| Compound ID |
Compound Name |
Compound Formula |
|
CP0039874
|
3-[(Benzyl-methyl-amino)-methyl]-7-(2,6-difluoro-benzyl)-2-(4-isobutyrylamino-phenyl)-4-oxo-4,7-dihydro-thieno[2,3-b]pyridine-5-carboxylic acid isopropyl ester; hydrochloride
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|
C37H37F2N3O4S
|
2
|
| 1 |
IC50 = 5.012 nM
|
|
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| 2 |
Ki = 0.1 nM
|
|
|
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CP0342019
|
5-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)quinoxaline
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|
C30H32N6
|
2
|
| 1 |
IC50 = 630.96 nM
|
|
|
| 2 |
Ki = 12.2 nM
|
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|
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CP0903004
|
2-(4-tert-Butylphenyl)-4-(4-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)piperazin-1-yl)-1H-benzo[d]imidazole
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|
C26H32FN7
|
2
|
| 1 |
IC50 = 794.33 nM
|
|
|
| 2 |
Ki = 13.8 nM
|
|
|
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CP0165712
|
5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)methyl)-N-(2,4,6-trimethoxyphenyl)furan-2-carboxamide
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|
C30H37NO5
|
2
|
| 1 |
IC50 = 1000 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0865066
|
1-((2R,4R,5S)-4-(4-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)-5-(hydroxymethyl)tetrahydrofuran-2-yl)-5-methylpyrimidine-2,4(1H,3H)-dione
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|
C34H41N9O4
|
2
|
| 1 |
IC50 = 1995.26 nM
|
|
|
| 2 |
Ki = 38 nM
|
|
|
|
CP0891070
|
4-(4-((1-(1H-benzo[d]imidazol-2-yl)-1H-1,2,3-triazol-4-yl)methyl)piperazin-1-yl)-2-(4-tertbutylphenyl)-1H-benzo[d]imidazole
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|
C31H33N9
|
2
|
| 1 |
IC50 = 5011.87 nM
|
|
|
| 2 |
Ki = 104 nM
|
|
|
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CP0864714
|
(2R,3S,4R,5R,6R)-5-Acetamido-2-(acetoxymethyl)-6-(4-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)tetrahydro-2H-pyran-3,4-diyl diacetate
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|
C38H48N8O8
|
2
|
| 1 |
IC50 = 7943.28 nM
|
|
|
| 2 |
Ki = 157 nM
|
|
|
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CP0862329
|
N-((2R,3S,4S,5R,6S)-2-(4-((4-(2-(4-tertbutylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)-4,5-dihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-3-yl)acetamide
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|
C32H42N8O5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
|
CP0864713
|
(2R,3R,4S,5S,6R)-2-(4-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C30H39N7O5
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
Ki > 1000 nM
|
|
|
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CP0864716
|
(S)-2-(tert-Butoxycarbonylamino)-3-(4-((4-(2-(4-tertbutylphenyl)-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)-1H-1,2,3-triazol-1-yl)propanoic acid
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|
C32H42N8O4
|
2
|
| 1 |
IC50 = 10000 nM
|
|
|
| 2 |
Ki = 186 nM
|
|
|
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CP0956942
|
2-(4-(tert-Butylphenyl)-4-(4-(2-fluoroethyl)piperazin-1-yl)-1H-benzo[d]imidazole
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|
C23H29FN4
|
2
|
| 1 |
IC50 = 12589.25 nM
|
|
|
| 2 |
Ki = 254 nM
|
|
|
|
CP0869631
|
2-(4-tert-Butylphenyl)-4-(4-((1-(4-fluorophenyl)-1H-1,2,3-triazol-4-yl)methyl)piperazin-1-yl)-1H-benzo[d]imidazole
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|
C30H32FN7
|
2
|
| 1 |
IC50 = 19952.62 nM
|
|
|
| 2 |
Ki = 410 nM
|
|
|
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CP0913820
|
2-(4-(tert-Butyl)phenyl)-4-(4-(prop-2-yn-1-yl)piperazin-1-yl)-1H-benzo[d]imidazole
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|
C24H28N4
|
2
|
| 1 |
IC50 = 19952.62 nM
|
|
|
| 2 |
Ki = 395 nM
|
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