| Compound ID |
Compound Name |
Compound Formula |
|
CP0063510
|
(S)-2-Amino-4-phosphono-butyric acid
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|
C4H10NO5P
|
3
|
| 1 |
EC50 = 70 nM
|
|
|
| 2 |
EC50 = 240 nM
|
|
|
| 3 |
EC50 = 300 nM
|
|
|
|
CP0392926
|
N-[3-chloro-4-(5-chloropyridin-2-yl)oxyphenyl]pyridine-2-carboxamide
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|
C17H11Cl2N3O2
|
1
|
| 1 |
EC50 = 125 nM
|
|
|
|
CP0106027
|
D-AP4
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|
C4H10NO5P
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0058507
|
(1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid
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|
C8H11NO6
|
1
|
| 1 |
EC50 = 680 nM
|
|
|
|
CP0288101
|
methyl 4-[3-[2-(4-acetamidophenyl)sulfanylacetyl]-2,5-dimethylpyrrol-1-yl]benzoate
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|
C24H24N2O4S
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0374296
|
(3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]ethanoic Acid
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|
C6H12NO6P
|
2
|
| 1 |
EC50 = 910 nM
|
|
|
| 2 |
EC50 = 2700 nM
|
|
|
|
CP0120365
|
5-methyl-N-(4-methylpyrimidin-2-yl)-4-(1H-pyrazol-4-yl)-1,3-thiazol-2-amine
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|
C12H12N6S
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0406804
|
US9212196, Derivative 26
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|
C13H18NO7PS
|
1
|
| 1 |
EC50 = 1230 nM
|
|
|
|
CP0475231
|
US9212196, Derivative 24
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|
C13H17N2O10P
|
1
|
| 1 |
EC50 = 1590 nM
|
|
|
|
CP0853331
|
(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-(hydroxymethyl)ethanoic Acid
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|
C6H12NO7P
|
1
|
| 1 |
EC50 = 2900 nM
|
|
|
|
CP0374295
|
(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)-methyl]butan-1,4-dioic Acid
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|
C9H16NO8P
|
2
|
| 1 |
EC50 = 3500 nM
|
|
|
| 2 |
EC50 = 38000 nM
|
|
|
|
CP0418091
|
US9212196, Derivative 5
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|
C14H19N2O11P
|
1
|
| 1 |
EC50 = 3720 nM
|
|
|
|
CP0907064
|
(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]propenoic acid
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|
C7H12NO6P
|
2
|
| 1 |
EC50 = 5100 nM
|
|
|
| 2 |
EC50 = 7200 nM
|
|
|
|
CP0096656
|
(1R,2S)-4-aminocyclopentane-1,2,4-tricarboxylic acid
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|
C8H11NO6
|
1
|
| 1 |
EC50 = 5100 nM
|
|
|
|
CP0377002
|
(S)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid
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|
C7H14NO6P
|
2
|
| 1 |
EC50 = 6600 nM
|
|
|
| 2 |
EC50 = 7800 nM
|
|
|
|
CP0464832
|
US9212196, Derivative 21
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|
C14H17F3NO8P
|
1
|
| 1 |
EC50 = 6860 nM
|
|
|
|
CP0418088
|
US9212196, Derivative 23
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|
C14H18NO10P
|
1
|
| 1 |
EC50 = 7400 nM
|
|
|
|
CP0400028
|
(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-chloropropanoic Acid
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|
C7H13ClNO6P
|
2
|
| 1 |
EC50 = 8100 nM
|
|
|
| 2 |
EC50 = 8300 nM
|
|
|
|
CP0418095
|
US9212196, Derivative 34
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|
C14H19FNO8P
|
1
|
| 1 |
EC50 = 9170 nM
|
|
|
|
CP0482641
|
3-(4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
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|
C16H14F3N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0402516
|
US9212196, Derivative 6
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|
C14H19FNO9P
|
1
|
| 1 |
EC50 = 10300 nM
|
|
|
|
CP0413237
|
US9212196, Derivative 25
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|
C13H17N2O9PS
|
1
|
| 1 |
EC50 = 11500 nM
|
|
|
|
CP0002355
|
(2S)-2-aminopentanedioic acid
Show/Hide
|
C5H9NO4
|
1
|
| 1 |
EC50 = 14010 nM
|
|
|
|
CP0418093
|
US9212196, Derivative 18
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|
C15H20NO11P
|
1
|
| 1 |
EC50 = 14100 nM
|
|
|
|
CP0418089
|
US9212196, Derivative 29
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|
C14H20NO8P
|
1
|
| 1 |
EC50 = 14300 nM
|
|
|
|
CP0374294
|
(3S)-4-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-butanoic Acid
Show/Hide
|
C8H16NO6P
|
2
|
| 1 |
EC50 = 18000 nM
|
|
|
| 2 |
EC50 = 19000 nM
|
|
|
|
CP0418086
|
US9212196, Derivative 3
Show/Hide
|
C14H20NO9P
|
1
|
| 1 |
EC50 = 18400 nM
|
|
|
|
CP0845512
|
(+/-)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid
Show/Hide
|
C7H14NO6P
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
|
CP0066050
|
(1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid
Show/Hide
|
C8H11NO6
|
1
|
| 1 |
EC50 = 20790 nM
|
|
|
|
CP0418097
|
US9212196, Derivative 10
Show/Hide
|
C15H22NO8P
|
1
|
| 1 |
EC50 = 21900 nM
|
|
|
|
CP0406806
|
US9212196, Derivative 19
Show/Hide
|
C15H22NO9P
|
1
|
| 1 |
EC50 = 25000 nM
|
|
|
|
CP0493272
|
US9212196, Derivative 4
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|
C15H22NO10P
|
1
|
| 1 |
EC50 = 27200 nM
|
|
|
|
CP0418098
|
US9212196, Derivative 28
Show/Hide
|
C13H16F2NO8P
|
1
|
| 1 |
EC50 = 27500 nM
|
|
|
|
CP0418087
|
US9212196, Derivative 13
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|
C13H20NO7P
|
1
|
| 1 |
EC50 = 28000 nM
|
|
|
|
CP0561457
|
US9212196, Derivative 8
Show/Hide
|
C14H19INO9P
|
1
|
| 1 |
EC50 = 28000 nM
|
|
|
|
CP0442807
|
US9212196, Derivative 2
Show/Hide
|
C13H18NO8P
|
1
|
| 1 |
EC50 = 29200 nM
|
|
|
|
CP0391280
|
3-[3-[(2-cyclopentyl-1-oxo-3H-isoindol-5-yl)oxymethyl]phenyl]-4-methoxybenzoic acid
Show/Hide
|
C28H27NO5
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0397657
|
2-chloro-5-[3-(2-cyclopentyl-1-oxo-3H-isoindol-5-yl)phenyl]benzoic acid
Show/Hide
|
C26H22ClNO3
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0397658
|
2-chloro-5-[3-[(2-cyclopropyl-3-oxo-1,2-benzothiazol-6-yl)oxymethyl]phenyl]benzoic acid
Show/Hide
|
C24H18ClNO4S
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0463911
|
US9212196, Derivative 22
Show/Hide
|
C13H18NO9P
|
1
|
| 1 |
EC50 = 34000 nM
|
|
|
|
CP0418096
|
US9212196, Derivative 35
Show/Hide
|
C14H19ClNO8P
|
1
|
| 1 |
EC50 = 38200 nM
|
|
|
|
CP0418092
|
US9212196, Derivative 7
Show/Hide
|
C14H19ClNO9P
|
1
|
| 1 |
EC50 = 44000 nM
|
|
|
|
CP0905965
|
(3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-ethylphosphonate
Show/Hide
|
C6H15NO7P2
|
1
|
| 1 |
EC50 = 48000 nM
|
|
|
|
CP0413236
|
US9212196, Derivative 12
Show/Hide
|
C14H20NO7P
|
1
|
| 1 |
EC50 = 48700 nM
|
|
|
|
CP0402517
|
US9212196, Derivative 11
Show/Hide
|
C14H18NO7P
|
1
|
| 1 |
EC50 = 49000 nM
|
|
|
|
CP0490836
|
(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-methylpropanoic Acid
Show/Hide
|
C8H16NO6P
|
1
|
| 1 |
EC50 = 53000 nM
|
|
|
|
CP0418094
|
US9212196, Derivative 20
Show/Hide
|
C14H17F3NO9P
|
1
|
| 1 |
EC50 = 55600 nM
|
|
|
|
CP0410794
|
(R)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid
Show/Hide
|
C7H14NO6P
|
1
|
| 1 |
EC50 = 58000 nM
|
|
|
|
CP0377001
|
(2S)-2-Amino-5-[(hydroxy)phosphinyl]pentanoic Acid
Show/Hide
|
C5H12NO4P
|
1
|
| 1 |
EC50 = 73000 nM
|
|
|
|
CP0514300
|
(3S)-3-[((3-Amino-3-carboxylate)propyl)(hydroxy)phosphinate]-2-(2-hydroxyethyl)propanoate
Show/Hide
|
C9H18NO7P
|
1
|
| 1 |
EC50 = 76000 nM
|
|
|
|
CP0920930
|
(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)hydroxymethyl]cyclopropane-1-carboxylic Acid hydrochloride
Show/Hide
|
C9H17ClNO7P
|
1
|
| 1 |
EC50 = 91000 nM
|
|
|
|
CP0902261
|
(3S)-4-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-furanone
Show/Hide
|
C8H14NO6P
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0932553
|
(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)-methyl]oxotetrahydrofuran-3-yl
Show/Hide
|
C9H16NO6P
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0418090
|
US9212196, Derivative 33
Show/Hide
|
C14H17F3NO7P
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0442808
|
US9212196, Derivative 30
Show/Hide
|
C13H18NO7P
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0475232
|
US9212196, Derivative 32
Show/Hide
|
C14H17F3NO8P
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0389571
|
6-(2,4-dimethylphenyl)-2-ethyl-6,7-dihydro-5H-1,3-benzoxazol-4-one
Show/Hide
|
C17H19NO2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0416254
|
7-(4-fluorophenyl)-2-[[2-(trifluoromethyl)pyridin-4-yl]oxymethyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
Show/Hide
|
C20H13F4N5O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
|
CP0416287
|
2-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-7-(4-fluorophenyl)thieno[3,2-b]pyridine-5-carboxamide
Show/Hide
|
C21H22FN3O2S
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
