Compound ID |
Compound Name |
Compound Formula |
CP0571091
|
[(3S)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-b]pyridazin-6-yl)phenyl]methanone
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|
C27H24N6O
|
1
|
1 |
IC50 = 2.3 nM
|
|
|
CP0550874
|
[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]-(4-piperidin-1-ylpiperidin-1-yl)methanone
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|
C33H33N5O
|
1
|
1 |
IC50 = 2.4 nM
|
|
|
CP0572219
|
[(3S)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
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|
C28H25N5O
|
1
|
1 |
IC50 = 2.5 nM
|
|
|
CP0569513
|
[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]-(4-morpholin-4-ylpiperidin-1-yl)methanone
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|
C32H31N5O2
|
1
|
1 |
IC50 = 4 nM
|
|
|
CP0550873
|
[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]-morpholin-4-ylmethanone
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|
C27H22N4O2
|
1
|
1 |
IC50 = 7 nM
|
|
|
CP0565075
|
[(3R)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
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|
C28H25N5O
|
1
|
1 |
IC50 = 7.7 nM
|
|
|
CP0550876
|
[(3R)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-b]pyridazin-6-yl)phenyl]methanone
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|
C27H24N6O
|
1
|
1 |
IC50 = 9.4 nM
|
|
|
CP0570182
|
[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]-piperazin-1-ylmethanone
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|
C27H23N5O
|
1
|
1 |
IC50 = 9.4 nM
|
|
|
CP0491640
|
4-(6-(4-(morpholine-4-carbonyl)phenyl)imidazo[1,2-a]pyridin-3-yl)benzonitrile
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|
C25H20N4O2
|
1
|
1 |
IC50 = 10.6 nM
|
|
|
CP0563463
|
(4-aminopiperidin-1-yl)-[4-(3-isoquinolin-6-ylimidazo[1,2-b]pyridazin-6-yl)phenyl]methanone
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|
C27H24N6O
|
1
|
1 |
IC50 = 14.5 nM
|
|
|
CP0569548
|
(4-aminopiperidin-1-yl)-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
Show/Hide
|
C28H25N5O
|
1
|
1 |
IC50 = 16.8 nM
|
|
|
CP0564225
|
[(3S)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyrazin-6-yl)phenyl]methanone
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|
C27H24N6O
|
1
|
1 |
IC50 = 27.3 nM
|
|
|
CP0569583
|
(4-aminopiperidin-1-yl)-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyrazin-6-yl)phenyl]methanone
Show/Hide
|
C27H24N6O
|
1
|
1 |
IC50 = 32.1 nM
|
|
|
CP0569550
|
[(3R)-3-aminopiperidin-1-yl]-[4-(3-isoquinolin-6-ylimidazo[1,2-a]pyrazin-6-yl)phenyl]methanone
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|
C27H24N6O
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0550877
|
piperazin-1-yl-[4-(3-quinolin-3-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
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|
C27H23N5O
|
1
|
1 |
IC50 = 67.6 nM
|
|
|
CP0563538
|
morpholin-4-yl-[4-(3-quinolin-3-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
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|
C27H22N4O2
|
1
|
1 |
IC50 = 153.7 nM
|
|
|
CP0550875
|
morpholin-4-yl-[4-(3-quinolin-6-ylimidazo[1,2-a]pyridin-6-yl)phenyl]methanone
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|
C27H22N4O2
|
1
|
1 |
IC50 = 370.8 nM
|
|
|