-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
Show/Hide
|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0385314
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H26N4O3S
|
1
|
| 1 |
IC50 = 1258.93 nM
|
|
|
|
CP0419711
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-pyrazol-1-ylbutan-2-yl]benzenesulfonamide
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|
C19H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
|
CP0427285
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(triazol-2-yl)butan-2-yl]benzenesulfonamide
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|
C18H24Cl2N6O3S
|
1
|
| 1 |
IC50 = 3162.28 nM
|
|
|
|
CP0445926
|
4-(2-cyanopyrrol-1-yl)-2-(1H-indol-4-ylsulfonylamino)-N,N-dimethylbutanamide
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|
C19H21N5O3S
|
1
|
| 1 |
IC50 = 3981.07 nM
|
|
|
|
CP0454709
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-pyrrol-1-ylbutan-2-yl]benzenesulfonamide
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|
C20H26Cl2N4O3S
|
1
|
| 1 |
IC50 = 3981.07 nM
|
|
|
|
CP0419706
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-pyrrolidin-1-ylbutan-2-yl]benzenesulfonamide
Show/Hide
|
C19H21Cl2N5O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0477747
|
2-[(4-amino-3,5-dichlorophenyl)sulfonylamino]-4-(2-cyanopyrrol-1-yl)-N,N-dimethylbutanamide
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|
C17H19Cl2N5O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0519192
|
4-amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamide
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|
C22H27Cl2N3O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0563704
|
4-amino-3,5-dichloro-N-[(2S)-4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
Show/Hide
|
C21H25Cl2N5O3S
|
1
|
| 1 |
IC50 = 15848.93 nM
|
|
|
|
CP0563705
|
4-amino-3,5-dichloro-N-[4-imidazol-1-yl-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H25Cl2N5O3S
|
1
|
| 1 |
IC50 > 19952.62 nM
|
|
|
|
CP0410849
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(1,2,4-triazol-1-yl)butan-2-yl]benzenesulfonamide
Show/Hide
|
C18H24Cl2N6O3S
|
1
|
| 1 |
IC50 > 19952.62 nM
|
|
|
|
CP0545419
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(triazol-1-yl)butan-2-yl]benzenesulfonamide
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|
C18H24Cl2N6O3S
|
1
|
| 1 |
IC50 > 19952.62 nM
|
|
|
|
CP0558399
|
4-amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
Show/Hide
|
C19H24Cl2N6O5S
|
1
|
| 1 |
IC50 > 19952.62 nM
|
|
|
