Brief Information of the Compound and Protein
Compound Name
7-[4-[ethyl(methyl)amino]butoxy]-3-[4-(2-piperidin-1-ylethoxy)phenyl]chromen-4-one
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PubChem ID
CID: 155560605
Canonical SMILES
CCN(C)CCCCOc1ccc2c(c1)occ(-c1ccc(OCCN3CCCCC3)cc1)c2=O
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Compound Formula C29H38N2O4
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000043 U2OS Homo sapiens (Human)  1
1
IC50 = 270 nM
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