Brief Information of the Compound and Protein
Compound Name
N-[2-[[cyclohexyl(2-hydroxyethyl)amino]methyl]-4-(hydroxymethyl)phenyl]-6-fluoro-8-(methylamino)-2-oxo-1H-quinoline-3-carboxamide
    Show/Hide
PubChem ID
CID: 146314041
Canonical SMILES
CNc1cc(F)cc2cc(C(=O)Nc3ccc(CO)cc3CN(CCO)C3CCCCC3)c(=O)[nH]c12
    Show/Hide
Compound Formula C27H33FN4O4
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Potassium channels
>
Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 2390 nM
   TI
   LI
   LO
   TS