| Compound ID |
Compound Name |
Compound Formula |
|
CP0170179
|
5-chloro-N-[4-(4-methylpiperazin-1-yl)phenyl]-4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine
Show/Hide
|
C22H22ClN7
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
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CP0101029
|
3-(4-methoxyphenyl)-N-[(4-methoxyphenyl)carbamothioyl]-1-phenylpyrazole-4-carboxamide
Show/Hide
|
C25H22N4O3S
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0870831
|
3-(4-Methoxyphenyl)-1-phenyl-N-(p-tolylcarbamothioyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C25H22N4O2S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0870830
|
N-((4-Chlorophenyl)carbamothioyl)-3-(4-methoxyphenyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19ClN4O2S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0898828
|
N-((4-Fluorophenyl)carbamothioyl)-3-(4-methoxyphenyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19FN4O2S
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0101028
|
3-(4-fluorophenyl)-N-[(4-methoxyphenyl)carbamothioyl]-1-phenylpyrazole-4-carboxamide
Show/Hide
|
C24H19FN4O2S
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0051785
|
3-(4-chlorophenyl)-N-[(4-methoxyphenyl)carbamothioyl]-1-phenylpyrazole-4-carboxamide
Show/Hide
|
C24H19ClN4O2S
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0919886
|
N-((4-Fluorophenyl)carbamothioyl)-1-phenyl-3-(p-tolyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19FN4OS
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0951266
|
3-(4-Chlorophenyl)-1-phenyl-N-(p-tolylcarbamothioyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19ClN4OS
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0899217
|
3-(4-Fluorophenyl)-1-phenyl-N-(p-tolylcarbamothioyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19FN4OS
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0864076
|
N-((4-Chlorophenyl)carbamothioyl)-3-(4-fluorophenyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H16ClFN4OS
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0053667
|
N-[(4-methoxyphenyl)carbamothioyl]-3-(4-methylphenyl)-1-phenylpyrazole-4-carboxamide
Show/Hide
|
C25H22N4O2S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0864077
|
3-(4-Fluorophenyl)-N-((4-fluorophenyl)carbamothioyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H16F2N4OS
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0908172
|
1-Phenyl-3-(p-tolyl)-N-(p-tolylcarbamothioyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C25H22N4OS
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0053665
|
N-[(4-methoxyphenyl)carbamothioyl]-1,3-diphenylpyrazole-4-carboxamide
Show/Hide
|
C24H20N4O2S
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0847864
|
3-(4-Chlorophenyl)-N-((4-chlorophenyl)carbamothioyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H16Cl2N4OS
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0899218
|
3-(4-Chlorophenyl)-N-((4-fluorophenyl)carbamothioyl)-1-phenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H16ClFN4OS
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0848142
|
N-((4-Chlorophenyl)carbamothioyl)-1-phenyl-3-(p-tolyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H19ClN4OS
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0860249
|
1,3-Diphenyl-N-(p-tolylcarbamothioyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H20N4OS
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0872301
|
N-((4-Chlorophenyl)carbamothioyl)-1,3-diphenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H17ClN4OS
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0860248
|
N-((4-Fluorophenyl)carbamothioyl)-1,3-diphenyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H17FN4OS
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0310598
|
3-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C14H10N4
|
1
|
| 1 |
IC50 = 314 nM
|
|
|
|
CP0001111
|
(2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]amino]butan-1-ol
Show/Hide
|
C19H26N6O
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0316807
|
N-[4-(4-methylpiperazin-1-yl)phenyl]-6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-amine
Show/Hide
|
C22H23N7
|
1
|
| 1 |
IC50 = 577 nM
|
|
|
|
CP0088578
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine
Show/Hide
|
C23H25N7O
|
1
|
| 1 |
IC50 = 1819 nM
|
|
|
|
CP0088579
|
1-[4-[3-methoxy-4-[[4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethanone
Show/Hide
|
C24H25N7O2
|
1
|
| 1 |
IC50 = 1995 nM
|
|
|
|
CP0073979
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine
Show/Hide
|
C24H27N7O
|
1
|
| 1 |
IC50 = 4473 nM
|
|
|
|
CP0072037
|
3-[2-[(E)-2-phenylethenyl]pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C19H14N4
|
1
|
| 1 |
IC50 = 5176 nM
|
|
|
|
CP0001206
|
2,6,9-Trisubstituted purine deriv. 26
Show/Hide
|
C15H18N6O
|
1
|
| 1 |
IC50 = 7000 nM
|
|
|
|
CP0514456
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(5-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine
Show/Hide
|
C24H27N7O
|
1
|
| 1 |
IC50 = 10476 nM
|
|
|
|
CP0388934
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-amine
Show/Hide
|
C23H25N7O
|
1
|
| 1 |
IC50 = 12295 nM
|
|
|
|
CP0072052
|
4-(1,7-dimethylpyrrolo[2,3-c]pyridin-3-yl)-N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]pyrimidin-2-amine
Show/Hide
|
C25H29N7O
|
1
|
| 1 |
IC50 = 13713 nM
|
|
|
|
CP0259635
|
1-[4-[3-methoxy-4-[[6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-yl]amino]phenyl]piperazin-1-yl]ethanone
Show/Hide
|
C24H25N7O2
|
1
|
| 1 |
IC50 = 14060 nM
|
|
|
|
CP0088580
|
1-[4-[3-methoxy-4-[[6-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-yl]amino]phenyl]piperazin-1-yl]ethanone
Show/Hide
|
C25H27N7O2
|
1
|
| 1 |
IC50 = 14789 nM
|
|
|
|
CP0084894
|
3-[2-(4-methylsulfonylphenyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C18H14N4O2S
|
1
|
| 1 |
IC50 = 16884 nM
|
|
|
|
CP0390051
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(7-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine
Show/Hide
|
C24H27N7O
|
1
|
| 1 |
IC50 = 17368 nM
|
|
|
|
CP0072040
|
6-(1H-indol-3-yl)-N-[4-(4-methylpiperazin-1-yl)phenyl]pyrimidin-4-amine
Show/Hide
|
C23H24N6
|
1
|
| 1 |
IC50 = 33215 nM
|
|
|
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CP0073977
|
3-(2-methylpyrimidin-4-yl)-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C12H10N4
|
1
|
| 1 |
IC50 = 38379 nM
|
|
|
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CP0072039
|
N-cyclopentyl-4-[4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-yl]benzamide
Show/Hide
|
C23H21N5O
|
1
|
| 1 |
IC50 = 45885 nM
|
|
|
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CP0380676
|
1-benzyl-3-(2-methylpyrimidin-4-yl)pyrrolo[2,3-c]pyridine
Show/Hide
|
C19H16N4
|
1
|
| 1 |
IC50 = 56703 nM
|
|
|
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CP0072038
|
7-methyl-3-[2-(4-methylsulfonylphenyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridine
Show/Hide
|
C19H16N4O2S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
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CP0283349
|
1-methyl-3-[2-(4-methylsulfonylphenyl)pyrimidin-4-yl]pyrrolo[2,3-c]pyridine
Show/Hide
|
C19H16N4O2S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
