Brief Information of the Cell Line and Protein
Cell Line ID: CL000017 , HeLa
Synonyms
HELA
Hela
He La
He-La
HeLa-CCL2
Henrietta Lacks cells
Helacyton gartleri
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT01286 , Bile acid receptor
Gene Name NR1H4
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID Q96RI1
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000017  Protein ID: PT01286
 
Compound ID Compound Name Compound Formula
CP0235782
6-chloro-2-(4-chloropyridin-2-yl)-N-[(4-methoxyphenyl)methyl]imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H16Cl2N4O
 1
1
EC50 = 0.3 nM
   TI
   LI
   LO
   TS
CP0306331
4-tert-butyl-N-[[4-(trifluoromethylsulfanyl)phenyl]methyl]benzamide
   Show/Hide
C19H20F3NOS
 1
1
EC50 = 0.4 nM
   TI
   LI
   LO
   TS
CP0394339
N-benzyl-2-(4-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H17ClN4
 1
1
EC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0849176
3-(3-o-tolyl-1,2,4-oxadiazol-5-yl)benzoic acid
   Show/Hide
C16H12N2O3
 1
1
EC50 = 7.2 nM
   TI
   LI
   LO
   TS
CP0548716
N-benzyl-2-(5-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H17ClN4
 1
1
EC50 = 7.4 nM
   TI
   LI
   LO
   TS
CP0143432
4-[[(4-tert-butylbenzoyl)amino]methyl]-3-fluorobenzoic acid
   Show/Hide
C19H20FNO3
 1
1
EC50 = 7.8 nM
   TI
   LI
   LO
   TS
CP0379834
3-[[2-[(4-tert-butylbenzoyl)amino]-4-methoxybenzoyl]amino]benzoic acid
   Show/Hide
C26H26N2O5
 1
1
EC50 = 8 nM
   TI
   LI
   LO
   TS
CP0558363
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-chlorobenzoic acid
   Show/Hide
C19H20ClNO3
 1
1
EC50 = 8.8 nM
   TI
   LI
   LO
   TS
CP0184082
4-tert-butyl-N-[[2-chloro-4-[(2,2,2-trifluoroacetyl)amino]phenyl]methyl]benzamide
   Show/Hide
C20H20ClF3N2O2
 1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
CP0566071
N-benzyl-2-(3-chlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H18ClN3
 1
1
EC50 = 16 nM
   TI
   LI
   LO
   TS
CP0474866
N-benzyl-6-methyl-2-pyridin-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H18N4
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0252290
4-tert-butyl-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
   Show/Hide
C19H23ClN2O3S
 2
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
2
EC50 = 20.4 nM
   TI
   LI
   LO
   TS
CP0394341
N-benzyl-2-(3,4-dichlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H17Cl2N3
 1
1
EC50 = 24 nM
   TI
   LI
   LO
   TS
CP0408116
N-benzyl-2-(3-chloro-4-fluorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H17ClFN3
 1
1
EC50 = 26 nM
   TI
   LI
   LO
   TS
CP0570143
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(2-hydroxypropan-2-yl)benzamide
   Show/Hide
C18H21ClN2O4S
 1
1
EC50 = 32 nM
   TI
   LI
   LO
   TS
CP0549531
N-[(4-amino-2-chlorophenyl)methyl]-4-tert-butylbenzamide
   Show/Hide
C18H21ClN2O
 2
1
EC50 = 40 nM
   TI
   LI
   LO
   TS
2
EC50 = 46 nM
   TI
   LI
   LO
   TS
CP0379495
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
   Show/Hide
C26H26N2O4
 1
1
EC50 = 42 nM
   TI
   LI
   LO
   TS
CP0566782
5-[[2-[(4-tert-butylbenzoyl)amino]-4-methylbenzoyl]amino]-2-methylbenzoic acid
   Show/Hide
C27H28N2O4
 1
1
EC50 = 43 nM
   TI
   LI
   LO
   TS
CP0365622
4-tert-butyl-N-[[4-(methanesulfonamido)phenyl]methyl]benzamide
   Show/Hide
C19H24N2O3S
 1
1
EC50 = 44 nM
   TI
   LI
   LO
   TS
CP0387199
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
   Show/Hide
C26H26N2O4
 1
1
EC50 = 45 nM
   TI
   LI
   LO
   TS
CP0387230
3-[[2-[(4-tert-butylbenzoyl)amino]-4-chlorobenzoyl]amino]benzoic acid
   Show/Hide
C25H23ClN2O4
 2
1
EC50 = 47 nM
   TI
   LI
   LO
   TS
2
EC50 = 120 nM
   TI
   LI
   LO
   TS
CP0399542
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methoxybenzoic acid
   Show/Hide
C26H26N2O5
 1
1
EC50 = 47 nM
   TI
   LI
   LO
   TS
CP0398525
3-[[4-bromo-2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
   Show/Hide
C25H23BrN2O4
 1
1
EC50 = 48 nM
   TI
   LI
   LO
   TS
CP0387200
3-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]propanoic acid
   Show/Hide
C27H28N2O4
 2
1
EC50 = 60 nM
   TI
   LI
   LO
   TS
2
EC50 = 64 nM
   TI
   LI
   LO
   TS
CP0398524
3-[[2-[(4-tert-butylbenzoyl)amino]-4-methylbenzoyl]amino]benzoic acid
   Show/Hide
C26H26N2O4
 1
1
EC50 = 61 nM
   TI
   LI
   LO
   TS
CP0419732
2-[(4-tert-butylbenzoyl)amino]-N-(3-carbamoylphenyl)benzamide
   Show/Hide
C25H25N3O3
 2
1
EC50 = 70 nM
   TI
   LI
   LO
   TS
2
EC50 = 74 nM
   TI
   LI
   LO
   TS
CP0414665
2-[(4-tert-butylbenzoyl)amino]-N-(3,4-dimethoxyphenyl)benzamide
   Show/Hide
C26H28N2O4
 1
1
EC50 = 71 nM
   TI
   LI
   LO
   TS
CP0457996
4-[1-[(4-tert-butylbenzoyl)amino]ethyl]benzoic acid
   Show/Hide
C20H23NO3
 1
1
EC50 = 76 nM
   TI
   LI
   LO
   TS
CP0408118
N-benzyl-2-(6-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H17ClN4
 1
1
EC50 = 80 nM
   TI
   LI
   LO
   TS
CP0436627
N-benzyl-6-methyl-2-(4-phenylphenyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C27H23N3
 1
1
EC50 = 81 nM
   TI
   LI
   LO
   TS
CP0399544
5-[[2-[(4-tert-butylbenzoyl)amino]-4-methoxybenzoyl]amino]-2-methylbenzoic acid
   Show/Hide
C27H28N2O5
 1
1
EC50 = 87 nM
   TI
   LI
   LO
   TS
CP0181580
4-tert-butyl-N-[(4-methylsulfanylphenyl)methyl]benzamide
   Show/Hide
C19H23NOS
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0454801
N-[(4-acetylphenyl)methyl]-4-tert-butylbenzamide
   Show/Hide
C20H23NO2
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0539159
5-[[2-[(4-tert-butylbenzoyl)amino]-4-chlorobenzoyl]amino]-2-methylbenzoic acid
   Show/Hide
C26H25ClN2O4
 1
1
EC50 = 110 nM
   TI
   LI
   LO
   TS
CP0881990
5-(4-methoxyphenyl)-3-o-tolyl-1,2,4-oxadiazole
   Show/Hide
C16H14N2O2
 1
1
EC50 = 120 nM
   TI
   LI
   LO
   TS
CP0143436
4-tert-butyl-N-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzamide
   Show/Hide
C19H21N5O
 1
1
EC50 = 120 nM
   TI
   LI
   LO
   TS
CP0378906
N-benzyl-6-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H21N3
 1
1
EC50 = 130 nM
   TI
   LI
   LO
   TS
CP0335294
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-fluorobenzoic acid
   Show/Hide
C19H20FNO3
 1
1
EC50 = 140 nM
   TI
   LI
   LO
   TS
CP0546183
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(trifluoromethyl)benzamide
   Show/Hide
C16H14ClF3N2O3S
 1
1
EC50 = 140 nM
   TI
   LI
   LO
   TS
CP0398725
2-bromo-5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
   Show/Hide
C25H23BrN2O4
 1
1
EC50 = 150 nM
   TI
   LI
   LO
   TS
CP0350531
4-tert-butyl-N-[(4-methoxyphenyl)methyl]benzamide
   Show/Hide
C19H23NO2
 1
1
EC50 = 150 nM
   TI
   LI
   LO
   TS
CP0049016
(4R)-4-[(1S,2S,5R,7S,8R,9R,10S,11S,14R,15R)-8-ethyl-5,9-dihydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-14-yl]pentanoic acid
   Show/Hide
C26H44O4
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0081889
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-methylbenzoic acid
   Show/Hide
C20H23NO3
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0143437
4-tert-butyl-N-[[4-(trifluoromethoxy)phenyl]methyl]benzamide
   Show/Hide
C19H20F3NO2
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0335295
4-tert-butyl-N-[(4-ethoxyphenyl)methyl]benzamide
   Show/Hide
C20H25NO2
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0559311
N-benzyl-6-chloro-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C18H14ClN3S
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0184079
4-[[(4-tert-butylbenzoyl)amino]methyl]-N,N-dimethylbenzamide
   Show/Hide
C21H26N2O2
 1
1
EC50 = 170 nM
   TI
   LI
   LO
   TS
CP0365623
4-tert-butyl-N-[(4-propan-2-yloxyphenyl)methyl]benzamide
   Show/Hide
C21H27NO2
 1
1
EC50 = 170 nM
   TI
   LI
   LO
   TS
CP0407802
N-benzyl-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C23H21N3O2
 1
1
EC50 = 170 nM
   TI
   LI
   LO
   TS
CP0436624
N-benzyl-2-(4-fluorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H18FN3
 1
1
EC50 = 170 nM
   TI
   LI
   LO
   TS
CP0506631
N-[(4-methoxyphenyl)methyl]-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3OS
 1
1
EC50 = 170 nM
   TI
   LI
   LO
   TS
CP0457728
N-benzyl-6-methyl-2-(3-methylphenyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H21N3
 1
1
EC50 = 180 nM
   TI
   LI
   LO
   TS
CP0533129
2-[(4-tert-butylbenzoyl)amino]-N-(3-methylsulfanylphenyl)benzamide
   Show/Hide
C25H26N2O2S
 1
1
EC50 = 200 nM
   TI
   LI
   LO
   TS
CP0539953
N-benzyl-6-phenyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C24H19N3S
 1
1
EC50 = 200 nM
   TI
   LI
   LO
   TS
CP0474863
N-benzyl-6-methyl-2-naphthalen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C25H21N3
 1
1
EC50 = 210 nM
   TI
   LI
   LO
   TS
CP0866880
4-(3-o-tolyl-1,2,4-oxadiazol-5-yl)benzoic acid
   Show/Hide
C16H12N2O3
 1
1
EC50 = 220 nM
   TI
   LI
   LO
   TS
CP0378905
N-benzyl-6-methyl-2-(4-methyl-1,3-thiazol-2-yl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H18N4S
 1
1
EC50 = 220 nM
   TI
   LI
   LO
   TS
CP0457716
6-methyl-N-[(4-methylphenyl)methyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3S
 1
1
EC50 = 220 nM
   TI
   LI
   LO
   TS
CP0396061
2-[(4-tert-butylbenzoyl)amino]-N-(3-cyanophenyl)benzamide
   Show/Hide
C25H23N3O2
 1
1
EC50 = 230 nM
   TI
   LI
   LO
   TS
CP0407804
6-methyl-N-(3-phenylpropyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H21N3S
 1
1
EC50 = 230 nM
   TI
   LI
   LO
   TS
CP0407801
N-benzyl-2-(4-chlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H18ClN3
 1
1
EC50 = 240 nM
   TI
   LI
   LO
   TS
CP0474861
N-benzyl-2-(3-methoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H21N3O
 1
1
EC50 = 250 nM
   TI
   LI
   LO
   TS
CP0553306
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-pyrrolidin-1-ylbenzamide
   Show/Hide
C19H22ClN3O3S
 1
1
EC50 = 250 nM
   TI
   LI
   LO
   TS
CP0365731
4-tert-butyl-N-[[4-[(2,2,2-trifluoroacetyl)amino]phenyl]methyl]benzamide
   Show/Hide
C20H21F3N2O2
 1
1
EC50 = 260 nM
   TI
   LI
   LO
   TS
CP0539023
N-benzyl-6-methyl-2-(2-methylphenyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H21N3
 1
1
EC50 = 260 nM
   TI
   LI
   LO
   TS
CP0388902
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-chlorobenzoic acid
   Show/Hide
C25H23ClN2O4
 1
1
EC50 = 280 nM
   TI
   LI
   LO
   TS
CP0477280
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
   Show/Hide
C25H24N2O4
 1
1
EC50 = 280 nM
   TI
   LI
   LO
   TS
CP0539082
N-benzyl-6-methyl-2-phenylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H19N3
 1
1
EC50 = 280 nM
   TI
   LI
   LO
   TS
CP0558982
N-benzyl-6-methyl-2-(2-phenylethyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C23H23N3
 1
1
EC50 = 310 nM
   TI
   LI
   LO
   TS
CP0454798
4-[[(3,4-dimethylbenzoyl)amino]methyl]benzoic acid
   Show/Hide
C17H17NO3
 1
1
EC50 = 320 nM
   TI
   LI
   LO
   TS
CP0539300
4-[[(4-tert-butylbenzoyl)amino]methyl]-N-methylbenzamide
   Show/Hide
C20H24N2O2
 1
1
EC50 = 340 nM
   TI
   LI
   LO
   TS
CP0919608
5-(4-bromophenyl)-3-phenyl-1,2,4-oxadiazole
   Show/Hide
C14H9BrN2O
 1
1
EC50 = 350 nM
   TI
   LI
   LO
   TS
CP0184342
3-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenyl]propanoic acid
   Show/Hide
C21H25NO3
 1
1
EC50 = 350 nM
   TI
   LI
   LO
   TS
CP0083256
4-[[(3,4-dimethoxybenzoyl)amino]methyl]benzoic acid
   Show/Hide
C17H17NO5
 1
1
EC50 = 370 nM
   TI
   LI
   LO
   TS
CP0143430
4-[[(4-tert-butylbenzoyl)amino]methyl]benzoic acid
   Show/Hide
C19H21NO3
 1
1
EC50 = 370 nM
   TI
   LI
   LO
   TS
CP0411575
2-[(4-tert-butylbenzoyl)amino]-N-(3-methoxyphenyl)benzamide
   Show/Hide
C25H26N2O3
 1
1
EC50 = 380 nM
   TI
   LI
   LO
   TS
CP0549530
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-propan-2-yloxybenzamide
   Show/Hide
C18H21ClN2O4S
 1
1
EC50 = 400 nM
   TI
   LI
   LO
   TS
CP0866881
5-(4-chlorophenyl)-3-p-tolyl-1,2,4-oxadiazole
   Show/Hide
C15H11ClN2O
 1
1
EC50 = 410 nM
   TI
   LI
   LO
   TS
CP0575759
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-piperidin-1-ylbenzamide
   Show/Hide
C20H24ClN3O3S
 1
1
EC50 = 410 nM
   TI
   LI
   LO
   TS
CP0419731
2-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C26H26N2O4
 1
1
EC50 = 420 nM
   TI
   LI
   LO
   TS
CP0546180
4-tert-butyl-N-[[2-chloro-4-(propan-2-ylsulfonylamino)phenyl]methyl]benzamide
   Show/Hide
C21H27ClN2O3S
 1
1
EC50 = 420 nM
   TI
   LI
   LO
   TS
CP0408117
N-benzyl-2-(4-bromophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C21H18BrN3
 1
1
EC50 = 430 nM
   TI
   LI
   LO
   TS
CP0083255
4-[[(4-phenylbenzoyl)amino]methyl]benzoic acid
   Show/Hide
C21H17NO3
 1
1
EC50 = 440 nM
   TI
   LI
   LO
   TS
CP0810328
7-(diethylamino)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-2H-chromen-2-one
   Show/Hide
C21H19N3O3
 1
1
EC50 = 460 nM
   TI
   LI
   LO
   TS
CP0559310
N-benzyl-2-thiophen-2-yl-6-(trifluoromethyl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H14F3N3S
 1
1
EC50 = 460 nM
   TI
   LI
   LO
   TS
CP0379833
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-fluorobenzoic acid
   Show/Hide
C25H23FN2O4
 1
1
EC50 = 480 nM
   TI
   LI
   LO
   TS
CP0456564
N-(3-acetylphenyl)-2-[(4-tert-butylbenzoyl)amino]benzamide
   Show/Hide
C26H26N2O3
 1
1
EC50 = 480 nM
   TI
   LI
   LO
   TS
CP0548715
N-benzyl-6-bromo-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C18H14BrN3S
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0284282
4-tert-butyl-N-[[2-chloro-4-(ethylsulfonylamino)phenyl]methyl]benzamide
   Show/Hide
C20H25ClN2O3S
 1
1
EC50 = 500 nM
   TI
   LI
   LO
   TS
CP0089615
3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(1-methylethyl)isoxazol-4-yl]methoxy}phenyl)ethenyl]benzoic acid
   Show/Hide
C28H22Cl3NO4
 1
1
EC50 = 510 nM
   TI
   LI
   LO
   TS
CP0394344
N-benzyl-6-methyl-2-pyridin-3-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H18N4
 1
1
EC50 = 520 nM
   TI
   LI
   LO
   TS
CP0849175
3,5-diphenyl-1,2,4-oxadiazole
   Show/Hide
C14H10N2O
 1
1
EC50 = 530 nM
   TI
   LI
   LO
   TS
CP0407805
N-benzyl-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N3S
 1
1
EC50 = 540 nM
   TI
   LI
   LO
   TS
CP0549525
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-[1-(trifluoromethyl)cyclopropyl]benzamide
   Show/Hide
C19H18ClF3N2O3S
 1
1
EC50 = 540 nM
   TI
   LI
   LO
   TS
CP0558983
N-benzyl-2-(furan-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N3O
 1
1
EC50 = 560 nM
   TI
   LI
   LO
   TS
CP0492060
4-(1-bicyclo[1.1.1]pentanyl)-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
   Show/Hide
C20H21ClN2O3S
 1
1
EC50 = 560 nM
   TI
   LI
   LO
   TS
CP0196829
4-[[(3-phenylbenzoyl)amino]methyl]benzoic acid
   Show/Hide
C21H17NO3
 1
1
EC50 = 670 nM
   TI
   LI
   LO
   TS
CP0387204
2-[3-[[2-[(4-phenylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C28H22N2O4
 1
1
EC50 = 700 nM
   TI
   LI
   LO
   TS
CP0572339
4-[[2-[[(E)-3-phenylprop-2-enoyl]amino]benzoyl]amino]butanoic acid
   Show/Hide
C20H20N2O4
 1
1
EC50 = 720 nM
   TI
   LI
   LO
   TS
CP0454799
2-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenoxy]acetic acid
   Show/Hide
C20H23NO4
 1
1
EC50 = 730 nM
   TI
   LI
   LO
   TS
CP0407803
7-methyl-N-(4-phenylbutyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H23N3S
 1
1
EC50 = 750 nM
   TI
   LI
   LO
   TS
CP0506632
3-benzyl-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridine
   Show/Hide
C19H16N2S
 1
1
EC50 = 810 nM
   TI
   LI
   LO
   TS
CP0394340
N-benzyl-6-methyl-2-thiophen-3-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N3S
 1
1
EC50 = 830 nM
   TI
   LI
   LO
   TS
CP0535248
N-benzyl-6-methoxy-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N3OS
 1
1
EC50 = 830 nM
   TI
   LI
   LO
   TS
CP0436626
N-benzyl-2-(3,4-dimethoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C23H23N3O2
 1
1
EC50 = 910 nM
   TI
   LI
   LO
   TS
CP0303425
4-tert-butyl-N-[(2-fluoro-4-sulfamoylphenyl)methyl]benzamide
   Show/Hide
C18H21FN2O3S
 1
1
EC50 = 970 nM
   TI
   LI
   LO
   TS
CP0403496
4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
   Show/Hide
C25H18N2O4
 1
1
EC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0539952
6-methyl-N-(2-phenylethyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3S
 1
1
EC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0546181
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(trifluoromethoxy)benzamide
   Show/Hide
C16H14ClF3N2O4S
 1
1
EC50 = 1090 nM
   TI
   LI
   LO
   TS
CP0396059
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-chlorobenzoic acid
   Show/Hide
C25H23ClN2O4
 1
1
EC50 = 1100 nM
   TI
   LI
   LO
   TS
CP0408119
N-benzyl-6-methyl-2-(1-methylpyrrol-2-yl)imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H20N4
 1
1
EC50 = 1100 nM
   TI
   LI
   LO
   TS
CP0474862
N-benzyl-6-methyl-2-[(E)-2-phenylethenyl]imidazo[1,2-a]pyridin-3-amine
   Show/Hide
C23H21N3
 1
1
EC50 = 1160 nM
   TI
   LI
   LO
   TS
CP0184169
4-[[(4-tert-butyl-3-methoxybenzoyl)amino]methyl]benzoic acid
   Show/Hide
C20H23NO4
 1
1
EC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0394343
N-benzyl-7-ethyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3S
 1
1
EC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0436628
N-benzyl-6-methyl-2-pyrazin-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N5
 1
1
EC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0575253
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(1,1-difluoroethyl)benzamide
   Show/Hide
C17H17ClF2N2O3S
 1
1
EC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0541210
N-benzyl-2-(4-methoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C22H21N3O
 1
1
EC50 = 1270 nM
   TI
   LI
   LO
   TS
CP0417144
4-[[[2-(naphthalene-2-carbonylamino)benzoyl]amino]methyl]benzoic acid
   Show/Hide
C26H20N2O4
 1
1
EC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0329861
4-tert-butyl-N-[(4-methylsulfinylphenyl)methyl]benzamide
   Show/Hide
C19H23NO2S
 1
1
EC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0539950
6-methyl-N-[(1S)-1-phenylethyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3S
 1
1
EC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0451683
4-[(naphthalene-2-carbonylamino)methyl]benzoic acid
   Show/Hide
C19H15NO3
 1
1
EC50 = 1360 nM
   TI
   LI
   LO
   TS
CP0081661
4-(4-tert-Butylphenylcarboxamidomethyl)benzenesulfonamide
   Show/Hide
C18H22N2O3S
 1
1
EC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0496466
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(dimethylamino)benzamide
   Show/Hide
C17H20ClN3O3S
 1
1
EC50 = 1460 nM
   TI
   LI
   LO
   TS
CP0387227
3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
   Show/Hide
C25H18N2O4
 1
1
EC50 = 1500 nM
   TI
   LI
   LO
   TS
CP0575254
4-tert-butyl-N-[[2-chloro-4-(cyclopropylsulfonylamino)phenyl]methyl]benzamide
   Show/Hide
C21H25ClN2O3S
 1
1
EC50 = 1500 nM
   TI
   LI
   LO
   TS
CP0303426
3-[[(4-tert-butylbenzoyl)amino]methyl]benzoic acid
   Show/Hide
C19H21NO3
 1
1
EC50 = 1700 nM
   TI
   LI
   LO
   TS
CP0436623
N-benzyl-2-(furan-3-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C19H17N3O
 1
1
EC50 = 1900 nM
   TI
   LI
   LO
   TS
CP0408115
N-benzyl-6-methyl-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H18N4
 1
1
EC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0396063
3-[[4-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
   Show/Hide
C22H14ClF3N2O4
 1
1
EC50 = 2100 nM
   TI
   LI
   LO
   TS
CP0500157
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-ethoxybenzamide
   Show/Hide
C17H19ClN2O4S
 1
1
EC50 = 2200 nM
   TI
   LI
   LO
   TS
CP0398732
3-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]propanoic acid
   Show/Hide
C24H19F3N2O4
 1
1
EC50 = 2300 nM
   TI
   LI
   LO
   TS
CP0387071
4-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]butanoic acid
   Show/Hide
C22H26N2O4
 1
1
EC50 = 2500 nM
   TI
   LI
   LO
   TS
CP0387205
2-[3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]phenyl]acetic acid
   Show/Hide
C26H20N2O4
 1
1
EC50 = 2500 nM
   TI
   LI
   LO
   TS
CP0445061
2-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C23H17F3N2O4
 1
1
EC50 = 2600 nM
   TI
   LI
   LO
   TS
CP0399541
2-[(4-tert-butylbenzoyl)amino]-N-[3-(2H-tetrazol-5-yl)phenyl]benzamide
   Show/Hide
C25H24N6O2
 1
1
EC50 = 2900 nM
   TI
   LI
   LO
   TS
CP0886015
5-(4-methoxyphenyl)-3-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazole
   Show/Hide
C16H11F3N2O2
 1
1
EC50 = 2900 nM
   TI
   LI
   LO
   TS
CP0331663
N-[(4-acetamidophenyl)methyl]-4-tert-butylbenzamide
   Show/Hide
C20H24N2O2
 1
1
EC50 = 2900 nM
   TI
   LI
   LO
   TS
CP0403497
2-[4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]phenyl]acetic acid
   Show/Hide
C26H20N2O4
 1
1
EC50 = 3100 nM
   TI
   LI
   LO
   TS
CP0541211
6-methyl-N-[(1R)-1-phenylethyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C20H19N3S
 1
1
EC50 = 3200 nM
   TI
   LI
   LO
   TS
CP0267212
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(1,1,2,2,2-pentafluoroethyl)benzamide
   Show/Hide
C17H14ClF5N2O3S
 1
1
EC50 = 3220 nM
   TI
   LI
   LO
   TS
CP0388903
3-[[5-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
   Show/Hide
C22H14ClF3N2O4
 1
1
EC50 = 3400 nM
   TI
   LI
   LO
   TS
CP0387232
3-[[2-[(4-bromobenzoyl)amino]benzoyl]amino]benzoic acid
   Show/Hide
C21H15BrN2O4
 1
1
EC50 = 3700 nM
   TI
   LI
   LO
   TS
CP0327641
4-[(4-tert-butylphenyl)carbamoylamino]benzoic acid
   Show/Hide
C18H20N2O3
 1
1
EC50 = 3800 nM
   TI
   LI
   LO
   TS
CP0393975
4-[[(4-tert-butylbenzoyl)amino]methyl]benzamide
   Show/Hide
C19H22N2O2
 1
1
EC50 = 3800 nM
   TI
   LI
   LO
   TS
CP0413032
4-tert-butyl-N-[(4-methylsulfonylphenyl)methyl]benzamide
   Show/Hide
C19H23NO3S
 1
1
EC50 = 3800 nM
   TI
   LI
   LO
   TS
CP0509519
N-benzyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
   Show/Hide
C18H15N3S
 1
1
EC50 = 4000 nM
   TI
   LI
   LO
   TS
CP0546185
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(2,2,2-trifluoroethyl)benzamide
   Show/Hide
C17H16ClF3N2O3S
 1
1
EC50 = 4000 nM
   TI
   LI
   LO
   TS
CP0380161
6-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]hexanoic acid
   Show/Hide
C24H24N2O4
 1
1
EC50 = 4400 nM
   TI
   LI
   LO
   TS
CP0546184
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-morpholin-4-ylbenzamide
   Show/Hide
C19H22ClN3O4S
 1
1
EC50 = 4400 nM
   TI
   LI
   LO
   TS
CP0379832
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-methoxybenzoic acid
   Show/Hide
C26H26N2O5
 1
1
EC50 = 4700 nM
   TI
   LI
   LO
   TS
CP0509140
3-[[2-(2,3-dihydro-1,4-benzodioxine-6-carbonylamino)benzoyl]amino]benzoic acid
   Show/Hide
C23H18N2O6
 1
1
EC50 = 4900 nM
   TI
   LI
   LO
   TS
CP0387068
3-[[2-[[3-fluoro-4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
   Show/Hide
C22H14F4N2O4
 1
1
EC50 = 5000 nM
   TI
   LI
   LO
   TS
CP0509141
3-[[2-[[(E)-3-phenylprop-2-enoyl]amino]benzoyl]amino]benzoic acid
   Show/Hide
C23H18N2O4
 1
1
EC50 = 5200 nM
   TI
   LI
   LO
   TS
CP0454800
4-tert-butyl-N-[(4-formylphenyl)methyl]benzamide
   Show/Hide
C19H21NO2
 1
1
EC50 = 5300 nM
   TI
   LI
   LO
   TS
CP0387228
4-[[2-[(4-ethylbenzoyl)amino]benzoyl]amino]butanoic acid
   Show/Hide
C20H22N2O4
 1
1
EC50 = 5800 nM
   TI
   LI
   LO
   TS
CP0413031
2-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenyl]acetic acid
   Show/Hide
C20H23NO3
 1
1
EC50 = 6400 nM
   TI
   LI
   LO
   TS
CP0387067
3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
   Show/Hide
C22H15F3N2O4
 1
1
EC50 = 6900 nM
   TI
   LI
   LO
   TS
CP0396062
2-[3-[[2-[[4-(trifluoromethylsulfanyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C23H17F3N2O4S
 1
1
EC50 = 7000 nM
   TI
   LI
   LO
   TS
CP0492702
methyl 4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]butanoate
   Show/Hide
C23H22N2O4
 1
1
EC50 = 7100 nM
   TI
   LI
   LO
   TS
CP0184078
4-[[(4-tert-butylbenzoyl)amino]methyl]-3-chlorobenzoic acid
   Show/Hide
C19H20ClNO3
 1
1
EC50 = 7500 nM
   TI
   LI
   LO
   TS
CP0403351
5-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]pentanoic acid
   Show/Hide
C23H22N2O4
 1
1
EC50 = 8300 nM
   TI
   LI
   LO
   TS
CP0387203
2-[3-[[2-[(4-methylsulfanylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
   Show/Hide
C23H20N2O4S
 1
1
EC50 = 8500 nM
   TI
   LI
   LO
   TS
CP0385188
4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]butanoic acid
   Show/Hide
C22H20N2O4
 2
1
EC50 = 8550 nM
   TI
   LI
   LO
   TS
2
EC50 = 8600 nM
   TI
   LI
   LO
   TS
CP0398523
3-[[2-(1,3-benzodioxole-5-carbonylamino)benzoyl]amino]benzoic acid
   Show/Hide
C22H16N2O6
 1
1
EC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0571435
4-(azetidin-1-yl)-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
   Show/Hide
C18H20ClN3O3S
 1
1
EC50 = 13000 nM
   TI
   LI
   LO
   TS
CP0002372
(4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R)-5,9-dihydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-14-yl]pentanoic acid
   Show/Hide
C24H40O4
 1
1
EC50 = 18000 nM
   TI
   LI
   LO
   TS
CP0392557
2-[4-[(4-tert-butyl-2-methoxybenzoyl)amino]phenyl]acetic acid
   Show/Hide
C20H23NO4
 2
1
IC50 = 1.3 nM
   TI
   LI
   LO
   TS
2
IC50 = 9.2 nM
   TI
   LI
   LO
   TS
CP0565305
2-[4-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
   Show/Hide
C19H21NO3
 1
1
IC50 = 76 nM
   TI
   LI
   LO
   TS
CP0396569
2-[4-[(4-tert-butylbenzoyl)amino]-2-methylphenyl]acetic acid
   Show/Hide
C20H23NO3
 1
1
IC50 = 80 nM
   TI
   LI
   LO
   TS
CP0513309
2-[2-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
   Show/Hide
C19H21NO3
 1
1
IC50 = 102 nM
   TI
   LI
   LO
   TS
CP0429349
2-[4-[(4-tert-butyl-2-hydroxybenzoyl)amino]phenyl]acetic acid
   Show/Hide
C19H21NO4
 1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS
CP0548250
2-[4-[(2-methoxy-5-phenylbenzoyl)amino]phenyl]acetic acid
   Show/Hide
C22H19NO4
 1
1
IC50 = 170 nM
   TI
   LI
   LO
   TS
CP0462122
2-[4-[(3-tert-butylbenzoyl)amino]phenyl]acetic acid
   Show/Hide
C19H21NO3
 1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS
CP0467757
2-[4-[(4-tert-butyl-3-methoxybenzoyl)amino]phenyl]acetic acid
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C20H23NO4
 1
1
IC50 = 220 nM
   TI
   LI
   LO
   TS
CP0411732
2-[4-[(3-phenylbenzoyl)amino]phenyl]acetic acid
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C21H17NO3
 1
1
IC50 = 280 nM
   TI
   LI
   LO
   TS
CP0487623
2-[3-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
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C19H21NO3
 2
1
IC50 = 350 nM
   TI
   LI
   LO
   TS
2
IC50 = 400 nM
   TI
   LI
   LO
   TS
CP0532536
3-[4-[(4-tert-butylbenzoyl)amino]phenyl]propanoic acid
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C20H23NO3
 1
1
IC50 = 630 nM
   TI
   LI
   LO
   TS
CP0429350
2-[4-(naphthalene-2-carbonylamino)phenyl]acetic acid
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C19H15NO3
 1
1
IC50 = 680 nM
   TI
   LI
   LO
   TS
CP0396571
4-[4-[(4-tert-butylbenzoyl)amino]phenyl]butanoic acid
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C21H25NO3
 1
1
IC50 = 700 nM
   TI
   LI
   LO
   TS
CP0549065
2-[4-(naphthalene-1-carbonylamino)phenyl]acetic acid
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C19H15NO3
 1
1
IC50 = 810 nM
   TI
   LI
   LO
   TS
CP0487621
2-[4-[(4-phenylbenzoyl)amino]phenyl]acetic acid
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C21H17NO3
 1
1
IC50 = 850 nM
   TI
   LI
   LO
   TS
CP0462123
2-[4-[(4-tert-butylbenzoyl)amino]phenyl]propanoic acid
   Show/Hide
C20H23NO3
 1
1
IC50 = 970 nM
   TI
   LI
   LO
   TS
CP0396568
2-[4-[(4-tert-butylbenzoyl)amino]-3-methylphenyl]acetic acid
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C20H23NO3
 1
1
IC50 = 1500 nM
   TI
   LI
   LO
   TS
CP0487622
2-[4-[benzyl-(4-tert-butylbenzoyl)amino]phenyl]acetic acid
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C26H27NO3
 1
1
IC50 = 2200 nM
   TI
   LI
   LO
   TS
CP0429348
2-[4-[(3-tert-butyl-2-methoxybenzoyl)amino]phenyl]acetic acid
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C20H23NO4
 1
1
IC50 = 3300 nM
   TI
   LI
   LO
   TS
CP0486448
2-[4-[(4-tert-butylbenzoyl)amino]-2-methoxyphenyl]acetic acid
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C20H23NO4
 1
1
IC50 = 3700 nM
   TI
   LI
   LO
   TS
CP0559369
2-[4-[(2-methoxy-3-phenylbenzoyl)amino]phenyl]acetic acid
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C22H19NO4
 1
1
IC50 = 5000 nM
   TI
   LI
   LO
   TS
CP0389938
2-[4-[(4-tert-butylbenzoyl)-methylamino]phenyl]acetic acid
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C20H23NO3
 1
1
IC50 = 8100 nM
   TI
   LI
   LO
   TS
CP0486449
2-[4-[[3-(3,5-dichlorophenyl)benzoyl]amino]phenyl]acetic acid
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C21H15Cl2NO3
 1
1
IC50 = 9100 nM
   TI
   LI
   LO
   TS
CP0379835
3-[[2-[(4-tert-butylbenzoyl)amino]-5-chlorobenzoyl]amino]benzoic acid
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C25H23ClN2O4
 1
1
IC50 = 12300 nM
   TI
   LI
   LO
   TS
CP0398526
3-[[2-[(4-tert-butylbenzoyl)amino]-5-methoxybenzoyl]amino]benzoic acid
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C26H26N2O5
 1
1
IC50 = 15100 nM
   TI
   LI
   LO
   TS
CP0942600
5-(4-methoxyphenyl)-3-phenyl-1,2,4-oxadiazole
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C15H12N2O2
 1
1
IC50 = 16400 nM
   TI
   LI
   LO
   TS
CP0392558
2-[4-[(2-naphthalen-2-ylacetyl)amino]phenyl]acetic acid
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C20H17NO3
 1
1
IC50 = 27000 nM
   TI
   LI
   LO
   TS