Compound ID |
Compound Name |
Compound Formula |
CP0235782
|
6-chloro-2-(4-chloropyridin-2-yl)-N-[(4-methoxyphenyl)methyl]imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H16Cl2N4O
|
1
|
1 |
EC50 = 0.3 nM
|
|
|
CP0306331
|
4-tert-butyl-N-[[4-(trifluoromethylsulfanyl)phenyl]methyl]benzamide
Show/Hide
|
C19H20F3NOS
|
1
|
1 |
EC50 = 0.4 nM
|
|
|
CP0394339
|
N-benzyl-2-(4-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H17ClN4
|
1
|
1 |
EC50 = 1.5 nM
|
|
|
CP0849176
|
3-(3-o-tolyl-1,2,4-oxadiazol-5-yl)benzoic acid
Show/Hide
|
C16H12N2O3
|
1
|
1 |
EC50 = 7.2 nM
|
|
|
CP0548716
|
N-benzyl-2-(5-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H17ClN4
|
1
|
1 |
EC50 = 7.4 nM
|
|
|
CP0143432
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-3-fluorobenzoic acid
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|
C19H20FNO3
|
1
|
1 |
EC50 = 7.8 nM
|
|
|
CP0379834
|
3-[[2-[(4-tert-butylbenzoyl)amino]-4-methoxybenzoyl]amino]benzoic acid
Show/Hide
|
C26H26N2O5
|
1
|
1 |
EC50 = 8 nM
|
|
|
CP0558363
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-chlorobenzoic acid
Show/Hide
|
C19H20ClNO3
|
1
|
1 |
EC50 = 8.8 nM
|
|
|
CP0184082
|
4-tert-butyl-N-[[2-chloro-4-[(2,2,2-trifluoroacetyl)amino]phenyl]methyl]benzamide
Show/Hide
|
C20H20ClF3N2O2
|
1
|
1 |
EC50 = 14 nM
|
|
|
CP0566071
|
N-benzyl-2-(3-chlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H18ClN3
|
1
|
1 |
EC50 = 16 nM
|
|
|
CP0474866
|
N-benzyl-6-methyl-2-pyridin-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H18N4
|
1
|
1 |
EC50 = 20 nM
|
|
|
CP0252290
|
4-tert-butyl-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
Show/Hide
|
C19H23ClN2O3S
|
2
|
1 |
EC50 = 20 nM
|
|
|
2 |
EC50 = 20.4 nM
|
|
|
CP0394341
|
N-benzyl-2-(3,4-dichlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H17Cl2N3
|
1
|
1 |
EC50 = 24 nM
|
|
|
CP0408116
|
N-benzyl-2-(3-chloro-4-fluorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H17ClFN3
|
1
|
1 |
EC50 = 26 nM
|
|
|
CP0570143
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(2-hydroxypropan-2-yl)benzamide
Show/Hide
|
C18H21ClN2O4S
|
1
|
1 |
EC50 = 32 nM
|
|
|
CP0549531
|
N-[(4-amino-2-chlorophenyl)methyl]-4-tert-butylbenzamide
Show/Hide
|
C18H21ClN2O
|
2
|
1 |
EC50 = 40 nM
|
|
|
2 |
EC50 = 46 nM
|
|
|
CP0379495
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C26H26N2O4
|
1
|
1 |
EC50 = 42 nM
|
|
|
CP0566782
|
5-[[2-[(4-tert-butylbenzoyl)amino]-4-methylbenzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C27H28N2O4
|
1
|
1 |
EC50 = 43 nM
|
|
|
CP0365622
|
4-tert-butyl-N-[[4-(methanesulfonamido)phenyl]methyl]benzamide
Show/Hide
|
C19H24N2O3S
|
1
|
1 |
EC50 = 44 nM
|
|
|
CP0387199
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C26H26N2O4
|
1
|
1 |
EC50 = 45 nM
|
|
|
CP0387230
|
3-[[2-[(4-tert-butylbenzoyl)amino]-4-chlorobenzoyl]amino]benzoic acid
Show/Hide
|
C25H23ClN2O4
|
2
|
1 |
EC50 = 47 nM
|
|
|
2 |
EC50 = 120 nM
|
|
|
CP0399542
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-methoxybenzoic acid
Show/Hide
|
C26H26N2O5
|
1
|
1 |
EC50 = 47 nM
|
|
|
CP0398525
|
3-[[4-bromo-2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C25H23BrN2O4
|
1
|
1 |
EC50 = 48 nM
|
|
|
CP0387200
|
3-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]propanoic acid
Show/Hide
|
C27H28N2O4
|
2
|
1 |
EC50 = 60 nM
|
|
|
2 |
EC50 = 64 nM
|
|
|
CP0398524
|
3-[[2-[(4-tert-butylbenzoyl)amino]-4-methylbenzoyl]amino]benzoic acid
Show/Hide
|
C26H26N2O4
|
1
|
1 |
EC50 = 61 nM
|
|
|
CP0419732
|
2-[(4-tert-butylbenzoyl)amino]-N-(3-carbamoylphenyl)benzamide
Show/Hide
|
C25H25N3O3
|
2
|
1 |
EC50 = 70 nM
|
|
|
2 |
EC50 = 74 nM
|
|
|
CP0414665
|
2-[(4-tert-butylbenzoyl)amino]-N-(3,4-dimethoxyphenyl)benzamide
Show/Hide
|
C26H28N2O4
|
1
|
1 |
EC50 = 71 nM
|
|
|
CP0457996
|
4-[1-[(4-tert-butylbenzoyl)amino]ethyl]benzoic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
EC50 = 76 nM
|
|
|
CP0408118
|
N-benzyl-2-(6-chloropyridin-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H17ClN4
|
1
|
1 |
EC50 = 80 nM
|
|
|
CP0436627
|
N-benzyl-6-methyl-2-(4-phenylphenyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C27H23N3
|
1
|
1 |
EC50 = 81 nM
|
|
|
CP0399544
|
5-[[2-[(4-tert-butylbenzoyl)amino]-4-methoxybenzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C27H28N2O5
|
1
|
1 |
EC50 = 87 nM
|
|
|
CP0181580
|
4-tert-butyl-N-[(4-methylsulfanylphenyl)methyl]benzamide
Show/Hide
|
C19H23NOS
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0454801
|
N-[(4-acetylphenyl)methyl]-4-tert-butylbenzamide
Show/Hide
|
C20H23NO2
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0539159
|
5-[[2-[(4-tert-butylbenzoyl)amino]-4-chlorobenzoyl]amino]-2-methylbenzoic acid
Show/Hide
|
C26H25ClN2O4
|
1
|
1 |
EC50 = 110 nM
|
|
|
CP0881990
|
5-(4-methoxyphenyl)-3-o-tolyl-1,2,4-oxadiazole
Show/Hide
|
C16H14N2O2
|
1
|
1 |
EC50 = 120 nM
|
|
|
CP0143436
|
4-tert-butyl-N-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzamide
Show/Hide
|
C19H21N5O
|
1
|
1 |
EC50 = 120 nM
|
|
|
CP0378906
|
N-benzyl-6-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C22H21N3
|
1
|
1 |
EC50 = 130 nM
|
|
|
CP0335294
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-fluorobenzoic acid
Show/Hide
|
C19H20FNO3
|
1
|
1 |
EC50 = 140 nM
|
|
|
CP0546183
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(trifluoromethyl)benzamide
Show/Hide
|
C16H14ClF3N2O3S
|
1
|
1 |
EC50 = 140 nM
|
|
|
CP0398725
|
2-bromo-5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C25H23BrN2O4
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0350531
|
4-tert-butyl-N-[(4-methoxyphenyl)methyl]benzamide
Show/Hide
|
C19H23NO2
|
1
|
1 |
EC50 = 150 nM
|
|
|
CP0049016
|
(4R)-4-[(1S,2S,5R,7S,8R,9R,10S,11S,14R,15R)-8-ethyl-5,9-dihydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-14-yl]pentanoic acid
Show/Hide
|
C26H44O4
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0081889
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-2-methylbenzoic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0143437
|
4-tert-butyl-N-[[4-(trifluoromethoxy)phenyl]methyl]benzamide
Show/Hide
|
C19H20F3NO2
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0335295
|
4-tert-butyl-N-[(4-ethoxyphenyl)methyl]benzamide
Show/Hide
|
C20H25NO2
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0559311
|
N-benzyl-6-chloro-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C18H14ClN3S
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0184079
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-N,N-dimethylbenzamide
Show/Hide
|
C21H26N2O2
|
1
|
1 |
EC50 = 170 nM
|
|
|
CP0365623
|
4-tert-butyl-N-[(4-propan-2-yloxyphenyl)methyl]benzamide
Show/Hide
|
C21H27NO2
|
1
|
1 |
EC50 = 170 nM
|
|
|
CP0407802
|
N-benzyl-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C23H21N3O2
|
1
|
1 |
EC50 = 170 nM
|
|
|
CP0436624
|
N-benzyl-2-(4-fluorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H18FN3
|
1
|
1 |
EC50 = 170 nM
|
|
|
CP0506631
|
N-[(4-methoxyphenyl)methyl]-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H19N3OS
|
1
|
1 |
EC50 = 170 nM
|
|
|
CP0457728
|
N-benzyl-6-methyl-2-(3-methylphenyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C22H21N3
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0533129
|
2-[(4-tert-butylbenzoyl)amino]-N-(3-methylsulfanylphenyl)benzamide
Show/Hide
|
C25H26N2O2S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0539953
|
N-benzyl-6-phenyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C24H19N3S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0474863
|
N-benzyl-6-methyl-2-naphthalen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C25H21N3
|
1
|
1 |
EC50 = 210 nM
|
|
|
CP0866880
|
4-(3-o-tolyl-1,2,4-oxadiazol-5-yl)benzoic acid
Show/Hide
|
C16H12N2O3
|
1
|
1 |
EC50 = 220 nM
|
|
|
CP0378905
|
N-benzyl-6-methyl-2-(4-methyl-1,3-thiazol-2-yl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C19H18N4S
|
1
|
1 |
EC50 = 220 nM
|
|
|
CP0457716
|
6-methyl-N-[(4-methylphenyl)methyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H19N3S
|
1
|
1 |
EC50 = 220 nM
|
|
|
CP0396061
|
2-[(4-tert-butylbenzoyl)amino]-N-(3-cyanophenyl)benzamide
Show/Hide
|
C25H23N3O2
|
1
|
1 |
EC50 = 230 nM
|
|
|
CP0407804
|
6-methyl-N-(3-phenylpropyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H21N3S
|
1
|
1 |
EC50 = 230 nM
|
|
|
CP0407801
|
N-benzyl-2-(4-chlorophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H18ClN3
|
1
|
1 |
EC50 = 240 nM
|
|
|
CP0474861
|
N-benzyl-2-(3-methoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C22H21N3O
|
1
|
1 |
EC50 = 250 nM
|
|
|
CP0553306
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-pyrrolidin-1-ylbenzamide
Show/Hide
|
C19H22ClN3O3S
|
1
|
1 |
EC50 = 250 nM
|
|
|
CP0365731
|
4-tert-butyl-N-[[4-[(2,2,2-trifluoroacetyl)amino]phenyl]methyl]benzamide
Show/Hide
|
C20H21F3N2O2
|
1
|
1 |
EC50 = 260 nM
|
|
|
CP0539023
|
N-benzyl-6-methyl-2-(2-methylphenyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C22H21N3
|
1
|
1 |
EC50 = 260 nM
|
|
|
CP0388902
|
5-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-2-chlorobenzoic acid
Show/Hide
|
C25H23ClN2O4
|
1
|
1 |
EC50 = 280 nM
|
|
|
CP0477280
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]benzoic acid
Show/Hide
|
C25H24N2O4
|
1
|
1 |
EC50 = 280 nM
|
|
|
CP0539082
|
N-benzyl-6-methyl-2-phenylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H19N3
|
1
|
1 |
EC50 = 280 nM
|
|
|
CP0558982
|
N-benzyl-6-methyl-2-(2-phenylethyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C23H23N3
|
1
|
1 |
EC50 = 310 nM
|
|
|
CP0454798
|
4-[[(3,4-dimethylbenzoyl)amino]methyl]benzoic acid
Show/Hide
|
C17H17NO3
|
1
|
1 |
EC50 = 320 nM
|
|
|
CP0539300
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-N-methylbenzamide
Show/Hide
|
C20H24N2O2
|
1
|
1 |
EC50 = 340 nM
|
|
|
CP0919608
|
5-(4-bromophenyl)-3-phenyl-1,2,4-oxadiazole
Show/Hide
|
C14H9BrN2O
|
1
|
1 |
EC50 = 350 nM
|
|
|
CP0184342
|
3-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenyl]propanoic acid
Show/Hide
|
C21H25NO3
|
1
|
1 |
EC50 = 350 nM
|
|
|
CP0083256
|
4-[[(3,4-dimethoxybenzoyl)amino]methyl]benzoic acid
Show/Hide
|
C17H17NO5
|
1
|
1 |
EC50 = 370 nM
|
|
|
CP0143430
|
4-[[(4-tert-butylbenzoyl)amino]methyl]benzoic acid
Show/Hide
|
C19H21NO3
|
1
|
1 |
EC50 = 370 nM
|
|
|
CP0411575
|
2-[(4-tert-butylbenzoyl)amino]-N-(3-methoxyphenyl)benzamide
Show/Hide
|
C25H26N2O3
|
1
|
1 |
EC50 = 380 nM
|
|
|
CP0549530
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-propan-2-yloxybenzamide
Show/Hide
|
C18H21ClN2O4S
|
1
|
1 |
EC50 = 400 nM
|
|
|
CP0866881
|
5-(4-chlorophenyl)-3-p-tolyl-1,2,4-oxadiazole
Show/Hide
|
C15H11ClN2O
|
1
|
1 |
EC50 = 410 nM
|
|
|
CP0575759
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-piperidin-1-ylbenzamide
Show/Hide
|
C20H24ClN3O3S
|
1
|
1 |
EC50 = 410 nM
|
|
|
CP0419731
|
2-[3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
|
C26H26N2O4
|
1
|
1 |
EC50 = 420 nM
|
|
|
CP0546180
|
4-tert-butyl-N-[[2-chloro-4-(propan-2-ylsulfonylamino)phenyl]methyl]benzamide
Show/Hide
|
C21H27ClN2O3S
|
1
|
1 |
EC50 = 420 nM
|
|
|
CP0408117
|
N-benzyl-2-(4-bromophenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C21H18BrN3
|
1
|
1 |
EC50 = 430 nM
|
|
|
CP0083255
|
4-[[(4-phenylbenzoyl)amino]methyl]benzoic acid
Show/Hide
|
C21H17NO3
|
1
|
1 |
EC50 = 440 nM
|
|
|
CP0810328
|
7-(diethylamino)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-2H-chromen-2-one
Show/Hide
|
C21H19N3O3
|
1
|
1 |
EC50 = 460 nM
|
|
|
CP0559310
|
N-benzyl-2-thiophen-2-yl-6-(trifluoromethyl)imidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C19H14F3N3S
|
1
|
1 |
EC50 = 460 nM
|
|
|
CP0379833
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-fluorobenzoic acid
Show/Hide
|
C25H23FN2O4
|
1
|
1 |
EC50 = 480 nM
|
|
|
CP0456564
|
N-(3-acetylphenyl)-2-[(4-tert-butylbenzoyl)amino]benzamide
Show/Hide
|
C26H26N2O3
|
1
|
1 |
EC50 = 480 nM
|
|
|
CP0548715
|
N-benzyl-6-bromo-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C18H14BrN3S
|
1
|
1 |
EC50 = 500 nM
|
|
|
CP0284282
|
4-tert-butyl-N-[[2-chloro-4-(ethylsulfonylamino)phenyl]methyl]benzamide
Show/Hide
|
C20H25ClN2O3S
|
1
|
1 |
EC50 = 500 nM
|
|
|
CP0089615
|
3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(1-methylethyl)isoxazol-4-yl]methoxy}phenyl)ethenyl]benzoic acid
Show/Hide
|
C28H22Cl3NO4
|
1
|
1 |
EC50 = 510 nM
|
|
|
CP0394344
|
N-benzyl-6-methyl-2-pyridin-3-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
|
C20H18N4
|
1
|
1 |
EC50 = 520 nM
|
|
|
CP0849175
|
3,5-diphenyl-1,2,4-oxadiazole
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C14H10N2O
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1
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1 |
EC50 = 530 nM
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CP0407805
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N-benzyl-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C19H17N3S
|
1
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1 |
EC50 = 540 nM
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CP0549525
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-[1-(trifluoromethyl)cyclopropyl]benzamide
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C19H18ClF3N2O3S
|
1
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1 |
EC50 = 540 nM
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CP0558983
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N-benzyl-2-(furan-2-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
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C19H17N3O
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1
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1 |
EC50 = 560 nM
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CP0492060
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4-(1-bicyclo[1.1.1]pentanyl)-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
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C20H21ClN2O3S
|
1
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1 |
EC50 = 560 nM
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CP0196829
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4-[[(3-phenylbenzoyl)amino]methyl]benzoic acid
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C21H17NO3
|
1
|
1 |
EC50 = 670 nM
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CP0387204
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2-[3-[[2-[(4-phenylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
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C28H22N2O4
|
1
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1 |
EC50 = 700 nM
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CP0572339
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4-[[2-[[(E)-3-phenylprop-2-enoyl]amino]benzoyl]amino]butanoic acid
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C20H20N2O4
|
1
|
1 |
EC50 = 720 nM
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CP0454799
|
2-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenoxy]acetic acid
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C20H23NO4
|
1
|
1 |
EC50 = 730 nM
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CP0407803
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7-methyl-N-(4-phenylbutyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C22H23N3S
|
1
|
1 |
EC50 = 750 nM
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CP0506632
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3-benzyl-6-methyl-2-thiophen-2-ylimidazo[1,2-a]pyridine
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C19H16N2S
|
1
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1 |
EC50 = 810 nM
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CP0394340
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N-benzyl-6-methyl-2-thiophen-3-ylimidazo[1,2-a]pyridin-3-amine
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C19H17N3S
|
1
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1 |
EC50 = 830 nM
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CP0535248
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N-benzyl-6-methoxy-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C19H17N3OS
|
1
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1 |
EC50 = 830 nM
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CP0436626
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N-benzyl-2-(3,4-dimethoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
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C23H23N3O2
|
1
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1 |
EC50 = 910 nM
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CP0303425
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4-tert-butyl-N-[(2-fluoro-4-sulfamoylphenyl)methyl]benzamide
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C18H21FN2O3S
|
1
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1 |
EC50 = 970 nM
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CP0403496
|
4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
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C25H18N2O4
|
1
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1 |
EC50 = 1000 nM
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CP0539952
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6-methyl-N-(2-phenylethyl)-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C20H19N3S
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1
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1 |
EC50 = 1000 nM
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CP0546181
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(trifluoromethoxy)benzamide
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C16H14ClF3N2O4S
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1
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1 |
EC50 = 1090 nM
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CP0396059
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3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-chlorobenzoic acid
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C25H23ClN2O4
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1
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1 |
EC50 = 1100 nM
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CP0408119
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N-benzyl-6-methyl-2-(1-methylpyrrol-2-yl)imidazo[1,2-a]pyridin-3-amine
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C20H20N4
|
1
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1 |
EC50 = 1100 nM
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CP0474862
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N-benzyl-6-methyl-2-[(E)-2-phenylethenyl]imidazo[1,2-a]pyridin-3-amine
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C23H21N3
|
1
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1 |
EC50 = 1160 nM
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CP0184169
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4-[[(4-tert-butyl-3-methoxybenzoyl)amino]methyl]benzoic acid
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C20H23NO4
|
1
|
1 |
EC50 = 1200 nM
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CP0394343
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N-benzyl-7-ethyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C20H19N3S
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1
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1 |
EC50 = 1200 nM
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CP0436628
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N-benzyl-6-methyl-2-pyrazin-2-ylimidazo[1,2-a]pyridin-3-amine
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C19H17N5
|
1
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1 |
EC50 = 1200 nM
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CP0575253
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(1,1-difluoroethyl)benzamide
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C17H17ClF2N2O3S
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1
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1 |
EC50 = 1200 nM
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CP0541210
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N-benzyl-2-(4-methoxyphenyl)-6-methylimidazo[1,2-a]pyridin-3-amine
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C22H21N3O
|
1
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1 |
EC50 = 1270 nM
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CP0417144
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4-[[[2-(naphthalene-2-carbonylamino)benzoyl]amino]methyl]benzoic acid
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C26H20N2O4
|
1
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1 |
EC50 = 1300 nM
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CP0329861
|
4-tert-butyl-N-[(4-methylsulfinylphenyl)methyl]benzamide
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C19H23NO2S
|
1
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1 |
EC50 = 1300 nM
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CP0539950
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6-methyl-N-[(1S)-1-phenylethyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
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C20H19N3S
|
1
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1 |
EC50 = 1300 nM
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CP0451683
|
4-[(naphthalene-2-carbonylamino)methyl]benzoic acid
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C19H15NO3
|
1
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1 |
EC50 = 1360 nM
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CP0081661
|
4-(4-tert-Butylphenylcarboxamidomethyl)benzenesulfonamide
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C18H22N2O3S
|
1
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1 |
EC50 = 1400 nM
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CP0496466
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(dimethylamino)benzamide
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C17H20ClN3O3S
|
1
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1 |
EC50 = 1460 nM
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CP0387227
|
3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]benzoic acid
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C25H18N2O4
|
1
|
1 |
EC50 = 1500 nM
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CP0575254
|
4-tert-butyl-N-[[2-chloro-4-(cyclopropylsulfonylamino)phenyl]methyl]benzamide
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C21H25ClN2O3S
|
1
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1 |
EC50 = 1500 nM
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CP0303426
|
3-[[(4-tert-butylbenzoyl)amino]methyl]benzoic acid
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C19H21NO3
|
1
|
1 |
EC50 = 1700 nM
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CP0436623
|
N-benzyl-2-(furan-3-yl)-6-methylimidazo[1,2-a]pyridin-3-amine
Show/Hide
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C19H17N3O
|
1
|
1 |
EC50 = 1900 nM
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CP0408115
|
N-benzyl-6-methyl-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
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C20H18N4
|
1
|
1 |
EC50 = 2000 nM
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CP0396063
|
3-[[4-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
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C22H14ClF3N2O4
|
1
|
1 |
EC50 = 2100 nM
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CP0500157
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-ethoxybenzamide
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C17H19ClN2O4S
|
1
|
1 |
EC50 = 2200 nM
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CP0398732
|
3-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]propanoic acid
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C24H19F3N2O4
|
1
|
1 |
EC50 = 2300 nM
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CP0387071
|
4-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]butanoic acid
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C22H26N2O4
|
1
|
1 |
EC50 = 2500 nM
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CP0387205
|
2-[3-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]phenyl]acetic acid
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C26H20N2O4
|
1
|
1 |
EC50 = 2500 nM
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CP0445061
|
2-[3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
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|
C23H17F3N2O4
|
1
|
1 |
EC50 = 2600 nM
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CP0399541
|
2-[(4-tert-butylbenzoyl)amino]-N-[3-(2H-tetrazol-5-yl)phenyl]benzamide
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C25H24N6O2
|
1
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1 |
EC50 = 2900 nM
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CP0886015
|
5-(4-methoxyphenyl)-3-(3-(trifluoromethyl)phenyl)-1,2,4-oxadiazole
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C16H11F3N2O2
|
1
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1 |
EC50 = 2900 nM
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CP0331663
|
N-[(4-acetamidophenyl)methyl]-4-tert-butylbenzamide
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C20H24N2O2
|
1
|
1 |
EC50 = 2900 nM
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CP0403497
|
2-[4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]phenyl]acetic acid
Show/Hide
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C26H20N2O4
|
1
|
1 |
EC50 = 3100 nM
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CP0541211
|
6-methyl-N-[(1R)-1-phenylethyl]-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
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C20H19N3S
|
1
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1 |
EC50 = 3200 nM
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CP0267212
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(1,1,2,2,2-pentafluoroethyl)benzamide
Show/Hide
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C17H14ClF5N2O3S
|
1
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1 |
EC50 = 3220 nM
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CP0388903
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3-[[5-chloro-2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
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C22H14ClF3N2O4
|
1
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1 |
EC50 = 3400 nM
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CP0387232
|
3-[[2-[(4-bromobenzoyl)amino]benzoyl]amino]benzoic acid
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C21H15BrN2O4
|
1
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1 |
EC50 = 3700 nM
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CP0327641
|
4-[(4-tert-butylphenyl)carbamoylamino]benzoic acid
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C18H20N2O3
|
1
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1 |
EC50 = 3800 nM
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CP0393975
|
4-[[(4-tert-butylbenzoyl)amino]methyl]benzamide
Show/Hide
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C19H22N2O2
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1
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1 |
EC50 = 3800 nM
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CP0413032
|
4-tert-butyl-N-[(4-methylsulfonylphenyl)methyl]benzamide
Show/Hide
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C19H23NO3S
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1
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1 |
EC50 = 3800 nM
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CP0509519
|
N-benzyl-2-thiophen-2-ylimidazo[1,2-a]pyridin-3-amine
Show/Hide
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C18H15N3S
|
1
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1 |
EC50 = 4000 nM
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CP0546185
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N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-(2,2,2-trifluoroethyl)benzamide
Show/Hide
|
C17H16ClF3N2O3S
|
1
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1 |
EC50 = 4000 nM
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CP0380161
|
6-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]hexanoic acid
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C24H24N2O4
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1
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1 |
EC50 = 4400 nM
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CP0546184
|
N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]-4-morpholin-4-ylbenzamide
Show/Hide
|
C19H22ClN3O4S
|
1
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1 |
EC50 = 4400 nM
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CP0379832
|
3-[[2-[(4-tert-butylbenzoyl)amino]benzoyl]amino]-4-methoxybenzoic acid
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|
C26H26N2O5
|
1
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1 |
EC50 = 4700 nM
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CP0509140
|
3-[[2-(2,3-dihydro-1,4-benzodioxine-6-carbonylamino)benzoyl]amino]benzoic acid
Show/Hide
|
C23H18N2O6
|
1
|
1 |
EC50 = 4900 nM
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CP0387068
|
3-[[2-[[3-fluoro-4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
|
C22H14F4N2O4
|
1
|
1 |
EC50 = 5000 nM
|
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CP0509141
|
3-[[2-[[(E)-3-phenylprop-2-enoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
|
C23H18N2O4
|
1
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1 |
EC50 = 5200 nM
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CP0454800
|
4-tert-butyl-N-[(4-formylphenyl)methyl]benzamide
Show/Hide
|
C19H21NO2
|
1
|
1 |
EC50 = 5300 nM
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CP0387228
|
4-[[2-[(4-ethylbenzoyl)amino]benzoyl]amino]butanoic acid
Show/Hide
|
C20H22N2O4
|
1
|
1 |
EC50 = 5800 nM
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CP0413031
|
2-[4-[[(4-tert-butylbenzoyl)amino]methyl]phenyl]acetic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
EC50 = 6400 nM
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CP0387067
|
3-[[2-[[4-(trifluoromethyl)benzoyl]amino]benzoyl]amino]benzoic acid
Show/Hide
|
C22H15F3N2O4
|
1
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1 |
EC50 = 6900 nM
|
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CP0396062
|
2-[3-[[2-[[4-(trifluoromethylsulfanyl)benzoyl]amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
|
C23H17F3N2O4S
|
1
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1 |
EC50 = 7000 nM
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CP0492702
|
methyl 4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]butanoate
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|
C23H22N2O4
|
1
|
1 |
EC50 = 7100 nM
|
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CP0184078
|
4-[[(4-tert-butylbenzoyl)amino]methyl]-3-chlorobenzoic acid
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|
C19H20ClNO3
|
1
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1 |
EC50 = 7500 nM
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CP0403351
|
5-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]pentanoic acid
Show/Hide
|
C23H22N2O4
|
1
|
1 |
EC50 = 8300 nM
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CP0387203
|
2-[3-[[2-[(4-methylsulfanylbenzoyl)amino]benzoyl]amino]phenyl]acetic acid
Show/Hide
|
C23H20N2O4S
|
1
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1 |
EC50 = 8500 nM
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CP0385188
|
4-[[2-(naphthalene-2-carbonylamino)benzoyl]amino]butanoic acid
Show/Hide
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C22H20N2O4
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2
|
1 |
EC50 = 8550 nM
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2 |
EC50 = 8600 nM
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CP0398523
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3-[[2-(1,3-benzodioxole-5-carbonylamino)benzoyl]amino]benzoic acid
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|
C22H16N2O6
|
1
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1 |
EC50 = 10000 nM
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CP0571435
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4-(azetidin-1-yl)-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
Show/Hide
|
C18H20ClN3O3S
|
1
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1 |
EC50 = 13000 nM
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CP0002372
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(4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R)-5,9-dihydroxy-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadecan-14-yl]pentanoic acid
Show/Hide
|
C24H40O4
|
1
|
1 |
EC50 = 18000 nM
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CP0392557
|
2-[4-[(4-tert-butyl-2-methoxybenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C20H23NO4
|
2
|
1 |
IC50 = 1.3 nM
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2 |
IC50 = 9.2 nM
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CP0565305
|
2-[4-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C19H21NO3
|
1
|
1 |
IC50 = 76 nM
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CP0396569
|
2-[4-[(4-tert-butylbenzoyl)amino]-2-methylphenyl]acetic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
IC50 = 80 nM
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CP0513309
|
2-[2-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C19H21NO3
|
1
|
1 |
IC50 = 102 nM
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CP0429349
|
2-[4-[(4-tert-butyl-2-hydroxybenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C19H21NO4
|
1
|
1 |
IC50 = 140 nM
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CP0548250
|
2-[4-[(2-methoxy-5-phenylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C22H19NO4
|
1
|
1 |
IC50 = 170 nM
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CP0462122
|
2-[4-[(3-tert-butylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C19H21NO3
|
1
|
1 |
IC50 = 190 nM
|
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CP0467757
|
2-[4-[(4-tert-butyl-3-methoxybenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C20H23NO4
|
1
|
1 |
IC50 = 220 nM
|
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CP0411732
|
2-[4-[(3-phenylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C21H17NO3
|
1
|
1 |
IC50 = 280 nM
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CP0487623
|
2-[3-[(4-tert-butylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C19H21NO3
|
2
|
1 |
IC50 = 350 nM
|
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|
2 |
IC50 = 400 nM
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CP0532536
|
3-[4-[(4-tert-butylbenzoyl)amino]phenyl]propanoic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
IC50 = 630 nM
|
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CP0429350
|
2-[4-(naphthalene-2-carbonylamino)phenyl]acetic acid
Show/Hide
|
C19H15NO3
|
1
|
1 |
IC50 = 680 nM
|
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CP0396571
|
4-[4-[(4-tert-butylbenzoyl)amino]phenyl]butanoic acid
Show/Hide
|
C21H25NO3
|
1
|
1 |
IC50 = 700 nM
|
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CP0549065
|
2-[4-(naphthalene-1-carbonylamino)phenyl]acetic acid
Show/Hide
|
C19H15NO3
|
1
|
1 |
IC50 = 810 nM
|
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CP0487621
|
2-[4-[(4-phenylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C21H17NO3
|
1
|
1 |
IC50 = 850 nM
|
|
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CP0462123
|
2-[4-[(4-tert-butylbenzoyl)amino]phenyl]propanoic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
IC50 = 970 nM
|
|
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CP0396568
|
2-[4-[(4-tert-butylbenzoyl)amino]-3-methylphenyl]acetic acid
Show/Hide
|
C20H23NO3
|
1
|
1 |
IC50 = 1500 nM
|
|
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CP0487622
|
2-[4-[benzyl-(4-tert-butylbenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C26H27NO3
|
1
|
1 |
IC50 = 2200 nM
|
|
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CP0429348
|
2-[4-[(3-tert-butyl-2-methoxybenzoyl)amino]phenyl]acetic acid
Show/Hide
|
C20H23NO4
|
1
|
1 |
IC50 = 3300 nM
|
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CP0486448
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2-[4-[(4-tert-butylbenzoyl)amino]-2-methoxyphenyl]acetic acid
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C20H23NO4
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1
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1 |
IC50 = 3700 nM
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CP0559369
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2-[4-[(2-methoxy-3-phenylbenzoyl)amino]phenyl]acetic acid
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C22H19NO4
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1
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1 |
IC50 = 5000 nM
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CP0389938
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2-[4-[(4-tert-butylbenzoyl)-methylamino]phenyl]acetic acid
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C20H23NO3
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1
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1 |
IC50 = 8100 nM
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CP0486449
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2-[4-[[3-(3,5-dichlorophenyl)benzoyl]amino]phenyl]acetic acid
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C21H15Cl2NO3
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1
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1 |
IC50 = 9100 nM
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CP0379835
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3-[[2-[(4-tert-butylbenzoyl)amino]-5-chlorobenzoyl]amino]benzoic acid
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C25H23ClN2O4
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1
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1 |
IC50 = 12300 nM
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CP0398526
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3-[[2-[(4-tert-butylbenzoyl)amino]-5-methoxybenzoyl]amino]benzoic acid
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C26H26N2O5
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1
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1 |
IC50 = 15100 nM
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CP0942600
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5-(4-methoxyphenyl)-3-phenyl-1,2,4-oxadiazole
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C15H12N2O2
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1
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1 |
IC50 = 16400 nM
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CP0392558
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2-[4-[(2-naphthalen-2-ylacetyl)amino]phenyl]acetic acid
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C20H17NO3
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1
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1 |
IC50 = 27000 nM
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