| Compound ID |
Compound Name |
Compound Formula |
|
CP0082712
|
4-Guanidino-benzoic acid 6-carbamimidoyl-naphthalen-2-yl ester
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|
C19H17N5O2
|
2
|
| 1 |
IC50 = 150 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0504742
|
(2-chloro-4-nitrophenyl) 4-(diaminomethylideneamino)benzoate
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|
C14H11ClN4O4
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0488678
|
methyl 6-[4-(diaminomethylideneamino)benzoyl]oxynaphthalene-2-carboxylate
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|
C20H17N3O4
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0040568
|
(4-nitrophenyl) 4-(diaminomethylideneamino)benzoate
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|
C14H12N4O4
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0078932
|
(4-methoxycarbonylphenyl) 4-(diaminomethylideneamino)benzoate
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|
C16H15N3O4
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0535287
|
(3-nitrophenyl) 4-(diaminomethylideneamino)benzoate
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|
C14H12N4O4
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0504743
|
(4-carbamoylphenyl) 4-(diaminomethylideneamino)benzoate
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|
C15H14N4O3
|
1
|
| 1 |
IC50 = 6800 nM
|
|
|
|
CP0234575
|
US9199927, camostat
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|
C20H22N4O5
|
1
|
| 1 |
IC50 = 32000 nM
|
|
|
|
CP0522205
|
methyl 6-[[4-(diaminomethylideneamino)phenyl]sulfonylamino]naphthalene-2-carboxylate
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|
C19H18N4O4S
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0523213
|
4-(diaminomethylideneamino)-N-phenylbenzamide
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|
C14H14N4O
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0530930
|
N-[4-(diaminomethylideneamino)phenyl]benzamide
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|
C14H14N4O
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0535286
|
2-[4-[(4-methylphenyl)sulfonylamino]phenyl]guanidine
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|
C14H16N4O2S
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0116398
|
3-[(2S)-3-oxo-3-[4-(piperidin-4-ylcarbonyl)piperazin-1-yl]-2-{[2,4,6-tris(propan-2-yl)benzene]sulfonamido}propyl]benzene-1-carboximidamide
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|
C35H52N6O4S
|
1
|
| 1 |
Ki = 5500 nM
|
|
|
|
CP0152554
|
2-(4-carbamimidoylanilino)-2-(7-ethyl-3-methyl-1-benzofuran-5-yl)-N-(1-methylimidazol-4-yl)sulfonylacetamide
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|
C24H26N6O4S
|
1
|
| 1 |
Ki = 7100 nM
|
|
|
|
CP0206875
|
3-[(2S)-2-(naphthalen-2-ylsulfonylamino)-3-oxo-3-(4-phenylpiperidin-1-yl)propyl]benzenecarboximidamide
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|
C31H32N4O3S
|
1
|
| 1 |
Ki = 10100 nM
|
|
|
|
CP0089706
|
N-benzyl-4-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]piperazine-1-carboxamide
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|
C32H34N6O4S
|
1
|
| 1 |
Ki = 14000 nM
|
|
|
|
CP0294929
|
N-[(4-bromophenyl)methyl]-4-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]piperazine-1-carboxamide
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|
C32H33BrN6O4S
|
1
|
| 1 |
Ki = 16200 nM
|
|
|
|
CP0186442
|
3-amidinophenylalanine deriv., 31
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|
C36H54N8O4S
|
1
|
| 1 |
Ki = 17000 nM
|
|
|
|
CP0185167
|
3-[(2S)-2-(naphthalen-2-ylsulfonylamino)-3-oxo-3-(4-phenylpiperazin-1-yl)propyl]benzenecarboximidamide
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|
C30H31N5O3S
|
1
|
| 1 |
Ki = 18200 nM
|
|
|
|
CP0116396
|
3-[(2S)-2-[(4-methylphenyl)sulfonylamino]-3-oxo-3-(4-phenylpiperidin-1-yl)propyl]benzenecarboximidamide
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|
C28H32N4O3S
|
1
|
| 1 |
Ki = 20000 nM
|
|
|
|
CP0206877
|
3-[(2S)-3-oxo-3-(4-phenylpiperazin-1-yl)-2-[[2,4,6-tri(propan-2-yl)phenyl]sulfonylamino]propyl]benzenecarboximidamide
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|
C35H47N5O3S
|
1
|
| 1 |
Ki = 22200 nM
|
|
|
|
CP0052965
|
benzyl 4-[(2S)-3-(3-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]propanoyl]piperazine-1-carboxylate
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|
C29H33N5O5S
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0052968
|
4-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]-N-hexylpiperazine-1-carboxamide
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|
C31H40N6O4S
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0152549
|
benzyl N-[(3R)-1-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]piperidin-3-yl]carbamate
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|
C33H35N5O5S
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0206874
|
3-[(2S)-3-[4-(1-benzothiophene-3-carbonyl)piperazin-1-yl]-2-(naphthalen-2-ylsulfonylamino)-3-oxopropyl]benzenecarboximidamide
Show/Hide
|
C33H31N5O4S2
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0334636
|
benzyl N-[(3S)-1-[(2S)-3-(3-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]propanoyl]piperidin-3-yl]carbamate
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|
C30H35N5O5S
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0347539
|
4-[(2S)-3-(3-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]propanoyl]-N-(2-phenylethyl)piperazine-1-carboxamide
Show/Hide
|
C30H36N6O4S
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
