| Compound ID |
Compound Name |
Compound Formula |
|
CP0634033
|
2-(3-acetamido-4-chlorophenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C21H18ClF3N6O2S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0636016
|
2-(3-acetamido-4-chlorophenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C20H19ClN6O2S
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0634034
|
2-(4-chloro-3-propionamidophenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C22H20ClF3N6O2S
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0634075
|
2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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|
C20H16ClF3N6O2S
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0634530
|
1-(3-acetamido-4-fluorophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)cyclopropanecarboxamide
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|
C20H17FN6O2S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0633748
|
2-(4-chloro-3-propionamidophenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C21H21ClN6O2S
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0634803
|
1-(4-chlorophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)cyclopropanecarboxamide
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|
C18H14ClN5OS
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0637465
|
2-(4-chloro-3-hydroxyphenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)acetamide
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|
C16H12ClN5O2S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0633664
|
2-chloro-N-ethyl-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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|
C22H20ClF3N6O2S
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0635370
|
1-(4-fluoro-3-propionamidophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)cyclopropanecarboxamide
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|
C21H19FN6O2S
|
1
|
| 1 |
IC50 = 4.6 nM
|
|
|
|
CP0634079
|
1-(4-chlorophenylamino)-N-(4-methyl-6H-thiazolo[5,4-e]indazol-2-yl)cyclopropanecarboxamide
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|
C19H16ClN5OS
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0633740
|
2-chloro-N-methyl-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
Show/Hide
|
C21H18ClF3N6O2S
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0633979
|
N-ethyl-2-fluoro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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|
C22H20F4N6O2S
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
|
CP0635232
|
5-(1-(6H-thiazolo[5,4-e]indazol-2-ylcarbamoyl)cyclopropylamino)-2-chloro-N-methylbenzamide
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|
C20H17ClN6O2S
|
1
|
| 1 |
IC50 = 7.5 nM
|
|
|
|
CP0634074
|
2-(4-chlorophenylamino)-3-hydroxy-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C17H14ClN5O2S
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0634519
|
2-(2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamido)acetic acid
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|
C22H18ClF3N6O4S
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0634525
|
4-(2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamido)butanoic acid
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|
C24H22ClF3N6O4S
|
1
|
| 1 |
IC50 = 7.7 nM
|
|
|
|
CP0634799
|
2-(3-hydroxyphenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C18H17N5O2S
|
1
|
| 1 |
IC50 = 7.8 nM
|
|
|
|
CP0637629
|
3-(2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamido)propanoic acid
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|
C23H20ClF3N6O4S
|
1
|
| 1 |
IC50 = 7.9 nM
|
|
|
|
CP0635785
|
2-(4-chlorophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C17H14ClN5OS
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0633741
|
2-(3-acetamido-4-fluorophenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C21H18F4N6O2S
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0633769
|
2-(3-acetamido-4-chlorophenylamino)-N-(6H-thiazolo[5,4-e]indazol-2-yl)acetamide
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|
C18H15ClN6O2S
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0633665
|
2-(4-chloro-3-hydroxyphenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C19H15ClF3N5O2S
|
1
|
| 1 |
IC50 = 8.7 nM
|
|
|
|
CP0636160
|
ethyl 5-(1-(6H-thiazolo[5,4-e]indazol-2-ylcarbamoyl)cyclopropylamino)-2-chlorobenzoate
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|
C21H18ClN5O3S
|
1
|
| 1 |
IC50 = 8.7 nM
|
|
|
|
CP0633766
|
2-(4-chlorophenylamino)-2-methyl-N-(6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C18H16ClN5OS
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0635003
|
2-chloro-N-cyclopropyl-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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|
C23H20ClF3N6O2S
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0633980
|
2-methyl-2-(3-sulfamoylphenylamino)-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C19H17F3N6O3S2
|
1
|
| 1 |
IC50 = 9.3 nM
|
|
|
|
CP0634484
|
2-(4-fluoro-3-propionamidophenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
Show/Hide
|
C22H20F4N6O2S
|
1
|
| 1 |
IC50 = 9.3 nM
|
|
|
|
CP0635002
|
2-(3-acetamido-4-chlorophenylamino)-2-phenyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)acetamide
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|
C25H18ClF3N6O2S
|
1
|
| 1 |
IC50 = 9.8 nM
|
|
|
|
CP0634518
|
N-(2-amino-2-oxoethyl)-2-chloro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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|
C22H19ClF3N7O3S
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0635368
|
2-(4-chloro-3-(2-oxo-2,3-dihydro-1H-imidazol-1-yl)phenylamino)-2-methyl-N-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-yl)propanamide
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|
C22H17ClF3N7O2S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
