Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
 Cell Line Info 
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT05269 , Gamma-aminobutyric acid receptor subunit alpha-2
 Protein Info 
Gene Name GABRA2
Organism Rattus norvegicus, Rat
Protein Classification Ion channel
Uniprot ID P23576
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006
 Cell Line Info 
 Protein ID: PT05269
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0000099
 Compound Info 
7-chloro-1-methyl-5-phenyl-3H-1,4-benzodiazepin-2-one
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C16H13ClN2O
  1
1
Ki = 15 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0000229
 Compound Info 
(R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide
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C19H15N3O4
  1
1
Ki = 85 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0003479
 Compound Info 
N-[(4-fluorophenyl)methyl]-2-(1H-indol-3-yl)-2-oxoacetamide
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C17H13FN2O2
  1
1
Ki = 118 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0003771
 Compound Info 
(R)-2-(5-nitro-1H-indol-3-yl)-2-oxo-N-(1-phenylethyl)acetamide
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C18H15N3O4
  1
1
Ki = 121 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002470
 Compound Info 
2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetamide
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C17H13N3O4
  1
1
Ki = 210 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0010590
 Compound Info 
(R/S)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide
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C20H17N3O5
  1
1
Ki = 231 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0009202
 Compound Info 
(R/S)-2-(5-nitro-1H-indol-3-yl)-N-(5-nitro-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide
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C19H14N4O6
  1
1
Ki = 513 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002158
 Compound Info 
(R/S)-2-(1H-indol-3-yl)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide
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C20H18N2O3
  1
1
Ki = 690 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0000163
 Compound Info 
Ambien
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C19H21N3O
  1
1
Ki = 765 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0009201
 Compound Info 
(R/S)-N-(5-fluoro-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide
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C19H14FN3O4
  1
1
Ki = 810 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0004581
 Compound Info 
(R)-2-(1H-indol-3-yl)-2-oxo-N-(1-phenylethyl)acetamide
   Show/Hide
C18H16N2O2
  1
1
Ki = 1550 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002684
 Compound Info 
N-[(4-methoxyphenyl)methyl]-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide
   Show/Hide
C18H15N3O5
  1
1
Ki = 1645 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0009784
 Compound Info 
2-(1H-Indol-3-yl)-N-(4-methoxy-benzyl)-2-oxo-acetamide
   Show/Hide
C18H16N2O3
  1
1
Ki = 1950 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0000228
 Compound Info 
2-(5-nitro-1H-indol-3-yl)-N-(4-nitrobenzyl)-2-oxoacetamide
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C17H12N4O6
  1
1
Ki = 2980 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002157
 Compound Info 
(R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(1H-indol-3-yl)-2-oxoacetamide
   Show/Hide
C19H16N2O2
  1
1
Ki = 3100 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS