| Compound ID |
Compound Name |
Compound Formula |
|
CP0051488
|
N-[2-[4-[(3S)-1-methylsulfonylpiperidin-3-yl]-1,3-thiazol-2-yl]-4-morpholin-4-ylphenyl]-1H-imidazole-2-carboxamide
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|
C23H28N6O4S2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0562564
|
N-[4-[2-(dimethylamino)ethoxy]-2-[4-[(3S)-1-methylsulfonylpiperidin-3-yl]-1,3-thiazol-2-yl]phenyl]-1H-imidazole-2-carboxamide
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|
C23H30N6O4S2
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0432863
|
N-[2-[4-[(2S)-4-methylsulfonylmorpholin-2-yl]-1,3-thiazol-2-yl]-4-morpholin-4-ylphenyl]-1H-imidazole-2-carboxamide
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|
C22H26N6O5S2
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0562563
|
N-[2-[4-[(3S)-1-methylsulfonylpiperidin-3-yl]-1,3-thiazol-2-yl]-4-piperazin-1-ylphenyl]-1H-imidazole-2-carboxamide
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|
C23H29N7O3S2
|
1
|
| 1 |
EC50 = 167 nM
|
|
|
|
CP0155152
|
N-[2-[4-[(3S)-1-methylsulfonylpiperidin-3-yl]-1,3-thiazol-2-yl]phenyl]-1H-imidazole-2-carboxamide
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|
C19H21N5O3S2
|
1
|
| 1 |
EC50 = 3600 nM
|
|
|
|
CP0402661
|
N-[2-[4-[(2S)-4-methylsulfonylmorpholin-2-yl]-1,3-thiazol-2-yl]phenyl]-1H-imidazole-2-carboxamide
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|
C18H19N5O4S2
|
1
|
| 1 |
EC50 = 4700 nM
|
|
|
|
CP0031719
|
(R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine
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|
C21H22Cl2FN5O
|
1
|
| 1 |
IC50 = 294 nM
|
|
|
|
CP0915359
|
(R)-6-chloro-3-(1-(4-methoxyphenyl)-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
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|
C21H21ClN6O
|
1
|
| 1 |
IC50 = 374 nM
|
|
|
|
CP0775775
|
(R)-6-chloro-3-(1-phenyl-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
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|
C20H19ClN6
|
1
|
| 1 |
IC50 = 668 nM
|
|
|
|
CP0775776
|
(R)-6-chloro-3-(1-(4-fluorophenyl)-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
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|
C20H18ClFN6
|
1
|
| 1 |
IC50 = 684 nM
|
|
|
|
CP0960720
|
(R)-4-(4-(6-chloro-5-(pyrrolidin-3-ylamino)-1H-indazol-3-yl)-1H-pyrazol-1-yl)benzonitrile
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|
C21H18ClN7
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0955678
|
(R)-6-chloro-3-(1-(4-methoxyphenyl)-1H-pyrazol-4-yl)-N-(5-azaspiro[2.4]heptan-7-yl)-1H-indazol-5-amine
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|
C23H23ClN6O
|
1
|
| 1 |
IC50 = 883 nM
|
|
|
|
CP0968870
|
(R)-3-(4-(6-chloro-5-(pyrrolidin-3-ylamino)-1H-indazol-3-yl)-1H-pyrazol-1-yl)benzonitrile
Show/Hide
|
C21H18ClN7
|
1
|
| 1 |
IC50 = 2020 nM
|
|
|
|
CP0955676
|
(R)-6-chloro-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
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|
C15H17ClN6
|
1
|
| 1 |
IC50 = 3130 nM
|
|
|
|
CP0958999
|
(R)-6-chloro-3-(1-(2-fluoroethyl)-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
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|
C16H18ClFN6
|
1
|
| 1 |
IC50 = 3460 nM
|
|
|
|
CP0950734
|
(R)-2-(4-(6-chloro-5-(pyrrolidin-3-ylamino)-1H-indazol-3-yl)-1H-pyrazol-1-yl)benzonitrile
Show/Hide
|
C21H18ClN7
|
1
|
| 1 |
IC50 = 3540 nM
|
|
|
|
CP0915358
|
(R)-6-chloro-3-(1-methyl-1H-pyrazol-4-yl)-N-(1-methylpyrrolidin-3-yl)-1H-indazol-5-amine
Show/Hide
|
C16H19ClN6
|
1
|
| 1 |
IC50 = 8960 nM
|
|
|
|
CP0775778
|
(R)-6-chloro-3-(1-(4-methoxyphenyl)-1H-pyrazol-4-yl)-N-(1-(oxetan-3-yl)pyrrolidin-3-yl)-1H-indazol-5-amine
Show/Hide
|
C24H25ClN6O2
|
1
|
| 1 |
IC50 = 11400 nM
|
|
|
|
CP0955675
|
(R)-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
Show/Hide
|
C15H18N6
|
1
|
| 1 |
IC50 = 20700 nM
|
|
|
|
CP0966819
|
(R)-6-chloro-3-(1-methyl-1H-pyrazol-4-yl)-N-(1-(oxetan-3-yl)pyrrolidin-3-yl)-1H-indazol-5-amine
Show/Hide
|
C18H21ClN6O
|
1
|
| 1 |
IC50 = 24700 nM
|
|
|
|
CP0955677
|
(R)-6-chloro-N-(1-cyclobutylpyrrolidin-3-yl)-3-(1-(trifluoromethyl)-1H-pyrazol-4-yl)-1H-indazol-5-amine
Show/Hide
|
C18H18ClF3N6O
|
1
|
| 1 |
IC50 = 26300 nM
|
|
|
|
CP0958808
|
(S)-3-(1-methyl-1H-pyrazol-4-yl)-N-(pyrrolidin-3-yl)-1H-indazol-5-amine
Show/Hide
|
C15H18N6
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
