Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[4-[(6-chloro-5-ethoxyindazol-2-yl)methyl]-1-oxophthalazin-2-yl]acetic acid
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 PubChem ID
CID: 150893832
Canonical SMILES
CCOc1cc2cn(Cc3nn(CC(O)=O)c(=O)c4ccccc34)nc2cc1Cl
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Compound Formula C20H17ClN4O4
Compound Structure
Protein Name
 Protein Info 
Sphingosine 1-phosphate receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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EDG receptor
Uniprot ID
O95136
Gene Name
S1PR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 113 nM
   TI
   LI
   LO
   TS
2
IC50 = 149 nM
   TI
   LI
   LO
   TS
CL000673 HFL1
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 23 nM
   TI
   LI
   LO
   TS
2
IC50 = 1620 nM
   TI
   LI
   LO
   TS