| Compound ID |
Compound Name |
Compound Formula |
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
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|
C10H12N2O
|
5
|
| 1 |
EC50 = 7 nM
|
|
|
| 2 |
EC50 = 15 nM
|
|
|
| 3 |
EC50 = 70 nM
|
|
|
| 4 |
Kd = 3.98 nM
|
|
|
| 5 |
Ki = 2.12 nM
|
|
|
|
CP0383842
|
1-[4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl]-1,3-dihydro-2Hindol-2-one
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|
C21H24N2O
|
2
|
| 1 |
EC50 = 310 nM
|
|
|
| 2 |
Ki = 7 nM
|
|
|
|
CP0133392
|
13-methyl-7-thia-5,13-diazapentacyclo[10.7.1.02,10.04,8.016,20]icosa-1(19),2,4(8),5,9,16(20),17-heptaen-6-amine
Show/Hide
|
C18H17N3S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 260 nM
|
|
|
|
CP0339668
|
(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)urea
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|
C18H19N3O
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
IC50 = 125 nM
|
|
|
|
CP0096286
|
(R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidin-1-ylsulfonyl)phenol
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|
C18H28N2O3S
|
5
|
| 1 |
IC50 = 0.93 nM
|
|
|
| 2 |
Ki = 0.34 nM
|
|
|
| 3 |
Ki = 0.71 nM
|
|
|
| 4 |
Ki = 1.26 nM
|
|
|
| 5 |
Ki = 1.9 nM
|
|
|
|
CP0031743
|
1H-imidazo[4,5-c]pyridine derivative
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|
C18H26N4O2S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0866569
|
SID50106969
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|
C23H27ClFN3O2
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0673446
|
2-Benzyl-N-(3-methoxyphenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-4-amine hydrochloride
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|
C22H25ClN4O
|
1
|
| 1 |
IC50 = 497 nM
|
|
|
|
CP0674236
|
2-Benzyl-N-(3-chlorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-4-amine hydrochloride
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|
C21H22Cl2N4
|
1
|
| 1 |
IC50 = 1003 nM
|
|
|
|
CP0417858
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylbenzenesulfonamide
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|
C20H27N3O2S
|
1
|
| 1 |
IC50 = 1006 nM
|
|
|
|
CP0867161
|
1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride
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|
C22H31ClN2O2
|
1
|
| 1 |
IC50 = 1050 nM
|
|
|
|
CP0673445
|
2-Benzyl-N-(3-fluorophenyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-4-amine hydrochloride
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|
C21H22ClFN4
|
1
|
| 1 |
IC50 = 1059 nM
|
|
|
|
CP0724162
|
2-Benzyl-N-phenyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine-4-amine hydrochloride
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|
C21H23ClN4
|
1
|
| 1 |
IC50 = 1564 nM
|
|
|
|
CP0377208
|
N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C21H23N3O2S
|
1
|
| 1 |
IC50 = 1582 nM
|
|
|
|
CP0864251
|
1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride
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|
C24H36Cl2N2O3
|
1
|
| 1 |
IC50 = 1840 nM
|
|
|
|
CP0417851
|
N-benzyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C28H29N3O2S
|
1
|
| 1 |
IC50 = 2044 nM
|
|
|
|
CP0416325
|
N-ethyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C23H27N3O2S
|
1
|
| 1 |
IC50 = 2059 nM
|
|
|
|
CP0873149
|
1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride
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|
C24H36Cl2N2O3
|
1
|
| 1 |
IC50 = 2340 nM
|
|
|
|
CP0398637
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-1-sulfonamide
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|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 2874 nM
|
|
|
|
CP0416326
|
N-(cyclopropylmethyl)-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C25H29N3O2S
|
1
|
| 1 |
IC50 = 3038 nM
|
|
|
|
CP0487098
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propylnaphthalene-2-sulfonamide
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|
C24H29N3O2S
|
1
|
| 1 |
IC50 = 3865 nM
|
|
|
|
CP0377202
|
N-methyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
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|
C22H25N3O2S
|
1
|
| 1 |
IC50 = 4425 nM
|
|
|
|
CP0873148
|
1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride
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|
C20H27Cl3N2O
|
1
|
| 1 |
IC50 = 5790 nM
|
|
|
|
CP0447211
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3-chloro-4-fluorobenzenesulfonamide
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|
C21H24ClFN4O3S
|
1
|
| 1 |
Ki = 0.1 nM
|
|
|
|
CP0443093
|
5-fluoro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methyl-1-benzothiophene-2-sulfonamide
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|
C25H27F2N3O3S2
|
1
|
| 1 |
Ki = 0.2 nM
|
|
|
|
CP0090070
|
6-{4-[2-(methylsulfanyl)phenyl]piperazin-1-yl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide
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|
C27H37N3OS
|
1
|
| 1 |
Ki = 0.22 nM
|
|
|
|
CP0510211
|
N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H24FN3O3S
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0486995
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-1-sulfonamide
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|
C25H26FN3O3S
|
1
|
| 1 |
Ki = 0.5 nM
|
|
|
|
CP0037955
|
METHIOTHEPIN
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|
C20H24N2S2
|
3
|
| 1 |
Ki = 0.5623 nM
|
|
|
| 2 |
Ki = 0.9 nM
|
|
|
| 3 |
Ki = 1 nM
|
|
|
|
CP0447122
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C22H26FN3O3S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0042265
|
2-{4-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-butyl}-isoindole-1,3-dione
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|
C23H27N3O3
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0393445
|
N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
|
C22H24ClN3O2S
|
1
|
| 1 |
Ki = 0.6 nM
|
|
|
|
CP0440055
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3,4-dichlorobenzenesulfonamide
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|
C21H24Cl2N4O3S
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0440753
|
5-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C25H27ClFN3O3S2
|
1
|
| 1 |
Ki = 0.7 nM
|
|
|
|
CP0395875
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H26FN3O3S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0440756
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H28N4O3S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0447214
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-1-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
Ki = 0.8 nM
|
|
|
|
CP0471903
|
2-[4-(4-phenylpiperazin-1-yl)butyl]-3H-thieno[3,2-d]pyrimidin-4-one
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|
C20H24N4OS
|
1
|
| 1 |
Ki = 0.85 nM
|
|
|
|
CP0440757
|
3-chloro-4-fluoro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C21H22ClF2N3O3S
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0443102
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
|
C19H22FN3O3S2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0489949
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-3-sulfonamide
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|
C23H24FN3O3S2
|
1
|
| 1 |
Ki = 0.9 nM
|
|
|
|
CP0483453
|
3-[4-[4-(2-methylphenyl)piperazin-1-yl]butyl]-1,3-benzothiazol-2-one
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|
C22H27N3OS
|
1
|
| 1 |
Ki = 0.99 nM
|
|
|
|
CP0393444
|
N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3-hydroxybenzenesulfonamide
Show/Hide
|
C21H22ClN3O3S
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0440062
|
N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
|
C21H24FN3O3S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0473171
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
|
C22H28N4O3S
|
1
|
| 1 |
Ki = 1.1 nM
|
|
|
|
CP0395881
|
3,4-dichloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C21H22Cl2FN3O3S
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
|
CP0443103
|
N-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]naphthalene-1-sulfonamide
Show/Hide
|
C24H24FN3O3S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0443105
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C22H23FN4O3S2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0447245
|
6-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H25ClFN3O3S2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0440755
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H28FN3O3S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0395874
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
|
C23H28FN3O3S
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0461294
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C24H26N4O2S2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0486986
|
N-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H24N4O2S2
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0307921
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H26FN3O3S2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0395869
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
|
C22H28N4O2S2
|
1
|
| 1 |
Ki = 1.6 nM
|
|
|
|
CP0468503
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C21H26N4O2S2
|
1
|
| 1 |
Ki = 1.7 nM
|
|
|
|
CP0379152
|
3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-benzothiazol-2-one
Show/Hide
|
C21H24ClN3OS
|
1
|
| 1 |
Ki = 1.72 nM
|
|
|
|
CP0461293
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H28N4O2S2
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0422308
|
3-[5-(4-phenylpiperazin-1-yl)pentanoylamino]thiophene-2-carboxamide
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|
C20H26N4O2S
|
1
|
| 1 |
Ki = 1.86 nM
|
|
|
|
CP0482709
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C21H23N5O2S3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0408139
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-3-hydroxybenzenesulfonamide
Show/Hide
|
C22H24ClN3O3S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0408141
|
N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3-fluorobenzenesulfonamide
Show/Hide
|
C21H21ClFN3O2S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0160735
|
OXITRIPTAN
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|
C11H12N2O3
|
1
|
| 1 |
Ki = 2.12 nM
|
|
|
|
CP0168742
|
2a-(4-(4-phenyl-5,6-dihydropyridin-1(2H)-yl)butyl)-2a,3,4,5-tetrahydrobenzo[cd]indol-2(1H)-one
Show/Hide
|
C26H30N2O
|
1
|
| 1 |
Ki = 2.14 nM
|
|
|
|
CP0440922
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H27FN4O3S2
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0418285
|
3-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazol-2-one
Show/Hide
|
C20H22N2OS
|
1
|
| 1 |
Ki = 2.84 nM
|
|
|
|
CP0383726
|
3-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-1,3-benzothiazol-2-one
Show/Hide
|
C24H31N3O2S
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0379154
|
3-[6-(4-phenylpiperazin-1-yl)hexyl]-1,3-benzothiazol-2-one
Show/Hide
|
C23H29N3OS
|
1
|
| 1 |
Ki = 2.96 nM
|
|
|
|
CP0429435
|
3-[5-[4-(2-ethoxyphenyl)piperazin-1-yl]pentyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-one
Show/Hide
|
C25H34N4O2S
|
1
|
| 1 |
Ki = 2.99 nM
|
|
|
|
CP0395870
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
|
C19H24N4O2S3
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0399032
|
6-chloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H27ClFN3O3S
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0447097
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C22H24FN5O3S
|
1
|
| 1 |
Ki = 3.2 nM
|
|
|
|
CP0395876
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C22H25N5O2S3
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0379157
|
benzimidazolone scaffold, 15d
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|
C21H26N4O2
|
1
|
| 1 |
Ki = 3.4 nM
|
|
|
|
CP0422047
|
3-methyl-2-[4-(4-phenylpiperazin-1-yl)butyl]-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C25H28N4OS
|
1
|
| 1 |
Ki = 3.43 nM
|
|
|
|
CP0458499
|
N-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
|
C20H24N4O2S2
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0461312
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H24FN3O3S2
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0481185
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C22H26N6O2S2
|
1
|
| 1 |
Ki = 4.1 nM
|
|
|
|
CP0447218
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1-benzothiophene-3-sulfonamide
Show/Hide
|
C24H26FN3O3S2
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0437880
|
N-benzyl-3-(4-benzylpiperazin-1-yl)propanamide
Show/Hide
|
C21H27N3O
|
1
|
| 1 |
Ki = 4.34 nM
|
|
|
|
CP0447213
|
3-chloro-4-fluoro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]benzenesulfonamide
Show/Hide
|
C22H24ClF2N3O3S
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0468506
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H27FN4O2S3
|
1
|
| 1 |
Ki = 4.6 nM
|
|
|
|
CP0463415
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C23H26ClN3O2S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0395873
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25ClN4O3S2
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0499522
|
3,4-dichloro-N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]benzenesulfonamide
Show/Hide
|
C22H24Cl2FN3O3S
|
1
|
| 1 |
Ki = 5.1 nM
|
|
|
|
CP0379318
|
3-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-1,3-benzothiazol-2-one
Show/Hide
|
C23H29N3O2S
|
1
|
| 1 |
Ki = 5.16 nM
|
|
|
|
CP0510212
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3-chloro-4-fluorobenzenesulfonamide
Show/Hide
|
C21H24ClFN4O2S2
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0447262
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C22H26N6O3S
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0399460
|
3-[5-[4-(2-methoxyphenyl)piperazin-1-yl]pentyl]-1,3-benzoxazol-2-one
Show/Hide
|
C23H29N3O3
|
1
|
| 1 |
Ki = 5.9 nM
|
|
|
|
CP0413409
|
4-chloro-N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C22H23Cl2N3O2S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0447217
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
|
C20H24FN3O3S2
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
|
CP0461305
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C21H24N6O2S2
|
1
|
| 1 |
Ki = 6.3 nM
|
|
|
|
CP0395872
|
N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
|
C25H27ClN4O3S
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0451848
|
3-[5-[4-(2-ethoxyphenyl)piperazin-1-yl]pentyl]quinazolin-4-one
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
Ki = 6.88 nM
|
|
|
|
CP0447123
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C21H24Cl2N4O2S2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0481334
|
benzimidazolone scaffold, 15m
Show/Hide
|
C22H27ClN4O
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0490098
|
methyl 3-[5-(4-phenylpiperazin-1-yl)pentanoylamino]thiophene-2-carboxylate
Show/Hide
|
C21H27N3O3S
|
1
|
| 1 |
Ki = 7.54 nM
|
|
|
|
CP0418286
|
3-[7-(4-phenylpiperazin-1-yl)heptyl]-1,3-benzothiazol-2-one
Show/Hide
|
C24H31N3OS
|
1
|
| 1 |
Ki = 7.58 nM
|
|
|
|
CP0386401
|
3-[7-[4-(2-methoxyphenyl)piperazin-1-yl]heptyl]-1,3-benzoxazol-2-one
Show/Hide
|
C25H33N3O3
|
1
|
| 1 |
Ki = 7.73 nM
|
|
|
|
CP0492525
|
3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-benzothiazol-2-one
Show/Hide
|
C22H27N3O2S
|
1
|
| 1 |
Ki = 7.77 nM
|
|
|
|
CP0388479
|
3-[5-[4-(2-ethoxyphenyl)piperazin-1-yl]pentyl]-2-methylquinazolin-4-one
Show/Hide
|
C26H34N4O2
|
1
|
| 1 |
Ki = 8.42 nM
|
|
|
|
CP0555203
|
3-[7-[4-(2-methoxyphenyl)piperazin-1-yl]heptyl]-1,3-benzothiazol-2-one
Show/Hide
|
C25H33N3O2S
|
1
|
| 1 |
Ki = 8.49 nM
|
|
|
|
CP0090148
|
N-[[2-(2-chlorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
|
C29H34ClN3O2
|
1
|
| 1 |
Ki = 8.69 nM
|
|
|
|
CP0468501
|
N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C22H23F4N3O4S
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0447124
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25ClN4O2S3
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0417892
|
5-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pentanamide
Show/Hide
|
C26H35N3O2
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0429556
|
N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C21H21ClFN3O2S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0490089
|
2-[3-(4-benzylpiperazin-1-yl)propylsulfanyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C24H26N4OS2
|
1
|
| 1 |
Ki = 9.08 nM
|
|
|
|
CP0391059
|
2-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C24H25ClN4OS
|
1
|
| 1 |
Ki = 9.42 nM
|
|
|
|
CP0506619
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3-chloro-4-fluorobenzenesulfonamide
Show/Hide
|
C20H22ClFN4O2S2
|
1
|
| 1 |
Ki = 9.5 nM
|
|
|
|
CP0466976
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H26N4O2S3
|
1
|
| 1 |
Ki = 9.9 nM
|
|
|
|
CP0510213
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3-chloro-4-fluorobenzenesulfonamide
Show/Hide
|
C20H22ClFN4O3S
|
1
|
| 1 |
Ki = 9.9 nM
|
|
|
|
CP0461307
|
5-fluoro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C24H25F2N3O3S2
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0510210
|
N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0393439
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C22H23ClFN3O2S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0379150
|
3-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-benzoxazol-2-one
Show/Hide
|
C22H27N3O3
|
1
|
| 1 |
Ki = 10.35 nM
|
|
|
|
CP0418281
|
3-[6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl]-1,3-benzoxazol-2-one
Show/Hide
|
C24H31N3O3
|
1
|
| 1 |
Ki = 11.68 nM
|
|
|
|
CP0451856
|
2-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-3H-quinazolin-4-one
Show/Hide
|
C23H27ClN4O
|
1
|
| 1 |
Ki = 11.9 nM
|
|
|
|
CP0408136
|
3-chloro-N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]benzenesulfonamide
Show/Hide
|
C22H23Cl2N3O2S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0415977
|
3-amino-2-[4-(4-phenylpiperazin-1-yl)butyl]-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C24H27N5OS
|
1
|
| 1 |
Ki = 12.2 nM
|
|
|
|
CP0413621
|
3-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]quinazolin-4-one
Show/Hide
|
C23H27ClN4O
|
1
|
| 1 |
Ki = 12.9 nM
|
|
|
|
CP0443106
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
|
C23H25FN4O3S2
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0461314
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C22H24N4O2S3
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0422311
|
2-[4-(4-phenylpiperazin-1-yl)butyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C24H26N4OS
|
1
|
| 1 |
Ki = 13.6 nM
|
|
|
|
CP0489950
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]imidazo[1,2-a]pyridine-3-sulfonamide
Show/Hide
|
C23H26FN5O3S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0513529
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-3-fluorobenzenesulfonamide
Show/Hide
|
C22H23ClFN3O2S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0481824
|
3-[6-(4-phenylpiperazin-1-yl)hexyl]-1,3-benzoxazol-2-one
Show/Hide
|
C23H29N3O2
|
1
|
| 1 |
Ki = 14.1 nM
|
|
|
|
CP0481184
|
N-[4-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C23H25F4N3O4S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0407585
|
1-(2-methoxyphenyl)-4-[[3-(2-methoxyphenyl)phenyl]methyl]piperazine
Show/Hide
|
C25H28N2O2
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0436651
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H26ClN3O2S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0528055
|
6-fluoro-3-[3-[3-(naphthalen-2-ylsulfonylmethyl)pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
|
C25H25FN2O3S
|
1
|
| 1 |
Ki = 15.49 nM
|
|
|
|
CP0129287
|
N-[[2-(2-chlorophenyl)phenyl]methyl]-6-[4-(2-methoxyphenyl)piperazin-1-yl]hexanamide
Show/Hide
|
C30H36ClN3O2
|
1
|
| 1 |
Ki = 15.9 nM
|
|
|
|
CP0393442
|
3-chloro-N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]benzenesulfonamide
Show/Hide
|
C21H21Cl2N3O2S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0468502
|
6-chloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H25ClFN3O3S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0475024
|
N-[3-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]naphthalene-1-sulfonamide
Show/Hide
|
C26H26ClN3O2S
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0551500
|
3-[3-[3-[(3-chloro-4-fluorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-6-fluoro-1,2-benzoxazole
Show/Hide
|
C21H21ClF2N2O3S
|
1
|
| 1 |
Ki = 18.62 nM
|
|
|
|
CP0447121
|
N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C22H25F3N4O3S2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0422048
|
2-[5-(4-phenylpiperazin-1-yl)pentyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C25H28N4OS
|
1
|
| 1 |
Ki = 19.3 nM
|
|
|
|
CP0483771
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-3,4-dichlorobenzenesulfonamide
Show/Hide
|
C20H22Cl2N4O2S2
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0483452
|
3-[5-(4-phenylpiperazin-1-yl)pentyl]-1,3-benzothiazol-2-one
Show/Hide
|
C22H27N3OS
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0429433
|
2-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3H-quinazolin-4-one
Show/Hide
|
C22H25ClN4O
|
1
|
| 1 |
Ki = 21.2 nM
|
|
|
|
CP0488674
|
3-[3-[3-[(3-chlorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-6-fluoro-1,2-benzoxazole
Show/Hide
|
C21H22ClFN2O3S
|
1
|
| 1 |
Ki = 21.38 nM
|
|
|
|
CP0532876
|
3-[3-[3-[(3,4-dichlorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-6-fluoro-1,2-benzoxazole
Show/Hide
|
C21H21Cl2FN2O3S
|
1
|
| 1 |
Ki = 21.88 nM
|
|
|
|
CP0386376
|
N-[[2-(3-methoxyphenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
|
C30H37N3O3
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0439674
|
1-{4-[4-(1-Naphthyl)piperazin-1-yl]butyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
|
C26H29N3O
|
2
|
| 1 |
Ki = 22 nM
|
|
|
| 2 |
Ki = 47 nM
|
|
|
|
CP0506649
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
|
C18H22N4O2S3
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0391061
|
2-[3-(4-phenylpiperazin-1-yl)propylsulfanyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
|
C23H24N4OS2
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0408275
|
4-[5-[4-(2-ethoxyphenyl)piperazin-1-yl]pentoxy]-6-phenylpyrimidine
Show/Hide
|
C27H34N4O2
|
1
|
| 1 |
Ki = 23.5 nM
|
|
|
|
CP0494824
|
3-(4-benzylpiperazin-1-yl)-1-(4-pyrimidin-2-ylpiperazin-1-yl)propan-1-one
Show/Hide
|
C22H30N6O
|
1
|
| 1 |
Ki = 23.5 nM
|
|
|
|
CP0474914
|
N-[2-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
|
C23H26ClN3O2S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0559856
|
3-(4-benzylpiperazin-1-yl)-1-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one
Show/Hide
|
C25H34N4O2
|
1
|
| 1 |
Ki = 24.2 nM
|
|
|
|
CP0395871
|
N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
|
C23H25FN4O2S3
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0418278
|
N-[[2-(4-chlorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
|
C29H34ClN3O2
|
1
|
| 1 |
Ki = 25.9 nM
|
|
|
|
CP0398830
|
5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[2-(2-methylphenyl)phenyl]methyl]pentanamide
Show/Hide
|
C30H37N3O2
|
1
|
| 1 |
Ki = 26.1 nM
|
|
|
|
CP0460661
|
1,3-bis(4-phenylpiperazin-1-yl)propan-1-one
Show/Hide
|
C23H30N4O
|
1
|
| 1 |
Ki = 26.2 nM
|
|
|
|
CP0546332
|
6-fluoro-3-[3-[3-[(3-methylphenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
|
C22H25FN2O3S
|
1
|
| 1 |
Ki = 26.3 nM
|
|
|
|
CP0379147
|
3-[4-(4-phenylpiperazin-1-yl)butyl]-1,3-benzoxazol-2-one
Show/Hide
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C21H25N3O2
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1
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| 1 |
Ki = 26.33 nM
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CP0422046
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2-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-3H-thieno[3,2-d]pyrimidin-4-one
Show/Hide
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C20H23ClN4OS
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1
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| 1 |
Ki = 27.8 nM
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CP0468504
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
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C21H23F3N4O3S2
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1
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| 1 |
Ki = 29 nM
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CP0393455
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N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]naphthalene-1-sulfonamide
Show/Hide
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C25H24ClN3O2S
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1
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| 1 |
Ki = 29 nM
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CP0437879
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3-(4-benzylpiperazin-1-yl)-1-(4-pyridin-2-ylpiperazin-1-yl)propan-1-one
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C23H31N5O
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1
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| 1 |
Ki = 29.5 nM
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CP0073285
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6-[4-[4-(2-hydroxyphenyl)piperazin-1-yl]butyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C29H33N7O3
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1
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| 1 |
Ki = 30 nM
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CP0429431
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5,6-dimethyl-2-[5-(4-phenylpiperazin-1-yl)pentyl]-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H30N4OS
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1
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| 1 |
Ki = 30.1 nM
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CP0567022
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N-[[2-(2-methoxyphenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C30H37N3O3
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1
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| 1 |
Ki = 31.4 nM
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CP0424211
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1-(4-(4-phenyl-1-piperazinyl)butyl)indolin-2-one
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C23H29N3O2
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1
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| 1 |
Ki = 32 nM
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CP0468855
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N-[3-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
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C26H26FN3O2S
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1
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| 1 |
Ki = 32 nM
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CP0537571
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N-[[2-(2,6-dimethoxyphenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C31H39N3O4
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1
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| 1 |
Ki = 32.4 nM
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CP0437876
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3-[4-(3-chlorophenyl)piperazin-1-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
Show/Hide
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C23H29ClN4O
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1
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| 1 |
Ki = 32.7 nM
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CP0447107
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N-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-6-chloronaphthalene-2-sulfonamide
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C25H27ClN4O2S2
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1
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| 1 |
Ki = 33 nM
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CP0395877
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-3,4-dichlorobenzenesulfonamide
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C20H22Cl2N4O3S
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1
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| 1 |
Ki = 34 nM
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CP0473172
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6-chloro-N-[3-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H23ClFN3O3S2
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1
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| 1 |
Ki = 34 nM
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CP0398831
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N-[[2-(3-fluorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C29H34FN3O2
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1
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| 1 |
Ki = 34.7 nM
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CP0567023
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N-[[2-(4-fluorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C29H34FN3O2
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1
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| 1 |
Ki = 34.7 nM
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CP0408274
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3-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-2-methylquinazolin-4-one
Show/Hide
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C24H29ClN4O
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1
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| 1 |
Ki = 35.1 nM
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CP0413622
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3-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]quinazolin-4-one
Show/Hide
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C23H27ClN4O
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1
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| 1 |
Ki = 35.8 nM
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CP0379148
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3-[4-(4-phenylpiperazin-1-yl)butyl]-1,3-benzothiazol-2-one
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C21H25N3OS
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1
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| 1 |
Ki = 36.48 nM
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CP0555190
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N-[[2-(2-fluorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C29H34FN3O2
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1
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| 1 |
Ki = 36.5 nM
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CP0424260
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3-(4-benzylpiperazin-1-yl)-1-[4-(4-chlorophenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C24H31ClN4O
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1
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| 1 |
Ki = 36.6 nM
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CP0282007
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6-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C29H32ClN7O2
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1
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| 1 |
Ki = 37 nM
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CP0555548
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5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(2-phenylphenyl)methyl]pentanamide
Show/Hide
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C29H35N3O2
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1
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| 1 |
Ki = 37.9 nM
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CP0468505
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-6-chloronaphthalene-2-sulfonamide
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C24H25ClN4O2S2
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1
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| 1 |
Ki = 38 nM
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CP0549990
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N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H24FN3O3S2
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1
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| 1 |
Ki = 38.02 nM
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CP0422306
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2-[3-(4-benzylpiperidin-1-yl)propylsulfanyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C25H27N3OS2
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1
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| 1 |
Ki = 40.1 nM
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CP0447126
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
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C21H23N5O3S2
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1
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| 1 |
Ki = 41 nM
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CP0418284
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3-[4-(4-benzylpiperazin-1-yl)butyl]-1,3-benzothiazol-2-one
Show/Hide
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C22H27N3OS
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1
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| 1 |
Ki = 41.93 nM
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CP0148485
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6-[5-[4-(2-hydroxyphenyl)piperazin-1-yl]pentyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C30H35N7O3
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1
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| 1 |
Ki = 43 nM
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CP0552785
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N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]naphthalene-2-sulfonamide
Show/Hide
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C25H26FN3O3S
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1
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| 1 |
Ki = 43.65 nM
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CP0398832
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6-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(2-phenylphenyl)methyl]hexanamide
Show/Hide
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C30H37N3O2
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1
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| 1 |
Ki = 43.7 nM
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CP0562208
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N-[[2-(4-methoxyphenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C30H37N3O3
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1
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| 1 |
Ki = 43.7 nM
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CP0471745
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2-[4-[4-(5-chloro-2-methoxyphenyl)piperazin-1-yl]butyl]-3H-thieno[3,2-d]pyrimidin-4-one
Show/Hide
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C21H25ClN4O2S
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1
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| 1 |
Ki = 43.8 nM
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CP0445786
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4-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentoxy]-6-phenylpyrimidine
Show/Hide
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C25H29ClN4O
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1
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| 1 |
Ki = 44.8 nM
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CP0504359
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3-[5-[4-(2-ethoxyphenyl)piperazin-1-yl]pentyl]-6-phenylpyrimidin-4-one
Show/Hide
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C27H34N4O2
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1
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| 1 |
Ki = 45.1 nM
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CP0559132
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3-[7-(4-phenylpiperazin-1-yl)heptyl]-1,3-benzoxazol-2-one
Show/Hide
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C24H31N3O2
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1
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| 1 |
Ki = 45.57 nM
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CP0418277
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N-[[2-(2-chlorophenyl)phenyl]methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]butanamide
Show/Hide
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C28H32ClN3O2
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1
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| 1 |
Ki = 46.6 nM
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CP0528049
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6-fluoro-3-[3-[3-[[4-(trifluoromethyl)phenyl]sulfonylmethyl]pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
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C22H22F4N2O3S
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1
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| 1 |
Ki = 46.77 nM
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CP0481825
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3-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1,3-benzothiazol-2-one
Show/Hide
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C21H24ClN3OS
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1
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| 1 |
Ki = 46.83 nM
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CP0553491
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5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[2-(3-methylphenyl)phenyl]methyl]pentanamide
Show/Hide
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C30H37N3O2
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1
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| 1 |
Ki = 47.6 nM
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CP0573889
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3-[3-[3-[(3,4-difluorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-6-fluoro-1,2-benzoxazole
Show/Hide
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C21H21F3N2O3S
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1
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| 1 |
Ki = 47.86 nM
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CP0534014
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6-fluoro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H23F2N3O3S2
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1
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| 1 |
Ki = 48.98 nM
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CP0443772
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3-(4-benzylpiperazin-1-yl)-1-[4-(2-chlorophenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C24H31ClN4O
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1
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| 1 |
Ki = 50.2 nM
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CP0393443
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4-chloro-N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]benzenesulfonamide
Show/Hide
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C21H21Cl2N3O2S
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1
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| 1 |
Ki = 51 nM
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CP0494823
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3-(4-benzylpiperazin-1-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
Show/Hide
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C24H32N4O
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1
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| 1 |
Ki = 52 nM
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CP0555765
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2-methyl-3-[5-(4-phenylpiperazin-1-yl)pentyl]quinazolin-4-one
Show/Hide
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C24H30N4O
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1
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| 1 |
Ki = 53.7 nM
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CP0482708
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N-[3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]propyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
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C22H23ClN4O2S3
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1
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| 1 |
Ki = 54 nM
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CP0437877
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3-(4-benzylpiperazin-1-yl)-1-[4-(3-chlorophenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C24H31ClN4O
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1
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| 1 |
Ki = 54.7 nM
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CP0468649
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2-[4-(4-benzylpiperazin-1-yl)butyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C25H28N4OS
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1
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| 1 |
Ki = 56.2 nM
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CP0395880
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-1,3-benzothiazole-4-sulfonamide
Show/Hide
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C22H25N5O3S2
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1
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| 1 |
Ki = 57 nM
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CP0398219
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3-[5-(4-phenylpiperazin-1-yl)pentyl]-1,3-benzoxazol-2-one
Show/Hide
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C22H27N3O2
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1
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| 1 |
Ki = 57.39 nM
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CP0188400
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9-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
Show/Hide
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C24H28ClN7O3
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1
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| 1 |
Ki = 61 nM
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CP0413408
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-hydroxybenzenesulfonamide
Show/Hide
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C23H26ClN3O3S
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1
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| 1 |
Ki = 61 nM
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CP0383839
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1-[5-(4-Phenylpiperazin-1-yl)pentyl]-1,3-dihydro-2H-indol-2-one
Show/Hide
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C23H29N3O
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1
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| 1 |
Ki = 63 nM
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CP0439675
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1-{5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C24H31N3O2
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1
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| 1 |
Ki = 63 nM
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CP0488673
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6-fluoro-3-[3-[3-[(4-fluorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
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C21H22F2N2O3S
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1
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| 1 |
Ki = 63.1 nM
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CP0567092
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4-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(2-phenylphenyl)methyl]butanamide
Show/Hide
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C28H33N3O2
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1
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| 1 |
Ki = 64.5 nM
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CP0472939
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3-chloro-N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]benzenesulfonamide
Show/Hide
|
C23H25Cl2N3O2S
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1
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| 1 |
Ki = 65 nM
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CP0455695
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2-[4-(4-benzylpiperidin-1-yl)butyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C26H29N3OS
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1
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| 1 |
Ki = 65.1 nM
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CP0562207
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5-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[[2-(4-methylphenyl)phenyl]methyl]pentanamide
Show/Hide
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C30H37N3O2
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1
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| 1 |
Ki = 66.1 nM
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CP0497344
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]thiophene-2-sulfonamide
Show/Hide
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C19H24N4O3S2
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1
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| 1 |
Ki = 67 nM
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CP0532871
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6-fluoro-3-[3-[3-[[3-(trifluoromethyl)phenyl]sulfonylmethyl]pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
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C22H22F4N2O3S
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1
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| 1 |
Ki = 67.61 nM
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CP0506462
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1-{5-[4-(1H)-benzimidazol-4-yl)piperazin-1-yl]pentyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C24H29N5O
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1
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| 1 |
Ki = 68 nM
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CP0542518
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2-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H29ClN4OS
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1
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| 1 |
Ki = 68.4 nM
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CP0493808
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1-{(2E)-4-[4-(1-Naphthyl)piperazin-1-yl]but-2-enyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C26H27N3O
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1
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| 1 |
Ki = 69 nM
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CP0497898
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1-{5-[4-(1-Naphthyl)piperazin-1-yl]pentyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C27H31N3O
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1
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| 1 |
Ki = 69 nM
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CP0408137
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N-[2-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
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C25H24ClN3O2S
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1
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| 1 |
Ki = 69 nM
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CP0403349
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
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C24H28ClN3O2S
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1
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| 1 |
Ki = 70 nM
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CP0424212
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1-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-indolin-2-one
Show/Hide
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C22H27N3O
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1
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| 1 |
Ki = 74 nM
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CP0455660
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2-[4-(4-benzylpiperidin-1-yl)butyl]-3H-thieno[3,2-d]pyrimidin-4-one
Show/Hide
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C22H27N3OS
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1
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| 1 |
Ki = 75.8 nM
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CP0463656
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C23H25ClFN3O2S
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1
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| 1 |
Ki = 80 nM
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CP0480970
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N-[2-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
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C25H24FN3O2S
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1
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| 1 |
Ki = 80 nM
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CP0420755
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3-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
Show/Hide
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C25H34N4O2
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1
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| 1 |
Ki = 80.3 nM
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CP0413623
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3-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H29ClN4OS
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1
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| 1 |
Ki = 88.5 nM
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CP0418283
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1-(5-(4-phenylpiperazin-1-yl)pentyl)benzo[cd]indol-2(1H)-one
Show/Hide
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C26H29N3O
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1
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| 1 |
Ki = 89 nM
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CP0408140
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4-chloro-N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]benzenesulfonamide
Show/Hide
|
C23H25Cl2N3O2S
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1
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| 1 |
Ki = 90 nM
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CP0436652
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-fluorobenzenesulfonamide
Show/Hide
|
C23H25ClFN3O2S
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1
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| 1 |
Ki = 91 nM
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CP0447212
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]thiophene-2-sulfonamide
Show/Hide
|
C18H22N4O3S2
|
1
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| 1 |
Ki = 94 nM
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CP0531207
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3-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentyl]-6-phenylpyrimidin-4-one
Show/Hide
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C25H29ClN4O
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1
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| 1 |
Ki = 94.7 nM
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CP0462037
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N-[3-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
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C23H26FN3O2S
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1
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| 1 |
Ki = 95 nM
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CP0528228
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N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-1-benzothiophene-3-sulfonamide
Show/Hide
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C23H24FN3O3S2
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1
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| 1 |
Ki = 95.5 nM
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CP0433461
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2-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-3H-quinazolin-4-one
Show/Hide
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C23H27ClN4O
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1
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| 1 |
Ki = 101 nM
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CP0552783
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6-fluoro-3-[3-[3-[(3-fluorophenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-1,2-benzoxazole
Show/Hide
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C21H22F2N2O3S
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1
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| 1 |
Ki = 102.33 nM
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CP0552784
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3-chloro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C21H23ClFN3O3S
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1
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| 1 |
Ki = 102.33 nM
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CP0522888
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1-[3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl]-1,3-dihydro-2H-indol-2-one
Show/Hide
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C20H22N2O
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1
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| 1 |
Ki = 105 nM
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CP0490087
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6-phenyl-2-[4-(4-phenylpiperazin-1-yl)butyl]-3H-thieno[3,2-d]pyrimidin-4-one
Show/Hide
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C26H28N4OS
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1
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| 1 |
Ki = 106 nM
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CP0474916
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
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C27H28ClN3O2S
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1
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| 1 |
Ki = 110 nM
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CP0389596
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6-[5-[4-(3,4-dichlorophenyl)piperazin-1-yl]pentyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C25H31Cl2N7O2
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1
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| 1 |
Ki = 111 nM
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CP0417895
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3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-6-fluoro-1,3-dihydroindol-2-one
Show/Hide
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C22H25ClFN3O
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1
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| 1 |
Ki = 118 nM
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CP0549301
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1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[4-(2-ethoxyphenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C25H33ClN4O2
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1
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| 1 |
Ki = 119 nM
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CP0548414
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
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C24H26N4O3S
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1
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| 1 |
Ki = 120 nM
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CP0393440
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N-[4-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
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C24H28FN3O2S
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1
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| 1 |
Ki = 120 nM
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CP0123095
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6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4-dimethyl-7-phenylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C30H34ClN7O2
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1
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| 1 |
Ki = 122 nM
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CP0073286
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6-[5-[4-(2-hydroxyphenyl)piperazin-1-yl]pentyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C25H33N7O3
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1
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| 1 |
Ki = 124 nM
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CP0488671
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6-chloro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H23ClFN3O3S2
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1
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| 1 |
Ki = 125.89 nM
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CP0528053
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3-chloro-4-fluoro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]benzenesulfonamide
Show/Hide
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C21H22ClF2N3O3S
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1
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| 1 |
Ki = 125.89 nM
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CP0422309
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2-[4-(4-benzylpiperazin-1-yl)butyl]-3H-thieno[3,2-d]pyrimidin-4-one
Show/Hide
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C21H26N4OS
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1
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| 1 |
Ki = 133 nM
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CP0393441
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N-[4-[4-(5-chloro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]naphthalene-1-sulfonamide
Show/Hide
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C27H28ClN3O2S
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1
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| 1 |
Ki = 140 nM
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CP0429434
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5,6-dimethyl-3-[5-(4-phenylpiperazin-1-yl)pentyl]thieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H30N4OS
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1
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| 1 |
Ki = 143 nM
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CP0382566
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4-phenyl-6-[5-(4-phenylpiperazin-1-yl)pentoxy]pyrimidine
Show/Hide
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C25H30N4O
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1
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| 1 |
Ki = 143 nM
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CP0530822
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2-[4-(4-phenylpiperazin-1-yl)butyl]-3H-quinazolin-4-one
Show/Hide
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C22H26N4O
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1
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| 1 |
Ki = 145 nM
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CP0433460
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2-[5-(4-benzylpiperazin-1-yl)pentyl]-6-methyl-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H30N4OS
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1
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| 1 |
Ki = 147 nM
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CP0486987
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C22H24N4O3S2
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1
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| 1 |
Ki = 150 nM
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CP0462036
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N-[3-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]naphthalene-2-sulfonamide
Show/Hide
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C27H28ClN3O2S
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1
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| 1 |
Ki = 150 nM
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CP0494035
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N-[3-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]propyl]-3-methylbenzenesulfonamide
Show/Hide
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C24H28ClN3O2S
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1
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| 1 |
Ki = 150 nM
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CP0371912
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2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinone
Show/Hide
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C23H29N3O2
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1
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| 1 |
Ki = 158 nM
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CP0534012
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6-chloro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]naphthalene-2-sulfonamide
Show/Hide
|
C25H25ClFN3O3S
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1
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| 1 |
Ki = 158.49 nM
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CP0459793
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1-[4-(4-Phenylpiperidin-1-yl)butyl]-1,3-dihydro-2H-indol-2-one
Show/Hide
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C23H28N2O
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1
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| 1 |
Ki = 160 nM
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CP0477293
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2-[5-[4-(3-chlorophenyl)piperazin-1-yl]pentanoylamino]benzamide
Show/Hide
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C22H27ClN4O2
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1
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| 1 |
Ki = 168 nM
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CP0494808
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N-benzyl-3-(benzylamino)propanamide
Show/Hide
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C17H20N2O
|
1
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| 1 |
Ki = 176 nM
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CP0488670
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N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-1-benzofuran-2-sulfonamide
Show/Hide
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C23H24FN3O4S
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1
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| 1 |
Ki = 177.83 nM
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CP0443099
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H26N4O3S2
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1
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| 1 |
Ki = 180 nM
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CP0472938
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N-[2-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]-3-methylbenzenesulfonamide
Show/Hide
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C22H24FN3O2S
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1
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| 1 |
Ki = 180 nM
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CP0376944
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4-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentoxy]-2-methylquinazoline
Show/Hide
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C24H29ClN4O
|
1
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| 1 |
Ki = 181 nM
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CP0504744
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2-[5-(4-benzylpiperidin-1-yl)pentyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
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C25H33N3OS
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1
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| 1 |
Ki = 185 nM
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CP0459570
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3-[4-(2-methoxyphenyl)piperazin-1-yl]-N-[(2-phenylphenyl)methyl]propanamide
Show/Hide
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C27H31N3O2
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1
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| 1 |
Ki = 186.5 nM
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CP0493810
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1-[4-(3-Phenylpiperidin-1-yl)butyl]-1,3-dihydro-2H-indol-2-one
Show/Hide
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C23H28N2O
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1
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| 1 |
Ki = 193 nM
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CP0477761
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1,5-bis(4-phenylpiperazin-1-yl)pentan-1-one
Show/Hide
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C25H34N4O
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1
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| 1 |
Ki = 197 nM
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CP0395878
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-5-fluoro-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C23H25FN4O3S2
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1
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| 1 |
Ki = 200 nM
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CP0493335
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2-[5-(4-Phenylpiperazin-1-yl)pentyl]isoindolin-1-one
Show/Hide
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C23H29N3O
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1
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| 1 |
Ki = 203 nM
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CP0551501
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3-[3-[3-[(3,4-dimethylphenyl)sulfonylmethyl]pyrrolidin-1-yl]propyl]-6-fluoro-1,2-benzoxazole
Show/Hide
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C23H27FN2O3S
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1
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| 1 |
Ki = 204.17 nM
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CP0557263
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3-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-one
Show/Hide
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C23H29ClN4OS
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1
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| 1 |
Ki = 213 nM
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CP0537737
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2-[5-(4-phenylpiperazin-1-yl)pentyl]-3H-quinazolin-4-one
Show/Hide
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C23H28N4O
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1
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| 1 |
Ki = 228 nM
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CP0123092
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6-[5-[4-(2-hydroxyphenyl)piperazin-1-yl]pentyl]-2,4-dimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C24H31N7O3
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1
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| 1 |
Ki = 230 nM
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CP0408135
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N-[4-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
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C27H28FN3O2S
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1
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| 1 |
Ki = 240 nM
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CP0506463
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1-{(2Z)-4-[4-(1-Naphthyl)piperazin-1-yl]but-2-enyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C26H27N3O
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1
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| 1 |
Ki = 250 nM
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CP0461296
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N-[4-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]butyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C22H25F3N4O4S
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1
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| 1 |
Ki = 270 nM
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CP0566533
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2-methyl-4-[5-(4-phenylpiperazin-1-yl)pentoxy]quinazoline
Show/Hide
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C24H30N4O
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1
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| 1 |
Ki = 276 nM
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CP0481834
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3-[5-(4-phenylpiperazin-1-yl)pentyl]quinazolin-4-one
Show/Hide
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C23H28N4O
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1
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| 1 |
Ki = 307 nM
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CP0445783
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3-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2-methylquinazolin-4-one
Show/Hide
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C24H29ClN4O
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1
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| 1 |
Ki = 327 nM
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CP0383841
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1-[2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl]-1,3-dihydro-2H-indol-2-one
Show/Hide
|
C19H20N2O
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1
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| 1 |
Ki = 350 nM
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CP0429430
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5,6-dimethyl-2-[4-(4-phenylpiperazin-1-yl)butyl]-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
|
C22H28N4OS
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1
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| 1 |
Ki = 357 nM
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CP0282006
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6-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C24H30ClN7O2
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1
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| 1 |
Ki = 361 nM
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CP0552163
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2-[5-(4-benzylpiperidin-1-yl)pentyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C27H31N3OS
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1
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| 1 |
Ki = 366 nM
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CP0497340
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-4-(trifluoromethoxy)benzenesulfonamide
Show/Hide
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C21H23F3N4O4S
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1
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| 1 |
Ki = 380 nM
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CP0447151
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N-[4-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]-3-methylbenzenesulfonamide
Show/Hide
|
C25H30ClN3O2S
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1
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| 1 |
Ki = 380 nM
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CP0121966
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6-[4-[4-(2,3-dimethylphenyl)piperazin-1-yl]butyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C26H35N7O2
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1
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| 1 |
Ki = 381 nM
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CP0037227
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7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-ol
Show/Hide
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C16H25NO
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1
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| 1 |
Ki = 388 nM
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CP0422307
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2-[5-(4-benzylpiperazin-1-yl)pentyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C26H30N4OS
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1
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| 1 |
Ki = 401 nM
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CP0553906
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N-[[2-(3-chlorophenyl)phenyl]methyl]-5-[4-(2-methoxyphenyl)piperazin-1-yl]pentanamide
Show/Hide
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C29H34ClN3O2
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1
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| 1 |
Ki = 405.3 nM
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CP0528047
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5-chloro-N-[(3S,5S)-1-[3-(6-fluoro-1,2-benzoxazol-3-yl)propyl]-5-methylpyrrolidin-3-yl]-3-methyl-1-benzothiophene-2-sulfonamide
Show/Hide
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C24H25ClFN3O3S2
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1
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| 1 |
Ki = 416.87 nM
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CP0494807
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3-[4-(4-chlorophenyl)piperazin-1-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
Show/Hide
|
C23H29ClN4O
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1
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| 1 |
Ki = 462 nM
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CP0118231
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9-[5-[4-(2-hydroxyphenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
Show/Hide
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C25H31N7O4
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1
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| 1 |
Ki = 473 nM
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CP0120218
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3-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]quinazolin-4-one
Show/Hide
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C22H25ClN4O
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1
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| 1 |
Ki = 502 nM
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CP0118234
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6-[4-[4-(2-hydroxyphenyl)piperazin-1-yl]butyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C24H31N7O3
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1
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| 1 |
Ki = 510 nM
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CP0408138
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N-[2-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]naphthalene-2-sulfonamide
Show/Hide
|
C26H26ClN3O2S
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1
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| 1 |
Ki = 520 nM
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CP0447152
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N-[4-[4-(5-chloro-2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-yl]butyl]naphthalene-2-sulfonamide
Show/Hide
|
C28H30ClN3O2S
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1
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| 1 |
Ki = 610 nM
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CP0376943
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6-phenyl-3-[5-(4-phenylpiperazin-1-yl)pentyl]pyrimidin-4-one
Show/Hide
|
C25H30N4O
|
1
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| 1 |
Ki = 613 nM
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CP0519720
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6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4,7-trimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C25H32ClN7O2
|
1
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| 1 |
Ki = 691 nM
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CP0486993
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-6-chloro-1-benzothiophene-2-sulfonamide
Show/Hide
|
C22H23ClN4O3S2
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1
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| 1 |
Ki = 900 nM
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CP0567737
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4-[5-(4-benzylpiperazin-1-yl)pentoxy]-6-phenylpyrimidine
Show/Hide
|
C26H32N4O
|
1
|
| 1 |
Ki = 990 nM
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CP0477292
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3-[5-(4-benzylpiperazin-1-yl)pentyl]quinazolin-4-one
Show/Hide
|
C24H30N4O
|
1
|
| 1 |
Ki = 1082 nM
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CP0488676
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2-[4-[4-(4-chlorophenyl)piperazin-1-yl]butyl]-3H-quinazolin-4-one
Show/Hide
|
C22H25ClN4O
|
1
|
| 1 |
Ki = 1135 nM
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CP0445632
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3-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-6-phenylpyrimidin-4-one
Show/Hide
|
C25H29ClN4O
|
1
|
| 1 |
Ki = 1310 nM
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CP0567738
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3-[5-(4-benzylpiperazin-1-yl)pentyl]-6-phenylpyrimidin-4-one
Show/Hide
|
C26H32N4O
|
1
|
| 1 |
Ki = 1328 nM
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CP0121965
|
6-[4-[4-(2-hydroxyphenyl)piperazin-1-yl]butyl]-2,4-dimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
|
C23H29N7O3
|
1
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| 1 |
Ki = 1364 nM
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CP0408273
|
4-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentoxy]-6-phenylpyrimidine
Show/Hide
|
C25H29ClN4O
|
1
|
| 1 |
Ki = 1377 nM
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CP0429432
|
2-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
Show/Hide
|
C23H29ClN4OS
|
1
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| 1 |
Ki = 1464 nM
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CP0462144
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3-[5-(4-benzylpiperazin-1-yl)pentyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-one
Show/Hide
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C24H32N4OS
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1
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| 1 |
Ki = 1650 nM
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CP0460660
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1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[4-(4-chlorophenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C23H28Cl2N4O
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1
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| 1 |
Ki = 2366 nM
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CP0497341
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N-[3-[4-(1,2-benzoxazol-3-yl)piperazin-1-yl]propyl]-6-chloronaphthalene-2-sulfonamide
Show/Hide
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C24H25ClN4O3S
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1
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| 1 |
Ki = 2500 nM
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CP0460659
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1,3-bis[4-(3-chlorophenyl)piperazin-1-yl]propan-1-one
Show/Hide
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C23H28Cl2N4O
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1
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| 1 |
Ki = 2761 nM
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CP0441366
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6-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-2,4-dimethylpurino[7,8-a]imidazole-1,3-dione
Show/Hide
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C24H30ClN7O2
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1
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| 1 |
Ki = 3636 nM
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CP0380574
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1-(2,3-dimethylphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C25H28N2
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1
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| 1 |
Ki > 10000 nM
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CP0380575
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1-(4-fluorophenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C23H23FN2
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1
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| 1 |
Ki > 10000 nM
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CP0393536
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1-(3,5-dimethylphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C25H28N2
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1
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| 1 |
Ki > 10000 nM
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CP0393537
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1-(2,5-dimethylphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C25H28N2
|
1
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| 1 |
Ki > 10000 nM
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CP0393538
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1-(2,4-dimethylphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C25H28N2
|
1
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| 1 |
Ki > 10000 nM
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CP0396272
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1-(4-chlorophenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C23H23ClN2
|
1
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| 1 |
Ki > 10000 nM
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CP0404874
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1-(3-fluorophenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C23H23FN2
|
1
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| 1 |
Ki > 10000 nM
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CP0408483
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1-(2-chlorophenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C23H23ClN2
|
1
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| 1 |
Ki > 10000 nM
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CP0449865
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1-(4-methoxyphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C24H26N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0481937
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1-(2-fluorophenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C23H23FN2
|
1
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| 1 |
Ki > 10000 nM
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CP0555819
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1-(3-methoxyphenyl)-4-[(2-phenylphenyl)methyl]piperazine
Show/Hide
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C24H26N2O
|
1
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| 1 |
Ki > 10000 nM
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CP0422266
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2-(2-aminoethylsulfanyl)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C12H11N3OS2
|
1
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| 1 |
Ki > 10000 nM
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CP0455431
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2-(2-pyrrolidin-1-ylethylsulfanyl)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C16H17N3OS2
|
1
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| 1 |
Ki > 10000 nM
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CP0471746
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2-[2-(dimethylamino)ethylsulfanyl]-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C14H15N3OS2
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1
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| 1 |
Ki > 10000 nM
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CP0552164
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2-(2-piperidin-1-ylethylsulfanyl)-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
Show/Hide
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C17H19N3OS2
|
1
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| 1 |
Ki > 10000 nM
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CP0371906
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2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1-isoindolinone
Show/Hide
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C22H27N3O
|
1
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| 1 |
Ki > 1000 nM
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CP0383840
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1-(4-{[4-(1-Naphthyl)piperazin-1-yl]methyl}benzyl)-1,3-dihydro-2H-indol-2-one
Show/Hide
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C30H29N3O
|
1
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| 1 |
Ki > 1000 nM
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CP0506464
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1-(3-{[4-(1-Naphthyl)piperazin-1-yl]methyl}benzyl)-1,3-dihydro-2H-indol-2-one
Show/Hide
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C30H29N3O
|
1
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| 1 |
Ki > 1000 nM
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CP0526645
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1-{4-[4-(1-Naphthyl)piperazin-1-yl]but-2-ynyl}-1,3-dihydro-2H-indol-2-one
Show/Hide
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C26H25N3O
|
1
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| 1 |
Ki > 1000 nM
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CP0113424
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9-[5-[4-(4-chlorophenyl)piperazin-1-yl]pentyl]-1,3-dimethylpurino[7,8-a]pyrimidine-2,4,8-trione
Show/Hide
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C25H30ClN7O3
|
1
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| 1 |
Ki > 1000 nM
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