Brief Information of the Compound and Protein
Compound Name
4-(4-cyclopropyl-2-piperidin-4-yl-1,3-thiazol-5-yl)-N-(2-methylpyridin-4-yl)pyrimidin-2-amine
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PubChem ID
CID: 155523740
Canonical SMILES
Cc1cc(Nc2nccc(n2)-c2sc(nc2C2CC2)C2CCNCC2)ccn1
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Compound Formula C21H24N6S
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 4200 nM
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