Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(2-(1H-indol-3-yl)-N-methylacetamido)-N-(4-isopropylphenyl)-2-phenylacetamide
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 PubChem ID
CID: 4695397
SID: 16612379
Canonical SMILES
CC(C)c1ccc(NC(=O)C(c2ccccc2)N(C)C(=O)Cc2c[nH]c3ccccc23)cc1
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Compound Formula C28H29N3O2
Compound Structure
Protein Name
 Protein Info 
Cystic fibrosis transmembrane conductance regulator
Protein Classification
Ion channel
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Other ion channel
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Chloride channel
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Cystic fibrosis transmembrane conductance regulator
Uniprot ID
P13569
Gene Name
CFTR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
EC50 = 390 nM
   TI
   LI
   LO
   TS
2
EC50 = 1250 nM
   TI
   LI
   LO
   TS
CL000259 FRT
 Cell Line Info 
Rattus norvegicus (Rat)  2
1
EC50 = 260 nM
   TI
   LI
   LO
   TS
2
EC50 = 990 nM
   TI
   LI
   LO
   TS