| Compound ID |
Compound Name |
Compound Formula |
|
CP0017650
|
8-(Phenylamino)-1-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H15F3N6O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0639837
|
8-[2-methoxy-5-(4-methylpiperazin-1-yl)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H28N8O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0018881
|
1-Methyl-8-[(2-methylphenyl)amino]-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H18N6O
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0026702
|
8-{[2-Methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H28N8O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0018224
|
8-[(2-Methoxyphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H18N6O2
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0018223
|
1-Methyl-8-{[3-(trifluoromethyl)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H15F3N6O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0017007
|
pyrazolo[4,3-h]quinazoline-3-carboxamide, 1
Show/Hide
|
C17H16N6O
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0020461
|
1-Methyl-8-{[2-(methylsulfanyl)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H18N6OS
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0026700
|
8-[(3-Acetylphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0017708
|
8-{[2-Acetyl-5-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C24H28N8O2
|
1
|
| 1 |
IC50 = 109 nM
|
|
|
|
CP0015510
|
1-Methyl-8-{[2-(methylamino)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H19N7O
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0025690
|
1-methyl-8-(phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid
Show/Hide
|
C17H15N5O2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0029110
|
8-[(2-Fluorophenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H15FN6O
|
1
|
| 1 |
IC50 = 125 nM
|
|
|
|
CP0018222
|
8-[(3-Methoxyphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H18N6O2
|
1
|
| 1 |
IC50 = 135 nM
|
|
|
|
CP0016541
|
1-Cyclohexyl-8-(phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]-quinazoline-3-carboxamide
Show/Hide
|
C22H24N6O
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0027872
|
8-[(2-Aminophenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H17N7O
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0019922
|
8-[(4-Acetylphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 = 197 nM
|
|
|
|
CP0025241
|
8-(Phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C16H14N6O
|
1
|
| 1 |
IC50 = 248 nM
|
|
|
|
CP0028619
|
8-[(4-Methoxyphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H18N6O2
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0017472
|
1-Methyl-8-[(2-phenoxyphenyl)amino]-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H20N6O2
|
1
|
| 1 |
IC50 = 278 nM
|
|
|
|
CP0025689
|
8-[(2-Acetylphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C19H18N6O2
|
1
|
| 1 |
IC50 = 346 nM
|
|
|
|
CP0025912
|
1-Methyl-8-{[2-(propan-2-yl)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C20H22N6O
|
1
|
| 1 |
IC50 = 365 nM
|
|
|
|
CP0025243
|
8-(Phenylamino)-1-(propan-2-yl)-4,5-dihydro-1H-pyrazolo[4,3-h]-quinazoline-3-carboxamide
Show/Hide
|
C19H20N6O
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0017652
|
1-Methyl-8-{[2-(trifluoromethyl)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H15F3N6O
|
1
|
| 1 |
IC50 = 432 nM
|
|
|
|
CP0027123
|
8-{[2-Acetyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C24H28N8O2
|
1
|
| 1 |
IC50 = 464 nM
|
|
|
|
CP0017651
|
1-Methyl-8-[(2-nitrophenyl)amino]-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H15N7O3
|
1
|
| 1 |
IC50 = 488 nM
|
|
|
|
CP0025242
|
1-Methyl-8-{[4-(trifluoromethyl)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H15F3N6O
|
1
|
| 1 |
IC50 = 872 nM
|
|
|
|
CP0018233
|
8-[(2-Benzylphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C24H22N6O
|
1
|
| 1 |
IC50 = 943 nM
|
|
|
|
CP0018232
|
1-Methyl-8-{[2-(phenylamino)phenyl]amino}-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H21N7O
|
1
|
| 1 |
IC50 = 949 nM
|
|
|
|
CP0026742
|
methyl 2-[(3-carbamoyl-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazolin-8-yl)amino]benzoate
Show/Hide
|
C19H18N6O3
|
1
|
| 1 |
IC50 = 1117 nM
|
|
|
|
CP0027122
|
8-(Biphenyl-2-ylamino)-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]-quinazoline-3-carboxamide
Show/Hide
|
C23H20N6O
|
1
|
| 1 |
IC50 = 1565 nM
|
|
|
|
CP0023011
|
1-Methyl-8-{[2-(phenylcarbonyl)phenyl]amino}-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C24H20N6O2
|
1
|
| 1 |
IC50 = 1969 nM
|
|
|
|
CP0025688
|
1-Methyl-8-{[2-(phenylsulfanyl)phenyl]amino}-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H20N6OS
|
1
|
| 1 |
IC50 = 2033 nM
|
|
|
|
CP0017471
|
8-{[2-Acetyl-3-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C24H28N8O2
|
1
|
| 1 |
IC50 = 2051 nM
|
|
|
|
CP0023674
|
8-[(2-Carbamoylphenyl)amino]-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C18H17N7O2
|
1
|
| 1 |
IC50 = 2076 nM
|
|
|
|
CP0018580
|
8-{[2-(Acetylamino)phenyl]amino}-1-methyl-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C19H19N7O2
|
1
|
| 1 |
IC50 = 2523 nM
|
|
|
|
CP0026741
|
1-Methyl-8-[(2-sulfamoylphenyl)amino]-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H17N7O3S
|
1
|
| 1 |
IC50 = 3733 nM
|
|
|
|
CP0016827
|
pyrazolo[4,3-h]quinazoline-3-carboxamide, 16
Show/Hide
|
C18H18N6O
|
1
|
| 1 |
IC50 = 4215 nM
|
|
|
|
CP0015588
|
1-Methyl-8-[(4-nitrophenyl)amino]-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H15N7O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0016540
|
1-Methyl-8-[(3-nitrophenyl)amino]-4,5-dihydro-1H-pyrazolo-[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C17H15N7O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0018215
|
pyrazolo[4,3-h]quinazoline-3-carboxamide, 20
Show/Hide
|
C23H20N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0018880
|
1-(1-Methylpiperidin-4-yl)-8-(phenylamino)-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C22H25N7O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0022208
|
8-(Phenylamino)-1-[2-(piperidin-1-yl)ethyl]-4,5-dihydro-1Hpyrazolo[4,3-h]quinazoline-3-carboxamide
Show/Hide
|
C23H27N7O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0023532
|
ethyl 8-anilino-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxylate
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0023794
|
pyrazolo[4,3-h]quinazoline-3-carboxamide, 17
Show/Hide
|
C20H20N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0025238
|
pyrazolo[4,3-h]quinazoline-3-carboxamide, 19
Show/Hide
|
C22H24N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0026701
|
1-Phenyl-8-(phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]-quinazoline-3-carboxamide
Show/Hide
|
C22H18N6O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
