Brief Information of the Compound and Protein
Compound Name
N-(1H-indol-5-ylmethyl)-3-[[4-(trifluoromethyl)phenoxy]methyl]azetidine-1-carboxamide
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Canonical SMILES
FC(F)(F)c1ccc(OCC2CN(C2)C(=O)NCc2ccc3[nH]ccc3c2)cc1
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Compound Formula C21H20F3N3O2
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 4600 nM
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