Compound ID |
Compound Name |
Compound Formula |
CP0868600
|
2-Thiouridine-5'-alpha,beta-methylene Diphosphate,bis-Triethylammonium Salt
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|
C16H31N3O10P2S
|
1
|
1 |
EC50 = 0.92 nM
|
|
|
CP0384686
|
((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methoxy)(hydroxy)phosphoryl)methylphosphonic acid
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|
C10H16N2O11P2
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0401576
|
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-(2-oxo-4-sulfanylidenepyrimidin-1-yl)oxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl] hydrogen phosphate
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|
C15H24N2O16P2S
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0874897
|
Diphosphoric Acid 1-beta-(3-Butynyl)Ester 2-(2-Thiouridine-5'-yl)ester, bis-Triethylammonium Salt
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|
C19H33N3O11P2S
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0858598
|
Diphosphoric Acid 1-beta-tert-Butyl Ester 2-(2-Thiouridine-5'-yl)ester, di Ammonium Salt
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|
C13H25N3O11P2S
|
1
|
1 |
EC50 = 32 nM
|
|
|
CP0917610
|
Diphosphoric Acid 1-beta-Ethyl Ester 2-(2-Thiouridine-5'-yl)-ester,di ammonium Salt
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|
C11H21N3O11P2S
|
1
|
1 |
EC50 = 39 nM
|
|
|
CP0918625
|
Diphosphoric Acid 1-beta-Propyl Ester 2-(2-Thiouridine-5'-yl)-ester, di ammonium Salt
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|
C12H23N3O11P2S
|
1
|
1 |
EC50 = 40 nM
|
|
|
CP0901965
|
Diphosphoric Acid 1-beta-Methyl Ester 2-(2-Thiouridine-5'-yl)-ester, di ammonium Salt
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|
C10H19N3O11P2S
|
1
|
1 |
EC50 = 56 nM
|
|
|
CP0439245
|
({[(2R,3S,4R,5R)-5-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3,4-dihydroxy-tetrahydro-furan-2-ylmethoxy]-hydroxy-phosphoryl}-difluoro-methyl)-phosphonic acid
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|
C10H14F2N2O11P2
|
1
|
1 |
EC50 = 63 nM
|
|
|
CP0864425
|
5-Iodouridine5'-Methylenediphosphate Triethylammonium salt
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|
C16H30IN3O11P2
|
1
|
1 |
EC50 = 140 nM
|
|
|
CP0398926
|
({[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(5-iodo-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-2-ylmethoxy]-hydroxy-phosphoryl}-difluoro-methyl)-phosphonic acid
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|
C10H13F2IN2O11P2
|
1
|
1 |
EC50 = 142 nM
|
|
|
CP0914501
|
Diphosphoric Acid 1-beta-Glycerol Ester 2-(Uridine-5'-yl)ester,bis-Triethylammonium Salt
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|
C18H35N3O14P2
|
1
|
1 |
EC50 = 167 nM
|
|
|
CP0916086
|
Diphosphoric Acid 1-beta-tert-Butyl Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C13H25N3O12P2
|
1
|
1 |
EC50 = 252 nM
|
|
|
CP0419133
|
4-Thio-UDP
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|
C9H14N2O11P2S
|
1
|
1 |
EC50 = 320 nM
|
|
|
CP0917612
|
Diphosphoric Acid 1-beta-(3-Butynyl)Ester 2-(Uridine-5'-yl)-ester, bis-Triethylammonium Salt
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|
C19H33N3O12P2
|
1
|
1 |
EC50 = 480 nM
|
|
|
CP0916051
|
Diphosphoric Acid 1-beta-Phenyl Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C15H21N3O12P2
|
1
|
1 |
EC50 = 768 nM
|
|
|
CP0894017
|
Diphosphoric Acid 1-beta-(4-Nitrophenyl)Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C15H20N4O14P2
|
1
|
1 |
EC50 = 1490 nM
|
|
|
CP0914500
|
Diphosphoric Acid 1-r-Glycerol Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C12H23N3O14P2
|
1
|
1 |
EC50 = 1600 nM
|
|
|
CP0901964
|
Diphosphoric Acid 1-beta-(3-Chlorophenyl)Ester 2-(Uridine-5'-yl)ester, di ammonium Salt
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|
C15H20ClN3O12P2
|
1
|
1 |
EC50 = 1800 nM
|
|
|
CP0888564
|
Diphosphoric Acid 1-beta-(4-Methoxyphenyl)Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C16H23N3O13P2
|
1
|
1 |
EC50 = 1900 nM
|
|
|
CP0888563
|
Diphosphoric Acid 1-beta-Methyl Ester 2-(Uridine-5'-yl)ester, di ammonium Salt
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|
C10H19N3O12P2
|
1
|
1 |
EC50 = 2730 nM
|
|
|
CP0844902
|
N4-Methoxycytidine 5'-Diphosphate triethylammonium Salt
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|
C16H32N4O12P2
|
1
|
1 |
EC50 = 3320 nM
|
|
|
CP0874895
|
[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-[(4E)-4-(methoxyimino)-2-oxo-1,2,3,4-tetrahydropyrimidin-1-yl]oxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy]phosphonic acid hydrochloride
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|
C10H18ClN3O12P2
|
1
|
1 |
EC50 = 3320 nM
|
|
|
CP0914213
|
[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(methoxyimino)-2-oxo-1,2,3,4-tetrahydropyrimidin-1-yl]oxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy]phosphonic acid
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|
C16H31N3O11P2
|
1
|
1 |
EC50 = 4580 nM
|
|
|
CP0874914
|
Diphosphoric Acid 1-beta-Cyclohexyl Ester 2-(Uridine-5'-yl)ester,di ammonium Salt
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|
C15H27N3O12P2
|
1
|
1 |
EC50 = 5160 nM
|
|
|
CP0918631
|
Diphosphoric Acid 1-beta-(2-Cyanoethyl)Ester 2-(Uridine-5'-yl)ester, di ammonium Salt
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|
C12H20N4O12P2
|
1
|
1 |
EC50 = 7460 nM
|
|
|
CP0435758
|
3-[(4-methylbenzoyl)amino]-5-(4-piperidin-4-ylphenyl)benzoic acid
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|
C26H26N2O3
|
1
|
1 |
IC50 = 1.77 nM
|
|
|
CP0569324
|
1-[(4-fluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H16FN3O3
|
1
|
1 |
IC50 = 1.93 nM
|
|
|
CP0032210
|
4-(4-piperidin-4-ylphenyl)-7-[4-(trifluoromethyl)phenyl]naphthalene-2-carboxylic acid
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|
C29H24F3NO2
|
1
|
1 |
IC50 = 1.98 nM
|
|
|
CP0546659
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(4-methoxyphenyl)acetamide
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|
C22H18N2O3
|
1
|
1 |
IC50 = 2 nM
|
|
|
CP0551452
|
3-(furan-3-yl)-5-[(4-methylbenzoyl)amino]benzoic acid
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|
C19H15NO4
|
1
|
1 |
IC50 = 2.18 nM
|
|
|
CP0558094
|
3-[(4-methylbenzoyl)amino]-5-(1H-pyrazol-5-yl)benzoic acid
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|
C18H15N3O3
|
1
|
1 |
IC50 = 2.63 nM
|
|
|
CP0563460
|
3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[(4-methylbenzoyl)amino]benzoic acid
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|
C20H18N2O4
|
1
|
1 |
IC50 = 2.95 nM
|
|
|
CP0575592
|
5-[(4-acetylbenzoyl)amino]-1-[(4-fluorophenyl)methyl]pyrazole-3-carboxylic acid
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|
C20H16FN3O4
|
1
|
1 |
IC50 = 3.81 nM
|
|
|
CP0572909
|
5-[(4-methylbenzoyl)amino]-1-[[4-(trifluoromethyl)phenyl]methyl]pyrazole-3-carboxylic acid
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|
C20H16F3N3O3
|
1
|
1 |
IC50 = 3.83 nM
|
|
|
CP0547328
|
5-[(4-methylbenzoyl)amino]-1-[(3,4,5-trifluorophenyl)methyl]pyrazole-3-carboxylic acid
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|
C19H14F3N3O3
|
1
|
1 |
IC50 = 4.01 nM
|
|
|
CP0568085
|
1-[(3,4-difluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H15F2N3O3
|
1
|
1 |
IC50 = 4.16 nM
|
|
|
CP0580107
|
5-[(4-ethylbenzoyl)amino]-1-[(4-fluorophenyl)methyl]pyrazole-3-carboxylic acid
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|
C20H18FN3O3
|
1
|
1 |
IC50 = 4.65 nM
|
|
|
CP0547330
|
1-[(4-cyanophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C20H16N4O3
|
1
|
1 |
IC50 = 4.66 nM
|
|
|
CP0546985
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-[4-(trifluoromethoxy)phenyl]acetamide
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|
C22H15F3N2O3
|
1
|
1 |
IC50 = 4.8 nM
|
|
|
CP0545529
|
5-[(4-methylbenzoyl)amino]-1-[[2-(trifluoromethyl)phenyl]methyl]pyrazole-3-carboxylic acid
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|
C20H16F3N3O3
|
1
|
1 |
IC50 = 4.83 nM
|
|
|
CP0533864
|
3-[(4-methylbenzoyl)amino]-5-phenylbenzoic acid
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|
C21H17NO3
|
1
|
1 |
IC50 = 4.85 nM
|
|
|
CP0580196
|
5-[(4-methylbenzoyl)amino]-1-[(4-nitrophenyl)methyl]pyrazole-3-carboxylic acid
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|
C19H16N4O5
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0575967
|
1-[(3-fluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H16FN3O3
|
1
|
1 |
IC50 = 5.39 nM
|
|
|
CP0577362
|
1-[(3,5-dimethylphenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C21H21N3O3
|
1
|
1 |
IC50 = 5.77 nM
|
|
|
CP0546984
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-[4-(trifluoromethyl)phenyl]acetamide
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|
C22H14ClF3N2O2
|
1
|
1 |
IC50 = 6.1 nM
|
|
|
CP0571384
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-(4-methylphenyl)acetamide
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|
C22H17ClN2O2
|
1
|
1 |
IC50 = 6.7 nM
|
|
|
CP0575995
|
1-[(4-chlorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H16ClN3O3
|
1
|
1 |
IC50 = 7.11 nM
|
|
|
CP0546657
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(4-methylphenyl)acetamide
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|
C22H18N2O2
|
1
|
1 |
IC50 = 8.7 nM
|
|
|
CP0545190
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-(4-methoxyphenyl)acetamide
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|
C22H17ClN2O3
|
1
|
1 |
IC50 = 9.2 nM
|
|
|
CP0578453
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(2-methylphenyl)acetamide
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|
C22H18N2O2
|
1
|
1 |
IC50 = 9.3 nM
|
|
|
CP0544882
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)-5-methylphenyl]-2-(3-methylphenyl)acetamide
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|
C23H19ClN2O2
|
1
|
1 |
IC50 = 9.7 nM
|
|
|
CP0566510
|
3-[(4-methylbenzoyl)amino]-5-thiophen-3-ylbenzoic acid
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|
C19H15NO3S
|
1
|
1 |
IC50 = 9.74 nM
|
|
|
CP0546980
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-[4-(trifluoromethoxy)phenyl]acetamide
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|
C22H14ClF3N2O3
|
1
|
1 |
IC50 = 9.8 nM
|
|
|
CP0546982
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-[4-(trifluoromethyl)phenyl]acetamide
Show/Hide
|
C22H15F3N2O2
|
1
|
1 |
IC50 = 11.5 nM
|
|
|
CP0567976
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
|
C22H18N2O3
|
1
|
1 |
IC50 = 12.2 nM
|
|
|
CP0571385
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(4-butoxyphenyl)acetamide
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|
C25H24N2O3
|
1
|
1 |
IC50 = 12.3 nM
|
|
|
CP0544881
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-[3-(trifluoromethoxy)phenyl]acetamide
Show/Hide
|
C22H14ClF3N2O3
|
1
|
1 |
IC50 = 12.6 nM
|
|
|
CP0578454
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-(3-chlorophenyl)acetamide
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|
C21H14Cl2N2O2
|
1
|
1 |
IC50 = 13.4 nM
|
|
|
CP0576752
|
2-[1-[(4-fluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazol-3-yl]acetic acid
Show/Hide
|
C20H18FN3O3
|
1
|
1 |
IC50 = 14.26 nM
|
|
|
CP0575968
|
5-[(4-methylbenzoyl)amino]-1-[[3-(trifluoromethyl)phenyl]methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C20H16F3N3O3
|
1
|
1 |
IC50 = 15.7 nM
|
|
|
CP0546661
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-[3-(trifluoromethoxy)phenyl]acetamide
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|
C22H15F3N2O3
|
1
|
1 |
IC50 = 16.2 nM
|
|
|
CP0546981
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-(2-methoxyphenyl)acetamide
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|
C22H17ClN2O3
|
1
|
1 |
IC50 = 17.1 nM
|
|
|
CP0577724
|
N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-(4-methylphenyl)acetamide
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|
C23H20N2O2
|
1
|
1 |
IC50 = 18.5 nM
|
|
|
CP0577531
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(3-methylphenyl)acetamide
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|
C22H18N2O2
|
1
|
1 |
IC50 = 21.8 nM
|
|
|
CP0577757
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-(3-methoxyphenyl)acetamide
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|
C22H17ClN2O3
|
1
|
1 |
IC50 = 23.8 nM
|
|
|
CP0572726
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(3-methoxyphenyl)acetamide
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|
C22H18N2O3
|
1
|
1 |
IC50 = 24.3 nM
|
|
|
CP0550137
|
N-[3-(1,3-benzoxazol-2-yl)phenyl]-2-(3-bromophenyl)acetamide
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|
C21H15BrN2O2
|
1
|
1 |
IC50 = 25.4 nM
|
|
|
CP0547030
|
N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]-2-[3-(trifluoromethyl)phenyl]acetamide
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|
C22H14ClF3N2O2
|
1
|
1 |
IC50 = 27.5 nM
|
|
|
CP0546983
|
2-(2-bromophenyl)-N-[3-(5-chloro-1,3-benzoxazol-2-yl)phenyl]acetamide
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|
C21H14BrClN2O2
|
1
|
1 |
IC50 = 32.9 nM
|
|
|
CP0543240
|
N-[3-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-2-[4-(trifluoromethyl)phenyl]acetamide
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|
C23H17F3N2O2
|
1
|
1 |
IC50 = 35.1 nM
|
|
|
CP0570113
|
1-[(3,5-difluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H15F2N3O3
|
1
|
1 |
IC50 = 40.95 nM
|
|
|
CP0544883
|
N-[4-(1-benzofuran-2-yl)phenyl]-2-(4-methylphenyl)acetamide
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|
C23H19NO2
|
1
|
1 |
IC50 = 42.4 nM
|
|
|
CP0579803
|
1-[(3-methoxyphenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
Show/Hide
|
C20H19N3O4
|
1
|
1 |
IC50 = 61.22 nM
|
|
|
CP0568773
|
1-[(4-acetylphenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C21H19N3O4
|
1
|
1 |
IC50 = 67 nM
|
|
|
CP0547331
|
1-(cyclopentylmethyl)-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C18H21N3O3
|
1
|
1 |
IC50 = 99.65 nM
|
|
|
CP0569319
|
1-[(2-fluorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H16FN3O3
|
1
|
1 |
IC50 = 110.9 nM
|
|
|
CP0567991
|
1-(cyclohexylmethyl)-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H23N3O3
|
1
|
1 |
IC50 = 135.7 nM
|
|
|
CP0564639
|
1-benzyl-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C19H17N3O3
|
1
|
1 |
IC50 = 170.8 nM
|
|
|
CP0545527
|
1-[(3-chlorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
Show/Hide
|
C19H16ClN3O3
|
1
|
1 |
IC50 = 227.3 nM
|
|
|
CP0578215
|
1-[(2-chlorophenyl)methyl]-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
Show/Hide
|
C19H16ClN3O3
|
1
|
1 |
IC50 = 245.1 nM
|
|
|
CP0573680
|
1-(cyclobutylmethyl)-5-[(4-methylbenzoyl)amino]pyrazole-3-carboxylic acid
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|
C17H19N3O3
|
1
|
1 |
IC50 = 369 nM
|
|
|
CP0580106
|
5-[(4-methylbenzoyl)amino]-1-[(2-methylphenyl)methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C20H19N3O3
|
1
|
1 |
IC50 = 531.5 nM
|
|
|