Brief Information of the Compound and Protein
Compound Name
2-[[(1R)-1-[4-[5-chloro-2-(5-oxo-4H-1,2,4-oxadiazol-3-yl)phenyl]phenyl]ethyl]-(cyclopropylmethyl)amino]-N-ethylsulfonyl-5-methyl-1,3-thiazole-4-carboxamide
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PubChem ID
CID: 168280867
Canonical SMILES
CCS(=O)(=O)NC(=O)c1nc(sc1C)N(CC1CC1)[C@H](C)c1ccc(cc1)-c1cc(Cl)ccc1-c1nc(=O)o[nH]1
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Compound Formula C27H28ClN5O5S2
Compound Structure
Protein Name
Chemerin-like receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Chemokine receptor-like
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Chemerin receptor
Uniprot ID
Q99788
Gene Name
CMKLR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000681 CAL-1 [Human melanoma] Homo sapiens (Human)  1
1
EC50 = 400 nM
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