| Compound ID |
Compound Name |
Compound Formula |
|
CP0389504
|
[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]-(oxolan-2-yl)methanone
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|
C24H32N4O4
|
2
|
| 1 |
EC50 = 0.4 nM
|
|
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| 2 |
EC50 = 24.6 nM
|
|
|
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CP0389498
|
[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]-thiophen-2-ylmethanone
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|
C24H28N4O3S
|
2
|
| 1 |
EC50 = 0.51 nM
|
|
|
| 2 |
EC50 = 8.2 nM
|
|
|
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CP0462496
|
[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]-phenylmethanone
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|
C26H30N4O3
|
2
|
| 1 |
EC50 = 0.6 nM
|
|
|
| 2 |
EC50 = 15.5 nM
|
|
|
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CP0391583
|
1-[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]-2,2-dimethylpropan-1-one
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|
C24H34N4O3
|
2
|
| 1 |
EC50 = 0.69 nM
|
|
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| 2 |
EC50 = 21.9 nM
|
|
|
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CP0389489
|
furan-2-yl-[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]methanone
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|
C24H28N4O4
|
2
|
| 1 |
EC50 = 0.88 nM
|
|
|
| 2 |
EC50 = 19.8 nM
|
|
|
|
CP0391584
|
1-[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]-2-phenoxyethanone
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|
C27H32N4O4
|
2
|
| 1 |
EC50 = 1.28 nM
|
|
|
| 2 |
EC50 = 18.2 nM
|
|
|
|
CP0109915
|
N-[[4-[(4-fluorophenyl)methylsulfamoyl]phenyl]carbamothioyl]-4-phenylbenzamide
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|
C27H22FN3O3S2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0109917
|
N-[[4-(furan-2-ylmethylsulfamoyl)phenyl]carbamothioyl]-4-phenylbenzamide
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|
C25H21N3O4S2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0558276
|
[(2R)-2-hydroxy-3-[hydroxy-[(2R,3R,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxyphosphoryl]oxypropyl] octadecanoate
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|
C27H53O12P
|
1
|
| 1 |
EC50 = 2.82 nM
|
|
|
|
CP0231660
|
N-[[4-(benzylsulfamoyl)phenyl]carbamothioyl]-4-phenylbenzamide
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|
C27H23N3O3S2
|
1
|
| 1 |
EC50 = 5.6 nM
|
|
|
|
CP0076591
|
4-phenyl-N-[[4-(phenylsulfamoyl)phenyl]carbamothioyl]benzamide
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|
C26H21N3O3S2
|
1
|
| 1 |
EC50 = 6.2 nM
|
|
|
|
CP0385457
|
N-[(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)methyl]-2-[4-(2-methoxyphenyl)piperazin-1-yl]acetamide
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|
C27H33N5O4
|
2
|
| 1 |
EC50 = 6.36 nM
|
|
|
| 2 |
EC50 = 28.4 nM
|
|
|
|
CP0076590
|
N-[[4-[(4-methoxyphenyl)methylsulfamoyl]phenyl]carbamothioyl]-4-phenylbenzamide
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|
C28H25N3O4S2
|
1
|
| 1 |
EC50 = 7.7 nM
|
|
|
|
CP0398848
|
cyclohexyl-[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)ethyl]piperazin-1-yl]methanone
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|
C26H36N4O3
|
2
|
| 1 |
EC50 = 8.67 nM
|
|
|
| 2 |
EC50 = 25.4 nM
|
|
|
|
CP0106955
|
N-[[4-[(4-methylphenyl)methylsulfamoyl]phenyl]carbamothioyl]-4-phenylbenzamide
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|
C28H25N3O3S2
|
1
|
| 1 |
EC50 = 12.4 nM
|
|
|
|
CP0141678
|
4-phenyl-N-[[4-(prop-2-enylsulfamoyl)phenyl]carbamothioyl]benzamide
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|
C23H21N3O3S2
|
1
|
| 1 |
EC50 = 19.4 nM
|
|
|
|
CP0389495
|
furan-2-yl-[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-1-yl)ethyl]piperazin-1-yl]methanone
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|
C24H28N4O4
|
1
|
| 1 |
EC50 = 19.6 nM
|
|
|
|
CP0403838
|
[(2R)-2-hydroxy-3-[hydroxy-[(2S,3S,5R,6S)-2,3,4,5,6-pentahydroxycyclohexyl]oxyphosphoryl]oxypropyl] (5Z,8Z,11Z,14Z)-icosa-5,8,11,14-tetraenoate
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|
C29H49O12P
|
1
|
| 1 |
EC50 = 20.24 nM
|
|
|
|
CP0389497
|
N-[(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-1-yl)methyl]-2-[4-(4-methoxyphenyl)piperazin-1-yl]acetamide
Show/Hide
|
C27H33N5O4
|
1
|
| 1 |
EC50 = 27.3 nM
|
|
|
|
CP0455151
|
N-[(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-1-yl)methyl]-2-(4-phenylpiperazin-1-yl)acetamide
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|
C26H31N5O3
|
1
|
| 1 |
EC50 = 27.7 nM
|
|
|
|
CP0398849
|
[4-[2-(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-1-yl)ethyl]piperazin-1-yl]-thiophen-2-ylmethanone
Show/Hide
|
C24H28N4O3S
|
1
|
| 1 |
EC50 = 29.3 nM
|
|
|
|
CP0389501
|
2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-N-[(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)methyl]acetamide
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|
C28H35N5O3
|
1
|
| 1 |
EC50 = 30.4 nM
|
|
|
|
CP0076589
|
N-[[4-(2-methylpropylsulfamoyl)phenyl]carbamothioyl]-4-phenylbenzamide
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|
C24H25N3O3S2
|
1
|
| 1 |
EC50 = 30.9 nM
|
|
|
|
CP0389486
|
N-[(7-methoxy-4,4-dimethylchromeno[4,3-c]pyrazol-2-yl)methyl]-2-(4-phenylpiperazin-1-yl)acetamide
Show/Hide
|
C26H31N5O3
|
1
|
| 1 |
EC50 = 31.5 nM
|
|
|
|
CP0076542
|
4-phenyl-N-[[4-(2-phenylethylsulfamoyl)phenyl]carbamothioyl]benzamide
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|
C28H25N3O3S2
|
1
|
| 1 |
EC50 = 39.2 nM
|
|
|
|
CP0109918
|
N-[[4-(dimethylsulfamoyl)phenyl]carbamothioyl]-4-phenylbenzamide
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|
C22H21N3O3S2
|
1
|
| 1 |
EC50 = 55.7 nM
|
|
|
|
CP0087158
|
4-phenyl-N-[[4-(propylsulfamoyl)phenyl]carbamothioyl]benzamide
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|
C23H23N3O3S2
|
1
|
| 1 |
EC50 = 175.7 nM
|
|
|
|
CP0043299
|
N-[[4-(4-methylpiperazin-1-yl)sulfonylphenyl]carbamothioyl]-4-phenylbenzamide
Show/Hide
|
C25H26N4O3S2
|
1
|
| 1 |
EC50 = 218 nM
|
|
|
|
CP0102214
|
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C22H21Cl2IN4O
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
|
CP0109916
|
N-[[4-(benzylcarbamoyl)phenyl]carbamothioyl]-4-phenylbenzamide
Show/Hide
|
C28H23N3O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0212238
|
4-phenyl-N-[[4-(2-phenylethylcarbamoyl)phenyl]carbamothioyl]benzamide
Show/Hide
|
C29H25N3O2S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0042287
|
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H19Cl2IN4O2
|
1
|
| 1 |
EC50 = 13600 nM
|
|
|
