| Compound ID |
Compound Name |
Compound Formula |
|
CP0120956
|
3-amino-5-chloro-N-cyclopropyl-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
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|
C13H14ClN3OS
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0120957
|
3-amino-5-chloro-4,6-dimethyl-N-(pyridin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxamide
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|
C16H15ClN4OS
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0066236
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-8-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0366351
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-5-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0873353
|
(R)-1-(3-chlorophenethyl)-3-((S)-2-phenyl-2-(piperidin-1-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
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|
C29H38ClN2O2+
|
1
|
| 1 |
IC50 < 0.03162 nM
|
|
|
|
CP0894034
|
(R)-1-(3-phenylpropyl)-3-((R)-2-(piperidin-1-yl)-2-(thiophen-2-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H39N2O2S+
|
1
|
| 1 |
IC50 < 0.03162 nM
|
|
|
|
CP0910842
|
(S)-4-(2-cyclopentyl-2-phenylpropanoyloxy)-1,1-dimethylpiperidinium bromide
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|
C21H32BrNO2
|
1
|
| 1 |
IC50 = 0.03162 nM
|
|
|
|
CP0823683
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-(2-methylpyridin-4-yl)propyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H41N2O2+
|
1
|
| 1 |
IC50 < 0.03162 nM
|
|
|
|
CP0848247
|
4-(2-cyclopentyl-2-phenylpropanoyloxy)-1,1-dimethylpiperidinium
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|
C21H32NO2+
|
1
|
| 1 |
IC50 = 0.03162 nM
|
|
|
|
CP0846002
|
(R)-1-(3-chlorophenethyl)-3-((R)-2-(piperidin-1-yl)-2-(thiophen-2-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36ClN2O2S+
|
1
|
| 1 |
IC50 < 0.03981 nM
|
|
|
|
CP0873355
|
(R)-1-(3-fluorophenethyl)-3-((S)-2-phenyl-2-(piperidin-1-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
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|
C29H38FN2O2+
|
1
|
| 1 |
IC50 < 0.03981 nM
|
|
|
|
CP0718665
|
(R)-1-(3-chlorophenethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
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|
C28H37ClNO2+
|
1
|
| 1 |
IC50 < 0.03981 nM
|
|
|
|
CP0823684
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-(pyridin-4-yl)propyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H39N2O2+
|
1
|
| 1 |
IC50 < 0.03981 nM
|
|
|
|
CP0666404
|
Tiotropium bromide
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|
C19H24BrNO5S2
|
5
|
| 1 |
IC50 = 0.05012 nM
|
|
|
| 2 |
IC50 < 0.05012 nM
|
|
|
| 3 |
IC50 = 0.35 nM
|
|
|
| 4 |
IC50 = 0.4 nM
|
|
|
| 5 |
Ki = 0.051 nM
|
|
|
|
CP0488353
|
[(3R)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H41N2O3+
|
1
|
| 1 |
IC50 = 0.05012 nM
|
|
|
|
CP0513346
|
[(3R)-1-[2-(5-chlorothiophen-2-yl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C27H36ClN2O2S+
|
1
|
| 1 |
IC50 = 0.05012 nM
|
|
|
|
CP0696953
|
Aclidinium bromide
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|
C26H30BrNO4S2
|
4
|
| 1 |
IC50 < 0.05012 nM
|
|
|
| 2 |
IC50 = 0.1259 nM
|
|
|
| 3 |
IC50 = 0.17 nM
|
|
|
| 4 |
Ki = 0.56 nM
|
|
|
|
CP0859113
|
(R)-1-phenethyl-3-((R)-2-(piperidin-1-yl)-2-(thiophen-2-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N2O2S+
|
1
|
| 1 |
IC50 < 0.05012 nM
|
|
|
|
CP0873354
|
(R)-1-(3-fluorophenethyl)-3-((R)-2-(piperidin-1-yl)-2-(thiophen-2-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36FN2O2S+
|
1
|
| 1 |
IC50 < 0.05012 nM
|
|
|
|
CP0924172
|
(R)-3-((S)-2-phenyl-2-(piperidin-1-yl)propanoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H41N2O2+
|
1
|
| 1 |
IC50 < 0.05012 nM
|
|
|
|
CP0666469
|
(R)-1-(3-(benzo[d]oxazol-2-yl)propyl)-8-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H39N2O3+
|
1
|
| 1 |
IC50 = 0.05012 nM
|
|
|
|
CP0821128
|
(R)-1-(3-(pyridin-4-yl)propyl)-3-(1-(thiophen-2-yl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N2O2S+
|
1
|
| 1 |
IC50 = 0.05012 nM
|
|
|
|
CP0375273
|
[(3R)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C28H39N2O3S+
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0428312
|
[(3R)-1-[3-(1-benzothiophen-2-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C32H41N2O2S+
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0456222
|
[(3R)-1-[2-(3-bromophenyl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38BrN2O2+
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0876196
|
(R)-1-(2-(5-methylthiophen-2-yl)ethyl)-3-((S)-2-phenyl-2-(piperidin-1-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H39N2O2S+
|
1
|
| 1 |
IC50 < 0.0631 nM
|
|
|
|
CP0821127
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(isoxazol-3-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C25H34N3O4+
|
1
|
| 1 |
IC50 < 0.0631 nM
|
|
|
|
CP0848245
|
(R)-quinuclidin-3-yl 1-phenylcycloheptanecarboxylate
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|
C21H29NO2
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0946249
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(5-methylthiophen-2-yl)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H38NO2S+
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0947380
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H40NO3+
|
1
|
| 1 |
IC50 = 0.0631 nM
|
|
|
|
CP0388362
|
[(3R)-1-(3-pyridin-4-ylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H40N3O2+
|
1
|
| 1 |
IC50 = 0.07943 nM
|
|
|
|
CP0428308
|
[(3R)-1-[3-(4-fluorophenoxy)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C28H38FN2O3S+
|
1
|
| 1 |
IC50 = 0.07943 nM
|
|
|
|
CP0682850
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((5-phenylisoxazol-3-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H37N2O3+
|
1
|
| 1 |
IC50 = 0.07943 nM
|
|
|
|
CP0682852
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38NO2+
|
1
|
| 1 |
IC50 = 0.07943 nM
|
|
|
|
CP0904563
|
(R)-quinuclidin-8-yl 1-(thiophen-2-yl)cycloheptanecarboxylate
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|
C19H27NO2S
|
1
|
| 1 |
IC50 = 0.07943 nM
|
|
|
|
CP0475076
|
[(3R)-1-[2-[(6-chloropyrazin-2-yl)amino]-2-oxoethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C25H33ClN5O3S+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0475078
|
[(3R)-1-[2-(3-fluoroanilino)-2-oxoethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C27H35FN3O3S+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0525093
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-piperidin-1-yl-2-thiophen-2-ylpropanoate
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|
C19H31N2O2S+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0904587
|
(R)-1-phenethyl-3-((S)-2-phenyl-2-(piperidin-1-yl)propanoyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H39N2O2+
|
1
|
| 1 |
IC50 < 0.1 nM
|
|
|
|
CP0682851
|
(R)-1-(2-(6-chloropyrazin-2-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H34ClN4O3+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0708598
|
(R)-1-(benzo[d]oxazol-2-ylmethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H35N2O3+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0935480
|
(R)-1-(2-(1H-pyrazol-3-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C25H35N4O3+
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0375270
|
[(3R)-1-[2-oxo-2-(pyridin-2-ylamino)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C28H37N4O3+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0375272
|
[(3R)-1-(2-amino-2-oxoethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C21H32N3O3S+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0456223
|
[(3R)-1-[2-(2-fluorophenyl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38FN2O2+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0525091
|
[(3R)-1-[3-(2-methylpyridin-4-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H42N3O2+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0428316
|
AHR-504
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|
C19H28NO3+
|
2
|
| 1 |
IC50 = 0.1259 nM
|
|
|
| 2 |
IC50 = 0.2512 nM
|
|
|
|
CP0819568
|
(R)-1-(2-(benzyloxy)ethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H40NO3+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0821126
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyrazin-2-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H35N4O3+
|
1
|
| 1 |
IC50 < 0.1259 nM
|
|
|
|
CP0829284
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(3-fluorophenylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H36FN2O3+
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0375274
|
[(3R)-1-[2-(2,3,3a,7a-tetrahydro-1-benzofuran-5-yl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H43N2O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0388364
|
[(3R)-1-[2-(2-fluorophenyl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C27H36FN2O2S+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0390608
|
[(3R)-1-[2-(4-fluorophenyl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38FN2O2+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0428307
|
[(3R)-1-[2-(1,2-oxazol-3-ylamino)-2-oxoethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C26H35N4O4+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0475083
|
[(3R)-1-(3-pyridin-4-ylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C27H38N3O2S+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0484741
|
[(3R)-1-[(6-methyl-1,3-benzoxazol-2-yl)methyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H38N3O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0666467
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(5-methylisoxazol-3-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H36N3O4+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0823237
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H36N3O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0829283
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyridazin-3-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H35N4O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0860996
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-(6-methylpyridin-3-yl)propyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H41N2O2+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0947381
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38NO3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0956968
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyrimidin-4-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H35N4O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0957206
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyridin-2-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36N3O3+
|
1
|
| 1 |
IC50 = 0.1585 nM
|
|
|
|
CP0705209
|
(3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 0.18 nM
|
|
|
|
CP0375268
|
[(3R)-1-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H38N3O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0375269
|
[(3R)-1-[2-oxo-2-(pyrazin-2-ylamino)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C27H36N5O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0375271
|
[(3R)-1-(2-anilino-2-oxoethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38N3O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0400727
|
[(3R)-1-[2-(3-fluoroanilino)-2-oxoethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H37FN3O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0433136
|
[(3R)-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H43N2O2+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0433137
|
[(3R)-1-(2-cyclohexylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C27H43N2O2S+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0458910
|
[(3R)-1-(2-anilino-2-oxoethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C27H36N3O3S+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0484742
|
[(3R)-1-(2-amino-2-oxoethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C23H34N3O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0524892
|
[(3R)-1-[2-(1,2-oxazol-3-ylamino)-2-oxoethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C24H33N4O4S+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
|
CP0525092
|
[(3R)-1-(2-naphthalen-2-ylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C33H41N2O2+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
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CP0666466
|
(R)-1-(2-(6-chloropyridazin-3-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H34ClN4O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
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CP0666468
|
(R)-1-(2-amino-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C22H33N2O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
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CP0956801
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyridin-3-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36N3O3+
|
1
|
| 1 |
IC50 = 0.1995 nM
|
|
|
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CP0666488
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H28BrNO3S2
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0911595
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0512720
|
US9233108, 9
Show/Hide
|
C41H44ClN5O8S2
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0917523
|
US9315463, 1
Show/Hide
|
C37H49N3O6S2
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0086732
|
(3R)-1-Azabicyclo[2.2.2]oct-3-ylhydroxy(di-2-thienyl)acetate
Show/Hide
|
C17H19NO3S2
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0851960
|
(3R)-3-{[(9-Methyl-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrNO4
|
1
|
| 1 |
IC50 = 0.24 nM
|
|
|
|
CP0918897
|
(3R)-3-{[Hydroxy(di-3-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30BrNO4S2
|
1
|
| 1 |
IC50 = 0.24 nM
|
|
|
|
CP0852883
|
(3R)-3-{[(2S)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.25 nM
|
|
|
|
CP0860527
|
GLYCOPYRROLATE
Show/Hide
|
C19H28BrNO3
|
2
|
| 1 |
IC50 = 0.2512 nM
|
|
|
| 2 |
Ki = 0.81 nM
|
|
|
|
CP0375276
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C21H33N2O2+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0428311
|
[(3R)-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C29H41N2O2S+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0458908
|
[(3R)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C28H35N4O3S+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0848246
|
1,1-dimethyl-4-(1-phenylcycloheptanecarbonyloxy)piperidinium
Show/Hide
|
C21H32NO2+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0860993
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(6-(trifluoromethyl)pyridin-3-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H35F3N3O3+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0936032
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(3-fluoropyridin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H35FN3O3+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0936033
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(phenylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H37N2O3+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0941910
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((3-phenylisoxazol-5-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H37N2O3+
|
1
|
| 1 |
IC50 = 0.2512 nM
|
|
|
|
CP0868133
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO4
|
1
|
| 1 |
IC50 = 0.28 nM
|
|
|
|
CP0846167
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0909075
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H35BrN2O2
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0527315
|
US9233108, 1
Show/Hide
|
C39H42N4O8S2
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0915656
|
US9315463, 25
Show/Hide
|
C40H46ClN3O8S2
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0431075
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-hydroxy(phenyl)2-thienylacetate
Show/Hide
|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0891026
|
(3R)-1-(2-Phenylethyl)-3-[(9H-xanthen-9-ylcarbonyl)oxy]-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0400729
|
[(3R)-1-[3-(1,3-benzoxazol-2-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H40N3O3+
|
1
|
| 1 |
IC50 = 0.3162 nM
|
|
|
|
CP0492601
|
[(3R)-1-[2-(4-methylphenoxy)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H41N2O3+
|
1
|
| 1 |
IC50 = 0.3162 nM
|
|
|
|
CP0525089
|
[(3R)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H37N4O3+
|
1
|
| 1 |
IC50 = 0.3162 nM
|
|
|
|
CP0525090
|
[(3R)-1-(3-pyridin-3-ylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H40N3O2+
|
1
|
| 1 |
IC50 = 0.3162 nM
|
|
|
|
CP0819567
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((5-phenyl-1,3,4-oxadiazol-2-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H36N3O3+
|
1
|
| 1 |
IC50 = 0.3162 nM
|
|
|
|
CP0868135
|
(3R)-3-[(Di-2-thienylacetyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30BrNO3S2
|
1
|
| 1 |
IC50 = 0.37 nM
|
|
|
|
CP0418147
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-cyclopentyl(hydroxy)2-thienylacetate
Show/Hide
|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.39 nM
|
|
|
|
CP0499035
|
(3R)-1-Heptyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H34BrNO3S2
|
1
|
| 1 |
IC50 = 0.39 nM
|
|
|
|
CP0458909
|
[(3R)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-piperidin-1-yl-2-thiophen-2-ylpropanoate
Show/Hide
|
C29H36N3O3S+
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0475082
|
[(3R)-1-[3-(1,3-benzothiazol-6-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H40N3O2S+
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0903772
|
(R)-1-(2-(1,2,4-thiadiazol-5-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C24H33N4O3S+
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0904560
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((1-phenyl-1H-pyrazol-3-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H38N3O2+
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0936031
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(2-methylpyrimidin-4-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N4O3+
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0402560
|
US9233108, 2
Show/Hide
|
C39H43N5O7S2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0402685
|
US9233108, 10
Show/Hide
|
C41H47ClN4O9S2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0483995
|
US9233108, 18
Show/Hide
|
C38H48N6O7S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0576434
|
US9233108, 5
Show/Hide
|
C40H43N5O7S2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0397014
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-hydroxy(phenyl)2-thienylacetate
Show/Hide
|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.42 nM
|
|
|
|
CP0874933
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.45 nM
|
|
|
|
CP0893211
|
(3R)-3-{[(2R)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.48 nM
|
|
|
|
CP0891718
|
(R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0412345
|
US9233108, 11
Show/Hide
|
C39H42N4O7S3
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0484743
|
[(3R)-1-[2-(2-phenylethoxy)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H43N2O3+
|
1
|
| 1 |
IC50 = 0.5012 nM
|
|
|
|
CP0860995
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-(1-methyl-1H-pyrazol-3-yl)propyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H40N3O2+
|
1
|
| 1 |
IC50 = 0.5012 nM
|
|
|
|
CP0935988
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(5-methylpyridin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38N3O3+
|
1
|
| 1 |
IC50 = 0.5012 nM
|
|
|
|
CP0851961
|
(3R)-3-[(2,2-Di-2-thienylpropanoyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.59 nM
|
|
|
|
CP0462649
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-methyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C18H22BrNO3S2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0456356
|
(R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0891721
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H35BrN2O2S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0895086
|
(R)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0906344
|
(R)-3-((3-fluorophenyl)(3,4,5-trifluorobenzyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H29BrF4N2O3
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0916859
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H33BrN2O2S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0402686
|
US9233108, 17
Show/Hide
|
C39H48N6O6S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0412344
|
US9233108, 4
Show/Hide
|
C40H44N4O6S2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0918903
|
(3R)-3-{[Hydroxy(diphenyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H34BrNO4
|
1
|
| 1 |
IC50 = 0.61 nM
|
|
|
|
CP0428309
|
[(3R)-1-[3-(4-fluorophenoxy)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H40FN2O3+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0458913
|
[(3R)-1-(4-methylpent-3-enyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C27H41N2O2+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0492602
|
[(3R)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H39N2O3+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0903771
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(5-fluoropyridin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H35FN3O3+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0906592
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyrimidin-5-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H35N4O3+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0936030
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(6-methylpyrazin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N4O3+
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0439371
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-cyclopentyl(hydroxy)2-thienylacetate
Show/Hide
|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0851406
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0859004
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H29BrN2O2S3
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0864661
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H29BrN2O3S2
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0917522
|
US9315463, 20
Show/Hide
|
C40H45ClN4O8S2
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0874051
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrNO4
|
1
|
| 1 |
IC50 = 0.71 nM
|
|
|
|
CP0369702
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carboxylate
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
IC50 = 0.76 nM
|
|
|
|
CP0400728
|
[(3R)-1-(2-phenylmethoxyethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H41N2O3+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0428315
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(azepin-1-yl)-2-phenylpropanoate
Show/Hide
|
C22H29N2O2+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0492607
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-phenyl-2-thiomorpholin-4-ylpropanoate
Show/Hide
|
C20H31N2O2S+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0848244
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(6-methylpyridin-3-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38N3O3+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0869443
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(6-methylpyridazin-3-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N4O3+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0913132
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(4-methylpyridin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38N3O3+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0935987
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(5-methylpyrazin-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N4O3+
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0847622
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H37BrN2O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0917225
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O3
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0847983
|
(R)-1-(3-phenoxypropyl)-3-(9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H33BrN2O3
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0402687
|
US9233108, 19
Show/Hide
|
C40H44N4O8S2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0217648
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate
Show/Hide
|
C21H23NO3
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0912371
|
(R)-1-(3-phenylpropyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrF3N2O2
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0462648
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9-hydroxy-9H-fluorene-9-carboxylate
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
IC50 = 0.92 nM
|
|
|
|
CP0920325
|
(3R)-3-{[(9-Methyl-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrNO3
|
1
|
| 1 |
IC50 = 0.96 nM
|
|
|
|
CP0456355
|
(R)-quinuclidin-3-yl phenyl(thiophen-3-ylmethyl)carbamate
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0846146
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H33BrN2O3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0456224
|
[(3R)-1-propan-2-yl-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C24H37N2O2+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0500232
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(4-methylpiperidin-1-yl)-2-phenylpropanoate
Show/Hide
|
C22H35N2O2+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0513344
|
[(3R)-1-[2-(3-methylphenoxy)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H41N2O3+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0524894
|
[(3R)-1-[2-oxo-2-(pyridazin-3-ylamino)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C27H36N5O3+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0861012
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(6-methylpyrimidin-4-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H37N4O3+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0956567
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-(2,6-dimethylpyridin-3-yl)propyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H43N2O2+
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0418170
|
US9233108, 15
Show/Hide
|
C44H46N4O8
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0858073
|
US9315463, 15
Show/Hide
|
C39H43ClN4O8S2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0891027
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 1.04 nM
|
|
|
|
CP0896422
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrNO5
|
1
|
| 1 |
IC50 = 1.04 nM
|
|
|
|
CP0441678
|
(2S)-N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-cyclopentyl-2-hydroxy-2-thiophen-2-ylacetamide
Show/Hide
|
C18H26N2O2S
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0964194
|
US9315463, 9
Show/Hide
|
C39H43ClN4O8S2
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0501199
|
(R)-quinuclidin-3-yl benzyl(phenyl)carbamate
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0912372
|
(R)-1-(2-phenoxyethyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrF3N2O3
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0472694
|
[9-[(3-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0488346
|
[(3R)-1-[2-oxo-2-(pyrimidin-4-ylamino)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C27H36N5O3+
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0488347
|
[(3R)-1-[2-(4-chlorophenoxy)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38ClN2O3+
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0492604
|
[(3R)-1-[3-(6-methylpyridin-3-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H42N3O2+
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0505922
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(4,4-difluoropiperidin-1-yl)-2-phenylpropanoate
Show/Hide
|
C21H31F2N2O2+
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0937434
|
US9315463, 2
Show/Hide
|
C38H43N3O7S2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0478198
|
(R)-quinuclidin-3-yl m-tolyl(2,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C22H23F3N2O2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0865543
|
US9233108, 6
Show/Hide
|
C40H46N4O8S2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0923220
|
US9315463, 22
Show/Hide
|
C40H43N5O9S2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0390751
|
(R)-quinuclidin-3-yl 3-fluorophenyl(3,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C21H20F4N2O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0524895
|
[(3R)-1-[2-(1H-indol-3-yl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H40N3O2+
|
1
|
| 1 |
IC50 = 1.585 nM
|
|
|
|
CP0894042
|
(3R)-3-(2-cyclopentyl-2-phenylpropanoyloxy)-1,1-dimethylpyrrolidinium bromide
Show/Hide
|
C20H30BrNO2
|
1
|
| 1 |
IC50 = 1.585 nM
|
|
|
|
CP0734482
|
US9315463, 12
Show/Hide
|
C39H43ClN4O9S2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0958034
|
US9315463, 18
Show/Hide
|
C38H40F2N4O7S2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0868134
|
(3R)-3-{[(2R)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 1.62 nM
|
|
|
|
CP0505031
|
(3R)-1-Heptyl-3-{[(9-hydroxy-9H-fluoren-9-yl)carbonyl]-oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H36BrNO3
|
1
|
| 1 |
IC50 = 1.68 nM
|
|
|
|
CP0502914
|
(R)-quinuclidin-3-yl pentyl(phenyl)carbamate
Show/Hide
|
C19H28N2O2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0070586
|
Ipratropium Bromide
Show/Hide
|
C20H30BrNO3
|
3
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
IC50 = 2.07 nM
|
|
|
| 3 |
Ki = 0.19 nM
|
|
|
|
CP0507579
|
US9315463, 26
Show/Hide
|
C38H43ClN4O10S2
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0864662
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O3S2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0923218
|
US9315463, 16
Show/Hide
|
C39H43FN4O8S2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0961367
|
US9315463, 13
Show/Hide
|
C40H45ClN4O8S2
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0387223
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2O2S2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0419358
|
US9233108, 8
Show/Hide
|
C39H44N4O8S2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0858072
|
US9315463, 10
Show/Hide
|
C38H41ClN4O7S2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0488363
|
(R)-quinuclidin-3-yl 3-fluorobenzyl(3-fluorophenyl)carbamate
Show/Hide
|
C21H22F2N2O2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0456220
|
[(3R)-1-[3-(2,6-dimethylpyridin-4-yl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H44N3O2+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0488355
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(4-chlorophenyl)-2-piperidin-1-ylpropanoate
Show/Hide
|
C21H32ClN2O2+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0848585
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(6-(trifluoromethyl)pyridazin-3-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H34F3N4O3+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0860994
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(6-(trifluoromethyl)pyridin-2-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H35F3N3O3+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0860997
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-methyl-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C21H32NO2+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0913133
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyridin-4-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36N3O3+
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0519466
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H28NO3S2+
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0470262
|
Ipratropium
Show/Hide
|
C20H30NO3+
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0572449
|
US9333195, 77
Show/Hide
|
C23H26NO3S3+
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0433135
|
[(3R)-1-[2-(4-fluorophenoxy)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C29H38FN2O3+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0433139
|
[(3R)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2R)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C30H41N2O3+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0488348
|
[(3R)-1-(3-pyrimidin-5-ylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C28H39N4O2+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0488349
|
[(3R)-1-(2-pyridin-3-ylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C28H38N3O2+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0492608
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-phenyl-2-pyrrolidin-1-ylpropanoate
Show/Hide
|
C20H31N2O2+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0904561
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(2-(pyrazine-2-carboxamido)ethylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H40N5O4+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0935481
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3-methoxybenzyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C28H38NO3+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0941916
|
(R)-1-(4-cyanophenethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H37N2O2+
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0561586
|
ATR
Show/Hide
|
C17H23NO3
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0482224
|
(R)-quinuclidin-3-yl phenethyl(phenyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0449982
|
US9233108, 20
Show/Hide
|
C40H46N4O8S2
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0915657
|
US9315463, 29
Show/Hide
|
C40H49ClN4O9S
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0577910
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H32NO3S2+
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0391432
|
(9-benzyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H29N3O2S
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0502913
|
(R)-quinuclidin-3-yl butyl(phenyl)carbamate
Show/Hide
|
C18H26N2O2
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0486070
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30NO4S2+
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0572447
|
US9333195, 8
Show/Hide
|
C28H32NO4S+
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0578599
|
US9333195, 78
Show/Hide
|
C24H28NO3S3+
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0502320
|
[9-[(3-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0375275
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] 2-phenyl-2-pyrrolidin-1-ylpropanoate
Show/Hide
|
C20H28N2O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0428310
|
[(3R)-1-(2-pyridin-4-yloxyethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C28H38N3O3+
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0458914
|
[(3R)-1-butyl-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C25H39N2O2+
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0496098
|
(1-methylpiperidin-4-yl) 2-phenyl-2-pyrrolidin-1-ylpropanoate
Show/Hide
|
C19H28N2O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0673968
|
SID50106181
Show/Hide
|
C21H26INO2
|
2
|
| 1 |
IC50 = 5.1 nM
|
|
|
| 2 |
Ki = 2.5 nM
|
|
|
|
CP0486073
|
(3R)-3-{[Hydroxy(di-3-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30NO4S2+
|
1
|
| 1 |
IC50 = 5.4 nM
|
|
|
|
CP0577361
|
US9333195, 53
Show/Hide
|
C26H29FNO4S2+
|
1
|
| 1 |
IC50 = 5.6 nM
|
|
|
|
CP0501201
|
(R)-quinuclidin-3-yl bis(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C18H22N2O2S2
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0910413
|
US9233108, 16
Show/Hide
|
C42H46N4O8
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0802380
|
quinuclidin-4-yl biphenyl-2-ylcarbamate hydrochloride
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0578220
|
(3R)-1-(2-Phenylethyl)-3-[(9H-xanthen-9-ylcarbonyl)oxy]-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30NO3+
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0513345
|
[(3R)-1-[2-(1-benzofuran-2-yl)ethyl]-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C31H39N2O3+
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0935479
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(3-(picolinamido)propylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C31H43N4O4+
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0490066
|
US9333195, 18
Show/Hide
|
C27H30NO5+
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0572448
|
US9333195, 20
Show/Hide
|
C28H32NO5+
|
1
|
| 1 |
IC50 = 6.8 nM
|
|
|
|
CP0578221
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30NO4+
|
1
|
| 1 |
IC50 = 6.9 nM
|
|
|
|
CP0572450
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30NO3+
|
1
|
| 1 |
IC50 = 7.6 nM
|
|
|
|
CP0399574
|
[9-[(2-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0488350
|
[(3R)-1-(3-cyanopropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C25H36N3O2+
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0957207
|
(R)-1-(2-(1,3,4-thiadiazol-2-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C24H33N4O3S+
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0486071
|
US9333195, 71
Show/Hide
|
C26H30NO5S2+
|
1
|
| 1 |
IC50 = 8.2 nM
|
|
|
|
CP0957327
|
US9315463, 28
Show/Hide
|
C42H51ClN4O9
|
1
|
| 1 |
IC50 = 8.5 nM
|
|
|
|
CP0500918
|
US9333195, 128
Show/Hide
|
C30H32NO4+
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0486072
|
US9333195, 84
Show/Hide
|
C26H30NO4S2+
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0454222
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C20H24ClN3O2S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0525094
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(dimethylamino)-2-phenylpropanoate
Show/Hide
|
C18H29N2O2+
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0956566
|
(R)-1-(2-(5-tert-butylisoxazol-3-ylamino)-2-oxoethyl)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C29H42N3O4+
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0494852
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32NO5+
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0869445
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-(oxazol-2-ylamino)-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C25H34N3O4+
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0494854
|
(3R)-3-{[(9-Methyl-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34NO4+
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0513355
|
US9333195, 126
Show/Hide
|
C31H34NO3+
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0577893
|
(3R)-3-[(Di-2-thienylacetyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30NO3S2+
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0477804
|
US9333195, 17
Show/Hide
|
C28H30NO4+
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0513354
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32NO4+
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0554633
|
US9333195, 114
Show/Hide
|
C31H32NO2+
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0390680
|
(R)-quinuclidin-3-yl benzyl(4-fluorophenyl)carbamate
Show/Hide
|
C21H23FN2O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0398693
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-diphenylacetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0513352
|
(3R)-3-{[Hydroxy(diphenyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H34NO4+
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0454223
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0454523
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-ethyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H26ClN3O2S
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0490067
|
US9333195, 74
Show/Hide
|
C24H29N2O3S2+
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0577912
|
US9333195, 127
Show/Hide
|
C29H30NO4+
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0459211
|
(R)-quinuclidin-3-yl butyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C17H26N2O2S
|
1
|
| 1 |
IC50 = 17.7 nM
|
|
|
|
CP0845813
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H33BrN2O2
|
1
|
| 1 |
IC50 = 17.7 nM
|
|
|
|
CP0459214
|
(R)-1-methyl-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C20H25BrN2O2S
|
1
|
| 1 |
IC50 = 18.6 nM
|
|
|
|
CP0379242
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9-hydroxyfluorene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 18.7 nM
|
|
|
|
CP0903846
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0470263
|
US9333195, 138
Show/Hide
|
C28H30NO4S+
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0447654
|
[9-[(2-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C22H28ClN3O2S
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0071487
|
BENZTROPINE
Show/Hide
|
C21H25NO
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0493177
|
US9333195, 7
Show/Hide
|
C31H36NO3+
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0375586
|
(R)-quinuclidin-3-yl benzyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C20H24N2O2S
|
1
|
| 1 |
IC50 = 22.5 nM
|
|
|
|
CP0554634
|
(3R)-3-{[(9-Methyl-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34NO3+
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0936029
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-((2-phenylthiazol-4-yl)methyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C30H37N2O2S+
|
1
|
| 1 |
IC50 = 25.12 nM
|
|
|
|
CP0413618
|
US9333195, 1
Show/Hide
|
C30H34NO3+
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0500917
|
US9333195, 109
Show/Hide
|
C28H28NO3S+
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0513353
|
US9333195, 99
Show/Hide
|
C30H30NO3+
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0528622
|
1-benzofuran-5-yl-[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]methanone
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0913134
|
(S)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-oxo-2-(pyridin-2-ylamino)ethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36N3O3+
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0882813
|
(R)-3-(2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 33.4 nM
|
|
|
|
CP0411467
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9H-xanthene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 37.3 nM
|
|
|
|
CP0906593
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(3,4-difluorobenzyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H34F2NO2+
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0956969
|
(R)-1-benzyl-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C27H36NO2+
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0398144
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(5-methylfuran-2-yl)methanone
Show/Hide
|
C21H25ClN2O3
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0868278
|
(R)-1-(3-(biphenyl-4-yloxy)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C37H39ClN2O3
|
1
|
| 1 |
IC50 = 60.2 nM
|
|
|
|
CP0508162
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(furan-2-yl)methanone
Show/Hide
|
C20H23ClN2O3
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0521412
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C20H23ClN2O2S
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0935343
|
(R)-1-(3-(1H-pyrrol-1-yl)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H34BrN3O2
|
1
|
| 1 |
IC50 = 64.4 nM
|
|
|
|
CP0459212
|
(R)-quinuclidin-3-yl phenyl(propyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 71.1 nM
|
|
|
|
CP0478197
|
(R)-quinuclidin-3-yl benzyl(p-tolyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 74.7 nM
|
|
|
|
CP0505885
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl 10,11-dihydro-5H-dibenzo-[a,d][7]annulene-5-carboxylate
Show/Hide
|
C23H25NO2
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0391428
|
[9-[(3-methylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-phenylmethanone
Show/Hide
|
C24H30N2O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0391429
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-[5-(hydroxymethyl)furan-2-yl]methanone
Show/Hide
|
C21H25ClN2O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0497828
|
[9-[(3-chlorophenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-phenylmethanone
Show/Hide
|
C23H27ClN2O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0904562
|
(R)-3-(1-(cyclopenta-1,3-dienyl)cycloheptanecarbonyloxy)-1-(2-morpholino-2-oxoethyl)-1-azoniabicyclo[2.2.2]octane
Show/Hide
|
C26H39N2O4+
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0398694
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2OS2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0454522
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(furan-3-yl)methanone
Show/Hide
|
C20H23ClN2O3
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0497829
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-phenylmethanone
Show/Hide
|
C23H28N2O
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0864660
|
(R)-3-(9-hydroxy-9H-fluorene-9-carboxamido)-1-(3-(methyl(phenyl)amino)propyl)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C31H36ClN3O2
|
1
|
| 1 |
IC50 = 130.5 nM
|
|
|
|
CP0846145
|
SOLIFENACIN SUCCINATE
Show/Hide
|
C27H32N2O6
|
1
|
| 1 |
IC50 = 130.8 nM
|
|
|
|
CP0391431
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,3-thiazol-4-yl)methanone
Show/Hide
|
C19H22ClN3O2S
|
1
|
| 1 |
IC50 = 158.49 nM
|
|
|
|
CP0488357
|
(1,1-dimethylpiperidin-1-ium-4-yl) 2-(dipropylamino)-2-phenylpropanoate
Show/Hide
|
C22H37N2O2+
|
1
|
| 1 |
IC50 = 158.49 nM
|
|
|
|
CP0469803
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-N-methyl-9H-xanthene-9-carboxamide
Show/Hide
|
C22H24N2O2
|
1
|
| 1 |
IC50 = 172.5 nM
|
|
|
|
CP0391430
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,2,5-thiadiazol-3-yl)methanone
Show/Hide
|
C18H21ClN4O2S
|
1
|
| 1 |
IC50 = 199.53 nM
|
|
|
|
CP0896423
|
(3R)-1-Benzyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H26BrNO3S2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0446893
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-phenylmethanone
Show/Hide
|
C22H25ClN2O2
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0513347
|
[(3R)-1-pentan-3-yl-1-azoniabicyclo[2.2.2]octan-3-yl] (2S)-2-phenyl-2-piperidin-1-ylpropanoate
Show/Hide
|
C26H41N2O2+
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0454220
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-thiophen-3-ylmethanone
Show/Hide
|
C21H26N2OS
|
1
|
| 1 |
IC50 = 316.23 nM
|
|
|
|
CP0435479
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(1,2-oxazol-3-yl)methanone
Show/Hide
|
C19H22ClN3O3
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0470009
|
[9-[(2-methylphenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C23H31N3O2S
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0502624
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-pyrimidin-2-ylmethanone
Show/Hide
|
C20H23ClN4O2
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0477682
|
1-[(2R)-4-(5-fluoro-3-methylpyridin-2-yl)-2-methylpiperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C24H27FN4O
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
|
CP0398464
|
2-hydroxy-N-[(3S)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl]-2,2-dithiophen-2-ylacetamide;bromide
Show/Hide
|
C26H31BrN2O3S2
|
1
|
| 1 |
IC50 = 599.3 nM
|
|
|
|
CP0390681
|
(R)-quinuclidin-3-yl isopropyl(phenyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 659.3 nM
|
|
|
|
CP0454221
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-(2-ethoxyphenyl)methanone
Show/Hide
|
C25H32N2O2
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0390678
|
(R)-quinuclidin-3-yl diphenylcarbamate
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
IC50 = 796.8 nM
|
|
|
|
CP0373153
|
2-chloro-N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzamide
Show/Hide
|
C19H21Cl2N3O
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0535342
|
N-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2O2S2
|
1
|
| 1 |
IC50 = 1069.4 nM
|
|
|
|
CP0477681
|
1-[(2S)-4-(5-fluoro-3-methylpyridin-2-yl)-2-methylpiperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C24H27FN4O
|
1
|
| 1 |
IC50 = 1258.93 nM
|
|
|
|
CP0469061
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2,3,4,5,6-pentafluorobenzamide
Show/Hide
|
C19H17ClF5N3O
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0401466
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 = 4200 nM
|
|
|
|
CP0514007
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C20H21ClF3N3O
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0372956
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2-methoxybenzamide
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
IC50 = 5600 nM
|
|
|
|
CP0372793
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]benzamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0372958
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-4-methoxybenzamide
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0469062
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,4-difluorobenzamide
Show/Hide
|
C19H20ClF2N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0493960
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0506234
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3-methylbenzamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0507717
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-4-methylbenzamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0055048
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-(furan-2-yl)methanone
Show/Hide
|
C21H26N2O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0398146
|
(2-tert-butyl-1,3-thiazol-4-yl)-[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]methanone
Show/Hide
|
C23H30ClN3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0475752
|
(9-benzyl-2,9-diazaspiro[5.5]undecan-2-yl)-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H27N3OS
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0502600
|
[9-[(4-chlorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl]-(2-methyl-1,3-thiazol-4-yl)methanone
Show/Hide
|
C21H26ClN3OS
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0504490
|
(9-benzyl-3,9-diazaspiro[5.5]undecan-3-yl)-pyridin-3-ylmethanone
Show/Hide
|
C22H27N3O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0528623
|
[9-[(4-chlorophenyl)methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-pyridin-3-ylmethanone
Show/Hide
|
C21H24ClN3O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0058454
|
BA-679-BR
Show/Hide
|
C19H22NO4S2+
|
1
|
| 1 |
Ki = 0.03162 nM
|
|
|
|
CP0461986
|
5-methyl-5-(3-phenoxyazetidin-1-yl)-2,2-diphenylhexanamide
Show/Hide
|
C28H32N2O2
|
1
|
| 1 |
Ki = 0.049 nM
|
|
|
|
CP0442108
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-2-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O6
|
1
|
| 1 |
Ki = 0.05012 nM
|
|
|
|
CP0550009
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]anilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C39H41N5O6
|
1
|
| 1 |
Ki = 0.07943 nM
|
|
|
|
CP0445804
|
[1-[3-[5-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]pentylamino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C37H45N5O6
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0116358
|
(R)-1-(9-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethylamino)nonyl)piperidin-4-yl biphenyl-2-ylcarbamate
Show/Hide
|
C38H48N4O5
|
1
|
| 1 |
Ki = 0.1259 nM
|
|
|
|
CP0384252
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxyanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O7
|
1
|
| 1 |
Ki = 0.1585 nM
|
|
|
|
CP0391031
|
5-[(3S)-3-(2-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.16 nM
|
|
|
|
CP0440301
|
5-[3-[(3-hydroxyphenyl)methoxy]azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.18 nM
|
|
|
|
CP0380830
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-N,2-dimethylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O6
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0398520
|
[1-[3-[2-chloro-4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]anilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C39H40ClN5O6
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0418735
|
[1-[3-[3-chloro-4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]anilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C39H40ClN5O6
|
1
|
| 1 |
Ki = 0.1995 nM
|
|
|
|
CP0199765
|
5-[3-(3-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0882281
|
Tiotropium bromide
Show/Hide
|
C19H22BrNO4S2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0392008
|
5-[(3S)-3-(3-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.21 nM
|
|
|
|
CP0495745
|
5-[3-(3-chloro-5-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H31ClN2O3
|
1
|
| 1 |
Ki = 0.22 nM
|
|
|
|
CP0387917
|
5-methyl-5-[(3S)-3-phenoxypyrrolidin-1-yl]-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O2
|
1
|
| 1 |
Ki = 0.25 nM
|
|
|
|
CP0387963
|
5-[3-(2-fluoro-3-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H31FN2O3
|
1
|
| 1 |
Ki = 0.26 nM
|
|
|
|
CP0440300
|
5-methyl-5-(4-phenoxypiperidin-1-yl)-2,2-diphenylhexanamide
Show/Hide
|
C30H36N2O2
|
1
|
| 1 |
Ki = 0.27 nM
|
|
|
|
CP0398267
|
[1-[3-[2-chloro-4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-5-methoxy-N-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H44ClN5O7
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0413266
|
[1-[3-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]cyclohexyl]amino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C39H47N5O6
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0441217
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-5-methoxy-2-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O7
|
1
|
| 1 |
Ki = 0.3162 nM
|
|
|
|
CP0540885
|
[(3R)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO3
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0552568
|
[1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO3
|
1
|
| 1 |
Ki = 0.44 nM
|
|
|
|
CP0080609
|
1-Cyclohexyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-piperidine
Show/Hide
|
C26H33NO3S
|
1
|
| 1 |
Ki = 0.48 nM
|
|
|
|
CP0384251
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxy-2-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O7
|
1
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| 1 |
Ki = 0.5012 nM
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CP0387964
|
5-[(3R)-3-(3-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
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C29H34N2O3
|
1
|
| 1 |
Ki = 0.51 nM
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CP0543095
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[1-[3-(4-chlorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
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C30H33BrClNO3
|
1
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| 1 |
Ki = 0.51 nM
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CP0673820
|
2-(2,2-diphenylacetoxy)-N,N,N-triethylethanaminiumiodide
Show/Hide
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C22H30INO2
|
1
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| 1 |
Ki = 0.543 nM
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CP0391062
|
5-[(3R)-3-(3-fluoro-5-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
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C29H33FN2O3
|
1
|
| 1 |
Ki = 0.56 nM
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CP0400417
|
5-[3-(3-fluoro-5-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
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C28H31FN2O3
|
1
|
| 1 |
Ki = 0.6 nM
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CP0418740
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxy-N-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O7
|
1
|
| 1 |
Ki = 0.631 nM
|
|
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CP0550008
|
[1-[3-[2-chloro-4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxyanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H42ClN5O7
|
1
|
| 1 |
Ki = 0.631 nM
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CP0550010
|
[1-[2-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]benzoyl]amino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C39H41N5O6
|
1
|
| 1 |
Ki = 0.631 nM
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CP0562060
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[1-(2-phenylsulfanylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C29H32BrNO3S
|
1
|
| 1 |
Ki = 0.65 nM
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CP0873360
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenethyl-pyrrolidinium bromide
Show/Hide
|
C28H32BrN3O
|
1
|
| 1 |
Ki = 0.67 nM
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CP0425074
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-propyl)-pyrrolidinium
Show/Hide
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C29H34N3O+
|
1
|
| 1 |
Ki = 0.7 nM
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CP0393464
|
5-[3-(2-fluoro-5-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
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C28H31FN2O3
|
1
|
| 1 |
Ki = 0.71 nM
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CP0475146
|
4-[1-[3-(3-hydroxyphenoxy)azetidin-1-yl]cyclopentyl]-2,2-diphenylbutanamide
Show/Hide
|
C30H34N2O3
|
1
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| 1 |
Ki = 0.73 nM
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CP0435668
|
1-methyl-3-(R)-[4,4-Bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-phenethyl-pyrrolidinium
Show/Hide
|
C28H30F2N3O+
|
1
|
| 1 |
Ki = 0.75 nM
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CP0475150
|
5-[(3S)-3-(4-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O3
|
1
|
| 1 |
Ki = 0.76 nM
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CP0413169
|
[1-[2-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]benzoyl]-methylamino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O6
|
1
|
| 1 |
Ki = 0.7943 nM
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CP0477680
|
6-[3-[3-(1,3-benzothiazol-7-ylsulfonyl)propanoyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridine-3-carbonitrile
Show/Hide
|
C22H21N5O3S2
|
1
|
| 1 |
Ki = 0.84 nM
|
|
|
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CP0472767
|
(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methyl-trimethylazanium;iodide
Show/Hide
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C20H32INO2
|
1
|
| 1 |
Ki = 0.8511 nM
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|
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CP0548236
|
[1-[3-(4-methylphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
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| 1 |
Ki = 0.86 nM
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CP0552567
|
[1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
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C29H32BrNO3
|
1
|
| 1 |
Ki = 0.86 nM
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CP0426656
|
[1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H34BrNO4
|
1
|
| 1 |
Ki = 0.88 nM
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CP0487381
|
[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 0.8913 nM
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CP0516427
|
1-[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 0.955 nM
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CP0398266
|
[1-[3-[3-[2-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]ethyl]anilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
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C40H43N5O6
|
1
|
| 1 |
Ki = 1 nM
|
|
|
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CP0516424
|
Flotros
Show/Hide
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C25H30ClNO3
|
1
|
| 1 |
Ki = 1.023 nM
|
|
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CP0526055
|
1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
|
| 1 |
Ki = 1.04 nM
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CP0528505
|
[1-[3-(3-fluorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrFNO3
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
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CP0550007
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methylanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O6
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
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CP0540884
|
[1-[3-[4-(trifluoromethoxy)phenyl]propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H33BrF3NO4
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
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CP0390370
|
1-[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H23NO2
|
1
|
| 1 |
Ki = 1.514 nM
|
|
|
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CP0481431
|
[1-[3-[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-2-methoxyanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O7
|
1
|
| 1 |
Ki = 1.585 nM
|
|
|
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CP0392023
|
5-methyl-5-[(3R)-3-phenoxypyrrolidin-1-yl]-2,2-diphenylhexanamide
Show/Hide
|
C29H34N2O2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
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CP0425077
|
1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-thiophen-3-ylethyl)-pyrrolidinium
Show/Hide
|
C26H26F2N3O2S+
|
1
|
| 1 |
Ki = 1.62 nM
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CP0548006
|
[1-[3-(4-fluorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrFNO3
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
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CP0505237
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenoxy-propyl)-pyrrolidinium
Show/Hide
|
C29H34N3O2+
|
1
|
| 1 |
Ki = 1.76 nM
|
|
|
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CP0425078
|
1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium
Show/Hide
|
C28H28F2N3O2+
|
1
|
| 1 |
Ki = 1.84 nM
|
|
|
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CP0435669
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
|
| 1 |
Ki = 1.89 nM
|
|
|
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CP0442398
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-oxo-2-phenyl-ethyl)-pyrrolidinium
Show/Hide
|
C28H30N3O2+
|
1
|
| 1 |
Ki = 1.89 nM
|
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CP0387962
|
5-[3-(4-chloro-3-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H31ClN2O3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
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CP0421654
|
[1-[3-(3-methylphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
|
| 1 |
Ki = 1.9 nM
|
|
|
|
CP0421081
|
1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 1.905 nM
|
|
|
|
CP0088670
|
Batefenterol
Show/Hide
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C40H42ClN5O7
|
1
|
| 1 |
Ki = 1.995 nM
|
|
|
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CP0418739
|
[1-[3-[3-[2-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]ethyl]-4-methoxyanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O7
|
1
|
| 1 |
Ki = 1.995 nM
|
|
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CP0400416
|
5-[(3S)-3-(4-chloro-3-hydroxyphenoxy)pyrrolidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C29H33ClN2O3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0109931
|
ATROPEN
Show/Hide
|
C17H23NO3
|
1
|
| 1 |
Ki = 2.18 nM
|
|
|
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CP0440288
|
5-[4-(3-hydroxyphenoxy)piperidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C30H36N2O3
|
1
|
| 1 |
Ki = 2.3 nM
|
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CP0412104
|
[1-[3-[4-(trifluoromethyl)phenyl]propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H33BrF3NO3
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
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CP0392021
|
5-[(3S)-3-phenoxypyrrolidin-1-yl]-2,2-diphenylpentanamide
Show/Hide
|
C27H30N2O2
|
1
|
| 1 |
Ki = 2.4 nM
|
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CP0552569
|
[1-[3-(4-bromophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33Br2NO3
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
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CP0435671
|
1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-2-ylethyl)-pyrrolidinium
Show/Hide
|
C27H27F2N4O2+
|
1
|
| 1 |
Ki = 2.61 nM
|
|
|
|
CP0412100
|
[1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C29H32BrNO4
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
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CP0405402
|
1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-[2-(3-fluoro-phenyl)-2-oxo-ethyl]-pyrrolidinium
Show/Hide
|
C28H27F3N3O2+
|
1
|
| 1 |
Ki = 3.01 nM
|
|
|
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CP0468712
|
S-[2-(diethylamino)ethyl] 2-hydroxy-2,2-diphenylethanethioate
Show/Hide
|
C20H25NO2S
|
1
|
| 1 |
Ki = 3.12 nM
|
|
|
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CP0379313
|
[1-[2-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-2,5-dimethylbenzoyl]amino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O6
|
1
|
| 1 |
Ki = 3.162 nM
|
|
|
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CP0203329
|
4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(piperidin-4-yl)piperidine
Show/Hide
|
C25H32N2O3S
|
1
|
| 1 |
Ki = 3.4 nM
|
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CP0167280
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid ethyl ester
Show/Hide
|
C28H36N2O5S
|
1
|
| 1 |
Ki = 3.7 nM
|
|
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CP0443935
|
[1-[3-(3-iodophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrINO3
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0850774
|
METHYLBENACTYZIUM BROMIDE
Show/Hide
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C21H28BrNO3
|
1
|
| 1 |
Ki = 4.25 nM
|
|
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CP0548005
|
[1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO3
|
1
|
| 1 |
Ki = 4.7 nM
|
|
|
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CP0855970
|
Mepenzolate
Show/Hide
|
C21H26BrNO3
|
1
|
| 1 |
Ki = 5.3 nM
|
|
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CP0436551
|
1-(bicyclo[2.2.1]hept-5-en-2-yl)-1-phenyl-3-(piperidin-1-yl)propan-1-ol
Show/Hide
|
C21H29NO
|
1
|
| 1 |
Ki = 5.95 nM
|
|
|
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CP0433352
|
3-(diethylamino)propyl (3S)-3-methyl-2-phenylpentanoate
Show/Hide
|
C19H31NO2
|
1
|
| 1 |
Ki = 5.97 nM
|
|
|
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CP0398268
|
[1-[2-[[4-[[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]methyl]-3-methoxybenzoyl]amino]ethyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C40H43N5O7
|
1
|
| 1 |
Ki = 6.31 nM
|
|
|
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CP0175835
|
Isoptpo Hyoscine
Show/Hide
|
C17H21NO4
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0528506
|
[1-[3-(3-chlorophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C30H33BrClNO3
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0491603
|
2-(diethylamino)ethyl 2-cyclohexyl-2-hydroxy-2-thiophen-2-ylacetate
Show/Hide
|
C18H29NO3S
|
1
|
| 1 |
Ki = 6.55 nM
|
|
|
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CP0511887
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(3-phenyl-oxiranylmethyl)-pyrrolidinium
Show/Hide
|
C29H32N3O2+
|
1
|
| 1 |
Ki = 6.66 nM
|
|
|
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CP0405401
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-benzyloxy-ethyl)-pyrrolidinium
Show/Hide
|
C29H34N3O2+
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
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CP0456644
|
5-[3-(2,4-dichloro-5-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H30Cl2N2O3
|
1
|
| 1 |
Ki = 7.3 nM
|
|
|
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CP0425073
|
1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
Show/Hide
|
C28H32N3O2+
|
1
|
| 1 |
Ki = 7.6 nM
|
|
|
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CP0540883
|
[1-[3-(4-methoxyphenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
Show/Hide
|
C31H36BrNO4
|
1
|
| 1 |
Ki = 7.8 nM
|
|
|
|
CP0398269
|
[1-[3-[5-[2-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]ethyl]-2-methoxyanilino]-3-oxopropyl]piperidin-4-yl] N-(2-phenylphenyl)carbamate
Show/Hide
|
C41H45N5O7
|
1
|
| 1 |
Ki = 7.943 nM
|
|
|
|
CP0420726
|
2-(diethylamino)ethyl 2-(1-hydroxycyclohexyl)-2-phenylacetate
Show/Hide
|
C20H31NO3
|
1
|
| 1 |
Ki = 8.37 nM
|
|
|
|
CP0379032
|
1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-phenylcarbamoylmethyl-pyrrolidinium
Show/Hide
|
C28H31N4O2+
|
1
|
| 1 |
Ki = 9.11 nM
|
|
|
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CP0209448
|
4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)-1-(propylsulfonyl)piperidine
Show/Hide
|
C28H38N2O5S2
|
1
|
| 1 |
Ki = 10.1 nM
|
|
|
|
CP0476223
|
5-[3-(2-hydroxyphenoxy)azetidin-1-yl]-5-methyl-2,2-diphenylhexanamide
Show/Hide
|
C28H32N2O3
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0433507
|
(1-methylpiperidin-4-yl) 3-hydroxy-2-[3-(trifluoromethyl)phenyl]propanoate
Show/Hide
|
C16H20F3NO3
|
1
|
| 1 |
Ki = 11.2 nM
|
|
|
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CP0002227
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SOLIFENACIN
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C23H26N2O2
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1
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| 1 |
Ki = 13.18 nM
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CP0564271
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[(2R,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H32INO2
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1
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| 1 |
Ki = 14.45 nM
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CP0438023
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[1-(5-phenylpentyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C32H38BrNO3
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1
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| 1 |
Ki = 17 nM
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CP0540887
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[1-[3-[3-(trifluoromethyl)phenyl]propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C31H33BrF3NO3
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1
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| 1 |
Ki = 19 nM
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CP0465680
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(3S)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
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C24H29NO3
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1
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| 1 |
Ki = 19.95 nM
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CP0543094
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[1-[3-(3-bromophenyl)propyl]-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C30H33Br2NO3
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1
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| 1 |
Ki = 20 nM
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CP0425076
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1-methyl-3-(R)-3-[4,4-bis-(4-fluoro-phenyl)-2-oxo-imidazolidin-1-yl]-1-(2-oxo-2-pyridin-3-ylethyl)-pyrrolidinium
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C27H27F2N4O2+
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1
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| 1 |
Ki = 22.9 nM
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CP0375774
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N,N-dimethyl-2-[3-(2-pyridin-2-ylpropan-2-yl)-1H-inden-2-yl]ethanamine
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C21H26N2
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1
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| 1 |
Ki = 25.7 nM
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CP0521081
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[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium
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C20H32NO2+
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1
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| 1 |
Ki = 30.9 nM
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CP0406396
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N,N-dimethyl-1-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methanamine
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C19H22N2
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1
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| 1 |
Ki = 31.62 nM
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CP0414398
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[(2R,5R)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H32INO2
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1
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| 1 |
Ki = 37.15 nM
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CP0540935
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2-[2-[6-[8-[6-[bis[2-oxo-2-(6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)ethyl]amino]hexyl-methylamino]octyl-methylamino]hexylamino]acetyl]-2,4,9,15-tetrazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-10-one
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C63H76N14O6
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1
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| 1 |
Ki = 38.02 nM
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CP0849141
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11-{2-[[(1S,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
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C28H34N4O10
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1
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| 1 |
Ki = 39.81 nM
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CP0849144
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11-{2-[[(1R,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
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C28H34N4O10
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1
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| 1 |
Ki = 40.74 nM
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CP0426657
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[1-(4-phenoxybutyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C31H36BrNO4
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1
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| 1 |
Ki = 41 nM
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CP0434673
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[1-(3-phenylmethoxypropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C31H36BrNO4
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1
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| 1 |
Ki = 42 nM
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CP0471590
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(3R)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
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C24H29NO3
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1
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| 1 |
Ki = 43.65 nM
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CP0473020
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[(2R,5S)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H32INO2
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1
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| 1 |
Ki = 43.65 nM
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CP0858320
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11-{2-[[(1R,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
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C28H34N4O10
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1
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| 1 |
Ki = 44.67 nM
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CP0056034
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11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one
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C19H21N5O2
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1
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| 1 |
Ki = 47.86 nM
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CP0849067
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11-{2-[[(1S,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
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C28H34N4O10
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1
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| 1 |
Ki = 48.98 nM
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CP0101233
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2-(4-Hydroxy-phenyl)-2-phenyl-propionic acid 2-diethylamino-ethyl ester
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C21H27NO3
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1
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| 1 |
Ki = 52.2 nM
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CP0468678
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2-[di(propan-2-yl)amino]ethyl 2-hydroxy-2,2-diphenylacetate
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C22H29NO3
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1
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| 1 |
Ki = 59 nM
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CP0225899
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AQ-RA 741
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C27H37N5O2
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1
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| 1 |
Ki = 63.1 nM
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CP0217520
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AF-DX 384
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C27H38N6O2
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1
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| 1 |
Ki = 66.07 nM
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CP0397949
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N,N-dimethyl-2-[3-[phenyl(pyridin-2-yl)methyl]-1H-inden-2-yl]ethanamine
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C25H26N2
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1
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| 1 |
Ki = 67.61 nM
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CP0475081
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1-[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
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C19H23NO2
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1
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| 1 |
Ki = 72.44 nM
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CP0540886
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(1-benzyl-1-azoniabicyclo[2.2.2]octan-3-yl) 2-hydroxy-2,2-diphenylacetate;bromide
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C28H30BrNO3
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1
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| 1 |
Ki = 81 nM
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CP0403962
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2-[6-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
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C20H23ClN2
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1
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| 1 |
Ki = 95.5 nM
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CP0489025
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(3S)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
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C24H29NO3
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1
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| 1 |
Ki = 104.71 nM
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CP0156301
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2-(diethylamino)ethyl 2-(4-chlorophenyl)sulfanylbenzoate
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C19H22ClNO2S
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1
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| 1 |
Ki = 109 nM
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CP0220544
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1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)butan-1-one
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C29H38N2O4S
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1
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| 1 |
Ki = 121.6 nM
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CP0516425
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[(2R)-5,5-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 134.9 nM
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CP0271112
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N,N-dimethyl-2-[3-[(1S)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
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C20H24N2
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1
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| 1 |
Ki = 138.04 nM
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CP0058613
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CAS_132947
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C64H77N13O6
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1
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| 1 |
Ki = 147.91 nM
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CP0428329
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8,8-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-8-azonia-bicyclo[3.2.1]octane
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C24H30N3O+
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1
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| 1 |
Ki = 153 nM
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CP0540888
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[(3S)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate;bromide
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C30H34BrNO3
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1
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| 1 |
Ki = 184 nM
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CP0220610
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Bietamiverine
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C19H30N2O2
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1
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| 1 |
Ki = 186 nM
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CP0420595
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6-methyl-5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridine-2-carboxamide
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C26H29F3N6OS
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1
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| 1 |
Ki = 186.21 nM
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CP0473019
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1-[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
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C19H29NO2
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1
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| 1 |
Ki = 186.21 nM
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CP0214556
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5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridine-2-carboxamide
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C25H27F3N6OS
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1
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| 1 |
Ki = 190.55 nM
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CP0398323
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N-[4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]cyclohexyl]acetamide
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C27H36F3N5OS
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1
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| 1 |
Ki = 229.09 nM
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CP0385601
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2-(diethylamino)ethyl 2,2-diphenylbutanoate
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C22H29NO2
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1
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| 1 |
Ki = 243 nM
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CP0368307
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5-[5-[3-[1-[2-fluoro-4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
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C23H26F4N6OS
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1
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| 1 |
Ki = 245.47 nM
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CP0425075
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1,1-dimethyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-piperidinium
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C22H28N3O+
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1
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| 1 |
Ki = 249 nM
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CP0432187
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2-(diethylamino)ethyl 2-(2,6-dimethylphenyl)-2-hydroxy-2-phenylacetate
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C22H29NO3
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1
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| 1 |
Ki = 254 nM
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CP0397929
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2-[5-fluoro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
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C20H23FN2
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1
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| 1 |
Ki = 263.03 nM
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CP0386733
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[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C24H27NO4
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1
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| 1 |
Ki = 269.15 nM
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CP0822547
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2-(2,2-diphenylacetoxy)-N,N-diethyl-Nmethylethanaminiumbromide
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C21H28BrNO2
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1
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| 1 |
Ki = 270 nM
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CP0875549
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1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-piperidinium iodide
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C22H30INO
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1
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| 1 |
Ki = 275.42 nM
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CP0380644
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4-methyl-5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
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C23H26F3N5OS
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1
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| 1 |
Ki = 275.42 nM
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CP0398325
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4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]thiadiazole
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C21H23F3N6S2
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1
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| 1 |
Ki = 275.42 nM
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CP0416602
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2-[6-chloro-3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]-N,N-dimethylethanamine
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C21H25ClN2
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1
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| 1 |
Ki = 281.84 nM
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CP0511888
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1-methyl-3-(R)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-benzyl-pyrrolidinium
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C27H30N3O+
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1
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| 1 |
Ki = 282 nM
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CP0449403
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N,N-dimethyl-2-[3-(1-phenylethyl)-1H-inden-2-yl]ethanamine
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C21H25N
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1
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| 1 |
Ki = 288.4 nM
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CP0179022
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2-[4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]phenyl]-1,3-oxazole
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C28H28F3N5OS
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1
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| 1 |
Ki = 302 nM
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CP0436921
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N,N-dimethyl-2-[3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]ethanamine
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C21H26N2
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1
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| 1 |
Ki = 309.03 nM
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CP0455599
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1,1-dimethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium
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C21H26N3O+
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1
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| 1 |
Ki = 310 nM
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CP0442399
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trimethyl-[2-(2-oxo-4,4-diphenylimidazolidin-1-yl)ethyl]azanium
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C20H26N3O+
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1
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| 1 |
Ki = 335 nM
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CP0398327
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1-methyl-4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridin-2-one
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C25H28F3N5OS
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1
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| 1 |
Ki = 354.81 nM
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CP0517270
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[(2R,5S,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 354.81 nM
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CP0511886
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1-methoxyethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
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C30H36N3O3+
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1
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| 1 |
Ki = 356 nM
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CP0851174
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1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium-4-yl]-1-methylpiperidin-1-ium diiodide
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C44H58I2N2O2
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1
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| 1 |
Ki = 371.54 nM
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CP0300572
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3-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]benzamide
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C26H28F3N5OS
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1
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| 1 |
Ki = 380.19 nM
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CP0842192
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2-(2,2-diphenylacetoxy)-N,N,Ntrimethylethanaminiumbromide
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C19H24BrNO2
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1
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| 1 |
Ki = 384 nM
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CP0386735
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[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C25H29NO4
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1
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| 1 |
Ki = 398.11 nM
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CP0390368
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[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C25H29NO4
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1
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| 1 |
Ki = 416.87 nM
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CP0398324
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5-[5-[3-[(2R,3R)-2-[2-fluoro-4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
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C23H25F4N5OS
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1
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| 1 |
Ki = 426.58 nM
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CP0398326
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4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]benzamide
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C26H28F3N5OS
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1
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| 1 |
Ki = 426.58 nM
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CP0122473
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1-methyl-5-[4-methyl-5-[3-[1-[4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridin-2-one
Show/Hide
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C25H29F3N6OS
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1
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| 1 |
Ki = 478.63 nM
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CP0403738
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2-[5-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
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C20H23ClN2
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1
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| 1 |
Ki = 501.19 nM
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CP0441146
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N,N-dimethyl-2-[6-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2
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1
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| 1 |
Ki = 501.19 nM
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CP0446158
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benzyl-dimethyl-[2-(2-oxo-4,4-diphenylimidazolidin-1-yl)ethyl]azanium
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C26H30N3O+
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1
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| 1 |
Ki = 507 nM
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CP0532167
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1-cyanomethyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-(2-phenoxy-ethyl)-pyrrolidinium
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C29H31N4O2+
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1
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| 1 |
Ki = 541 nM
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CP0380642
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5-[5-[3-[(2S,3R)-2-[2-fluoro-4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
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C23H25F4N5OS
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1
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| 1 |
Ki = 549.54 nM
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CP0372485
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N,N-dimethyl-3-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]propan-1-amine
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C21H26N2
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1
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| 1 |
Ki = 575.44 nM
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CP0378875
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1-benzyl-1-methyl-4-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-piperidinium
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C28H32N3O+
|
1
|
| 1 |
Ki = 612 nM
|
|
|
|
CP0410687
|
(3R)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 616.6 nM
|
|
|
|
CP0891232
|
Alamethicin
Show/Hide
|
C92H150N22O25
|
1
|
| 1 |
Ki = 619 nM
|
|
|
|
CP0392151
|
N,N-dimethyl-2-[3-(1-pyridin-2-ylbutyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C22H28N2
|
1
|
| 1 |
Ki = 630.96 nM
|
|
|
|
CP0134104
|
5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-3H-pyridin-2-one
Show/Hide
|
C24H26F3N5OS
|
1
|
| 1 |
Ki = 630.96 nM
|
|
|
|
CP0851172
|
4-(4-hydroxy-4,4-diphenylbutyl)piperazine-1,4-diium dichloride
Show/Hide
|
C20H28Cl2N2O
|
1
|
| 1 |
Ki = 660.69 nM
|
|
|
|
CP0398322
|
4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-3H-pyridin-2-one
Show/Hide
|
C24H26F3N5OS
|
1
|
| 1 |
Ki = 676.08 nM
|
|
|
|
CP0462407
|
4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]piperidine-1-carboxamide
Show/Hide
|
C25H33F3N6OS
|
1
|
| 1 |
Ki = 676.08 nM
|
|
|
|
CP0436507
|
N-(2-fluoroethyl)-N-methyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H25FN2
|
1
|
| 1 |
Ki = 707.95 nM
|
|
|
|
CP0139207
|
9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
|
C23H24N2O4
|
1
|
| 1 |
Ki = 724.44 nM
|
|
|
|
CP0851169
|
1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)piperidin-1-ium-4-yl]piperidin-1-ium dichloride
Show/Hide
|
C42H54Cl2N2O2
|
1
|
| 1 |
Ki = 724.44 nM
|
|
|
|
CP0379030
|
1-benzyl-1-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-pyrrolidinium
Show/Hide
|
C27H30N3O+
|
1
|
| 1 |
Ki = 727 nM
|
|
|
|
CP0403951
|
N-methyl-N-[[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methyl]propan-2-amine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 741.31 nM
|
|
|
|
CP0479764
|
N-[3-[1-[2-(8-chloro-6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-2-oxoethyl]piperidin-4-yl]propyl]-N-ethyl-2,2-dimethylpentanamide
Show/Hide
|
C31H42ClN5O3
|
1
|
| 1 |
Ki = 776.25 nM
|
|
|
|
CP0380480
|
(2R,3S)-5-[3-[[4-methyl-5-(oxan-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptane
Show/Hide
|
C24H31F3N4OS
|
1
|
| 1 |
Ki = 891.25 nM
|
|
|
|
CP0372479
|
N,N-diethyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C22H28N2
|
1
|
| 1 |
Ki = 954.99 nM
|
|
|
|
CP0472768
|
trimethyl-[[(2R,5R)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 977.24 nM
|
|
|
|
CP0406408
|
N,N-dimethyl-2-[5-methylsulfanyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2S
|
1
|
| 1 |
Ki = 1047.13 nM
|
|
|
|
CP0404647
|
4-[4-methyl-5-[3-[1-[4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1H-pyridin-2-one
Show/Hide
|
C24H27F3N6OS
|
1
|
| 1 |
Ki = 1096.48 nM
|
|
|
|
CP0487380
|
trimethyl-[[(2R,5S)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C26H30INO2
|
1
|
| 1 |
Ki = 1096.48 nM
|
|
|
|
CP0851168
|
DIPHENIDOL HYDROCHLORIDE
Show/Hide
|
C21H28ClNO
|
1
|
| 1 |
Ki = 1122.02 nM
|
|
|
|
CP0458157
|
4-methyl-5-[4-methyl-5-[3-[(2S,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
|
C23H26F3N5OS
|
1
|
| 1 |
Ki = 1148.15 nM
|
|
|
|
CP0372477
|
2-[6-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
Ki = 1174.9 nM
|
|
|
|
CP0420656
|
(2R,3S)-5-[3-[[4-methyl-5-(2-methylpyridin-3-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptane
Show/Hide
|
C25H28F3N5S
|
1
|
| 1 |
Ki = 1230.27 nM
|
|
|
|
CP0066235
|
4-methyl-5-[4-methyl-5-[3-(1-phenyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl)propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
|
C22H28N6OS
|
1
|
| 1 |
Ki = 1258.93 nM
|
|
|
|
CP0479629
|
[(2R,5S)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO3S
|
1
|
| 1 |
Ki = 1318.26 nM
|
|
|
|
CP0479715
|
[(2R,6R)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO3S
|
1
|
| 1 |
Ki = 1318.26 nM
|
|
|
|
CP0425606
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-(4-methoxy-phenyl)-ethyl ester; oxalic acid
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
Ki = 1370 nM
|
|
|
|
CP0364090
|
5-[3-[[4-methyl-5-(oxan-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-1-phenyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole
Show/Hide
|
C23H33N5OS
|
1
|
| 1 |
Ki = 1445.44 nM
|
|
|
|
CP0398329
|
5-[5-[3-[(2S,3R)-2-[4-fluoro-2-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H25F4N5OS
|
1
|
| 1 |
Ki = 1479.11 nM
|
|
|
|
CP0397931
|
N,N-dimethyl-2-[3-(pyridin-2-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C19H22N2
|
1
|
| 1 |
Ki = 1548.82 nM
|
|
|
|
CP0410686
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 1548.82 nM
|
|
|
|
CP0516426
|
[(2R,5R,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 1548.82 nM
|
|
|
|
CP0386734
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 1621.81 nM
|
|
|
|
CP0415329
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 1698.24 nM
|
|
|
|
CP0472770
|
trimethyl-[[(2R,6R)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 1698.24 nM
|
|
|
|
CP0487384
|
[(2R,5R)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C21H28INO2
|
1
|
| 1 |
Ki = 1698.24 nM
|
|
|
|
CP0862110
|
N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N3-dimethylpropane-1,3-diaminium chloride
Show/Hide
|
C37H48Cl2N2O2
|
1
|
| 1 |
Ki = 1737.8 nM
|
|
|
|
CP0372527
|
2-[1-[2-(2-piperidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
|
C23H28N2
|
1
|
| 1 |
Ki = 1778.28 nM
|
|
|
|
CP0449839
|
N-methyl-N-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]propan-2-amine
Show/Hide
|
C22H28N2
|
1
|
| 1 |
Ki = 1819.7 nM
|
|
|
|
CP0372523
|
2-[1-[2-(2-pyrrolidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
|
C22H26N2
|
1
|
| 1 |
Ki = 1905.46 nM
|
|
|
|
CP0479714
|
trimethyl-[[(2R,5R)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C26H30INO2
|
1
|
| 1 |
Ki = 1995.26 nM
|
|
|
|
CP0237860
|
4-methyl-5-[4-methyl-5-[3-[(2S,3R)-2-phenyl-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
|
C22H27N5OS
|
1
|
| 1 |
Ki = 2041.74 nM
|
|
|
|
CP0455598
|
trimethyl-[3-(2-oxo-4,4-diphenylimidazolidin-1-yl)propyl]azanium
Show/Hide
|
C21H28N3O+
|
1
|
| 1 |
Ki = 2065 nM
|
|
|
|
CP0445692
|
5-[5-[3-[(2S,3S)-2-[4-fluoro-2-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H25F4N5OS
|
1
|
| 1 |
Ki = 2089.3 nM
|
|
|
|
CP0317889
|
5-[3-[(4-methyl-5-pyridin-3-yl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1-[2-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole
Show/Hide
|
C24H27F3N6S
|
1
|
| 1 |
Ki = 2187.76 nM
|
|
|
|
CP0487382
|
[(2R,5R)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C21H28INO2
|
1
|
| 1 |
Ki = 2238.72 nM
|
|
|
|
CP0479720
|
[(2R,6R)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO4S
|
1
|
| 1 |
Ki = 2344.23 nM
|
|
|
|
CP0473022
|
[(2R,5S)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C21H28INO2
|
1
|
| 1 |
Ki = 2398.83 nM
|
|
|
|
CP0492466
|
N,N-dimethyl-2-[5-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 2511.89 nM
|
|
|
|
CP0405400
|
8-benzyl-8-methyl-3-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-8-azonia-bicyclo[3.2.1]octane
Show/Hide
|
C30H34N3O+
|
1
|
| 1 |
Ki = 2535 nM
|
|
|
|
CP0386736
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 2630.27 nM
|
|
|
|
CP0404155
|
4-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]morpholine
Show/Hide
|
C22H26N2O
|
1
|
| 1 |
Ki = 2754.23 nM
|
|
|
|
CP0418483
|
2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H25NO3
|
1
|
| 1 |
Ki = 2840 nM
|
|
|
|
CP0453180
|
1-methyl-3-(S)-(2-oxo-4,4-diphenyl-imidazolidin-1-yl)-1-benzyl pyrrolidinium
Show/Hide
|
C27H30N3O+
|
1
|
| 1 |
Ki = 3158 nM
|
|
|
|
CP0403766
|
2-[5-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O
|
1
|
| 1 |
Ki = 3162.28 nM
|
|
|
|
CP0139209
|
N,N-dimethyl-2-[3-[(1R)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 3388.44 nM
|
|
|
|
CP0913741
|
4-(1,1-dimethylpiperidin-1-ium-4-yl)-1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium diiodide
Show/Hide
|
C29H44I2N2O
|
1
|
| 1 |
Ki = 3630.78 nM
|
|
|
|
CP0425883
|
3-(4-methoxyphenyl)propyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 4070 nM
|
|
|
|
CP0875550
|
4-(4-Hydroxy-4,4-diphenyl-butyl)-1,1-dimethyl-piperazin-1-ium iodide
Show/Hide
|
C22H31IN2O
|
1
|
| 1 |
Ki = 4073.8 nM
|
|
|
|
CP0473017
|
trimethyl-[[(2R,5S)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
|
1
|
| 1 |
Ki = 4466.84 nM
|
|
|
|
CP0437455
|
[(2R,5S,6S)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 4677.35 nM
|
|
|
|
CP0425882
|
2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(2-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H24FNO3
|
1
|
| 1 |
Ki = 4890 nM
|
|
|
|
CP0862120
|
1-(4-hydroxy-4,4-diphenylbutyl)-4-(1-methylpiperidin-1-ium-4-yl)piperidin-1-ium dichloride
Show/Hide
|
C27H40Cl2N2O
|
1
|
| 1 |
Ki = 5248.07 nM
|
|
|
|
CP0862114
|
1,4-Bis-(4-hydroxy-4,4-diphenyl-butyl)-1-methyl-piperazin-1-ium iodide
Show/Hide
|
C37H45IN2O2
|
1
|
| 1 |
Ki = 5495.41 nM
|
|
|
|
CP0473018
|
[(2R,5R)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO4S
|
1
|
| 1 |
Ki = 7244.36 nM
|
|
|
|
CP0479717
|
trimethyl-[[(2R,5R)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C14H22INO2
|
1
|
| 1 |
Ki = 7244.36 nM
|
|
|
|
CP0851171
|
4-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperazine-1,4-diium dichloride
Show/Hide
|
C21H30Cl2N2O
|
1
|
| 1 |
Ki = 7413.1 nM
|
|
|
|
CP0851173
|
1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-4-phenyl-piperazin-1-ium iodide
Show/Hide
|
C27H33IN2O
|
1
|
| 1 |
Ki = 7585.78 nM
|
|
|
|
CP0164673
|
2,2-Diphenyl-propionic acid 2-diethylamino-ethyl ester
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
Ki = 7760 nM
|
|
|
|
CP0851569
|
1-(3,5-dichlorophenyl)piperazine
Show/Hide
|
C10H12Cl2N2
|
1
|
| 1 |
Ki = 7943.28 nM
|
|
|
|
CP0399353
|
N,N-dimethyl-2-[3-(pyridin-3-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C19H22N2
|
1
|
| 1 |
Ki = 8128.31 nM
|
|
|
|
CP0424269
|
2-(dimethylamino)ethyl 3-(pyridin-3-ylmethyl)-1H-indene-2-carboxylate
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 8128.31 nM
|
|
|
|
CP0404384
|
2-(dimethylamino)ethyl 3-(pyridin-2-ylmethyl)-1H-indene-2-carboxylate
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 8912.51 nM
|
|
|
|
CP0381409
|
11-[2-[(4aS,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0381581
|
11-[2-[(4aR,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0010653
|
2-{1-[2-(2,3-Dihydro-benzofuran-5-yl)-ethyl]-pyrrolidin-3-yl}-2,2-diphenyl-acetamide (Darifenacin)
Show/Hide
|
C28H30N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
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CP0387007
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[(2R,5S)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO4S
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1
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| 1 |
Ki > 10000 nM
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CP0421082
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trimethyl-[[(2R,5S)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C14H22INO2
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1
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| 1 |
Ki > 10000 nM
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CP0472769
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trimethyl-[[(2R,6S)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
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C20H26INO2S
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1
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| 1 |
Ki > 10000 nM
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CP0473016
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[(2R,5S)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C21H28INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479627
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trimethyl-[[(2R,5S)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479628
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trimethyl-[[(2R,5R)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479654
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trimethyl-[[(2R,6R)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479708
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[(2R,6S)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
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1
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| 1 |
Ki > 10000 nM
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CP0479711
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trimethyl-[[(2R,6S)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0491695
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[(2R,6S)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki > 10000 nM
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CP0516423
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[(2R,5R)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki > 10000 nM
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CP0505786
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N,N-dimethyl-2-[3-(pyridin-4-ylmethyl)-1H-inden-2-yl]ethanamine
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C19H22N2
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1
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| 1 |
Ki = 11748.98 nM
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CP0862121
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N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N3,N3-tetramethylpropane-1,3-diaminium iodide
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C39H52I2N2O2
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1
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| 1 |
Ki = 12302.69 nM
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CP0386732
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C24H27NO4
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1
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| 1 |
Ki = 14454.4 nM
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CP0069240
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4-(piperazin-1-yl)-1H-indole
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C12H15N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0184743
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4-methyl-2-piperazin-1-ylquinoline
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C14H17N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0364794
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1-(2,3-dichlorophenyl)piperazine
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C10H12Cl2N2
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1
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| 1 |
Ki > 19952.62 nM
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CP0404254
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N-[2-(dimethylamino)ethyl]-3-(pyridin-2-ylmethyl)-1H-indene-2-carboxamide
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 23988.33 nM
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CP0484746
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H27NO3
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1
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| 1 |
Ki = 31100 nM
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CP0862112
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N1,N2-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N2,N2-tetramethylethane-1,2-diaminium iodide
Show/Hide
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C38H50I2N2O2
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1
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| 1 |
Ki = 43651.58 nM
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CP0416829
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N-[2-(dimethylamino)ethyl]-3-(pyridin-3-ylmethyl)-1H-indene-2-carboxamide
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 48977.88 nM
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CP0862118
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1-(4-Hydroxy-4,4-diphenyl-butyl)-4-phenyl-piperazin-1-ium chloride
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C26H31ClN2O
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1
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| 1 |
Ki = 70794.58 nM
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CP0862116
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1,4-bis(4-hydroxy-4,4-diphenylbutyl)piperazine-1,4-diium dichloride
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C36H44Cl2N2O2
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1
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| 1 |
Ki = 87096.36 nM
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CP0418482
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2-naphthalen-1-ylethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C25H25NO2
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1
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| 1 |
Ki > 100000 nM
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CP0425884
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2-(3,4-dimethoxyphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H27NO4
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1
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| 1 |
Ki > 100000 nM
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CP0471231
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2-(3,4-dimethoxyphenyl)ethyl 4-(3-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H26FNO4
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1
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| 1 |
Ki > 100000 nM
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