| Compound ID |
Compound Name |
Compound Formula |
|
CP0006058
|
2-amino-N-[(1S)-1-[8-[2-(1-methylpyrazol-4-yl)ethynyl]-1-oxo-2-phenylisoquinolin-3-yl]ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
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|
C30H24N8O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0019791
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-(methanesulfonamido)-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C20H24N4O4S2
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0019793
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-(methylsulfamoyl)-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C20H24N4O4S2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0012179
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-methyl-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C20H23N3O2S
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0024001
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-(2-methoxyethylsulfonylamino)-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C22H28N4O5S2
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0031524
|
N-[5-[7-chloro-2-[(1S)-1-cyclopropylethyl]-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C19H20ClN3O2S
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0017013
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-methylsulfonyl-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C20H23N3O4S2
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0017098
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-1-oxo-7-sulfamoyl-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C19H22N4O4S2
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0019794
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-(2-methoxyethylsulfamoyl)-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C22H28N4O5S2
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0353655
|
4-amino-6-[[(1S)-1-(6-methyl-4-oxo-3-phenylquinolizin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile
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|
C23H20N6O
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0017012
|
N-[5-[7-chloro-2-[(1S)-1-cyclopropylethyl]-1-oxo-3H-isoindol-5-yl]-1,3-thiazol-2-yl]acetamide
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|
C18H18ClN3O2S
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0026318
|
5-chloro-3-phenyl-2-[(1S)-1-(7H-purin-6-ylamino)ethyl]quinazolin-4-one
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|
C21H16ClN7O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0024003
|
N-[5-[7-chloro-2-[(1R)-1-cyclopropylethyl]-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0077387
|
N-[4-methyl-5-(2-pyridin-3-yl-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
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|
C14H12N4O2S
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0136524
|
2,4-diamino-6-[[(1S)-1-(7-fluoro-4-oxo-3-phenylquinolizin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile
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|
C22H18FN7O
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0276259
|
N-[4-methyl-5-[2-(2,2,2-trifluoroethyl)-1,3-oxazol-5-yl]-1,3-thiazol-2-yl]acetamide
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|
C11H10F3N3O2S
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0219705
|
2-amino-4-[[(1S)-1-[7-fluoro-1-(4-fluorophenyl)-4-oxo-3-phenylquinolizin-2-yl]ethyl]amino]-6-methylpyrimidine-5-carbonitrile
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|
C29H22F2N6O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0077385
|
N-[5-(2-tert-butyl-1,3-oxazol-5-yl)-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C13H17N3O2S
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0252714
|
N-[5-[3-(3-hydroxy-2,2-dimethylbutyl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C14H20N4O3S
|
1
|
| 1 |
IC50 = 155 nM
|
|
|
|
CP0176936
|
2,4-diamino-6-[[(1S)-1-[7-fluoro-1-(4-fluorophenyl)-4-oxo-3-phenylquinolizin-2-yl]ethyl]amino]pyrimidine-5-carbonitrile
Show/Hide
|
C28H21F2N7O
|
1
|
| 1 |
IC50 = 177 nM
|
|
|
|
CP0134073
|
N-[5-[3-(3-hydroxy-2,2-dimethylpropyl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C13H18N4O3S
|
1
|
| 1 |
IC50 = 191 nM
|
|
|
|
CP0224694
|
N-[4-methyl-5-(2-methylsulfonyl-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
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|
C10H11N3O4S2
|
1
|
| 1 |
IC50 = 222 nM
|
|
|
|
CP0134074
|
N-[5-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C12H16N4O2S
|
1
|
| 1 |
IC50 = 231 nM
|
|
|
|
CP0224695
|
N-[5-[2-(3-hydroxypiperidin-1-yl)-1,3-oxazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H18N4O3S
|
1
|
| 1 |
IC50 = 237 nM
|
|
|
|
CP0019790
|
N-[5-[2-[(1S)-1-cyclopropylethyl]-7-(3-hydroxypropylsulfonyl)-1-oxo-3H-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C22H27N3O5S2
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0262745
|
N-[4-methyl-5-[3-(2,2,2-trifluoroethyl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C10H9F3N4O2S
|
1
|
| 1 |
IC50 = 278 nM
|
|
|
|
CP0245832
|
N-[4-methyl-5-(2-pyridin-3-ylsulfanyl-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
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|
C14H12N4O2S2
|
1
|
| 1 |
IC50 = 279 nM
|
|
|
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CP0067381
|
N-[5-[3-(3-hydroxypiperidin-1-yl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C13H17N5O3S
|
1
|
| 1 |
IC50 = 294 nM
|
|
|
|
CP0122221
|
N-[4-methyl-5-(2-methylsulfanyl-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C10H11N3O2S2
|
1
|
| 1 |
IC50 = 322 nM
|
|
|
|
CP0245831
|
N-[5-[2-(2-hydroxypropan-2-yl)-1,3-oxazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C12H15N3O3S
|
1
|
| 1 |
IC50 = 369 nM
|
|
|
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CP0016620
|
3-amino-6-[2-[(1S)-1-cyclopropylethyl]-7-methyl-1-oxo-3H-isoindol-5-yl]-N-methylpyrazine-2-carboxamide
Show/Hide
|
C20H23N5O2
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0017099
|
2-[(1S)-1-cyclopropylethyl]-7-methyl-5-(5H-pyrrolo[2,3-b]pyrazin-2-yl)-3H-isoindol-1-one
Show/Hide
|
C20H20N4O
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0122220
|
N-[4-methyl-5-[2-(pyridin-3-ylamino)-1,3-oxazol-5-yl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H13N5O2S
|
1
|
| 1 |
IC50 = 431 nM
|
|
|
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CP0252713
|
N-[4-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C12H14N4O3S
|
1
|
| 1 |
IC50 = 558 nM
|
|
|
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CP0284911
|
N-[4-methyl-5-(2-morpholin-4-yl-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C13H16N4O3S
|
1
|
| 1 |
IC50 = 599 nM
|
|
|
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CP0024002
|
5-(2-aminopyrimidin-5-yl)-7-chloro-2-[(1S)-1-cyclopropylethyl]-3H-isoindol-1-one
Show/Hide
|
C17H17ClN4O
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
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CP0057640
|
N-[5-[2-[(6-chloropyridin-3-yl)amino]-1,3-oxazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H12ClN5O2S
|
1
|
| 1 |
IC50 = 1040 nM
|
|
|
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CP0316180
|
N-[5-[2-(dimethylamino)-1,3-oxazol-5-yl]-4-methyl-1,3-thiazol-2-yl]acetamide
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|
C11H14N4O2S
|
1
|
| 1 |
IC50 = 1222 nM
|
|
|
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CP0473312
|
7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino)-9-(tetrahydro-2H-pyran-4-yl)-7,9-dihydro-8H-purin-8-one
Show/Hide
|
C18H20N8O2
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
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CP0077388
|
N-[4-methyl-5-(2-pyridin-3-yloxy-1,3-oxazol-5-yl)-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C14H12N4O3S
|
1
|
| 1 |
IC50 = 1666 nM
|
|
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CP0030807
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3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-amine
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
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CP0029667
|
5-(3-aminopyrazin-2-yl)-2-[(1S)-1-cyclopropylethyl]-7-methyl-3H-isoindol-1-one
Show/Hide
|
C18H20N4O
|
1
|
| 1 |
IC50 = 7943.28 nM
|
|
|
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CP0221106
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3-[[5-(2-acetamido-4-methyl-1,3-thiazol-5-yl)-1,3-oxazol-2-yl]amino]benzoic acid
Show/Hide
|
C16H14N4O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0335247
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3-[[5-(2-acetamido-4-methyl-1,3-thiazol-5-yl)-1,3-oxazol-2-yl]methyl]benzoic acid
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|
C17H15N3O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0016012
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4-[3-amino-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]-N,N-dimethylpyrazole-1-sulfonamide
Show/Hide
|
C21H23N9O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0033023
|
N-[4-methyl-5-(7-methyl-1-oxo-2,3-dihydroisoindol-5-yl)-1,3-thiazol-2-yl]acetamide
Show/Hide
|
C15H15N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0702721
|
(S)-2-(1-((9H-Purin-6-yl)amino)ethyl)-7-fluoro-3-phenyl-4H-quinolizin-4-one
Show/Hide
|
C22H17FN6O
|
1
|
| 1 |
IC50 > 3000 nM
|
|
|
