| Compound ID |
Compound Name |
Compound Formula |
|
CP0511766
|
1-[2-[(E)-[2-(2,4-dichlorophenyl)phenyl]methylideneamino]oxyethyl]-3,6-dihydro-2H-pyridine-5-carboxylic acid
Show/Hide
|
C21H20Cl2N2O3
|
3
|
| 1 |
IC50 = 5.129 nM
|
|
|
| 2 |
IC50 = 5.37 nM
|
|
|
| 3 |
Ki = 5.129 nM
|
|
|
|
CP0426741
|
1-[2-[(E)-[2-(2,4-dichlorophenyl)phenyl]methylideneamino]oxyethyl]-3,6-dihydro-2H-pyridine-5-carboxylic acid;hydrochloride
Show/Hide
|
C21H21Cl3N2O3
|
2
|
| 1 |
IC50 = 5.37 nM
|
|
|
| 2 |
Ki = 5.129 nM
|
|
|
|
CP0378790
|
(R)-1-{2-[2,2-Bis-(3-methyl-thiophen-2-yl)-vinyloxy]-ethyl}-piperidine-3-carboxylic acid; hydrochloride
Show/Hide
|
C20H25NO3S2
|
1
|
| 1 |
IC50 = 14.13 nM
|
|
|
|
CP0402837
|
1-[2-[(E)-[3-(2,4-dichlorophenyl)thiophen-2-yl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
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|
C19H21Cl3N2O3S
|
2
|
| 1 |
IC50 = 28.18 nM
|
|
|
| 2 |
Ki = 11.75 nM
|
|
|
|
CP0438345
|
(3R)-1-[2-[(E)-[2-(2-chloro-4-fluorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23Cl2FN2O3
|
2
|
| 1 |
IC50 = 32.36 nM
|
|
|
| 2 |
Ki = 2.818 nM
|
|
|
|
CP0221365
|
(R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)piperidine-3-carboxylic acid hydrochloride
Show/Hide
|
C20H25NO2S2
|
6
|
| 1 |
IC50 = 37.15 nM
|
|
|
| 2 |
IC50 = 131.83 nM
|
|
|
| 3 |
Ki = 27.54 nM
|
|
|
| 4 |
Ki = 37.15 nM
|
|
|
| 5 |
Ki = 38.9 nM
|
|
|
| 6 |
Ki = 54.95 nM
|
|
|
|
CP0402841
|
1-[2-[(E)-[2-(2,4-dichlorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23Cl3N2O3
|
2
|
| 1 |
IC50 = 38.9 nM
|
|
|
| 2 |
Ki = 10.47 nM
|
|
|
|
CP0384440
|
1-[2-[(E)-[2-(2,4-difluorophenyl)phenyl]methylideneamino]oxyethyl]-3,6-dihydro-2H-pyridine-5-carboxylic acid;hydrochloride
Show/Hide
|
C21H21ClF2N2O3
|
2
|
| 1 |
IC50 = 56.23 nM
|
|
|
| 2 |
Ki = 4.467 nM
|
|
|
|
CP0384438
|
(3R)-1-[2-[(E)-[2-(2,4-dichlorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23Cl3N2O3
|
2
|
| 1 |
IC50 = 60.26 nM
|
|
|
| 2 |
Ki = 5.888 nM
|
|
|
|
CP0387090
|
1-[2-[(2E)-2-[[2-(2,4-dichlorophenyl)phenyl]methylidene]hydrazinyl]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C21H23Cl2N3O2
|
2
|
| 1 |
IC50 = 61.24 nM
|
|
|
| 2 |
Ki = 8.054 nM
|
|
|
|
CP0440032
|
1-[2-[(E)-[2-(2-chloro-4-fluorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23Cl2FN2O3
|
2
|
| 1 |
IC50 = 66.07 nM
|
|
|
| 2 |
Ki = 10 nM
|
|
|
|
CP0402836
|
1-[2-[(E)-[2-(2,4-difluorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23ClF2N2O3
|
2
|
| 1 |
IC50 = 85.11 nM
|
|
|
| 2 |
Ki = 13.8 nM
|
|
|
|
CP0416830
|
(3R)-1-[4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 97.72 nM
|
|
|
|
CP0537534
|
(3R)-1-[2-[2-(2-benzylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
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|
C23H29NO3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0564770
|
1-[4-(2-phenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23NO2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0426740
|
(3R)-1-[2-[(E)-[2-(2,4-difluorophenyl)phenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H23ClF2N2O3
|
2
|
| 1 |
IC50 = 102.33 nM
|
|
|
| 2 |
Ki = 5.888 nM
|
|
|
|
CP0416804
|
1-[4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
|
CP0876464
|
(E)-1-(2-(2-((4'-chloro-2'-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23ClFN3O2
|
2
|
| 1 |
IC50 = 126.18 nM
|
|
|
| 2 |
Ki = 24.72 nM
|
|
|
|
CP0880744
|
(E)-1-(2-(2-((2',4'-difluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23F2N3O2
|
2
|
| 1 |
IC50 = 128.53 nM
|
|
|
| 2 |
Ki = 35.56 nM
|
|
|
|
CP0043886
|
1-[2-(benzhydrylideneamino)oxyethyl]-3,6-dihydro-2H-pyridine-5-carboxylic acid
Show/Hide
|
C21H22N2O3
|
3
|
| 1 |
IC50 = 147.91 nM
|
|
|
| 2 |
IC50 <= 530 nM
|
|
|
| 3 |
Kd = 26.5 nM
|
|
|
|
CP0575675
|
1-[(E)-4-(2-phenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H25NO2
|
1
|
| 1 |
IC50 = 162.18 nM
|
|
|
|
CP0392411
|
1-[(E)-5,5-diphenylpent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H27NO2
|
2
|
| 1 |
IC50 = 165.96 nM
|
|
|
| 2 |
Ki = 30.9 nM
|
|
|
|
CP0543641
|
1-[2-[(E)-[2-(2,4-dichlorophenyl)-5-fluorophenyl]methylideneamino]oxyethyl]piperidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H22Cl3FN2O3
|
2
|
| 1 |
IC50 = 169.82 nM
|
|
|
| 2 |
Ki = 16.98 nM
|
|
|
|
CP0476254
|
(3R)-1-[4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 181.97 nM
|
|
|
|
CP0519707
|
1-[4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 229.09 nM
|
|
|
|
CP0848808
|
(E)-1-(2-(2-((2',4',6'-trifluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H22F3N3O2
|
2
|
| 1 |
IC50 = 254.68 nM
|
|
|
| 2 |
Ki = 30.62 nM
|
|
|
|
CP0398819
|
(3R)-1-[2-[2-[4-(naphthalen-1-yldiazenyl)phenyl]ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H29N3O3
|
2
|
| 1 |
IC50 = 269.15 nM
|
|
|
| 2 |
IC50 = 794.33 nM
|
|
|
|
CP0851602
|
(E)-1-(2-(2-((2'-chloro-4'-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23ClFN3O2
|
2
|
| 1 |
IC50 = 291.74 nM
|
|
|
| 2 |
Ki = 14.62 nM
|
|
|
|
CP0382886
|
1-[2-[(Z)-2-[5-fluoro-2-[(2-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 302 nM
|
|
|
|
CP0387840
|
1-[2-[(Z)-2-[5-fluoro-2-[(3-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 302 nM
|
|
|
|
CP0387842
|
1-[2-[(Z)-2-[4-fluoro-2-(4-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 338.84 nM
|
|
|
|
CP0449847
|
1-[2-[(Z)-2-(2-benzylphenyl)ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0398820
|
(3R)-1-[2-[2-[3-(naphthalen-1-yldiazenyl)phenyl]ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H29N3O3
|
2
|
| 1 |
IC50 = 407.38 nM
|
|
|
| 2 |
IC50 = 1659.59 nM
|
|
|
|
CP0392774
|
(3R)-1-[4-(4-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 416.87 nM
|
|
|
|
CP0392775
|
(3R)-1-[4-(3-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 416.87 nM
|
|
|
|
CP0410624
|
1-(5,5,5-triphenylpent-3-ynyl)piperidine-3-carboxylic acid
Show/Hide
|
C29H29NO2
|
2
|
| 1 |
IC50 = 426.58 nM
|
|
|
| 2 |
Ki = 91.2 nM
|
|
|
|
CP0879098
|
(E)-1-(2-(2-((2'-chlorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H24ClN3O2
|
2
|
| 1 |
IC50 = 478.63 nM
|
|
|
| 2 |
Ki = 65.46 nM
|
|
|
|
CP0886428
|
(E)-1-(2-(2-((2'-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H24FN3O2
|
2
|
| 1 |
IC50 = 528.45 nM
|
|
|
| 2 |
Ki = 121.9 nM
|
|
|
|
CP0399440
|
1-[2-[(Z)-2-[4-fluoro-2-[(2-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0486228
|
1-[4-(4-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 645.65 nM
|
|
|
|
CP0037615
|
1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxylic acid
Show/Hide
|
C22H25NO2
|
2
|
| 1 |
IC50 = 691.83 nM
|
|
|
| 2 |
Ki = 186.21 nM
|
|
|
|
CP0857264
|
(R)-1-(4,4-diphenylbut-3-enyl)piperidine-3-carboxylic acid hydrochloride
Show/Hide
|
C22H26ClNO2
|
1
|
| 1 |
IC50 = 691.83 nM
|
|
|
|
CP0449846
|
1-[2-[(Z)-2-[4-fluoro-2-(2-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 758.58 nM
|
|
|
|
CP0387088
|
1-[(E)-5-[2-(2,4-dichlorophenyl)phenyl]pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25Cl2NO2
|
2
|
| 1 |
IC50 = 769.13 nM
|
|
|
| 2 |
Ki = 117.49 nM
|
|
|
|
CP0432402
|
1-[2-[(Z)-2-[4-fluoro-2-(3-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0398821
|
(3R)-1-[2-[2-[4-(naphthalen-1-yldiazenyl)phenyl]ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H29N3O3
|
1
|
| 1 |
IC50 = 794.33 nM
|
|
|
|
CP0909026
|
(E)-1-(2-(2-((2',4'-dimethylbiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H29N3O2
|
2
|
| 1 |
IC50 = 835.6 nM
|
|
|
| 2 |
Ki = 73.28 nM
|
|
|
|
CP0521061
|
1-[4-(3-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 891.25 nM
|
|
|
|
CP0886429
|
(E)-1-(2-(2-((4'-chlorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H24ClN3O2
|
2
|
| 1 |
IC50 = 972.75 nM
|
|
|
| 2 |
Ki = 172.98 nM
|
|
|
|
CP0848813
|
(E)-1-(2-(2-((2',6'-difluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23F2N3O2
|
2
|
| 1 |
IC50 = 997.7 nM
|
|
|
| 2 |
Ki = 130.92 nM
|
|
|
|
CP0480748
|
(3R)-1-[4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0474167
|
1-[(Z)-5,5,5-triphenylpent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C29H31NO2
|
2
|
| 1 |
IC50 = 1000 nM
|
|
|
| 2 |
Ki = 512.86 nM
|
|
|
|
CP0397571
|
1-[2-[(Z)-2-[5-fluoro-2-[(4-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 1096.48 nM
|
|
|
|
CP0396477
|
1-[2-[(Z)-2-[4-fluoro-2-[(4-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 1174.9 nM
|
|
|
|
CP0848805
|
(E)-1-(2-(2-((2'-chloro-4-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23ClFN3O2
|
2
|
| 1 |
IC50 = 1233.1 nM
|
|
|
| 2 |
Ki = 104.47 nM
|
|
|
|
CP0416808
|
(3R)-1-[4-(4-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 1445.44 nM
|
|
|
|
CP0871607
|
(E)-1-(2-(2-((2',3'-difluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23F2N3O2
|
2
|
| 1 |
IC50 = 1499.68 nM
|
|
|
| 2 |
Ki = 204.17 nM
|
|
|
|
CP0886420
|
(E)-1-(2-(2-((2'-methylbiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O2
|
2
|
| 1 |
IC50 = 1563.15 nM
|
|
|
| 2 |
Ki = 215.77 nM
|
|
|
|
CP0513090
|
(3R)-1-[2-[2-[3-(naphthalen-1-yldiazenyl)phenyl]ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H29N3O3
|
1
|
| 1 |
IC50 = 1659.59 nM
|
|
|
|
CP0851604
|
(E)-1-(2-(2-((2',4-difluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23F2N3O2
|
2
|
| 1 |
IC50 = 1725.84 nM
|
|
|
| 2 |
Ki = 264.24 nM
|
|
|
|
CP0872755
|
(E)-1-(2-(2-((4'-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H24FN3O2
|
2
|
| 1 |
IC50 = 1794.73 nM
|
|
|
| 2 |
Ki = 284.45 nM
|
|
|
|
CP0376462
|
1-[2-[(E)-2-[4-fluoro-2-(4-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 1862.09 nM
|
|
|
|
CP0452841
|
1-[2-[2-(4-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
2
|
| 1 |
IC50 = 1905.46 nM
|
|
|
| 2 |
IC50 = 4570.88 nM
|
|
|
|
CP0390623
|
1-[2-[(E)-[2-(2-fluoro-6-methoxyphenyl)phenyl]methylideneamino]oxyethyl]pyrrolidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C21H24ClFN2O4
|
2
|
| 1 |
IC50 = 1905.46 nM
|
|
|
| 2 |
Ki = 407.38 nM
|
|
|
|
CP0416810
|
1-[4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 1949.84 nM
|
|
|
|
CP0851603
|
(E)-1-(2-(2-((4'-chloro-4-fluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23ClFN3O2
|
2
|
| 1 |
IC50 = 1958.84 nM
|
|
|
| 2 |
Ki = 234.42 nM
|
|
|
|
CP0549068
|
(3R)-1-(3-fluoren-9-ylidenepropyl)piperidine-3-carboxylic acid
Show/Hide
|
C22H23NO2
|
1
|
| 1 |
IC50 = 1995.26 nM
|
|
|
|
CP0397783
|
(2S)-2-[(2R)-1-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl]pyrrolidin-2-yl]-2-hydroxyacetic acid
Show/Hide
|
C20H25NO3S2
|
2
|
| 1 |
IC50 = 2137.96 nM
|
|
|
| 2 |
Ki = 102.33 nM
|
|
|
|
CP0848806
|
(E)-1-(2-(2-((2'-fluoro-6'-methoxybiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C22H26FN3O3
|
2
|
| 1 |
IC50 = 2249.05 nM
|
|
|
| 2 |
Ki = 442.59 nM
|
|
|
|
CP0379824
|
(2S)-2-[(2R)-1-(4,4-diphenylbut-3-enyl)pyrrolidin-2-yl]-2-hydroxyacetic acid
Show/Hide
|
C22H25NO3
|
2
|
| 1 |
IC50 = 2290.87 nM
|
|
|
| 2 |
Ki = 144.54 nM
|
|
|
|
CP0391421
|
1-[2-[(E)-[2-(2,4-dichlorophenyl)phenyl]methylideneamino]oxyethyl]pyrrolidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C20H21Cl3N2O3
|
2
|
| 1 |
IC50 = 2290.87 nM
|
|
|
| 2 |
Ki = 389.05 nM
|
|
|
|
CP0560522
|
1-[4-(4-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
|
1
|
| 1 |
IC50 = 2570.4 nM
|
|
|
|
CP0525723
|
1-[2-[(Z)-2-[5-fluoro-2-(3-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 2630.27 nM
|
|
|
|
CP0397521
|
1-[2-[(E)-2-[4-fluoro-2-[(2-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 2691.53 nM
|
|
|
|
CP0886427
|
(E)-1-(2-(2-((2',4'-bis(trifluoromethyl)biphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H23F6N3O2
|
2
|
| 1 |
IC50 = 2824.88 nM
|
|
|
| 2 |
Ki = 170.22 nM
|
|
|
|
CP0905398
|
(E)-1-(5-(2',4'-difluorobiphenyl-2-yl)pent-4-enyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO2
|
2
|
| 1 |
IC50 = 2837.92 nM
|
|
|
| 2 |
Ki = 591.56 nM
|
|
|
|
CP0928983
|
(E)-1-(2-(2-(2-(thiophen-2-yl)benzylidene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C19H23N3O2S
|
2
|
| 1 |
IC50 = 2870.78 nM
|
|
|
| 2 |
Ki = 590.2 nM
|
|
|
|
CP0397522
|
1-[2-[(Z)-2-[5-fluoro-2-(2-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 3019.95 nM
|
|
|
|
CP0476251
|
1-[5-[4-(naphthalen-1-yldiazenyl)phenyl]pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H27N3O2
|
1
|
| 1 |
IC50 = 3019.95 nM
|
|
|
|
CP0410387
|
1-[2-[2-(3-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
2
|
| 1 |
IC50 = 3162.28 nM
|
|
|
| 2 |
IC50 = 4168.69 nM
|
|
|
|
CP0851611
|
(E)-1-(2-(2-((3',4'-difluorobiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H23F2N3O2
|
2
|
| 1 |
IC50 = 3318.94 nM
|
|
|
| 2 |
Ki = 625.17 nM
|
|
|
|
CP0879100
|
(E)-1-(5-(2'-fluorobiphenyl-2-yl)pent-4-enyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H26FNO2
|
2
|
| 1 |
IC50 = 3334.26 nM
|
|
|
| 2 |
Ki = 647.14 nM
|
|
|
|
CP0411793
|
(2R)-2-[(2R)-1-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl]pyrrolidin-2-yl]-2-hydroxyacetic acid
Show/Hide
|
C20H25NO3S2
|
2
|
| 1 |
IC50 = 3388.44 nM
|
|
|
| 2 |
Ki = 1071.52 nM
|
|
|
|
CP0868760
|
(E)-1-(2-(2-((4'-methylbiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O2
|
2
|
| 1 |
IC50 = 3404.08 nM
|
|
|
| 2 |
Ki = 473.15 nM
|
|
|
|
CP0848809
|
(E)-1-(5-(2'-chlorobiphenyl-2-yl)pent-4-enyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H26ClNO2
|
2
|
| 1 |
IC50 = 3564.51 nM
|
|
|
| 2 |
Ki = 833.68 nM
|
|
|
|
CP0424089
|
1-[4,4-bis(4-methoxyphenyl)but-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C24H27NO4
|
2
|
| 1 |
IC50 = 3715.35 nM
|
|
|
| 2 |
Ki = 1096.48 nM
|
|
|
|
CP0889397
|
(E)-1-(5-(2'-chloro-4'-fluorobiphenyl-2-yl)pent-4-enyl)piperidine-3-carboxylic acid
Show/Hide
|
C23H25ClFNO2
|
2
|
| 1 |
IC50 = 3990.25 nM
|
|
|
| 2 |
Ki = 312.61 nM
|
|
|
|
CP0363584
|
4-((4,4-bis(3-methylthiophen-2-yl)but-3-enyl)(methyl)amino)-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol
Show/Hide
|
C22H26N2O2S2
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0486232
|
1-[5-(3-phenyldiazenylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 = 4073.8 nM
|
|
|
|
CP0508407
|
1-[(E)-4,4,4-tris(1-benzofuran-5-yl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C34H29NO5
|
2
|
| 1 |
IC50 = 4073.8 nM
|
|
|
| 2 |
Ki = 2137.96 nM
|
|
|
|
CP0324831
|
2-pyrrolidin-3-ylacetic acid
Show/Hide
|
C6H11NO2
|
1
|
| 1 |
IC50 = 4073.8 nM
|
|
|
|
CP0482503
|
1-[2-[(E)-2-(2-benzylphenyl)ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
IC50 = 4168.69 nM
|
|
|
|
CP0556642
|
1-[2-[2-(3-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
1
|
| 1 |
IC50 = 4168.69 nM
|
|
|
|
CP0416803
|
(3R)-1-[4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 4265.8 nM
|
|
|
|
CP0449849
|
1-[2-[(E)-2-[4-fluoro-2-[(4-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 4570.88 nM
|
|
|
|
CP0846185
|
(rac)-3-[(4,4-Diphenylbut-3-enyl)amino]butanoic acid
Show/Hide
|
C20H23NO2
|
1
|
| 1 |
IC50 = 4570.88 nM
|
|
|
|
CP0513091
|
1-[2-[2-(4-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
1
|
| 1 |
IC50 = 4570.88 nM
|
|
|
|
CP0521060
|
1-[4-(3-phenyldiazenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
IC50 = 4786.3 nM
|
|
|
|
CP0435653
|
1-[2-[(E)-[2-(2-chloro-4-fluorophenyl)phenyl]methylideneamino]oxyethyl]pyrrolidine-3-carboxylic acid;hydrochloride
Show/Hide
|
C20H21Cl2FN2O3
|
2
|
| 1 |
IC50 = 4786.3 nM
|
|
|
| 2 |
Ki = 691.83 nM
|
|
|
|
CP0519708
|
1-[5-[4-(naphthalen-1-yldiazenyl)phenyl]pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H27N3O2
|
1
|
| 1 |
IC50 = 4897.79 nM
|
|
|
|
CP0851612
|
(E)-1-(2-(2-(biphenyl-2-ylmethylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C21H25N3O2
|
2
|
| 1 |
IC50 = 4920.4 nM
|
|
|
| 2 |
Ki = 651.63 nM
|
|
|
|
CP0398822
|
1-[2-[2-(2-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
1
|
| 1 |
IC50 = 5495.41 nM
|
|
|
|
CP0415304
|
1-[2-[2-(2-phenyldiazenylphenyl)ethoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H27N3O3
|
2
|
| 1 |
IC50 = 5495.41 nM
|
|
|
| 2 |
IC50 = 10715.19 nM
|
|
|
|
CP0521062
|
1-[(E)-5-(4-phenyldiazenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H27N3O2
|
1
|
| 1 |
IC50 = 5754.4 nM
|
|
|
|
CP0476252
|
1-[4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H27N3O2
|
1
|
| 1 |
IC50 = 5888.44 nM
|
|
|
|
CP0476253
|
1-[5-[4-(naphthalen-1-yldiazenyl)phenyl]pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
IC50 = 6165.95 nM
|
|
|
|
CP0549067
|
4-amino-N-[(4-chlorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H34ClN3O
|
2
|
| 1 |
IC50 = 6309.57 nM
|
|
|
| 2 |
IC50 = 25118.86 nM
|
|
|
|
CP0549069
|
4-amino-N-[(4-fluorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H34FN3O
|
2
|
| 1 |
IC50 = 6309.57 nM
|
|
|
| 2 |
IC50 = 10964.78 nM
|
|
|
|
CP0476249
|
1-[4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H25N3O2
|
1
|
| 1 |
IC50 = 6456.54 nM
|
|
|
|
CP0486227
|
1-[(E)-5-[4-(naphthalen-1-yldiazenyl)phenyl]pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
IC50 = 6456.54 nM
|
|
|
|
CP0451186
|
4-amino-N-[(2-chlorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H34ClN3O
|
2
|
| 1 |
IC50 = 6606.93 nM
|
|
|
| 2 |
IC50 = 13489.63 nM
|
|
|
|
CP0387841
|
1-[2-[(E)-2-[5-fluoro-2-[(3-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 6760.83 nM
|
|
|
|
CP0380468
|
1-[2-[(Z)-2-(2-benzoylphenyl)ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25NO4
|
1
|
| 1 |
IC50 = 7079.46 nM
|
|
|
|
CP0487035
|
5-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-4,5,6,7-tetrahydro-1,2-benzoxazol-3-one
Show/Hide
|
C22H26N2O2S2
|
1
|
| 1 |
IC50 = 7079.46 nM
|
|
|
|
CP0000066
|
4-amino-n-[2,3-3H]butyric acid
Show/Hide
|
C4H9NO2
|
1
|
| 1 |
IC50 = 7244.36 nM
|
|
|
|
CP0418966
|
4-amino-N-[(4-methylphenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C31H37N3O
|
1
|
| 1 |
IC50 = 7244.36 nM
|
|
|
|
CP0872754
|
(E)-1-(2-(2-((4'-fluoro-2'-methoxybiphenyl-2-yl)methylene)hydrazinyl)ethyl)piperidine-3-carboxylic acid
Show/Hide
|
C22H26FN3O3
|
2
|
| 1 |
IC50 = 7345.14 nM
|
|
|
| 2 |
Ki = 760.33 nM
|
|
|
|
CP0486229
|
1-[4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H27N3O2
|
1
|
| 1 |
IC50 = 7413.1 nM
|
|
|
|
CP0423069
|
1-[2-[(Z)-2-[5-fluoro-2-(4-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 7585.78 nM
|
|
|
|
CP0392773
|
1-[5-(4-phenyldiazenylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 = 7585.78 nM
|
|
|
|
CP0511795
|
4-amino-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2-chlorophenyl)methyl]butanamide
Show/Hide
|
C26H32ClN3OS2
|
2
|
| 1 |
IC50 = 7585.78 nM
|
|
|
| 2 |
Ki = 11748.98 nM
|
|
|
|
CP0311493
|
(2S,3S)-1-(benzylamino)-3-(3,3-diphenylpropylamino)-4-phenylbutan-2-ol
Show/Hide
|
C32H36N2O
|
1
|
| 1 |
IC50 = 7590 nM
|
|
|
|
CP0406400
|
(2R,4R)-2-(4-benzhydrylidenepiperidin-1-yl)-N-benzyl-4-hydroxypentanamide
Show/Hide
|
C30H34N2O2
|
1
|
| 1 |
IC50 = 7762.47 nM
|
|
|
|
CP0396652
|
1-[2-[(E)-2-[5-fluoro-2-(2-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 8128.31 nM
|
|
|
|
CP0531417
|
4-amino-N-benzyl-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H35N3O
|
2
|
| 1 |
IC50 = 8128.31 nM
|
|
|
| 2 |
IC50 = 16595.87 nM
|
|
|
|
CP0390166
|
1-[4,4-bis(4-methoxyphenyl)-5-phenylpent-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H33NO4
|
2
|
| 1 |
IC50 = 8317.64 nM
|
|
|
| 2 |
Ki = 2137.96 nM
|
|
|
|
CP0059522
|
(R)-Piperidine-3-carboxylic acid
Show/Hide
|
C6H11NO2
|
1
|
| 1 |
IC50 = 8511.38 nM
|
|
|
|
CP0171598
|
(RS)-nipecotic acid
Show/Hide
|
C6H11NO2
|
4
|
| 1 |
IC50 = 8511.38 nM
|
|
|
| 2 |
IC50 = 13182.57 nM
|
|
|
| 3 |
IC50 = 13304.54 nM
|
|
|
| 4 |
Ki = 58210.32 nM
|
|
|
|
CP0419669
|
4-amino-2-[4,4-diphenylbut-3-enyl(methyl)amino]-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C29H35N3O
|
2
|
| 1 |
IC50 = 8511.38 nM
|
|
|
| 2 |
Ki = 9120.11 nM
|
|
|
|
CP0846188
|
(rac)-3-({2-[2-(10H-Phenothiazin-10-yl)ethoxy]ethyl}amino)butanoic acid
Show/Hide
|
C20H24N2O3S
|
1
|
| 1 |
IC50 = 8709.64 nM
|
|
|
|
CP0411928
|
1-[(E)-4-[4-(naphthalen-1-yldiazenyl)phenyl]but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H27N3O2
|
1
|
| 1 |
IC50 = 8709.64 nM
|
|
|
|
CP0425215
|
4-acetamido-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2-chlorophenyl)methyl]butanamide
Show/Hide
|
C28H34ClN3O2S2
|
1
|
| 1 |
IC50 = 8709.64 nM
|
|
|
|
CP0396476
|
1-[2-[(E)-2-[5-fluoro-2-[(4-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 8912.51 nM
|
|
|
|
CP0511793
|
4-amino-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]butanamide
Show/Hide
|
C26H32ClN3OS2
|
2
|
| 1 |
IC50 = 9332.54 nM
|
|
|
| 2 |
Ki = 19952.62 nM
|
|
|
|
CP0534671
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C26H31ClN2O2S2
|
1
|
| 1 |
IC50 = 9332.54 nM
|
|
|
|
CP0391942
|
2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C29H31FN2O2
|
2
|
| 1 |
IC50 = 9772.37 nM
|
|
|
| 2 |
Ki = 11481.54 nM
|
|
|
|
CP0435652
|
2-(2,4,6-trifluorophenyl)benzaldehyde
Show/Hide
|
C13H7F3O
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0480746
|
1-[(E)-4-(4-phenyldiazenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H25N3O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0486231
|
1-[5-[3-(naphthalen-1-yldiazenyl)phenyl]pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0517070
|
N-[(4-chlorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H33ClN2O2
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0390468
|
1-(3-carbazol-9-ylpropyl)-4-(2-methoxyphenyl)piperidin-4-ol
Show/Hide
|
C27H30N2O2
|
1
|
| 1 |
IC50 = 10232.93 nM
|
|
|
|
CP0410008
|
1-[2-[(E)-2-[5-fluoro-2-[(2-fluorophenyl)methyl]phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25F2NO3
|
1
|
| 1 |
IC50 = 10232.93 nM
|
|
|
|
CP0484399
|
1-[(E)-4-(1-benzothiophen-5-yl)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H33NO4S
|
2
|
| 1 |
IC50 = 10232.93 nM
|
|
|
| 2 |
Ki = 3311.31 nM
|
|
|
|
CP0499667
|
N-benzyl-2-[4,4-diphenylbut-3-enyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
|
C28H32N2O2
|
1
|
| 1 |
IC50 = 10471.29 nM
|
|
|
|
CP0432401
|
1-[2-[(E)-2-[4-fluoro-2-(2-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
|
1
|
| 1 |
IC50 = 10715.19 nM
|
|
|
|
CP0548359
|
N-[(2S,3R)-4-[(3-tert-butylphenyl)methylamino]-3-hydroxy-1-phenylbutan-2-yl]-2,2-diphenylacetamide
Show/Hide
|
C35H40N2O2
|
1
|
| 1 |
IC50 = 10960 nM
|
|
|
|
CP0434412
|
4-amino-2-(4-benzhydrylidenepiperidin-1-yl)-N-benzylbutanamide
Show/Hide
|
C29H33N3O
|
2
|
| 1 |
IC50 = 10964.78 nM
|
|
|
| 2 |
Ki = 16595.87 nM
|
|
|
|
CP0440818
|
4-amino-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C29H32FN3O
|
2
|
| 1 |
IC50 = 10964.78 nM
|
|
|
| 2 |
Ki = 25118.86 nM
|
|
|
|
CP0506689
|
4-amino-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-chlorophenyl)methyl]butanamide
Show/Hide
|
C29H32ClN3O
|
2
|
| 1 |
IC50 = 10964.78 nM
|
|
|
| 2 |
Ki = 23988.33 nM
|
|
|
|
CP0390211
|
1-[4-(1-benzothiophen-5-yl)-4,4-bis(4-methoxyphenyl)but-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H31NO4S
|
2
|
| 1 |
IC50 = 10964.78 nM
|
|
|
| 2 |
Ki = 1905.46 nM
|
|
|
|
CP0419707
|
4-amino-N-[(2-chlorophenyl)methyl]-2-[4,4-diphenylbut-3-enyl(methyl)amino]butanamide
Show/Hide
|
C28H32ClN3O
|
3
|
| 1 |
IC50 = 10964.78 nM
|
|
|
| 2 |
IC50 = 12882.5 nM
|
|
|
| 3 |
Ki = 10964.78 nM
|
|
|
|
CP0440820
|
4-amino-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C30H35N3O
|
2
|
| 1 |
IC50 = 11220.18 nM
|
|
|
| 2 |
Ki = 29512.09 nM
|
|
|
|
CP0443496
|
4-amino-2-(4-benzhydrylpiperidin-1-yl)-N-[(4-chlorophenyl)methyl]butanamide
Show/Hide
|
C29H34ClN3O
|
2
|
| 1 |
IC50 = 11220.18 nM
|
|
|
| 2 |
Ki = 30199.52 nM
|
|
|
|
CP0392372
|
1-[(E)-4,4,5-tris(4-methoxyphenyl)pent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H37NO5
|
2
|
| 1 |
IC50 = 11220.18 nM
|
|
|
| 2 |
Ki = 3090.3 nM
|
|
|
|
CP0486489
|
4-amino-N-benzyl-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]butanamide
Show/Hide
|
C26H33N3OS2
|
2
|
| 1 |
IC50 = 11481.54 nM
|
|
|
| 2 |
Ki = 24547.09 nM
|
|
|
|
CP0542549
|
4-amino-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C27H35N3OS2
|
2
|
| 1 |
IC50 = 11481.54 nM
|
|
|
| 2 |
Ki = 18197.01 nM
|
|
|
|
CP0458153
|
3-[1-[5-[9-(4-methoxyphenyl)fluoren-9-yl]oxypentyl]imidazol-2-yl]propanoic acid
Show/Hide
|
C31H32N2O4
|
1
|
| 1 |
IC50 = 11748.98 nM
|
|
|
|
CP0487050
|
4-amino-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C26H32FN3OS2
|
2
|
| 1 |
IC50 = 11748.98 nM
|
|
|
| 2 |
Ki = 21877.62 nM
|
|
|
|
CP0893161
|
5-n-Dodecylaminomethyl-2-methoxyphenol
Show/Hide
|
C20H35NO2
|
1
|
| 1 |
IC50 = 12302.69 nM
|
|
|
|
CP0481429
|
4-amino-2-[4,4-diphenylbutyl(methyl)amino]-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C29H37N3O
|
2
|
| 1 |
IC50 = 12302.69 nM
|
|
|
| 2 |
Ki = 15488.17 nM
|
|
|
|
CP0476250
|
1-[5-[3-(naphthalen-1-yldiazenyl)phenyl]pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H27N3O2
|
1
|
| 1 |
IC50 = 12302.69 nM
|
|
|
|
CP0534831
|
1-[(E)-4-[3-(naphthalen-1-yldiazenyl)phenyl]but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C26H27N3O2
|
1
|
| 1 |
IC50 = 12302.69 nM
|
|
|
|
CP0511786
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2,4-difluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C26H30F2N2O2S2
|
1
|
| 1 |
IC50 = 12302.69 nM
|
|
|
|
CP0419668
|
4-amino-N-[(2-chlorophenyl)methyl]-2-[4,4-diphenylbutyl(methyl)amino]butanamide
Show/Hide
|
C28H34ClN3O
|
2
|
| 1 |
IC50 = 12589.25 nM
|
|
|
| 2 |
Ki = 21379.62 nM
|
|
|
|
CP0458152
|
(E)-3-[1-[5-[9-(4-methoxyphenyl)fluoren-9-yl]oxypentyl]imidazol-2-yl]prop-2-enoic acid
Show/Hide
|
C31H30N2O4
|
1
|
| 1 |
IC50 = 12589.25 nM
|
|
|
|
CP0546564
|
4-amino-N-[(4-chlorophenyl)methyl]-2-[4,4-diphenylbut-3-enyl(methyl)amino]butanamide
Show/Hide
|
C28H32ClN3O
|
2
|
| 1 |
IC50 = 12882.5 nM
|
|
|
| 2 |
Ki = 11220.18 nM
|
|
|
|
CP0487038
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C27H34N2O2S2
|
1
|
| 1 |
IC50 = 12882.5 nM
|
|
|
|
CP0886721
|
(rac)-3-({2-[2-(10,11-Dihydro-5H-dibenzo[b,f]azepin-5-yl)ethoxy]ethyl}amino)butanoic acid
Show/Hide
|
C22H28N2O3
|
1
|
| 1 |
IC50 = 13182.57 nM
|
|
|
|
CP0404028
|
2-(4-benzhydrylpiperidin-1-yl)-N-benzyl-4-hydroxybutanamide
Show/Hide
|
C29H34N2O2
|
1
|
| 1 |
IC50 = 13182.57 nM
|
|
|
|
CP0397318
|
4-amino-2-(4-benzhydrylpiperidin-1-yl)-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C30H37N3O
|
2
|
| 1 |
IC50 = 13182.57 nM
|
|
|
| 2 |
Ki = 16595.87 nM
|
|
|
|
CP0560437
|
1-[4,4,5-tris(4-methoxyphenyl)pent-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H35NO5
|
2
|
| 1 |
IC50 = 13182.57 nM
|
|
|
| 2 |
Ki = 1905.46 nM
|
|
|
|
CP0047120
|
1,2,3,6-tetrahydropyridine-5-carboxylic acid;hydrochloride
Show/Hide
|
C6H9NO2
|
1
|
| 1 |
IC50 = 13489.63 nM
|
|
|
|
CP0397316
|
4-amino-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(2-chlorophenyl)methyl]butanamide
Show/Hide
|
C29H32ClN3O
|
2
|
| 1 |
IC50 = 13489.63 nM
|
|
|
| 2 |
Ki = 10471.29 nM
|
|
|
|
CP0392600
|
1-[(E)-5,5-bis(4-methoxyphenyl)pent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C25H31NO4
|
2
|
| 1 |
IC50 = 13489.63 nM
|
|
|
| 2 |
Ki = 3235.94 nM
|
|
|
|
CP0511790
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-3-hydroxy-N-[[4-(trifluoromethyl)phenyl]methyl]propanamide
Show/Hide
|
C26H29F3N2O2S2
|
1
|
| 1 |
IC50 = 13489.63 nM
|
|
|
|
CP0561677
|
1-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]piperidine-3-carboxylic acid
Show/Hide
|
C24H27NO2
|
1
|
| 1 |
IC50 = 13489.63 nM
|
|
|
|
CP0396968
|
4-amino-2-[4,4-diphenylbut-3-enyl(methyl)amino]-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C28H32FN3O
|
2
|
| 1 |
IC50 = 13803.84 nM
|
|
|
| 2 |
Ki = 15848.93 nM
|
|
|
|
CP0481294
|
4-amino-2-(4-benzhydrylpiperidin-1-yl)-N-[(2-chlorophenyl)methyl]butanamide
Show/Hide
|
C29H34ClN3O
|
2
|
| 1 |
IC50 = 13803.84 nM
|
|
|
| 2 |
Ki = 25703.96 nM
|
|
|
|
CP0480750
|
1-[5-[3-(naphthalen-1-yldiazenyl)phenyl]pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H27N3O2
|
1
|
| 1 |
IC50 = 13803.84 nM
|
|
|
|
CP0534668
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C26H31ClN2O2S2
|
1
|
| 1 |
IC50 = 13803.84 nM
|
|
|
|
CP0567514
|
(2R)-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C26H31ClN2O2S2
|
2
|
| 1 |
IC50 = 13803.84 nM
|
|
|
| 2 |
Ki = 25703.96 nM
|
|
|
|
CP0418968
|
4-acetamido-N-[(4-methylphenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C33H39N3O2
|
1
|
| 1 |
IC50 = 13803.84 nM
|
|
|
|
CP0561678
|
4-acetamido-N-[(4-fluorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C32H36FN3O2
|
1
|
| 1 |
IC50 = 13803.84 nM
|
|
|
|
CP0858008
|
(2RS)-2-Amino-2-{(2RS)-1-[4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl]-pyrrolidine-2-yl}aceticacid ditrifluoroaceticacid
Show/Hide
|
C22H27F3N2O4S2
|
2
|
| 1 |
IC50 = 14125.38 nM
|
|
|
| 2 |
Ki = 17378.01 nM
|
|
|
|
CP0389351
|
(3S)-1-[(E)-4-(1-benzothiophen-5-yl)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H33NO4S
|
2
|
| 1 |
IC50 = 14125.38 nM
|
|
|
| 2 |
Ki = 7244.36 nM
|
|
|
|
CP0432317
|
1-[(E)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C24H29NO4
|
2
|
| 1 |
IC50 = 14125.38 nM
|
|
|
| 2 |
Ki = 3715.35 nM
|
|
|
|
CP0418965
|
4-hydroxy-N-[(4-methylphenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C31H36N2O2
|
1
|
| 1 |
IC50 = 14125.38 nM
|
|
|
|
CP0418439
|
1-[4,4,4-tris(4-methoxyphenyl)but-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H33NO5
|
2
|
| 1 |
IC50 = 14454.4 nM
|
|
|
| 2 |
Ki = 4365.16 nM
|
|
|
|
CP0480747
|
1-[5-(3-phenyldiazenylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H25N3O2
|
1
|
| 1 |
IC50 = 14454.4 nM
|
|
|
|
CP0406397
|
2-(4-benzhydrylidenepiperidin-1-yl)-N-benzyl-4-hydroxybutanamide
Show/Hide
|
C29H32N2O2
|
2
|
| 1 |
IC50 = 14791.08 nM
|
|
|
| 2 |
Ki = 9120.11 nM
|
|
|
|
CP0549749
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-fluorophenyl)methyl]-3-hydroxypropanamide
Show/Hide
|
C25H29FN2O2S2
|
2
|
| 1 |
IC50 = 15135.61 nM
|
|
|
| 2 |
Ki = 51286.14 nM
|
|
|
|
CP0542548
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C26H31FN2O2S2
|
1
|
| 1 |
IC50 = 15488.17 nM
|
|
|
|
CP0419670
|
4-amino-2-(4-benzhydrylpiperidin-1-yl)-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C29H34FN3O
|
2
|
| 1 |
IC50 = 15848.93 nM
|
|
|
| 2 |
Ki = 33884.42 nM
|
|
|
|
CP0443480
|
4-amino-N-[(2-chlorophenyl)methyl]-2-(4,4-diphenylbut-3-enylamino)butanamide
Show/Hide
|
C27H30ClN3O
|
1
|
| 1 |
IC50 = 15848.93 nM
|
|
|
|
CP0390314
|
1-[5,5,5-tris(4-methoxyphenyl)pent-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H35NO5
|
2
|
| 1 |
IC50 = 15848.93 nM
|
|
|
| 2 |
Ki = 2754.23 nM
|
|
|
|
CP0421179
|
1-[(E)-4,4-bis(4-methoxyphenyl)-5-phenylpent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H35NO4
|
2
|
| 1 |
IC50 = 15848.93 nM
|
|
|
| 2 |
Ki = 4677.35 nM
|
|
|
|
CP0542547
|
N-benzyl-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-4-hydroxybutanamide
Show/Hide
|
C26H32N2O2S2
|
1
|
| 1 |
IC50 = 15848.93 nM
|
|
|
|
CP0404033
|
(2R,4R)-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-fluorophenyl)methyl]-4-hydroxypentanamide
Show/Hide
|
C30H33FN2O2
|
2
|
| 1 |
IC50 = 16218.1 nM
|
|
|
| 2 |
Ki = 42657.95 nM
|
|
|
|
CP0419714
|
4-amino-N-[(4-chlorophenyl)methyl]-2-(4,4-diphenylbut-3-enylamino)butanamide
Show/Hide
|
C27H30ClN3O
|
2
|
| 1 |
IC50 = 16595.87 nM
|
|
|
| 2 |
Ki = 16218.1 nM
|
|
|
|
CP0434410
|
4-amino-2-[4,4-diphenylbutyl(methyl)amino]-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C28H34FN3O
|
2
|
| 1 |
IC50 = 16595.87 nM
|
|
|
| 2 |
Ki = 21379.62 nM
|
|
|
|
CP0848859
|
(rac)-3-({2-[2-(5H-Dibenzo[b,f]azepin-5-yl)ethoxy]ethyl}amino)butanoic acid
Show/Hide
|
C22H26N2O3
|
1
|
| 1 |
IC50 = 17378.01 nM
|
|
|
|
CP0469004
|
4-amino-N-[(4-chlorophenyl)methyl]-2-[4,4-diphenylbutyl(methyl)amino]butanamide
Show/Hide
|
C28H34ClN3O
|
2
|
| 1 |
IC50 = 17378.01 nM
|
|
|
| 2 |
Ki = 17782.79 nM
|
|
|
|
CP0536724
|
1-[(E)-4,4,4-tris(1,3-benzodioxol-5-yl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H29NO8
|
2
|
| 1 |
IC50 = 17782.79 nM
|
|
|
| 2 |
Ki = 6309.57 nM
|
|
|
|
CP0511787
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[2-(4-fluorophenyl)ethyl]-4-hydroxybutanamide
Show/Hide
|
C27H33FN2O2S2
|
1
|
| 1 |
IC50 = 17782.79 nM
|
|
|
|
CP0514837
|
2-(4-benzhydrylpiperidin-1-yl)-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C29H33FN2O2
|
1
|
| 1 |
IC50 = 18197.01 nM
|
|
|
|
CP0852115
|
5-[(4,4-Diphenylbut-3-enylamino)methyl]-2-methoxyphenol
Show/Hide
|
C24H25NO2
|
1
|
| 1 |
IC50 = 18620.87 nM
|
|
|
|
CP0397315
|
4-amino-N-benzyl-2-[4,4-diphenylbut-3-enyl(methyl)amino]butanamide
Show/Hide
|
C28H33N3O
|
2
|
| 1 |
IC50 = 18620.87 nM
|
|
|
| 2 |
Ki = 12589.25 nM
|
|
|
|
CP0216114
|
1-(3-(9H-carbazol-9-yl)propyl)-4-(4-methoxyphenyl)piperidin-4-ol
Show/Hide
|
C27H30N2O2
|
1
|
| 1 |
IC50 = 19000 nM
|
|
|
|
CP0391947
|
N-[(2-chlorophenyl)methyl]-2-[4,4-diphenylbut-3-enyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
|
C28H31ClN2O2
|
1
|
| 1 |
IC50 = 19054.61 nM
|
|
|
|
CP0478937
|
2-(4-benzhydrylpiperidin-1-yl)-N-[(2-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C29H33ClN2O2
|
1
|
| 1 |
IC50 = 19498.45 nM
|
|
|
|
CP0419709
|
4-amino-2-(4-benzhydrylpiperidin-1-yl)-N-benzylbutanamide
Show/Hide
|
C29H35N3O
|
2
|
| 1 |
IC50 = 19498.45 nM
|
|
|
| 2 |
Ki = 32359.37 nM
|
|
|
|
CP0497374
|
4-amino-2-(4,4-diphenylbut-3-enylamino)-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C28H33N3O
|
2
|
| 1 |
IC50 = 19498.45 nM
|
|
|
| 2 |
Ki = 10964.78 nM
|
|
|
|
CP0519706
|
1-[(E)-5-[3-(naphthalen-1-yldiazenyl)phenyl]pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
IC50 = 19498.45 nM
|
|
|
|
CP0511768
|
2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-3-hydroxy-N-[(4-methylphenyl)methyl]propanamide
Show/Hide
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C26H32N2O2S2
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2
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| 1 |
IC50 = 19952.62 nM
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| 2 |
Ki = 38904.51 nM
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CP0531419
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N-benzyl-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
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C30H34N2O2
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1
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| 1 |
IC50 = 19952.62 nM
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CP0848860
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3-({2-[2-(10,11-Dihydro-5H-dibenzo[b,f]azepin-5-yl)ethoxy]ethyl}amino)propanoic acid
Show/Hide
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C21H26N2O3
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1
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| 1 |
IC50 = 20417.38 nM
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CP0392642
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1-[(E)-4,4,4-tris(4-methylphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C31H35NO2
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2
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| 1 |
IC50 = 20417.38 nM
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| 2 |
Ki = 5495.41 nM
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CP0425243
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2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]-3-hydroxypropanamide
Show/Hide
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C25H29ClN2O2S2
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1
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| 1 |
IC50 = 20417.38 nM
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CP0487037
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(2R)-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]-3-hydroxypropanamide
Show/Hide
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C25H29ClN2O2S2
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2
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| 1 |
IC50 = 20417.38 nM
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| 2 |
Ki = 18620.87 nM
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CP0882771
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3-((dodecylamino)methyl)phenol
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C19H33NO
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1
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| 1 |
IC50 = 20892.96 nM
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CP0515301
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1-[2-[(E)-2-[5-fluoro-2-(4-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C23H23F2NO4
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1
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| 1 |
IC50 = 20892.96 nM
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CP0419713
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4-amino-2-(4-benzhydrylpiperazin-1-yl)-N-[(2-chlorophenyl)methyl]butanamide
Show/Hide
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C28H33ClN4O
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1
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| 1 |
IC50 = 20892.96 nM
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CP0517072
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N-[(2-chlorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propyl]amino]butanamide
Show/Hide
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C30H31ClN2O2
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1
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| 1 |
IC50 = 20892.96 nM
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CP0392373
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1-[(E)-5,5,5-triphenylpent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C29H31NO2
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2
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| 1 |
IC50 = 21379.62 nM
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| 2 |
Ki = 9772.37 nM
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CP0406399
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2-[4,4-diphenylbut-3-enyl(methyl)amino]-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
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C28H31FN2O2
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1
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| 1 |
IC50 = 21877.62 nM
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CP0418969
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N-[(4-fluorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
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C30H33FN2O2
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1
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| 1 |
IC50 = 21877.62 nM
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CP0517071
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N-[(4-fluorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propyl]amino]butanamide
Show/Hide
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C30H31FN2O2
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1
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| 1 |
IC50 = 21877.62 nM
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CP0531416
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N-benzyl-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propyl]amino]butanamide
Show/Hide
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C30H32N2O2
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1
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| 1 |
IC50 = 21877.62 nM
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CP0391946
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2-[4,4-diphenylbut-3-enyl(methyl)amino]-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
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C29H34N2O2
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1
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| 1 |
IC50 = 22387.21 nM
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CP0469003
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4-amino-N-benzyl-2-[4,4-diphenylbutyl(methyl)amino]butanamide
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C28H35N3O
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2
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| 1 |
IC50 = 22387.21 nM
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| 2 |
Ki = 30902.95 nM
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CP0476255
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(3R)-1-[4-(3-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C22H23N3O2
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1
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| 1 |
IC50 = 22387.21 nM
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CP0475887
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1-[4-(1,3-benzodioxol-5-yl)-4,4-bis(4-methoxyphenyl)but-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C31H31NO6
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2
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| 1 |
IC50 = 22908.68 nM
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| 2 |
Ki = 4897.79 nM
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CP0427513
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(3R,5S)-5-[[(2E)-2-[(5-naphthalen-1-ylfuran-2-yl)methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
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C22H23N3O3
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2
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| 1 |
IC50 = 22908.68 nM
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| 2 |
Ki = 213.8 nM
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CP0391938
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N-[(4-chlorophenyl)methyl]-2-[4,4-diphenylbut-3-enyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
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C28H31ClN2O2
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1
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| 1 |
IC50 = 23442.29 nM
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CP0404073
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N-[(4-chlorophenyl)methyl]-2-(4,4-diphenylbutylamino)-4-hydroxybutanamide
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C27H31ClN2O2
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2
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| 1 |
IC50 = 23442.29 nM
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| 2 |
Ki = 56234.13 nM
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CP0396966
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4-amino-2-(4-benzhydrylpiperazin-1-yl)-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
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C28H33FN4O
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2
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| 1 |
IC50 = 23442.29 nM
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| 2 |
Ki = 66069.34 nM
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CP0416806
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1-[5-(4-phenyldiazenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
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C23H27N3O2
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1
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| 1 |
IC50 = 23442.29 nM
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CP0391940
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(2R,4S)-2-(4-benzhydrylidenepiperidin-1-yl)-N-benzyl-4-hydroxypentanamide
Show/Hide
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C30H34N2O2
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1
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| 1 |
IC50 = 23988.33 nM
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CP0391941
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2-(4-benzhydrylpiperidin-1-yl)-N-[(4-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
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C29H33ClN2O2
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1
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| 1 |
IC50 = 23988.33 nM
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CP0418984
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N-benzyl-2-[3-fluoren-9-ylidenepropyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
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C28H30N2O2
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1
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| 1 |
IC50 = 23988.33 nM
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CP0452679
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(3R,4R)-4-[(E)-6-(2-phenylphenyl)hex-5-enyl]piperidine-3-carboxylic acid
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C24H29NO2
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2
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| 1 |
IC50 = 24490.63 nM
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| 2 |
Ki = 27415.74 nM
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CP0474183
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(3R,4S)-4-[(E)-5-(2-benzylphenyl)pent-4-enyl]-1-methylpiperidine-3-carboxylic acid
Show/Hide
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C25H31NO2
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2
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| 1 |
IC50 = 24717.24 nM
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| 2 |
Ki = 39902.49 nM
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CP0525722
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1-[2-[(E)-2-(2-benzoylphenyl)ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C23H25NO4
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1
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| 1 |
IC50 = 25118.86 nM
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CP0397774
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(2R)-2-[(2R)-1-(4,4-diphenylbut-3-enyl)pyrrolidin-2-yl]-2-hydroxyacetic acid
Show/Hide
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C22H25NO3
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2
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| 1 |
IC50 = 25118.86 nM
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| 2 |
Ki = 3890.45 nM
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CP0390210
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1-[4,4-bis(4-methoxyphenyl)-4-thiophen-3-ylbut-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C28H29NO4S
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2
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| 1 |
IC50 = 25118.86 nM
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| 2 |
Ki = 5248.07 nM
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CP0486230
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1-[5-(3-phenyldiazenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
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C23H27N3O2
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1
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| 1 |
IC50 = 25118.86 nM
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CP0451185
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N-[(2-chlorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C30H33ClN2O2
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1
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| 1 |
IC50 = 25118.86 nM
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CP0317626
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N-[(2S,3R)-4-(2,2-dimethylpropylamino)-3-hydroxy-1-phenylbutan-2-yl]-2,2-diphenylacetamide
Show/Hide
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C29H36N2O2
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1
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| 1 |
IC50 = 25120 nM
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CP0876647
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5-({2-[Tris-(4-methoxyphenyl)methoxy]ethylamino}-methyl)-2-methoxyphenol
Show/Hide
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C32H35NO6
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1
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| 1 |
IC50 = 25703.96 nM
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CP0481317
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4-amino-2-(4-benzhydrylpiperazin-1-yl)-N-[(4-chlorophenyl)methyl]butanamide
Show/Hide
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C28H33ClN4O
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1
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| 1 |
IC50 = 25703.96 nM
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CP0480749
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1-[5-(4-phenyldiazenylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C23H25N3O2
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1
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| 1 |
IC50 = 25703.96 nM
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CP0516616
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(3R,4S)-4-[5-(2-benzylphenyl)pent-4-ynyl]-1-methylpiperidine-3-carboxylic acid
Show/Hide
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C25H29NO2
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2
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| 1 |
IC50 = 25941.79 nM
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| 2 |
Ki = 28575.91 nM
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CP0557706
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(2R,3S)-1-(2,2-dimethylpropylamino)-3-(2,2-diphenylethylamino)-4-phenylbutan-2-ol
Show/Hide
|
C29H38N2O
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1
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| 1 |
IC50 = 26300 nM
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CP0510729
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3-[1-[2-[(E)-3-[9-(4-methoxyphenyl)fluoren-9-yl]prop-2-enoxy]ethyl]imidazol-2-yl]propanoic acid
Show/Hide
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C31H30N2O4
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1
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| 1 |
IC50 = 26302.68 nM
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CP0452678
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(3R,4S)-1-methyl-4-[(E)-4-(2-phenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H27NO2
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2
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| 1 |
IC50 = 26546.06 nM
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| 2 |
Ki = 14256.08 nM
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CP0870533
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2-({2-[Tris-(4-methoxyphenyl)methoxy]ethylamino}-methyl)phenol
Show/Hide
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C31H33NO5
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1
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| 1 |
IC50 = 26915.35 nM
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CP0397317
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4-amino-2-(4,4-diphenylbut-3-enylamino)-N-[(4-fluorophenyl)methyl]butanamide
Show/Hide
|
C27H30FN3O
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2
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| 1 |
IC50 = 27542.29 nM
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| 2 |
Ki = 22908.68 nM
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CP0531381
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4-hydroxy-N-[(4-methylphenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propyl]amino]butanamide
Show/Hide
|
C31H34N2O2
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1
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| 1 |
IC50 = 27542.29 nM
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CP0481430
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4-amino-2-(4-benzhydrylpiperazin-1-yl)-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
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C29H36N4O
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2
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| 1 |
IC50 = 28183.83 nM
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| 2 |
Ki = 63095.73 nM
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CP0392371
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1-[(E)-4-(1,3-benzodioxol-5-yl)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H33NO6
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2
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| 1 |
IC50 = 28183.83 nM
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| 2 |
Ki = 8709.64 nM
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CP0423415
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4-acetamido-N-[(4-chlorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C32H36ClN3O2
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1
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| 1 |
IC50 = 28183.83 nM
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CP0893160
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3-[(4,4-Diphenylbut-3-enylamino)methyl]phenol
Show/Hide
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C23H23NO
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1
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| 1 |
IC50 = 28840.32 nM
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CP0552385
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4-acetamido-N-[(2-chlorophenyl)methyl]-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C32H36ClN3O2
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1
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| 1 |
IC50 = 28840.32 nM
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CP0564259
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4-acetamido-N-benzyl-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidene)propyl]amino]butanamide
Show/Hide
|
C32H37N3O2
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1
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| 1 |
IC50 = 28840.32 nM
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CP0397572
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1-[2-[(E)-2-[5-fluoro-2-(3-fluorobenzoyl)phenyl]ethenoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C23H23F2NO4
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1
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| 1 |
IC50 = 29512.09 nM
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CP0404034
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2-(4-benzhydrylpiperidin-1-yl)-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C30H36N2O2
|
1
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| 1 |
IC50 = 30199.52 nM
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CP0542545
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2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-4-hydroxy-N-(1-phenylethyl)butanamide
Show/Hide
|
C27H34N2O2S2
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1
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| 1 |
IC50 = 30199.52 nM
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CP0399451
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4-amino-N-benzyl-2-(4,4-diphenylbut-3-enylamino)butanamide
Show/Hide
|
C27H31N3O
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2
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| 1 |
IC50 = 30902.95 nM
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| 2 |
Ki = 17378.01 nM
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CP0422689
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1-[(Z)-5,5,5-tris(4-methoxyphenyl)pent-3-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C32H37NO5
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2
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| 1 |
IC50 = 30902.95 nM
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| 2 |
Ki = 23442.29 nM
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CP0531382
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2-[3-fluoren-9-ylidenepropyl(methyl)amino]-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C29H32N2O2
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1
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| 1 |
IC50 = 31622.78 nM
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CP0416802
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1-[4-(3-phenyldiazenylphenyl)but-3-ynyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N3O2
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1
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| 1 |
IC50 = 32359.37 nM
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CP0876645
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2-[(4,4-Diphenylbut-3-enylamino)methyl]phenol
Show/Hide
|
C23H23NO
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1
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| 1 |
IC50 = 33113.11 nM
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CP0404032
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N-[(2-chlorophenyl)methyl]-2-(4,4-diphenylbutylamino)-4-hydroxybutanamide
Show/Hide
|
C27H31ClN2O2
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2
|
| 1 |
IC50 = 33113.11 nM
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| 2 |
Ki = 46773.51 nM
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CP0451184
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N-[(2-chlorophenyl)methyl]-2-[3-fluoren-9-ylidenepropyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
|
C28H29ClN2O2
|
1
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| 1 |
IC50 = 33113.11 nM
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CP0524040
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2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-chlorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
|
C29H31ClN2O2
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2
|
| 1 |
IC50 = 33884.42 nM
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| 2 |
Ki = 75857.76 nM
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CP0545753
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N-[(2S,3S)-4-(benzylamino)-3-hydroxy-1-phenylbutan-2-yl]-2,2-diphenylacetamide
Show/Hide
|
C31H32N2O2
|
1
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| 1 |
IC50 = 34670 nM
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CP0433301
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(2R,4S)-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-fluorophenyl)methyl]-4-hydroxypentanamide
Show/Hide
|
C30H33FN2O2
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1
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| 1 |
IC50 = 34673.69 nM
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CP0848172
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(2SR)-2-Amino-2-[(2RS)-1-(4,4-diphenylbut-3-en-1-yl)pyrrolidine-2-yl]aceticacid ditrifluoroaceticacid
Show/Hide
|
C24H27F3N2O4
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1
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| 1 |
IC50 = 34673.69 nM
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CP0516614
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(3R,4S)-1-methyl-4-[(E)-5-(2-phenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C24H29NO2
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2
|
| 1 |
IC50 = 34753.62 nM
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| 2 |
Ki = 72443.6 nM
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CP0846186
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3-({2-[2-(10H-Phenothiazin-10-yl)ethoxy]ethyl}amino)propanoic acid
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
IC50 = 35481.34 nM
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CP0424090
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1-(5,5,5-triphenylpent-2-ynyl)piperidine-3-carboxylic acid
Show/Hide
|
C29H29NO2
|
2
|
| 1 |
IC50 = 35481.34 nM
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| 2 |
Ki = 14454.4 nM
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CP0427518
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(3R,5R)-5-[2-[(2E)-2-[[5-(2,4-dichlorophenyl)furan-2-yl]methylidene]hydrazinyl]ethyl]piperidine-3-carboxylic acid
Show/Hide
|
C19H21Cl2N3O3
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2
|
| 1 |
IC50 = 35481.34 nM
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| 2 |
Ki = 478.63 nM
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CP0425213
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N-benzyl-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-3-hydroxypropanamide
Show/Hide
|
C25H30N2O2S2
|
1
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| 1 |
IC50 = 35481.34 nM
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CP0472306
|
(3R,4S)-4-[(E)-4-(2-benzylphenyl)but-3-enyl]-1-methylpiperidine-3-carboxylic acid
Show/Hide
|
C24H29NO2
|
2
|
| 1 |
IC50 = 36728.23 nM
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| 2 |
Ki = 39810.72 nM
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CP0391944
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2-[4,4-diphenylbutyl(methyl)amino]-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
|
C29H36N2O2
|
2
|
| 1 |
IC50 = 37153.52 nM
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| 2 |
Ki = 81283.05 nM
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CP0406398
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N-[(2-chlorophenyl)methyl]-2-[4,4-diphenylbutyl(methyl)amino]-4-hydroxybutanamide
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C28H33ClN2O2
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1
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| 1 |
IC50 = 37153.52 nM
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CP0458156
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3-[1-[2-[2-[9-(4-methoxyphenyl)fluoren-9-yl]oxyethoxy]ethyl]imidazol-2-yl]propanoic acid
Show/Hide
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C30H30N2O5
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1
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| 1 |
IC50 = 37153.52 nM
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CP0575676
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1-[4-(4-phenyldiazenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
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C22H25N3O2
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1
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| 1 |
IC50 = 37153.52 nM
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CP0531383
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2-[3-fluoren-9-ylidenepropyl(methyl)amino]-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
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C28H29FN2O2
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1
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| 1 |
IC50 = 37153.52 nM
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CP0474182
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(3R,4S)-1-methyl-4-[5-(2-phenylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
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C24H27NO2
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1
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| 1 |
IC50 = 37411.06 nM
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CP0391937
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2-(4-benzhydrylidenepiperidin-1-yl)-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
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C30H34N2O2
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2
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| 1 |
IC50 = 38018.94 nM
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| 2 |
Ki = 43651.58 nM
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CP0520051
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1-[(E)-4-(3-phenyldiazenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
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C22H25N3O2
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1
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| 1 |
IC50 = 38018.94 nM
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CP0570428
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1-[(E)-5-(3-phenyldiazenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
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C23H27N3O2
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1
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| 1 |
IC50 = 38018.94 nM
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CP0418415
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1-[(Z)-4,4-bis(4-methoxyphenyl)-5-phenylpent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C31H35NO4
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2
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| 1 |
IC50 = 38018.94 nM
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| 2 |
Ki = 41686.94 nM
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CP0391945
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N-[(4-chlorophenyl)methyl]-2-[4,4-diphenylbutyl(methyl)amino]-4-hydroxybutanamide
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C28H33ClN2O2
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1
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| 1 |
IC50 = 38904.51 nM
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CP0404072
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2-(4,4-diphenylbutylamino)-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
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C27H31FN2O2
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1
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| 1 |
IC50 = 38904.51 nM
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CP0489513
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1-[(E)-4,4-bis(4-methoxyphenyl)-4-thiophen-3-ylbut-2-enyl]piperidine-3-carboxylic acid
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C28H31NO4S
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2
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| 1 |
IC50 = 38904.51 nM
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| 2 |
Ki = 12882.5 nM
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CP0386960
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(3S)-1-[(E)-4,4,4-tris(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C31H35NO5
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3
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| 1 |
IC50 = 39810 nM
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| 2 |
IC50 = 39810.72 nM
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| 3 |
Ki = 46773.51 nM
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CP0564670
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N-[(2S,3R)-4-(cyclopropylmethylamino)-3-hydroxy-1-phenylbutan-2-yl]-3,3-diphenylpropanamide
Show/Hide
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C29H34N2O2
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1
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| 1 |
IC50 = 39810 nM
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CP0392370
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1-[(E)-4,4,4-triphenylbut-2-enyl]piperidine-3-carboxylic acid
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C28H29NO2
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2
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| 1 |
IC50 = 40738.03 nM
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| 2 |
Ki = 8317.64 nM
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CP0479786
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1-[(Z)-5,5,5-triphenylpent-3-enyl]piperidine-3-carboxylic acid
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C29H31NO2
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2
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| 1 |
IC50 = 40738.03 nM
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| 2 |
Ki = 7413.1 nM
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CP0516615
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(3R,4R)-4-[5-(2-benzylphenyl)pent-4-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C24H27NO2
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2
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| 1 |
IC50 = 40831.94 nM
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| 2 |
Ki = 31045.6 nM
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CP0427517
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(3R,5S)-5-[[(2E)-2-[[5-[2-chloro-4-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
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C19H19ClF3N3O3
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2
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| 1 |
IC50 = 41686.94 nM
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| 2 |
Ki = 446.68 nM
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CP0473950
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1-[(Z)-5,5,5-tris(4-methoxyphenyl)pent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C32H37NO5
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2
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| 1 |
IC50 = 41686.94 nM
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| 2 |
Ki = 23988.33 nM
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CP0451187
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N-[(4-chlorophenyl)methyl]-2-[3-fluoren-9-ylidenepropyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
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C28H29ClN2O2
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1
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| 1 |
IC50 = 42657.95 nM
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CP0920888
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3-({2-[Tris-(4-methoxyphenyl)methoxy]ethylamino}-methyl)phenol
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C31H33NO5
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1
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| 1 |
IC50 = 43651.58 nM
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CP0443479
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4-amino-2-(4-benzhydrylpiperazin-1-yl)-N-benzylbutanamide
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C28H34N4O
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1
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| 1 |
IC50 = 44668.36 nM
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CP0427512
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(3R,5R)-5-[2-[(2E)-2-[[5-[2-chloro-4-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C20H21ClF3N3O3
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2
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| 1 |
IC50 = 44668.36 nM
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| 2 |
Ki = 616.6 nM
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CP0393111
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1-[(E)-4,4,4-tris(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C31H35NO5
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2
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| 1 |
IC50 = 47863.01 nM
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| 2 |
Ki = 14791.08 nM
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CP0858007
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(2RS)-2-Amino-2-{[(2RS)-1-(4,4-diphenylbut-3-en-1-yl)]pyrrolidine-2-yl}aceticacid ditrifluoroaceticacid
Show/Hide
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C24H27F3N2O4
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1
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| 1 |
IC50 = 48977.88 nM
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CP0848861
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SID118229
Show/Hide
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C4H9NO2
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1
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| 1 |
IC50 = 50118.72 nM
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CP0920887
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2-[(3,3-Diphenylpropylamino)methyl]phenol
Show/Hide
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C22H23NO
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1
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| 1 |
IC50 = 52480.75 nM
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CP0393112
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1-[5,5,5-tris(4-methoxyphenyl)pent-2-ynyl]piperidine-3-carboxylic acid
Show/Hide
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C32H35NO5
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2
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| 1 |
IC50 = 52480.75 nM
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| 2 |
Ki = 37153.52 nM
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CP0433304
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(2R,4S)-2-(4-benzhydrylidenepiperidin-1-yl)-4-hydroxy-N-[(4-methylphenyl)methyl]pentanamide
Show/Hide
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C31H36N2O2
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1
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| 1 |
IC50 = 53703.18 nM
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CP0404030
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2-(4,4-diphenylbutylamino)-4-hydroxy-N-[(4-methylphenyl)methyl]butanamide
Show/Hide
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C28H34N2O2
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2
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| 1 |
IC50 = 54954.09 nM
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| 2 |
Ki = 51286.14 nM
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CP0457739
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1-[(E)-5,5,5-tris(4-methoxyphenyl)pent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C32H37NO5
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2
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| 1 |
IC50 = 54954.09 nM
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| 2 |
Ki = 34673.69 nM
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CP0511789
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2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]-4-hydroxypentanamide
Show/Hide
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C27H33ClN2O2S2
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1
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| 1 |
IC50 = 57543.99 nM
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CP0893162
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2-((dodecylamino)methyl)phenol
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C19H33NO
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1
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| 1 |
IC50 = 58884.37 nM
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CP0491778
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N-benzyl-2-[4,4-diphenylbutyl(methyl)amino]-4-hydroxybutanamide
Show/Hide
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C28H34N2O2
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1
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| 1 |
IC50 = 58884.37 nM
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CP0443985
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(3R,4S)-4-[(E)-4-(2-phenylphenyl)but-3-enyl]piperidine-3-carboxylic acid
Show/Hide
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C22H25NO2
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2
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| 1 |
IC50 = 60534.09 nM
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| 2 |
Ki = 33189.45 nM
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CP0523056
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N-benzyl-2-(4,4-diphenylbutylamino)-4-hydroxybutanamide
Show/Hide
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C27H32N2O2
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1
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| 1 |
IC50 = 61659.5 nM
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CP0459814
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(3R,4R)-4-[(E)-5-(2-benzylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
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C24H29NO2
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2
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| 1 |
IC50 = 64120.96 nM
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| 2 |
Ki = 68076.94 nM
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CP0390316
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(3S)-1-[2-[(4-methoxy-2-methylphenyl)-bis(4-methoxyphenyl)methoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C31H37NO6
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2
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| 1 |
IC50 = 64565.42 nM
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| 2 |
IC50 = 64570 nM
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CP0391939
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(2R,4S)-2-(4-benzhydrylidenepiperidin-1-yl)-N-[(4-chlorophenyl)methyl]-4-hydroxypentanamide
Show/Hide
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C30H33ClN2O2
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1
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| 1 |
IC50 = 66069.34 nM
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CP0407628
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(3R,4R)-4-[(E)-5-(2-phenylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
Show/Hide
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C23H27NO2
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1
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| 1 |
IC50 = 66834.39 nM
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CP0390312
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1-[2-[bis(4-methoxy-2-methylphenyl)-(4-methoxyphenyl)methoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C32H39NO6
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2
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| 1 |
IC50 = 67608.3 nM
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| 2 |
Ki = 38018.94 nM
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CP0542519
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pyrrolidine-3-carboxylic acid
Show/Hide
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C5H9NO2
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1
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| 1 |
IC50 = 67608.3 nM
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CP0555015
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N-[(4-chlorophenyl)methyl]-4-hydroxy-2-[methyl-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,9,11,13-heptaenylidene)propyl]amino]butanamide
Show/Hide
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C30H31ClN2O2
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1
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| 1 |
IC50 = 69183.1 nM
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CP0455056
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3-[1-[(Z)-4-[9-(4-methoxyphenyl)fluoren-9-yl]oxybut-2-enyl]imidazol-2-yl]propanoic acid
Show/Hide
|
C30H28N2O4
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1
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| 1 |
IC50 = 70794.58 nM
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CP0437989
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1-[(E)-4-hydroxy-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C24H29NO5
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1
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| 1 |
IC50 = 70794.58 nM
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CP0524552
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1-[(Z)-4,4,4-tris(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C31H35NO5
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2
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| 1 |
IC50 = 72443.6 nM
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| 2 |
Ki = 17782.79 nM
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CP0418964
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(3S)-1-[2-[[4-(4-formylphenyl)phenyl]-bis(4-methoxyphenyl)methoxy]ethyl]piperidine-3-carboxylic acid
Show/Hide
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C36H37NO6
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1
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| 1 |
IC50 = 72443.6 nM
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CP0044059
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(S)-Piperidine-3-carboxylic acid
Show/Hide
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C6H11NO2
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1
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| 1 |
IC50 = 74131.02 nM
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CP0050744
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5-Amino-Pentanoic Acid
Show/Hide
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C5H11NO2
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1
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| 1 |
IC50 = 74131.02 nM
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CP0446684
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3-[1-(4,4-diphenylbut-3-enyl)imidazol-2-yl]propanoic acid
Show/Hide
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C22H22N2O2
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1
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| 1 |
IC50 = 74131.02 nM
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CP0422688
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1-[(Z)-4,4,5-tris(4-methoxyphenyl)pent-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C32H37NO5
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2
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| 1 |
IC50 = 74131.02 nM
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| 2 |
Ki = 25703.96 nM
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CP0403231
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(3R,4S)-4-[(E)-6-(2-phenylphenyl)hex-5-enyl]piperidine-3-carboxylic acid
Show/Hide
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C24H29NO2
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2
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| 1 |
IC50 = 75509.22 nM
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| 2 |
Ki = 71779.43 nM
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CP0419764
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2-[3-[5-[9-(4-methoxyphenyl)fluoren-9-yl]oxypentyl]imidazol-4-yl]acetic acid
Show/Hide
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C30H30N2O4
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1
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| 1 |
IC50 = 79432.82 nM
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CP0440313
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1-[(Z)-4,4-bis(4-methoxyphenyl)-4-thiophen-3-ylbut-2-enyl]piperidine-3-carboxylic acid
Show/Hide
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C28H31NO4S
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1
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| 1 |
IC50 = 79432.82 nM
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CP0427515
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(3R,5S)-5-[[(2E)-2-[[5-[2-chloro-5-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C19H19ClF3N3O3
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2
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| 1 |
IC50 = 81283.05 nM
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| 2 |
Ki = 467.74 nM
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CP0081174
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(S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piperidine-3-carboxylic acid
Show/Hide
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C30H35NO6
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3
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| 1 |
IC50 = 85000 nM
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| 2 |
IC50 = 85113.8 nM
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| 3 |
Ki = 27542.29 nM
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CP0444847
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2,6-Difluoro-3-({2-[tris-(4-methoxyphenyl)methoxy]ethylamino}methyl)phenol
Show/Hide
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C31H31F2NO5
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1
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| 1 |
IC50 = 85113.8 nM
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CP0876646
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3-[(3,3-Diphenylpropylamino)methyl]phenol
Show/Hide
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C22H23NO
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1
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| 1 |
IC50 = 87096.36 nM
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CP0543361
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N-[(2S,3S)-3-hydroxy-4-[(2-methoxyphenyl)methylamino]-1-phenylbutan-2-yl]-2,2-diphenylacetamide
Show/Hide
|
C32H34N2O3
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1
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| 1 |
IC50 = 87100 nM
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CP0479787
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1-[(Z)-4-(1,3-benzodioxol-5-yl)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
Show/Hide
|
C31H33NO6
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2
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| 1 |
IC50 = 95499.26 nM
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| 2 |
Ki = 53703.18 nM
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CP0524041
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2-[4,4-diphenylbutyl(methyl)amino]-N-[(4-fluorophenyl)methyl]-4-hydroxybutanamide
Show/Hide
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C28H33FN2O2
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1
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| 1 |
IC50 = 97723.72 nM
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CP0848173
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(2SR)-2-Amino-2-{(2RS)-1-[4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl]pyrrolidine-2-yl}aceticacid ditrifluoroaceticacid
Show/Hide
|
C22H27F3N2O4S2
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2
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| 1 |
IC50 = 100000 nM
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| 2 |
Ki = 37153.52 nM
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CP0419765
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3-[1-[3-[9-(4-methoxyphenyl)fluoren-9-yl]oxypropyl]imidazol-2-yl]propanoic acid
Show/Hide
|
C29H28N2O4
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1
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| 1 |
IC50 = 100000 nM
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CP0427519
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(3R,5S)-5-[[(2E)-2-[[5-[3,5-bis(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C20H19F6N3O3
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1
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| 1 |
Ki = 245.47 nM
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CP0427509
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(3R,5S)-5-[[(2E)-2-[[5-(2,4-dichlorophenyl)furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C18H19Cl2N3O3
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1
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| 1 |
Ki = 645.65 nM
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CP0470585
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(3R,5S)-5-[[(2E)-2-[[5-[3-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C19H20F3N3O3
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1
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| 1 |
Ki = 707.95 nM
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CP0470587
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(3R,5S)-5-[[(2E)-2-[(2-naphthalen-2-ylpyrimidin-5-yl)methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C22H23N5O2
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1
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| 1 |
Ki = 933.25 nM
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CP0427506
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(3R,5S)-5-[[(2E)-2-[(3-phenoxyphenyl)methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C20H23N3O3
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1
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| 1 |
Ki = 954.99 nM
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CP0470584
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(3R,5S)-5-[[(2E)-2-[[5-(2-chlorophenyl)furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C18H20ClN3O3
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1
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| 1 |
Ki = 1230.27 nM
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CP0470586
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(3R,5S)-5-[[(2E)-2-[[5-[4-fluoro-3-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C19H19F4N3O3
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1
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| 1 |
Ki = 1258.93 nM
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CP0518719
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(3R,5S)-5-[[(2E)-2-[[5-(2-bromophenyl)furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C18H20BrN3O3
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1
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| 1 |
Ki = 1445.44 nM
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CP0427510
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(3R,5S)-5-[[(2E)-2-[[5-(4-chloro-2-nitrophenyl)furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C18H19ClN4O5
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1
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| 1 |
Ki = 1479.11 nM
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CP0427508
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(3R,5S)-5-[[(2E)-2-[[5-(3-chlorophenyl)furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C18H20ClN3O3
|
1
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| 1 |
Ki = 1862.09 nM
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CP0534222
|
(3R,5S)-5-[[(2E)-2-[[5-[2-(trifluoromethyl)phenyl]furan-2-yl]methylidene]hydrazinyl]methyl]piperidine-3-carboxylic acid
Show/Hide
|
C19H20F3N3O3
|
1
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| 1 |
Ki = 2290.87 nM
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CP0459768
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1-[(Z)-4,4-bis(4-methoxyphenyl)but-2-enyl]piperidine-3-carboxylic acid
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C24H29NO4
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1
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| 1 |
Ki = 26302.68 nM
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CP0421182
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1-[(E)-4,4-bis(4-methoxyphenyl)-4-(1,3-thiazol-2-yl)but-2-enyl]piperidine-3-carboxylic acid
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C27H30N2O4S
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1
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| 1 |
Ki = 33884.42 nM
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CP0452680
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(3R,4R)-4-[(E)-6-(2-benzylphenyl)hex-5-enyl]piperidine-3-carboxylic acid
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C25H31NO2
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1
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| 1 |
Ki = 35399.73 nM
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CP0560514
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(2S)-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(2-chlorophenyl)methyl]-4-hydroxybutanamide
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C26H31ClN2O2S2
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1
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| 1 |
Ki = 38018.94 nM
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CP0474184
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(3R,4S)-4-[(E)-5-(2-benzylphenyl)pent-4-enyl]piperidine-3-carboxylic acid
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C24H29NO2
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1
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| 1 |
Ki = 77090.35 nM
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CP0424088
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1-[4,4-bis(4-methoxyphenyl)-4-(1,3-thiazol-2-yl)but-2-ynyl]piperidine-3-carboxylic acid
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C27H28N2O4S
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1
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| 1 |
Ki = 77624.71 nM
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CP0425217
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(2S)-2-[4,4-bis(3-methylthiophen-2-yl)but-3-enyl-methylamino]-N-[(4-chlorophenyl)methyl]-3-hydroxypropanamide
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C25H29ClN2O2S2
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1
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| 1 |
Ki = 87096.36 nM
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