Compound ID |
Compound Name |
Compound Formula |
CP0261899
|
2-butoxy-N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]quinoline-4-carboxamide
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|
C25H23F3N4O2
|
1
|
1 |
EC50 = 700 nM
|
|
|
CP0489389
|
(4-benzhydrylpiperazin-1-yl)-(1,5-dimethylpyrazol-3-yl)methanone
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|
C23H26N4O
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0573764
|
N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-4-(4-phenylphenyl)butanamide
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|
C27H24F3N3O
|
1
|
1 |
EC50 = 1200 nM
|
|
|
CP0578023
|
4-amino-5-chloro-2-methoxy-N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide
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|
C19H16ClF3N4O2
|
1
|
1 |
EC50 = 3000 nM
|
|
|
CP0000847
|
(2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-methyl-3,6,17-triazatetracyclo[8.7.0.0^{3,8}.0^{11,16}]heptadeca-1(10),11(16),12,14-tetraene-4,7-dione
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|
C22H19N3O4
|
1
|
1 |
EC50 = 5000 nM
|
|
|
CP0576788
|
4-(4-hydroxyphenyl)-N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]piperazine-1-carboxamide
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|
C22H22F3N5O2
|
1
|
1 |
EC50 = 5000 nM
|
|
|
CP0489388
|
N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]acetamide
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|
C13H12F3N3O
|
1
|
1 |
EC50 = 11000 nM
|
|
|
CP0280111
|
1-amino-3-naphthalen-1-yloxypropan-2-ol
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|
C13H15NO2
|
2
|
1 |
EC50 = 19400 nM
|
|
|
2 |
EC50 = 43000 nM
|
|
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
1 |
EC50 = 32000 nM
|
|
|
2 |
EC50 = 37000 nM
|
|
|
CP0072327
|
(2R)-1-(1-naphthalenyloxy)-3-(propan-2-ylamino)-2-propanol;hydrochloride
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|
C16H21NO2
|
1
|
1 |
EC50 = 40000 nM
|
|
|
CP0011846
|
1-(2-(2-hydroxy-3-(propylamino)propoxy)phenyl)-3-phenylpropan-1-one
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|
C21H27NO3
|
1
|
1 |
EC50 = 47000 nM
|
|
|
CP0571911
|
3-naphthalen-1-yloxy-N-propan-2-ylpropan-1-amine
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|
C16H21NO
|
1
|
1 |
EC50 = 50000 nM
|
|
|
CP0559367
|
2-methoxy-3-naphthalen-1-yloxy-N-propan-2-ylpropan-1-amine
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|
C17H23NO2
|
1
|
1 |
EC50 = 52000 nM
|
|
|
CP0951183
|
2,3,4,9-tetrahydro-1H-carbazol-3-amine
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|
C12H14N2
|
2
|
1 |
EC50 = 67000 nM
|
|
|
2 |
EC50 > 100000 nM
|
|
|
CP0072120
|
(-)-(S)-Propranolol
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|
C16H21NO2
|
1
|
1 |
EC50 = 72000 nM
|
|
|
CP0065986
|
2,3,4,9-Tetrahydro-1H-beta-carboline
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|
C11H12N2
|
2
|
1 |
EC50 = 74000 nM
|
|
|
2 |
EC50 > 100000 nM
|
|
|
CP0567410
|
1-naphthalen-1-yloxy-3-propan-2-yloxypropan-2-ol
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|
C16H20O3
|
1
|
1 |
EC50 = 83000 nM
|
|
|
CP0577376
|
1-[methyl(propan-2-yl)amino]-3-naphthalen-1-yloxypropan-2-ol
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|
C17H23NO2
|
1
|
1 |
EC50 > 100000 nM
|
|
|