| Compound ID |
Compound Name |
Compound Formula |
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CP0458164
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2-[[3-(4-cyanophenyl)-10-hydroxy-12-oxo-7-(trifluoromethoxy)-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carbonyl]amino]acetic acid
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|
C22H14F3N3O7
|
1
|
| 1 |
IC50 = 5.1 nM
|
|
|
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CP0437857
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2-[[4-hydroxy-2-oxo-1-[[4-(trifluoromethoxy)phenyl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C18H15F3N2O7
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
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CP0517636
|
2-[[4-hydroxy-2-oxo-1-[(1-phenylpyrazol-3-yl)methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C20H18N4O6
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
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CP0439910
|
2-[[4-hydroxy-2-oxo-1-[[2-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C15H12F3N3O6S
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
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CP0521144
|
2-[[1-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C17H15ClN2O6
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
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CP0426003
|
2-[[4-hydroxy-2-oxo-1-[(2,4,5-trifluorophenyl)methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C17H13F3N2O6
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
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CP0533783
|
2-[[1-(1,3-benzoxazol-2-ylmethyl)-4-hydroxy-2-oxo-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C18H15N3O7
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0533798
|
2-[[10-hydroxy-12-oxo-3-[6-(trifluoromethyl)pyridin-3-yl]-1,4-diazatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carbonyl]amino]acetic acid
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|
C20H15F3N4O5
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
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CP0492051
|
2-[[4-hydroxy-2-oxo-1-[[4-(trifluoromethyl)-1,3-thiazol-2-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C15H12F3N3O6S
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
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CP0142820
|
2-[[4-hydroxy-2-oxo-1-[[4-(trifluoromethyl)phenyl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C18H15F3N2O6
|
1
|
| 1 |
IC50 = 8.2 nM
|
|
|
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CP0434449
|
2-[[1-[(2,4-difluorophenyl)methyl]-4-hydroxy-2-oxo-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C17H14F2N2O6
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0559017
|
2-[[10-hydroxy-12-oxo-2-[6-(trifluoromethyl)pyridin-3-yl]-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carbonyl]amino]acetic acid
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|
C20H14F3N3O6
|
1
|
| 1 |
IC50 = 8.9 nM
|
|
|
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CP0426000
|
2-[[4-hydroxy-2-oxo-1-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C17H14F3N3O6
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0426002
|
2-[[4-hydroxy-2-oxo-1-[[5-(trifluoromethyl)pyrazin-2-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C16H13F3N4O6
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0470792
|
2-[[10-hydroxy-12-oxo-3-[4-(trifluoromethyl)phenyl]-4-thia-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carbonyl]amino]acetic acid
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|
C21H15F3N2O5S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0458167
|
2-[[1-(1,3-benzothiazol-2-ylmethyl)-4-hydroxy-2-oxo-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonyl]amino]acetic acid
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|
C19H17N3O6S
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
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CP0136665
|
N-[bis(4-methoxyphenyl)methyl]-6-oxo-2-pyridazin-3-yl-1H-pyrimidine-5-carboxamide
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|
C24H21N5O4
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
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CP0470796
|
2-[[7-chloro-4-hydroxy-2-oxo-1-[[4-(trifluoromethyl)phenyl]methyl]quinoline-3-carbonyl]amino]acetic acid
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|
C20H14ClF3N2O5
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
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CP0519246
|
2-[[4-hydroxy-1-[[4-(2-hydroxypropan-2-yl)phenyl]methyl]-2-oxo-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C20H22N2O7
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
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CP0426423
|
2-[[4-hydroxy-2-oxo-1-[[2-(trifluoromethyl)pyrimidin-5-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C16H13F3N4O6
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
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CP0533799
|
2-[[1-[(4-cyano-2-fluorophenyl)methyl]-4-hydroxy-2-oxo-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonyl]amino]acetic acid
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|
C19H16FN3O6
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
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CP0425999
|
2-[[10-hydroxy-2-(4-methoxyphenyl)-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13),10-tetraene-11-carbonyl]amino]acetic acid
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|
C21H18N2O7
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
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CP0426422
|
2-[[4-hydroxy-2-oxo-1-[[5-(trifluoromethyl)pyrimidin-2-yl]methyl]-5,7-dihydrofuro[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C16H13F3N4O6
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
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CP0533800
|
2-[[1-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonyl]amino]acetic acid
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|
C18H17ClN2O6
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
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CP0437858
|
2-[[4-hydroxy-2-oxo-1-[[4-(trifluoromethyl)phenyl]methyl]-6,8-dihydro-5H-pyrano[3,4-b]pyridine-3-carbonyl]amino]acetic acid
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|
C19H17F3N2O6
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
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CP0492050
|
2-[[4-hydroxy-2-oxo-1-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonyl]amino]acetic acid
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|
C18H16F3N3O6
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
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CP0492049
|
2-[[4-hydroxy-2-oxo-1-[[4-(trifluoromethyl)phenyl]methyl]-7,8-dihydro-5H-pyrano[4,3-b]pyridine-3-carbonyl]amino]acetic acid
Show/Hide
|
C19H17F3N2O6
|
1
|
| 1 |
IC50 = 51 nM
|
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