Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-ethyl-2-fluoro-5-(2-methyl-1-oxo-1-(4-(trifluoromethyl)-6H-thiazolo[5,4-e]indazol-2-ylamino)propan-2-ylamino)benzamide
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 PubChem ID
CID: 57951272
Canonical SMILES
CCNC(=O)c1cc(NC(C)(C)C(=O)Nc2nc3c(C(F)(F)F)cc4[nH]ncc4c3s2)ccc1F
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Compound Formula C22H20F4N6O2S
Compound Structure
Protein Name
 Protein Info 
Beta-adrenergic receptor kinase 1
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
AGC protein kinase group
>
AGC protein kinase GRK family
>
AGC protein kinase BARK subfamily
Uniprot ID
P25098
Gene Name
GRK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9
 Cell Line Info 
Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 6.4 nM
   TI
   LI
   LO
   TS