Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01177 , Serine/threonine-protein kinase ULK2
Gene Name ULK2
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID Q8IYT8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01177
 
Compound ID Compound Name Compound Formula
CP0515043
N2-(1H-benzo[d]imidazol-6-yl)-N4-cyclopropyl-5-(trifluoromethyl)pyrimidine-2,4-diamine
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C15H13F3N6
 1
1
IC50 = 703 nM
   TI
   LI
   LO
   TS
CP0489042
US10266549, Example 349
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C16H17F3N4O2
 1
1
IC50 = 1158 nM
   TI
   LI
   LO
   TS
CP0515037
N4-cyclopropyl-N2-(quinolin-6-yl)-5-(trifluoromethyl) pyrimidine-2,4-diamine
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C17H14F3N5
 1
1
IC50 = 1647 nM
   TI
   LI
   LO
   TS
CP0540134
US10266549, Example 304a
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C14H14F3N5
 1
1
IC50 = 1687 nM
   TI
   LI
   LO
   TS
CP0495717
N4-cyclopropyl-N2-(5-methoxypyridin-3-yl)-5-(trifluoromethyl) pyrimidine-2,4-diamine
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C14H14F3N5O
 1
1
IC50 = 1885 nM
   TI
   LI
   LO
   TS
CP0537630
US10266549, Example 208a
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C15H12F3N5O
 1
1
IC50 = 4256 nM
   TI
   LI
   LO
   TS
CP0331654
2-(5-Bromo-2-(3,4,5-trimethoxyphenylamino)pyrimidin-4-yloxy)-N-methylbenzamide
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C21H21BrN4O5
 1
1
IC50 = 4578 nM
   TI
   LI
   LO
   TS