Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT04908 , Transient receptor potential cation channel subfamily M member 2
Gene Name TRPM2
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID O94759
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT04908
 
Compound ID Compound Name Compound Formula
CP0553199
ethyl 2-[3-[4-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydro-4H-cyclohepta[c]pyrazol-1-yl]acetate
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C19H21F3N2O2
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0008872
Scalaradial
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C27H40O4
 1
1
IC50 = 210 nM
   TI
   LI
   LO
   TS
CP0548392
2-[[(E)-3-[4-(3-nitrophenyl)phenyl]prop-2-enoyl]amino]benzoic acid
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C22H16N2O5
 1
1
IC50 = 398 nM
   TI
   LI
   LO
   TS
CP0418925
5-bromo-2-[[(E)-3-(4-phenylphenyl)prop-2-enoyl]amino]benzoic acid
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C22H16BrNO3
 1
1
IC50 = 410 nM
   TI
   LI
   LO
   TS
CP0547790
4-methyl-2-[[(E)-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid
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C22H25NO3
 1
1
IC50 = 467 nM
   TI
   LI
   LO
   TS
CP0418957
2-[[(E)-3-[4-[3-(trifluoromethyl)phenyl]phenyl]prop-2-enoyl]amino]benzoic acid
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C23H16F3NO3
 1
1
IC50 = 788 nM
   TI
   LI
   LO
   TS
CP0485134
2-[[(E)-3-[4-(3-fluorophenyl)phenyl]prop-2-enoyl]amino]benzoic acid
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C22H16FNO3
 1
1
IC50 = 830 nM
   TI
   LI
   LO
   TS
CP0418958
5-methyl-2-[[(E)-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid
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C22H25NO3
 1
1
IC50 = 987 nM
   TI
   LI
   LO
   TS
CP0083490
2-(Diphenylboryloxy)Ethanamine
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C14H16BNO
 1
1
IC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0409040
2-[[(E)-3-(4-pentylphenyl)prop-2-enoyl]amino]benzoic acid
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C21H23NO3
 1
1
IC50 = 1700 nM
   TI
   LI
   LO
   TS
CP0293205
2-((E)-3-Biphenyl-4-yl-acryloylamino)-benzoic acid
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C22H17NO3
 1
1
IC50 = 2560 nM
   TI
   LI
   LO
   TS
CP0030899
1-[(2-chlorophenyl)-diphenylmethyl]imidazole
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C22H17ClN2
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0057530
ECONAZOLE
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C18H15Cl3N2O
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0865093
6-Bromo-8-methyl-2-(3-(naphthalen-1-yl)-1H-pyrazol-4-yl)-2,3-dihydroquinazolin-4(1H)-one
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C22H17BrN4O
 1
1
IC50 = 3700 nM
   TI
   LI
   LO
   TS
CP0036697
2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid
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C14H10F3NO2
 1
1
IC50 = 70000 nM
   TI
   LI
   LO
   TS
CP0280422
2-(3-methylanilino)benzoic acid
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C14H13NO2
 1
1
IC50 = 76000 nM
   TI
   LI
   LO
   TS