| Compound ID |
Compound Name |
Compound Formula |
|
CP0217203
|
GS-4997
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|
C24H24FN7O
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
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CP0447844
|
2-[6-[4-[(2R)-1-hydroxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-6-propan-2-yloxy-3H-isoindol-1-one
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|
C21H23N5O3
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
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CP0096218
|
N-[4-(6,7-dimethoxycinnolin-4-yl)oxyphenyl]-4-oxo-1-propan-2-ylquinoline-3-carboxamide
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|
C29H26N4O5
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0447843
|
6-[[(2S)-4-methylmorpholin-2-yl]methoxy]-2-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-3H-isoindol-1-one
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|
C24H28N6O3
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
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CP0462192
|
2-[6-[4-[(2R)-1-hydroxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-6-(2-methoxyethoxy)-3H-isoindol-1-one
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|
C21H23N5O4
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
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CP0471228
|
6-(2-methoxyethoxy)-2-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-3H-isoindol-1-one
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|
C21H23N5O3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0573677
|
2-[6-[4-[(2R)-1-hydroxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C18H17N5O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0240812
|
2-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-3H-isoindol-1-one
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|
C18H17N5O
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0572183
|
2-[6-[4-(1-fluoropropan-2-yl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C18H16FN5O
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
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CP0462188
|
6-propan-2-yloxy-2-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-3H-isoindol-1-one
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|
C21H23N5O2
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0563062
|
4-(1-methylpyrazol-4-yl)-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C23H22N8O
|
1
|
| 1 |
IC50 = 19.6 nM
|
|
|
|
CP0471159
|
2-[6-[4-[(2S)-butan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C19H19N5O
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
|
CP0572603
|
3-[3-[6-(3-oxo-1H-isoindol-2-yl)pyridin-2-yl]-1,2,4-triazol-4-yl]butanenitrile
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|
C19H16N6O
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
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CP0548376
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-7-pyridin-4-yl-1H-indole-2-carboxamide
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|
C24H21N7O
|
1
|
| 1 |
IC50 = 23.1 nM
|
|
|
|
CP0552271
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-5-(1H-pyrazol-4-yl)-1H-indole-2-carboxamide
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|
C22H20N8O
|
1
|
| 1 |
IC50 = 31.6 nM
|
|
|
|
CP0541727
|
2-[6-[4-[(2S)-1-hydroxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C18H17N5O2
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0548375
|
6-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C20H20N6O
|
1
|
| 1 |
IC50 = 32.8 nM
|
|
|
|
CP0548007
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-6-(1H-pyrazol-4-yl)-1H-indole-2-carboxamide
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|
C22H20N8O
|
1
|
| 1 |
IC50 = 37.5 nM
|
|
|
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CP0572757
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-7-(1H-pyrazol-4-yl)-1H-indole-2-carboxamide
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|
C22H20N8O
|
1
|
| 1 |
IC50 = 38.9 nM
|
|
|
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CP0572184
|
2-[6-[4-(4-hydroxybutan-2-yl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C19H19N5O2
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
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CP0568676
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C19H18N6O
|
1
|
| 1 |
IC50 = 41.4 nM
|
|
|
|
CP0181251
|
2-fluoro-4-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
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|
C18H18FN5O
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0458751
|
2-[6-[4-[(2R)-butan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C19H19N5O
|
1
|
| 1 |
IC50 = 50.12 nM
|
|
|
|
CP0548378
|
6-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C20H20N6O2
|
1
|
| 1 |
IC50 = 54.3 nM
|
|
|
|
CP0953731
|
(R)-N-(6-(4-(1-hydroxypropan-2-yl)-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-1H-indole-2-carboxamide
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|
C19H18N6O2
|
1
|
| 1 |
IC50 = 65.5 nM
|
|
|
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CP0537395
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-6-pyridin-3-yl-1H-indole-2-carboxamide
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|
C24H21N7O
|
1
|
| 1 |
IC50 = 68.5 nM
|
|
|
|
CP0548380
|
6-[1-(oxan-4-yl)pyrazol-4-yl]-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C27H28N8O2
|
1
|
| 1 |
IC50 = 73.7 nM
|
|
|
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CP0568504
|
3-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C20H20N6O
|
1
|
| 1 |
IC50 = 88.2 nM
|
|
|
|
CP0552355
|
7-chloro-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C19H17ClN6O
|
1
|
| 1 |
IC50 = 89.6 nM
|
|
|
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CP0961250
|
6-(1-(1-ethoxyethyl)-1H-pyrazol-4-yl)-N-(6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-yl)-1H-indole-2-carboxamide
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|
C26H28N8O2
|
1
|
| 1 |
IC50 = 91.1 nM
|
|
|
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CP0548377
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
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|
C18H17N7O
|
1
|
| 1 |
IC50 = 125.1 nM
|
|
|
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CP0564198
|
3-(furan-3-yl)-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C23H20N6O2
|
1
|
| 1 |
IC50 = 142.8 nM
|
|
|
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CP0552588
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-benzofuran-2-carboxamide
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|
C19H17N5O2
|
1
|
| 1 |
IC50 = 151.6 nM
|
|
|
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CP0551834
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-7-thiophen-3-yl-1H-indole-2-carboxamide
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|
C23H20N6OS
|
1
|
| 1 |
IC50 = 153.3 nM
|
|
|
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CP0568503
|
7-acetamido-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1H-indole-2-carboxamide
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|
C21H21N7O2
|
1
|
| 1 |
IC50 = 240.1 nM
|
|
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CP0559851
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
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|
C17H17N5O
|
1
|
| 1 |
IC50 = 398.11 nM
|
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CP0537394
|
N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1,3-benzothiazole-2-carboxamide
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|
C18H16N6OS
|
1
|
| 1 |
IC50 = 506 nM
|
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CP0552269
|
1-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]indole-2-carboxamide
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|
C20H20N6O
|
1
|
| 1 |
IC50 = 743 nM
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CP0471229
|
2-[6-[4-(oxetan-2-ylmethyl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3H-isoindol-1-one
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|
C19H17N5O2
|
1
|
| 1 |
IC50 = 794.33 nM
|
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CP0558183
|
3-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-benzofuran-2-carboxamide
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|
C20H19N5O2
|
1
|
| 1 |
IC50 = 1106 nM
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CP0154571
|
5-(4-cyclopropylimidazol-1-yl)-2-fluoro-4-methyl-N-pyridin-2-ylbenzamide
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|
C19H17FN4O
|
1
|
| 1 |
IC50 = 6309.57 nM
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CP0563061
|
3-methyl-N-[3-(tetrazol-1-yl)phenyl]-1-benzofuran-2-carboxamide
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|
C17H13N5O2
|
1
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| 1 |
IC50 = 16700 nM
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