Compound ID |
Compound Name |
Compound Formula |
CP0041262
|
5-chloro-2-[(4-methylpiperazin-1-yl)carbonyl]-1H-indole
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|
C14H16ClN3O
|
1
|
1 |
EC50 = 2.399 nM
|
|
|
CP0173066
|
2,4-diamino-5,6-disubstituted pyrimidine, 11
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|
C18H23N5
|
1
|
1 |
EC50 = 4.365 nM
|
|
|
CP0094765
|
14-fluoro-6-(piperazin-1-yl)-3,5-diazatricyclo[9.4.0.0^{2,7}]pentadeca-1(15),2(7),3,5,11,13-hexaen-4-amine
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|
C17H20FN5
|
1
|
1 |
EC50 = 4.786 nM
|
|
|
CP0205085
|
2,4-diamino-5,6-disubstituted pyrimidine, 10
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|
C17H21N5
|
1
|
1 |
EC50 = 5.754 nM
|
|
|
CP0173068
|
2,4-diamino-5,6-disubstituted pyrimidine, 12
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|
C17H21N5
|
1
|
1 |
EC50 = 9.12 nM
|
|
|
CP0173069
|
5-chloro-2-(piperazin-1-ylcarbonyl)-1H-indole
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|
C13H14ClN3O
|
1
|
1 |
EC50 = 17.78 nM
|
|
|
CP0198951
|
2,4-diamino-5,6-disubstituted pyrimidine, 9
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|
C17H21N5
|
1
|
1 |
EC50 = 18.2 nM
|
|
|
CP0044460
|
N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
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|
C15H24N4S
|
1
|
1 |
EC50 = 28.18 nM
|
|
|
CP0229853
|
2,4-diamino-5,6-disubstituted pyrimidine, 14
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|
C19H25N5
|
1
|
1 |
EC50 = 45.71 nM
|
|
|
CP0388279
|
4-[(1E,3E)-4-[1-[4-(1H-imidazol-5-yl)butyl]-2,6-dimethylpyridin-1-ium-4-yl]buta-1,3-dienyl]-N,N-dimethylaniline;2,2,2-trifluoroacetate;2,2,2-trifluoroacetic acid
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|
C30H34F6N4O4
|
1
|
1 |
EC50 = 50.12 nM
|
|
|
CP0036920
|
2-(1H-imidazol-4-yl)ethan-1-amine
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|
C5H9N3
|
1
|
1 |
EC50 = 94 nM
|
|
|
CP0286034
|
2-Aminopyrimidine analog., 25
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|
C15H16N6
|
1
|
1 |
EC50 = 102.33 nM
|
|
|
CP0068173
|
2-Aminopyrimidine analog., 4
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|
C16H18N6
|
1
|
1 |
EC50 = 123.03 nM
|
|
|
CP0382899
|
1-cyano-2-[[(1S,3S)-3-(1H-imidazol-5-yl)cyclopentyl]methyl]-3-(2-phenylsulfanylethyl)guanidine
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|
C19H24N6S
|
1
|
1 |
EC50 = 166 nM
|
|
|
CP0377316
|
1-cyano-3-[[(1S,3S)-3-(1H-imidazol-5-yl)cyclopentyl]methyl]-2-methylguanidine
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|
C12H18N6
|
1
|
1 |
EC50 = 538 nM
|
|
|
CP0377318
|
1-cyano-2-[[(1R,3R)-3-(1H-imidazol-5-yl)cyclopentyl]methyl]-3-(2-phenylsulfanylethyl)guanidine
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|
C19H24N6S
|
1
|
1 |
EC50 = 589 nM
|
|
|
CP0823737
|
SID50106398
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|
C5H11Cl2N3
|
1
|
1 |
EC50 = 2344.23 nM
|
|
|
CP0382908
|
1-cyano-3-[[(1R,3R)-3-(1H-imidazol-5-yl)cyclopentyl]methyl]-2-methylguanidine
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|
C12H18N6
|
1
|
1 |
EC50 = 3631 nM
|
|
|
CP0224333
|
4-[(E)-2-(3-chlorophenyl)ethenyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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|
C16H19ClN6
|
1
|
1 |
Ki = 854 nM
|
|
|