| Compound ID |
Compound Name |
Compound Formula |
|
CP0131851
|
1-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]-3-[6-(triazol-2-yl)-5-(trifluoromethyl)pyridin-3-yl]urea
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|
C18H15ClF3N9O2
|
1
|
| 1 |
IC50 = 0.023 nM
|
|
|
|
CP0190644
|
1-[2-chloro-7-(1-cyclopropyl-2-methoxyethyl)pyrazolo[1,5-a]pyrimidin-6-yl]-3-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]urea
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|
C20H19Cl2N9O2
|
1
|
| 1 |
IC50 = 0.028 nM
|
|
|
|
CP0158299
|
1-[7-[(1S)-1-methoxyethyl]-2-methylpyrazolo[1,5-a]pyrimidin-6-yl]-3-[5-(trifluoromethyl)pyridin-3-yl]urea
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|
C17H17F3N6O2
|
1
|
| 1 |
IC50 = 0.052 nM
|
|
|
|
CP0351408
|
1-[2-chloro-7-(oxolan-2-yl)pyrazolo[1,5-a]pyrimidin-6-yl]-3-[6-(triazol-2-yl)-5-(trifluoromethyl)pyridin-3-yl]urea
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|
C19H15ClF3N9O2
|
1
|
| 1 |
IC50 = 0.094 nM
|
|
|
|
CP0509410
|
1-[4-[4-(aminomethyl)pyrazol-1-yl]-3-chlorophenyl]-3-(2-chloro-7-propan-2-ylpyrazolo[1,5-a]pyrimidin-6-yl)urea
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|
C20H20Cl2N8O
|
1
|
| 1 |
IC50 = 0.134 nM
|
|
|
|
CP0199102
|
1-(2-chloro-7-propan-2-ylpyrazolo[1,5-a]pyrimidin-6-yl)-3-[6-(1,1-dioxo-1,2-thiazolidin-2-yl)-5-(trifluoromethyl)pyridin-3-yl]urea
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|
C19H19ClF3N7O3S
|
1
|
| 1 |
IC50 = 0.248 nM
|
|
|
|
CP0431592
|
1-(3-bromopyridin-2-yl)-N-(3-chloro-4-methoxyphenyl)-2-methylpiperidine-4-carboxamide
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|
C19H21BrClN3O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0074453
|
1-(3-chloropyridin-2-yl)-N-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]piperidine-4-carboxamide
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|
C18H17Cl2N7O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0402090
|
(2R,4R)-1-(3-bromopyridin-2-yl)-N-(3-chloro-4-methoxyphenyl)-2-methylpiperidine-4-carboxamide
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|
C19H21BrClN3O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0402170
|
N-(3-chloro-4-methoxyphenyl)-2-methyl-1-(3-methylpyridin-2-yl)piperidine-4-carboxamide
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|
C20H24ClN3O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0536081
|
1-(3-aminopyridin-2-yl)-N-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]piperidine-4-carboxamide
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|
C18H19ClN8O
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0258300
|
1-[2-chloro-7-[(3S,5S)-3,5-dimethylmorpholin-4-yl]pyrazolo[1,5-a]pyrimidin-6-yl]-3-[2-(trifluoromethyl)pyridin-4-yl]urea
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|
C19H19ClF3N7O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0382831
|
N-(3-chloro-4-methoxyphenyl)-1-(3-methylpyridin-2-yl)piperidine-4-carboxamide
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|
C19H22ClN3O2
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
|
CP0431590
|
N-(3-chloro-4-methoxyphenyl)-1-thieno[3,2-c]pyridin-4-ylpiperidine-4-carboxamide
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|
C20H20ClN3O2S
|
1
|
| 1 |
IC50 = 2340 nM
|
|
|
