Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT03053 , Cysteinyl leukotriene receptor 2
Gene Name CYSLTR2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9NS75
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT03053
 
Compound ID Compound Name Compound Formula
CP0400409
4-(3-carboxypropyl)-8-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
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C31H33NO7
 1
1
IC50 = 0.31 nM
   TI
   LI
   LO
   TS
CP0524590
4-[8-[[4-(4-phenylbutoxy)benzoyl]amino]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C30H32N6O5
 1
1
IC50 = 0.49 nM
   TI
   LI
   LO
   TS
CP0481627
4-(3-carboxypropyl)-8-[[4-(5-phenylpentoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
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C31H34N2O7
 1
1
IC50 = 0.62 nM
   TI
   LI
   LO
   TS
CP0379304
(2S)-4-(3-carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H32N2O7
 1
1
IC50 = 0.87 nM
   TI
   LI
   LO
   TS
CP0408242
4-[1-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acid
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C34H34ClNO5
 1
1
IC50 = 0.88 nM
   TI
   LI
   LO
   TS
CP0448955
2-[1-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]acetic acid
   Show/Hide
C32H30ClNO5
 1
1
IC50 = 0.89 nM
   TI
   LI
   LO
   TS
CP0382282
4-[1-(carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,6-trifluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H32F3NO5
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0382284
4-[1-(carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,4,5-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H31F4NO5
 1
1
IC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0487602
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(2,3,6-trifluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C32H30F3NO5
 1
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
CP0411554
4-[1-(carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H31F4NO5
 1
1
IC50 = 2.2 nM
   TI
   LI
   LO
   TS
CP0379267
4-(3-carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H32N2O7
 2
1
IC50 = 2.3 nM
   TI
   LI
   LO
   TS
2
IC50 = 2.5 nM
   TI
   LI
   LO
   TS
CP0379269
4-[8-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C31H33N5O4
 1
1
IC50 = 3.4 nM
   TI
   LI
   LO
   TS
CP0494801
4-[1-(3-carboxypropyl)-2-methyl-7-[2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethynyl]indol-3-yl]butanoic acid
   Show/Hide
C35H33F4NO5
 1
1
IC50 = 3.6 nM
   TI
   LI
   LO
   TS
CP0566585
4-[1-(carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,5,6-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H31F4NO5
 1
1
IC50 = 3.7 nM
   TI
   LI
   LO
   TS
CP0379718
3-[(3-carboxycyclohexyl)carbamoyl]-4-[3-[4-(4-cyclohexyloxybutoxy)phenyl]propoxy]benzoic acid
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C34H45NO8
 2
1
IC50 = 3.8 nM
   TI
   LI
   LO
   TS
2
IC50 = 38 nM
   TI
   LI
   LO
   TS
CP0484535
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
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C33H34ClNO5
 1
1
IC50 = 4.6 nM
   TI
   LI
   LO
   TS
CP0428421
4-[1-(carboxymethyl)-2-methyl-7-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H35NO5
 1
1
IC50 = 4.7 nM
   TI
   LI
   LO
   TS
CP0418315
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C34H36ClNO5
 1
1
IC50 = 5.1 nM
   TI
   LI
   LO
   TS
CP0381577
4-[1-(3-carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H38ClNO5
 1
1
IC50 = 5.5 nM
   TI
   LI
   LO
   TS
CP0429311
4-[2-(benzenesulfonylcarbamoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C36H37N3O8S
 1
1
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
CP0529629
4-(3-carboxypropyl)-8-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C31H33NO6
 1
1
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
CP0382287
3-[1-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]propanoic acid
   Show/Hide
C33H32ClNO5
 1
1
IC50 = 5.7 nM
   TI
   LI
   LO
   TS
CP0408240
4-[1-(carboxymethyl)-7-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C32H33NO6
 1
1
IC50 = 6 nM
   TI
   LI
   LO
   TS
CP0408236
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C34H36FNO5
 1
1
IC50 = 7.2 nM
   TI
   LI
   LO
   TS
CP0380609
4-[1-(3-carboxypropyl)-7-[2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H38FNO5
 1
1
IC50 = 8.8 nM
   TI
   LI
   LO
   TS
CP0456062
4-[1-(3-carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-4-fluoro-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H37ClFNO5
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0432238
4-[1-(3-carboxypropyl)-4-fluoro-2-methyl-7-[2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethynyl]indol-3-yl]butanoic acid
   Show/Hide
C35H32F5NO5
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0484534
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C33H34FNO5
 1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0418562
4-[8-[2-[4-(4-phenylbutoxy)phenyl]ethyl]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C31H35N5O4
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0382290
4-[3-(2-carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]butanoic acid
   Show/Hide
C35H36ClNO5
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0484536
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(2-methoxyphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C34H37NO6
 1
1
IC50 = 15 nM
   TI
   LI
   LO
   TS
CP0481625
4-(3-carboxypropyl)-8-[[4-(3-phenoxypropoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C29H30N2O8
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0386772
4-(3-carboxypropyl)-8-[2-[4-(4-phenylbutoxy)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C31H35NO6
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0386773
4-[2-(methylsulfonylcarbamoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C31H35N3O8S
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0553496
4-(3-carboxypropyl)-8-[[4-(4-phenoxybutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H32N2O8
 1
1
IC50 = 17 nM
   TI
   LI
   LO
   TS
CP0448956
4-[1-(2-carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C35H36ClNO5
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS
CP0428430
4-[1-(carboxymethyl)-7-[(E)-2-[4-[4-(3-chlorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C32H32ClNO5
 1
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
CP0408239
4-[3-(carboxymethyl)-4-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]indol-1-yl]butanoic acid
   Show/Hide
C32H33NO6
 2
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
2
IC50 = 27 nM
   TI
   LI
   LO
   TS
CP0382286
4-[1-(carboxymethyl)-7-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]indol-3-yl]butanoic acid
   Show/Hide
C32H33NO5
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
CP0427949
4-[1-(3-carboxypropyl)-4-fluoro-7-[2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H37F2NO5
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
CP0524589
4-(3-carboxypropyl)-8-[[4-(4-phenylbutoxy)phenyl]methoxy]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H33NO7
 1
1
IC50 = 30 nM
   TI
   LI
   LO
   TS
CP0382291
5-[3-(3-carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acid
   Show/Hide
C37H40ClNO5
 1
1
IC50 = 30 nM
   TI
   LI
   LO
   TS
CP0456063
4-[1-(3-carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-5-fluoro-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H37ClFNO5
 1
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
CP0408238
4-[1-(3-carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-6-fluoro-2-methylindol-3-yl]butanoic acid
   Show/Hide
C36H37ClFNO5
 1
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
CP0379714
3-[(3-carboxycyclohexyl)carbamoyl]-4-[3-[4-(4-phenoxybutoxy)phenyl]propoxy]benzoic acid
   Show/Hide
C34H39NO8
 1
1
IC50 = 53 nM
   TI
   LI
   LO
   TS
CP0481626
(2R)-4-(3-carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H32N2O7
 1
1
IC50 = 55 nM
   TI
   LI
   LO
   TS
CP0484537
4-[3-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]butanoic acid
   Show/Hide
C34H34ClNO5
 1
1
IC50 = 55 nM
   TI
   LI
   LO
   TS
CP0448958
5-[3-(2-carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acid
   Show/Hide
C36H38ClNO5
 1
1
IC50 = 60 nM
   TI
   LI
   LO
   TS
CP0498608
4-(3-carboxypropyl)-8-[[4-(3-phenylpropoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C29H30N2O7
 1
1
IC50 = 68 nM
   TI
   LI
   LO
   TS
CP0384755
3-(3-carboxypropoxy)-8-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]quinoxaline-2-carboxylic acid
   Show/Hide
C31H30N2O7
 1
1
IC50 = 75 nM
   TI
   LI
   LO
   TS
CP0531079
3-[1-(2-carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]propanoic acid
   Show/Hide
C34H34ClNO5
 1
1
IC50 = 78 nM
   TI
   LI
   LO
   TS
CP0382289
3-[3-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]propanoic acid
   Show/Hide
C33H32ClNO5
 1
1
IC50 = 96 nM
   TI
   LI
   LO
   TS
CP0494291
4-(4-carboxybutyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C31H34N2O7
 1
1
IC50 = 170 nM
   TI
   LI
   LO
   TS
CP0533704
5-[3-(carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acid
   Show/Hide
C35H36ClNO5
 1
1
IC50 = 248 nM
   TI
   LI
   LO
   TS
CP0551481
4-(5-carboxypentyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C32H36N2O7
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0508488
4-[(4S,5R,6E,8E,10Z,13Z)-1-carboxy-4-hydroxynonadeca-6,8,10,13-tetraen-5-yl]sulfanylbenzoic acid
   Show/Hide
C27H36O5S
 1
1
IC50 = 300 nM
   TI
   LI
   LO
   TS
CP0400410
1-(3-carboxypropyl)-4-oxo-5-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]quinoline-3-carboxylic acid
   Show/Hide
C32H31NO7
 1
1
IC50 = 370 nM
   TI
   LI
   LO
   TS
CP0379268
4-[2-(hydroxymethyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C30H34N2O6
 1
1
IC50 = 410 nM
   TI
   LI
   LO
   TS
CP0455907
4-(3-carboxypropanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H30N2O8
 1
1
IC50 = 890 nM
   TI
   LI
   LO
   TS
CP0511154
4-(5-carboxypentanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C32H34N2O8
 1
1
IC50 = 890 nM
   TI
   LI
   LO
   TS
CP0379712
4-(3-carboxypropyl)-8-[[4-(2-phenoxyethoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C28H28N2O8
 1
1
IC50 = 1500 nM
   TI
   LI
   LO
   TS
CP0455908
4-(4-carboxybutanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C31H32N2O8
 1
1
IC50 = 1800 nM
   TI
   LI
   LO
   TS
CP0455909
4-acetyl-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C28H28N2O6
 1
1
IC50 = 3600 nM
   TI
   LI
   LO
   TS
CP0379709
4-butanoyl-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C30H32N2O6
 1
1
IC50 = 3700 nM
   TI
   LI
   LO
   TS
CP0418561
4-[8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acid
   Show/Hide
C29H32N2O5
 1
1
IC50 = 4300 nM
   TI
   LI
   LO
   TS
CP0489186
8-[[4-(4-phenylbutoxy)benzoyl]amino]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C26H26N2O5
 1
1
IC50 = 4600 nM
   TI
   LI
   LO
   TS
CP0379707
8-[[4-(4-phenylbutoxy)benzoyl]amino]-4-propanoyl-2,3-dihydro-1,4-benzoxazine-2-carboxylic acid
   Show/Hide
C29H30N2O6
 1
1
IC50 = 5200 nM
   TI
   LI
   LO
   TS
CP0551497
(Z)-2-cyano-N-[2-(4-cyanobenzoyl)-5-[(E)-4-(diethylamino)-4-oxobut-2-en-2-yl]-1-benzofuran-3-yl]-3-hydroxybut-2-enamide
   Show/Hide
C29H26N4O5
 1
1
IC50 = 7700 nM
   TI
   LI
   LO
   TS
CP0380350
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-7-methoxy-1H-indole-2-carboxylic acid
   Show/Hide
C30H22ClN3O4
 1
1
IC50 = 15000 nM
   TI
   LI
   LO
   TS
CP0380616
3-[[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl]carbamoyl]-1H-indole-2-carboxylic acid
   Show/Hide
C27H18ClN3O3
 1
1
IC50 = 23000 nM
   TI
   LI
   LO
   TS
CP0380618
CHEBI:6993
   Show/Hide
C35H35ClNNaO3S
 1
1
IC50 = 27000 nM
   TI
   LI
   LO
   TS
CP0380375
4-chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C29H19Cl2N3O3
 1
1
IC50 = 36000 nM
   TI
   LI
   LO
   TS
CP0959286
Pranlukast hemihydrate
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C27H25N5O5
 1
1
IC50 = 43000 nM
   TI
   LI
   LO
   TS
CP0399551
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-5-fluoro-1H-indole-2-carboxylic acid
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C29H19ClFN3O3
 1
1
IC50 = 46000 nM
   TI
   LI
   LO
   TS
CP0508763
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-5-methoxy-1H-indole-2-carboxylic acid
   Show/Hide
C30H22ClN3O4
 1
1
IC50 = 46000 nM
   TI
   LI
   LO
   TS
CP0531289
3-[3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxopropyl]-1H-indole-2-carboxylic acid
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C29H22ClN3O3
 1
1
IC50 = 50000 nM
   TI
   LI
   LO
   TS
CP0045344
4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol-3-ylmethyl)-3-methoxy-N-o-tolylsulfonylbenzamide
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C31H33N3O6S
 1
1
IC50 = 58000 nM
   TI
   LI
   LO
   TS
CP0399550
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C29H20ClN3O3
 1
1
IC50 = 58000 nM
   TI
   LI
   LO
   TS
CP0399347
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-4,6-difluoro-1H-indole-2-carboxylic acid
   Show/Hide
C29H18ClF2N3O3
 1
1
IC50 = 76000 nM
   TI
   LI
   LO
   TS
CP0390349
6-chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C29H19Cl2N3O3
 1
1
IC50 = 87000 nM
   TI
   LI
   LO
   TS
CP0380376
4,6-dichloro-3-[(E)-3-cyclohexyloxy-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C18H17Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0380377
4,6-dichloro-3-[(E)-3-oxo-3-(4-phenylbutoxy)prop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C22H19Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0380619
4,6-dichloro-3-[(E)-3-[[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl]methoxy]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C30H19Cl3N2O4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0399548
4,6-dichloro-3-[(E)-3-oxo-3-phenoxyprop-1-enyl]-1H-indole-2-carboxylic acid
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C18H11Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0407630
4,6-dichloro-3-[(E)-3-oxo-3-(3-phenylpropoxy)prop-1-enyl]-1H-indole-2-carboxylic acid
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C21H17Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0414693
4,6-dichloro-3-[(E)-3-(4-cyanobutoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C17H14Cl2N2O4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0414695
7-chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C29H19Cl2N3O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0429281
4,6-dichloro-3-[(E)-3-oxo-3-phenylmethoxyprop-1-enyl]-1H-indole-2-carboxylic acid
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C19H13Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0447690
4,6-dichloro-3-[(E)-3-oxo-3-pentoxyprop-1-enyl]-1H-indole-2-carboxylic acid
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C17H17Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0447691
[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl]methyl (E)-3-(4,6-dichloro-1H-indol-3-yl)prop-2-enoate
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C29H19Cl3N2O2
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0451909
4,6-dichloro-3-[(E)-3-(4-methylpentoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C18H19Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0451911
4,6-dichloro-3-[(E)-3-(cyclohexylmethoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C19H19Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0458738
4,6-dichloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C29H18Cl3N3O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0459655
3-[(E)-3-[[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl]methoxy]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
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C30H21ClN2O4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0469615
3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-6-methoxy-1H-indole-2-carboxylic acid
   Show/Hide
C30H22ClN3O4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0531290
5-chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C29H19Cl2N3O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0538956
4,6-dichloro-3-[(E)-3-oxo-3-(2-phenylethoxy)prop-1-enyl]-1H-indole-2-carboxylic acid
   Show/Hide
C20H15Cl2NO4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS