Brief Information of the Compound and Protein
Compound Name
N-[[(2R)-6-[dideuterio(tetrahydropyran-4-yl)methyl]-6-azaspiro[2.5]octan-2-yl]methyl]-6-(2,3,5-trifluorophenyl)pyridazin-3-amine
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PubChem ID
CID: 168296352
Canonical SMILES
[2H]C([2H])(C1CCOCC1)N1CCC2(CC1)C[C@H]2CNc1ccc(-c2cc(F)cc(F)c2F)nn1
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Compound Formula C24H29F3N4O
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08172
Gene Name
CHRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3000 nM
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